Search results for "TRIP"

showing 10 items of 2134 documents

Voltage- and Agonist-Induced Activation of Smooth Muscle of the Human Upper Urinary Tract: Different Mechanisms

1985

Smooth muscles are such a remarkably diverse group of tissues that the difference in properties between any two of them may be as great as between a smooth muscle and a striated muscle. With this diversity it is not surprising that the ways in which different stimuli initiate contraction are also extremely varied and interesting although we still know very little about the details of the mechanisms involved. In an attempt to shed some light on the cellular contraction cycle of smooth muscle of the human upper urinary tract, this article will focus on two topics: 1. Previous findings in smooth muscle research will be summarized and discussed briefly as they are pertinent to an understanding …

AgonistTONIC CONTRACTIONContraction (grammar)Smooth musclemedicine.drug_classMuscle stripmedicineExtracellular potassiumBiologyNeurosciencePhasic contractionUpper urinary tract
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ATP and endogenous agonists inhibit evoked [3H]-noradrenaline release in rat iris via A1 and P2y-like purinoceptors.

1993

Effects of ATP, adenosine and purinoceptor antagonists on field stimulation-evoked (3 Hz, 2 min) [3H]-noradrenaline overflow were investigated in the rat isolated iris. ATP and adenosine inhibited the evoked overflow of [3H]-noradrenaline. 1,3-Dipropyl-8-cyclopentylxanthine (DPCPX) shifted the concentration-response curve of ATP to the right in a concentration-dependent manner, but with a potency (-log KB = 7.88) much lower than expected for an A1 adenosine receptor. In the continuous presence of DPCPX, the ATP-induced prejunctional inhibition was unaffected by suramin (100 mumol/l) and DIDS (4,4'-diisothiocyanatostilbene-2,2'-disulfonic acid, 50 mumol/l) but was antagonized by the P2Y-rece…

Agonistmedicine.medical_specialtyAdenosinemedicine.drug_classSuraminIrisSuraminBiologyP2 receptor44'-Diisothiocyanostilbene-22'-Disulfonic AcidIn Vitro TechniquesSynaptic Transmissionchemistry.chemical_compoundNorepinephrineAdenosine TriphosphateInternal medicinemedicinePurinergic P2 Receptor AntagonistsAnimalsRats WistarPharmacologyProtein Synthesis InhibitorsReceptors Purinergic P2TriazinesPurinergic receptorReceptors Purinergic P1General MedicineAdenosine receptorAdenosineElectric StimulationRatsEndocrinologychemistryPurinergic P1 Receptor AntagonistsDIDSXanthinesAutoreceptormedicine.drugNaunyn-Schmiedeberg's archives of pharmacology
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Evidence for the presence of P2y and P2x receptors with different functions in mouse stomach.

2005

To clarify the function of P2 receptor subtypes in mouse stomach, the motor responses to ATP, alpha,beta-methyleneATP (alpha,beta-MeATP), P2X receptor agonist, 2-methylthioATP (2-MeSATP), P2Y receptor agonist, and the effects of the desensitisation of P2X receptors with alpha,beta-MeATP and of P2Y receptors with ADPbetaS were analysed recording the endoluminal pressure from whole-organ. ATP-induced relaxation was antagonised by suramin, non-selective P2 receptor antagonist, by desensitisation of P2Y receptors with ADPbetaS, and increased by desensitisation of P2X receptors with alpha,beta-MeATP. alpha,beta-MeATP produced biphasic responses: relaxation, reduced by P2X- or P2Y desensitisation…

Agonistmedicine.medical_specialtyP2Y receptorRelaxationContraction (grammar)medicine.drug_classSuraminMuscle RelaxationTetrodotoxinP2 receptorBiologyIn Vitro TechniquesSettore BIO/09 - Fisiologiachemistry.chemical_compoundMiceAdenosine TriphosphateInternal medicinemedicineAnimalsReceptorPharmacologyContractionDose-Response Relationship DrugReceptors Purinergic P2Mouse stomachStomachAntagonistP2Y receptorThionucleotidesATPAdenosine DiphosphateMice Inbred C57BLEndocrinologychemistryP2X receptorReceptors Purinergic P2XTetrodotoxinmedicine.drugMuscle ContractionEuropean journal of pharmacology
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Suitability of 1-hexyl-3-methylimidazolium ionic liquids for the analysis of pharmaceutical formulations containing tricyclic antidepressants

2018

Abstract The reversed-phase chromatographic behaviour of six tricyclic antidepressants (amitryptiline, clomipramine, doxepin, imipramine, nortryptiline and maprotiline) was examined in this work with acetonitrile-water mobile phases, in the absence and presence of the ionic liquids 1-hexyl-3-methylimidazolium chloride and 1-hexyl-3-methylimidazolium tetrafluoroborate, which have interesting features for the separation of basic compounds, in terms of peak shape combined with reduced retention. Tricyclic antidepressants are low polarity drugs that strongly associate to the alkyl chains of conventional stationary phases. They are also positively charged in the usual working pH range (2–8) in r…

AmitriptylineDrug CompoundingIonic LiquidsNortriptyline02 engineering and technologyAntidepressive Agents Tricyclic01 natural sciencesBiochemistryChlorideAnalytical Chemistrychemistry.chemical_compoundLimit of DetectionBoratesmedicineSample preparationMaprotilineAcetonitrileAlkylchemistry.chemical_classificationChromatography Reverse-PhaseChromatography010401 analytical chemistryOrganic ChemistryImidazolesGeneral Medicine021001 nanoscience & nanotechnologyDoxepin0104 chemical scienceschemistryIonic liquidSpectrophotometry UltravioletDoxepin0210 nano-technologymedicine.drugTricyclicJournal of Chromatography A
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First experimental proof of asymmetric charge transfer in ICP-MS/MS (ICP-QQQ-MS) through isotopically enriched oxygen as cell gas

2014

The quantification of a variety of elements in the field of ICP-MS is restricted by isobaric interferences. The recent development of ICP-MS/MS (“triple quadrupole” configuration) offers a new way to solve the problem of the detection of such elements affected by interferences because the signal caused by either the analyte or the isobaric interference can be shifted to another m/z through reactions with the cell gas (oxygen, ammonia or hydrogen). This system consists of two quadrupoles (Q1 and Q2) with a collision/reaction cell in between. When using the MS/MS mode of this configuration it becomes possible to restrict the ions entering the cell to a defined m/z and therefore get a better i…

AnalyteHydrogenAnalytical chemistrychemistry.chemical_elementOxygenAnalytical ChemistryTriple quadrupole mass spectrometerIonAmmoniachemistry.chemical_compoundchemistryIsobaric processInductively coupled plasma mass spectrometrySpectroscopyJournal of Analytical Atomic Spectrometry
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Ultra high performance liquid chromatography-time-of-flight high resolution mass spectrometry in the analysis of hexabromocyclododecane diastereomers…

2014

An efficient ultra high performance liquid chromatography (UHPLC)-time-of-flight high resolution mass spectrometry (TOF-HRMS) method was elaborated for the determination of hexabromocyclododecane (HBCD) diastereomers in fish samples and compared against UHPLC-Orbitrap-HRMS and UHPLC-triple quadrupole (QqQ) tandem MS (MS/MS) techniques. The TOF-HRMS analyzer was operated at high resolution (>10000 full width at half maximum (FWHM)) with scanning the m/z range from 600 to 700, to achieve picogram quantitation limits. The effects of various operational parameters on the instrumental response were systematically investigated. Evaluation of the influence of sample clean-up procedure steps on sig…

Analytical chemistryTandem mass spectrometryOrbitrapBiochemistryMass SpectrometryAnalytical Chemistrylaw.inventionMatrix (chemical analysis)Gel permeation chromatographychemistry.chemical_compoundColumn chromatographylawTandem Mass SpectrometryAnimalsMuscle SkeletalChromatography High Pressure LiquidHexabromocyclododecaneChromatographyEelsOrganic ChemistryFishesReproducibility of ResultsGeneral MedicineRepeatabilityTriple quadrupole mass spectrometerHydrocarbons BrominatedchemistryWater Pollutants ChemicalEnvironmental MonitoringJournal of chromatography. A
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New n-type molecular semiconductor–doped insulator (MSDI) heterojunctions combining a triphenodioxazine (TPDO) and the lutetium bisphthalocyanine (Lu…

2018

International audience; Molecular semiconductor–doped insulator (MSDI) heterojunctions were designed using a new family of sublayers, namely triphenodioxazines (TPDO). The device obtained by combining the tetracyano triphenodioxazine bearing two triisopropylsilylethynyl moieties as a sublayer with the lutetium bisphthalocyanine (LuPc2) as a top layer showed a nonlinear current–voltage characteristic independent of the sign of the polarization, which is the signature of MSDI heterojunctions. Thus, a TPDO was used in a chemical sensor for the first time. Despite LuPc2 being the only material exposed to the atmosphere, the positive response of the device under ammonia revealed the key role pla…

Analytical chemistrychemistry.chemical_element02 engineering and technology010402 general chemistryConductometric transducer01 natural sciencesAmmoniachemistry.chemical_compoundMolecular semiconductorAmmonia[CHIM.ANAL]Chemical Sciences/Analytical chemistryMaterials ChemistryTriphenodioxazineElectrical and Electronic EngineeringMolecular materialsInstrumentationChemistrybusiness.industryDopingMetals and AlloysHeterojunction021001 nanoscience & nanotechnologyCondensed Matter PhysicsLutetiumChemical sensor0104 chemical sciencesSurfaces Coatings and FilmsElectronic Optical and Magnetic Materials[SPI.TRON]Engineering Sciences [physics]/ElectronicsMolecular materialsPositive responseHeterojunctionsOptoelectronics0210 nano-technologybusiness
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Influence of metallic silver and of platinum-silver bimetallic deposits on the photocatalytic activity of titania (anatase and rutile) in organic and…

1998

Abstract The influence of deposited silver upon the photocatalytic activity of titania in the rutile and anatase allotropic forms has been studied in three different reactions. The common feature found for these three reactions was an electron transfer from illuminated TiO 2 to silver particles. In the first reaction (platinum photodeposition). it has been shown that the initial presence of metallic silver orientates the localization of subsequent Pt photodeposits with, in particular, a 100% selectivity to Pt deposition on top of silver particles or agglomerates previously deposited on anatase. In the second reaction (2-propanol oxidation), Ag deposit was found beneficial for the activity o…

AnataseChemistryGeneral Chemical EngineeringGeneral Physics and Astronomychemistry.chemical_elementGeneral ChemistryPhotochemistryCatalysisMetalRutilevisual_artPhotocatalysisvisual_art.visual_art_mediumDehydrogenationPlatinumBimetallic stripJournal of Photochemistry and Photobiology A: Chemistry
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Partial photoelectrocatalytic oxidation of 3-pyridinemethanol by Pt, Au and Pd loaded TiO2 nanotubes on Ti plate

2021

Abstract The photoelectrocatalytic (PEC) oxidation of 3-pyridinemethanol to 3-pyridinemethanal and vitamin B3 was investigated by using Pt, Au and Pd loaded (as single or bimetallic) nanotube structured TiO2 on Ti plate in water under UVA irradiation. Nanotube structured TiO2 on Ti plate samples were prepared as anode by anodic oxidation method in ethylene glycol solution in different times, and then they were calcined at 500 °C to be obtained in crystalline form. The anodes were loaded with noble metals by electrochemical reduction method and characterized by XRD, XPS, SEM, and photocurrent techniques. The TiO2 on the plates was in the anatase phase. The loaded metals were in metallic form…

AnataseNanotubeMaterials science02 engineering and technologyGeneral Chemistry010402 general chemistry021001 nanoscience & nanotechnologyElectrochemistry01 natural sciencesCatalysis0104 chemical scienceslaw.inventionMetalchemistry.chemical_compoundchemistrylawvisual_artvisual_art.visual_art_mediumPhotocatalysisCalcination0210 nano-technologyBimetallic stripEthylene glycolNuclear chemistry
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I CARCINOMI TRIPLO-NEGATIVI DELLA MAMMELLA: caratterizzazione morfologica e immunoistochimica della stromatogenesi tumorale, del contesto immunologic…

2021

Androgen receptortriple-negativeCarcinoma della mammellaBreast carcinomaimmune-checkpointstromatogenesi neoplasticatumor stromatogenesisSettore MED/08 - Anatomia PatologicaTNBCtriplo-negativirecettore androgenicheckpoint immunologici
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