Search results for "Terpenoid"

showing 10 items of 221 documents

Arthrinins A–D: Novel diterpenoids and further constituents from the sponge derived fungus Arthrinium sp.

2011

Bioassay-guided fractionation of a methanolic extract of the fungus Arthrinium sp., isolated from the Mediterranean sponge Geodia cydonium, afforded 10 natural products including five new diterpenoids, arthrinins A-D (1-4) and myrocin D (5). In addition, five known compounds were obtained, which included myrocin A (6), norlichexanthone (7), anomalin A (8), decarboxycitrinone (9) and 2,5-dimethyl-7-hydroxychromone (10). The structures of all isolated compounds were unambiguously elucidated based on extensive 1D and 2D NMR and HR-MS analyzes. The absolute configuration of arthrinins A-D (1-4) was established by the convenient Mosher method performed in NMR tubes and by interpretation of the R…

Vascular Endothelial Growth Factor AClinical BiochemistryPharmaceutical ScienceAntineoplastic AgentsBiochemistryMiceAscomycotaCell Line TumorNeoplasmsDrug DiscoveryAnimalsHumansMTT assayCytotoxicityProtein Kinase InhibitorsMolecular BiologyNeovascularization PathologicKinaseChemistryOrganic ChemistryTerpenoidIn vitroPoriferaEndothelial stem cellVascular endothelial growth factor ABiochemistryCell cultureMolecular MedicineDiterpenesProtein KinasesBioorganic & Medicinal Chemistry
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Cytotoxic glycosides from the roots of Weigela x “Bristol Ruby”

2019

International audience; Seven oleanane-type glycosides were extracted and isolated by various chromatographic methods from the roots of Weigela x "Bristol Ruby" (1-7), six previously undescribed (1-6) and a known one (7). Their structures were assigned by spectroscopic analysis mainly 2D NMR and mass spectrometry (ESIMS). Selected triterpenoid glycosides (1-3, 6, 7) displayed a good cytotoxic activity against a mouse colon cancer cell line CT26.

WeigelaCytotoxicityPhytochemicalsOleanolic acid glycosidesMass spectrometryPlant Roots01 natural sciencesCaprifoliaceaeMiceTriterpenoidCell Line TumorDrug Discovery[SDV.IDA]Life Sciences [q-bio]/Food engineeringAnimalsCytotoxic T cellGlycosidesOleanolic AcidCytotoxicityCaprifoliaceaePharmacologychemistry.chemical_classificationChromatographyMolecular Structurebiology010405 organic chemistryGlycosideGeneral MedicineWeigela x “Bristol Ruby”biology.organism_classificationAntineoplastic Agents PhytogenicTriterpenesNMR3. Good health0104 chemical sciences010404 medicinal & biomolecular chemistrychemistryTwo-dimensional nuclear magnetic resonance spectroscopy
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Identification of bound alcohols in soil humic acids by gas chromatography-mass spectrometry

2000

International audience; Humic acids are complex, partly macromolecular, yellow-brownish substances occurring in soils, waters and sediments. In order to shed some light on their molecular structure, crop humic acids were cleaved by alkaline hydrolysis (KOH). The products were fractionated by thin layer chromatography to give mono-alcohols which were analysed as acetate derivatives by gas chromatography coupled to mass spectrometry. Linear alcohols, sterols, stanols and plant-derived triterpenoid alcohols were identified by co-injection of pure standards and by comparison with literature data. These findings imply that alcohols could have been incorporated into the humic matrix by esterifica…

[SDE] Environmental SciencescampesterolKOH hydrolysisstanols[SDV]Life Sciences [q-bio]TLCFatty alcoholBrassicasterolAlkaline hydrolysis (body disposal)chemical degradation[SDV.SA.SDS]Life Sciences [q-bio]/Agricultural sciences/Soil study010402 general chemistryMass spectrometry01 natural sciencescomplex mixtureskerogenchemistry.chemical_compoundsterolstigmasterolOrganic chemistrySpectroscopyChromatographyhuminChemistryhumic substancesamyrin010401 analytical chemistrybrassicasterolcholesterolGeneral MedicineAtomic and Molecular Physics and OpticsThin-layer chromatography0104 chemical sciences[SDV] Life Sciences [q-bio]CHIMIE ANALYTIQUEsitosteroln-alkanols[SDE]Environmental SciencesHumintriterpenoidGas chromatographyGas chromatography–mass spectrometryGC-MSfatty alcohol
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Isolation and caracterisation of saponins from three plants of Araliaceae and Dracaenaceae families and evaluation of their cytotoxic activities on t…

2010

The interest of the substances from natural origin, potentially antitumor led us to interest in triterpenoid and steroidal saponins of plants from the African biodiversity belonging to the Araliaceae and Dracaenaceae families of plants. Indeed, of the former studies undertaken on some plants of these two families led to obtaining complex and original molecules having excellent cytotoxic, immuno-modulating, anti-inflammatory properties. Within sight of these results we undertook pharmaco-chemical investigations on Cussonia arborea (Araliaceae), Dracaena deisteliana, and Dracaena arborea (Dracaenaceae), medicinal plants usually used in african traditional pharmacopeia to treat various disease…

[SDV.SA] Life Sciences [q-bio]/Agricultural sciences[ SDV.BV ] Life Sciences [q-bio]/Vegetal Biology[SDV.MHEP] Life Sciences [q-bio]/Human health and pathologyCytotoxicityCussonia arboreaDracaena arboreaDracaena deistelianaTriterpenoid saponinsDracaenaceaeSaponines triterpéniquesSaponines stéroïdiquesCytotoxicité[ SDV.MHEP ] Life Sciences [q-bio]/Human health and pathology[SDV.BV] Life Sciences [q-bio]/Vegetal BiologyAraliaceae[ SDV.SA ] Life Sciences [q-bio]/Agricultural sciencesSteroidal saponins
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Pyrolysis-gas chromatography : mass spectrometry analysis of di- and triterpenoids

2017

The objective of this work was to study a specific class of extractives existing in lignocellulosic biomass and more precisely in wood materials, and their thermochemical behavior during pyrolysis. The focus was centered on the class of terpenes and terpenoids; specifically two model compounds, abietic acid and betulinol, were chosen to represent the subclasses of di- and triterpenoids, respectively. The model compounds were investigated via pyrolysis-gas chromatography/mass spectrometry (Py-GC/MS) and the main objective was to study their product profiles and characteristic fragmentations, as well as the influence of specific variables (pyrolysis temperature and time) on pyrolysis products…

abietic acidterpeenitterpenoidsbetulinolkuivatislausPy-GC/MSpyrolysistriterpeenit
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Composition and antimicrobial activity of the essential oil of Achillea falcata L. (Asteraceae).

2005

The composition of the essential oil from aerial parts of Achillea falcata L. (Asteraceae) growing wild in Lebanon was analysed by GC and GC–MS; 58 compounds, representing 94.4% of the oil, were identified. Isomers of the cyclobutane ethanol, 1-methyl-2-(1-methylethenyl), grandisol (21.4%) and fragranol (16.8%) were the main components of the oil. Also abundant were artemisia ketone (5.2%), terpinen-4-ol (4.5%) and 1,8-cineole (4.0%). The essential oil shows inhibitory activity mainly against Gram-positive bacteria.

antimicrobial activityGrandisolbiologyAchilleaMonoterpeneAchillea falcataGeneral ChemistrySettore CHIM/06 - Chimica OrganicaAsteraceaeAsteraceaebiology.organism_classificationSesquiterpenegrandisolTerpenoidessential oillaw.inventionfragranolchemistry.chemical_compoundchemistrylawBotanyEssential oilFood ScienceAntibacterial agent
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Secondary metabolites of the lichen-associated fungus Apiospora montagnei

2017

Abstract The endolichenic fungus Apiospora montagnei isolated from the lichen Cladonia sp. was cultured on solid rice medium, yielding the new diterpenoid libertellenone L (1), the new pyridine alkaloid, 23-O-acetyl-N-hydroxyapiosporamide (2) and the new xanthone derivative 8-hydroxy-3-hydroxymethyl-9-oxo-9H-xanthene-1-carboxylic acid methyl ether (3) together with 19 known compounds (4–22). The structures of the new compounds were elucidated by 1D and 2D NMR spectra as well as by HRESIMS data. The absolute configuration of the new 6,7-seco-libertellenone derivative 1 was determined by single-crystal X-ray diffraction. Four additional known compounds 23–26 were isolated when NaCl or NH4Cl w…

biology010405 organic chemistryStereochemistryAlkaloidOrganic ChemistryAbsolute configurationEtherbiology.organism_classification01 natural sciencesBiochemistryTerpenoid0104 chemical sciences010404 medicinal & biomolecular chemistrychemistry.chemical_compoundchemistryDrug DiscoveryXanthoneOrganic chemistryApiosporaTwo-dimensional nuclear magnetic resonance spectroscopyDerivative (chemistry)Tetrahedron Letters
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Triterpenoid saponins from Polycarpaea corymbosa Lamk. var. eriantha Hochst.

2013

Abstract Four triterpenoid saponins (1–4) were isolated from Polycarpaea corymbosa Lamk. var. eriantha Hochst along with the known apoanagallosaponin IV (5). Their structures were elucidated by spectroscopic data analysis. Among the compounds 1, 3–5 which were evaluated for their cytotoxicity against three tumor cell lines (SW480, DU145 and EMT6), compound 1 exhibited cytotoxicity with IC50 values ranging from 4.61 to 22.61 μM, which was greater than that of etoposide. Compound 2 was tested only against SW480 and a cardiomyoblast cell line (H9c2), and was inactive.

biologyChemistryCaryophyllaceaeTumor cellsCaryophyllaceaePlant ScienceGeneral MedicineHorticultureSaponinsbiology.organism_classificationBiochemistryAntineoplastic Agents PhytogenicTriterpenesInhibitory Concentration 50TriterpenoidDU145Cell Line TumorPolycarpaea corymbosaBotanyIc50 valuesHumansCytotoxicityMolecular BiologyPhytochemistry
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Norisoprenoids from Centaurea aspera and C. salmantica

1993

Abstract From aerial parts of Centaurea aspera var. subinermis a new homoderivative of the grasshopper ketone has been isolated. Its structure was deter

biologyChemistryPlant ScienceGeneral MedicineHorticulturebiology.organism_classificationNorisoprenoidsBiochemistryTerpenoidGrasshopper ketoneCentaureaCentaurea asperaBotanySpectral analysisDehydrovomifoliolMolecular BiologyPhytochemistry
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Terpenoid composition and chemotaxonomic aspects of Miocene amber from the Koroglu Mountains, Turkey

2014

Abstract A recently discovered fossil resin from Koroglu Mountain in Turkey has been analyzed by gas chromatography–mass spectrometry and pyrolysis gas chromatography–mass spectrometry to determine its structural class and botanical origin. The sesqui- and diterpenoids contained in the amber extract were used as chemosystematic markers when compared with terpenoids in extant conifers. The pyrolysis products were dominated by labdanoid derived bicyclic products together with succinic acid indicating Class Ia type amber. The biomarker compositions of the resin comprise mainly sesqui- and diterpenoids, and lack triterpenoids. This distribution suggests a gymnosperm, and more specifically a con…

biologyCupressaceaebiology.organism_classificationTerpenoidAnalytical Chemistrychemistry.chemical_compoundFuel TechnologyGymnospermBiomarker (petroleum)chemistryChemotaxonomySuccinic acidPinaceaeBotanyAbietaneJournal of Analytical and Applied Pyrolysis
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