Search results for "choline"

showing 10 items of 1138 documents

Robust Conditional Independence maps of single-voxel Magnetic Resonance Spectra to elucidate associations between brain tumours and metabolites.

2020

The aim of the paper is two-fold. First, we show that structure finding with the PC algorithm can be inherently unstable and requires further operational constraints in order to consistently obtain models that are faithful to the data. We propose a methodology to stabilise the structure finding process, minimising both false positive and false negative error rates. This is demonstrated with synthetic data. Second, to apply the proposed structure finding methodology to a data set comprising single-voxel Magnetic Resonance Spectra of normal brain and three classes of brain tumours, to elucidate the associations between brain tumour types and a range of observed metabolites that are known to b…

False discovery rateB VitaminsMagnetic Resonance SpectroscopyComputer scienceDirected Acyclic GraphsBiochemistry030218 nuclear medicine & medical imaging0302 clinical medicineMetabolitesMedicine and Health SciencesAmino AcidsQANeurological Tumors0303 health sciencesMultidisciplinaryDirected GraphsOrganic CompoundsBrain NeoplasmsQRTotal Cell CountingBrainMutual informationVitaminsLipidsChemistryConditional independenceOncologyNeurologyPhysical SciencesEngineering and TechnologyMedicineMeningiomaAlgorithmManagement EngineeringAlgorithmsResearch ArticleComputer and Information SciencesScienceCell Enumeration TechniquesGlycineFeature selectionCholinesResearch and Analysis MethodsSynthetic data03 medical and health sciencesInsuranceRobustness (computer science)HumansMetabolomics030304 developmental biologyRisk ManagementOrganic ChemistryChemical CompoundsBayesian networkBiology and Life SciencesCancers and NeoplasmsProteinsBayes TheoremDirected acyclic graphR1MetabolismAliphatic Amino AcidsGraph TheoryMathematicsPLoS ONE
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Liver fatty acid composition in the spontaneously diabetic BB rat.

1991

The purpose of the present experiment was to investigate if the modulation by insulin of liver microsomal desaturase activities in the spontaneously diabetic adult male Bio-Breeding (BB) rat, with destructive insulitis resembling the lesions described in the human Type I (insulin-dependent) diabetes, corresponds to modifications in fatty acid composition, reflect of changes in fatty acid desaturation. We observed no significant differences between BB rats, during the hyper-(48 h), the normo-(17 h) and the hypo-glycemic (3 h) periods which followed the insulin injection, and control rats for the fatty acid composition of liver total lipids, phosphatidylethanolamines, phosphatidylcholines, tr…

Fatty Acid DesaturasesMalemedicine.medical_specialtymedicine.medical_treatmentLinoleic acidArachidonic AcidsBiologyDiabetes Mellitus ExperimentalLinoleic Acidchemistry.chemical_compoundDiabetes mellitusInternal medicinemedicineAnimalsInsulinRats Inbred BBTriglycerideschemistry.chemical_classificationArachidonic AcidCholesterolInsulinPhosphatidylethanolaminesFatty AcidsFatty acidGeneral Medicinemedicine.diseaseLipid MetabolismRatsEndocrinologychemistryLinoleic AcidsLiverMicrosomeMicrosomes LiverPhosphatidylcholinesArachidonic acidCholesterol EstersInsulitisArchives internationales de physiologie, de biochimie et de biophysique
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Shape transitions of giant liposomes induced by an anisotropic spontaneous curvature

2000

International audience; We explore how a magnetic field breaks the symmetry of an initially spherical giant liposome filled with a magnetic colloid. The condition of rotational symmetry along the field axis leads either to a prolate or to an oblate ellipsoid. We demonstrate that an electrostatic interaction between the nanoparticles and the membrane triggers the shape transition. PACS numbers: 75.

Field (physics)Static ElectricityRotational symmetryFOS: Physical sciencesNanoparticle02 engineering and technologyCondensed Matter - Soft Condensed Matter[CHIM.INOR]Chemical Sciences/Inorganic chemistryCurvatureFerric Compounds01 natural sciencesMagneticsColloid0103 physical sciencesColloids010306 general physicsAnisotropyDebye lengthPhysicsCondensed matter physicsOsmolar Concentration[CHIM.MATE]Chemical Sciences/Material chemistryModels Theoretical021001 nanoscience & nanotechnologyGiant liposomesSymmetry (physics)Magnetic field[CHIM.POLY]Chemical Sciences/PolymersClassical mechanicsLiposomesMagnetic nanoparticlesPhosphatidylcholinesSoft Condensed Matter (cond-mat.soft)AnisotropySpontaneous curvature0210 nano-technology[PHYS.COND.CM-SCM]Physics [physics]/Condensed Matter [cond-mat]/Soft Condensed Matter [cond-mat.soft]Physical Review E
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The role of metallothionein and selenium in metal detoxification in the liver of deep-sea fish from the NW Mediterranean Sea

2014

8 pages, 1 figure, 5 tables

Fish ProteinsMaleEnvironmental Engineeringchemistry.chemical_elementMetal toxicityZincBiologyMetal detoxificationMass Spectrometrychemistry.chemical_compoundSeleniumMediterranean seaMetals HeavyLactate dehydrogenaseDeep sea fishMediterranean SeaAnimalsEnvironmental ChemistryMetallothioneinMuscle SkeletalWaste Management and DisposalL-Lactate DehydrogenaseFishesPollutionMercury (element)ZincchemistryLiverSpainEnvironmental chemistryInactivation MetabolicAcetylcholinesteraseFemaleMetallothioneinDeep-sea fishBiomarkersWater Pollutants ChemicalSeleniumEnvironmental MonitoringPolarography
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Chemistry and functional properties in prevention of neurodegenerative disorders of five Cistus species essential oils.

2013

The chemical composition of Cistus creticus, Cistus salvifolius, Cistus libanotis, Cistus monspeliensis and Cistus villosus essential oils has been examined by GC and GC–MS analysis. Height-nine constituents were identified in C. salvifolius oil, sixty in C. creticus, fifty-six in C. libanotis, fifty-four in C. villosus, forty-five in C. monspeliensis. Although the five species belong to the same genus, the composition showed interesting differences. Essential oils were screened also for their potential antioxidant effects (by DPPH, ABTS, FRAP and b-carotene bleaching test) and their acetylcholinesterase (AChE) and butyrylcholinesterase (BChE) inhibitory activity, useful for prevention and …

Fish ProteinsTunisiaDPPHCistuCistus libanotisToxicologyEssential oilAntioxidantslaw.inventionchemistry.chemical_compoundNutraceuticalAntioxidant activitylawCistusBotanyOils VolatileAnimalsGC–MSSettore BIO/15 - Biologia FarmaceuticaCistus monspeliensisHorsesEssential oilNootropic AgentsABTSbiologyTraditional medicineChemistryCistusSettore CHIM/06 - Chimica OrganicaGeneral MedicineFree Radical Scavengersbiology.organism_classificationFlavoring AgentsPlant LeavesCistus creticusNeuroprotective AgentsItalyButyrylcholinesteraseDietary SupplementsElectrophorusEthnopharmacologyAcetylcholinesteraseCholinesterase inhibitory activityCholinesterase InhibitorsMedicine TraditionalGC-MSFood ScienceFood and chemical toxicology : an international journal published for the British Industrial Biological Research Association
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Improved automated synthesis of [18F]fluoroethylcholine as a radiotracer for cancer imaging.

2007

[(18)F]Fluoroethylcholine has been recently introduced as a promising (18)F-labelled analogue of [(11)C]choline which had been previously described as a tracer for metabolic cancer imaging with positron emission tomography (PET). Due to the practical advantages of using the longer-lived radioisotope (18)F (t(1/2)=110 min), offering the opportunity of a more widespread clinical application, we established a reliable, fully automated synthesis for its production using a modified, commercially available module. [(18)F]Fluoroethylcholine was prepared from N,N-dimethylaminoethanol by iodide catalyzed alkylation with 1-[(18)F]fluoro-2-tosylethane as alkylating agent, resulting in a total radioche…

Fluorine RadioisotopesClinical BiochemistryIodidePharmaceutical ScienceCancer imagingAlkylationBiochemistryChemical synthesisSensitivity and SpecificityCholineNeoplasmsDrug DiscoverymedicineMolecular BiologyChromatography High Pressure LiquidFluoroethylcholinechemistry.chemical_classificationmedicine.diagnostic_test18F-FluoroethylcholineMolecular StructureChemistryOrganic ChemistryRadiochemistryBiochemistryFully automatedPositron emission tomographyMolecular MedicineBioorganicmedicinal chemistry
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Effects of extra-fine inhaled beclomethasone/formoterol on both large and small airways in asthma

2010

Background: Airway inflammation in asthma involves both large and small airways, and the combination of inhaled corticosteroids (ICS) and long acting beta-2 agonists (LABA) is the mainstay of therapy. Available inhaled combinations differ in terms of drug delivery to the lung and the ability to reach small airways. Aim: To evaluate whether treatment with an extra-fine inhaled combination provides additional effects vs a nonextra-fine combination on airway function. Methods: After a 1- to 4-week run-in period, patients with asthma were randomized to a double blind, double dummy, 12-week treatment with either extra-fine beclomethasone/formoterol (BDP/F) 400/24 lg daily or fluticasone propiona…

Fluticasone-Salmeterol Drug CombinationInhalationClosing capacitybusiness.industryImmunologyrespiratory systemmedicine.diseaseFluticasone propionaterespiratory tract diseasesAnesthesiamedicineImmunology and AllergyMethacholineSalmeterolFormoterolbusinessAsthmamedicine.drugAllergy
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Chapter 17 Muscarinic receptors and cell signalling

1996

Publisher Summary Cells have developed signal transduction mechanisms in order to communicate with the cell exterior. Acetylcholine as an external signal is recognized by nicotinic and muscarinic receptors. This chapter presents various muscarinic receptors belonging to the superfamily of G protein-coupled receptors consisting of seven transmembrane (TM) helices tightly packed in a ring-like structure and arranged in a counter-clockwise fashion. Agonist binding leads to a conformational change of the receptor, thereby activating associated G proteins. Muscarinic stimulation of G proteins leads to the activation or inhibition of ion channels, such as K + and Ca 2+ channels, the activation of…

G proteinHeterotrimeric G proteinMuscarinic acetylcholine receptor M5Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M1BiologyG protein-gated ion channelRhodopsin-like receptorsG protein-coupled receptorCell biology
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Functional evidence for GABA as modulator of the contractility of the longitudinal muscle in mouse duodenum: Role of GABAA and GABAC receptors

2007

We investigated, in vitro, the effects of gamma-aminobutyric acid (GABA) on the spontaneous mechanical activity of the longitudinal smooth muscle in mouse duodenum. GABA induced an excitatory effect, consisting in an increase in the basal tone, which was antagonized by the GABA(A)-receptor antagonist, bicuculline, potentiated by (1,2,5,6-Tetrahydropyridin-4-yl)methylphosphinic acid hydrate (TPMPA), a GABA(C)-receptor antagonist and it was not affected by phaclofen, a GABA(B)-receptor antagonist. Muscimol, GABA(A) receptor agonist, induced a contractile effect markedly reduced by bicuculline, tetrodotoxin (TTX), hexamethonium and atropine. Cis-4-aminocrotonic acid (CACA), a specific GABA(C) …

GABA receptorsAgonistmedicine.medical_specialtyDuodenumPyridinesmedicine.drug_classIn Vitro TechniquesBicucullineInhibitory postsynaptic potentialSettore BIO/09 - FisiologiaGABAA-rho receptorGABA AntagonistsMiceGABACellular and Molecular Neurosciencechemistry.chemical_compoundPhaclofenReceptors GABAInternal medicineIntestinal motilitymedicineAnimalsDrug InteractionsGABA Agonistsgamma-Aminobutyric AcidPharmacologyDose-Response Relationship DrugMuscimolGABAA receptorCytarabineMuscle SmoothBicucullinePhosphinic AcidsMice Inbred C57BLEndocrinologyReceptors GABA-Bnervous systemchemistryMuscimolCholinergic excitatory nerveNANC inhibitory nerveHexamethoniumMouse duodenumMuscle Contractionmedicine.drugNeuropharmacology
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Neuroinflammation and acetylcholinesterase overexpression as the main targets for low doses of GABA-A receptor agonists in Alzheimer's disease rat mo…

2018

GABA-A Receptor Agonistschemistry.chemical_compoundChemistryApplied MathematicsGeneral MathematicsLow doseRat modelDiseasePharmacologyAcetylcholinesteraseNeuroinflammationProceedings for Annual Meeting of The Japanese Pharmacological Society
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