Search results for "ganglio"

showing 10 items of 362 documents

Corrigendum to: α-Conotoxins EpI and AuIB switch subtype selectivity and activity in native versus recombinant nicotinic acetylcholine receptors (FEB…

2003

Corrigendum to: K-Conotoxins EpI and AuIB switch subtype selectivity and activity in native versus recombinant nicotinic acetylcholine receptors (FEBS 27779) [FEBS Letters 554 (2003) 219^223]C Annette Nickea;1, Marek Samochockib, Marion L. Loughnana, Paramjit S. Bansala, Alfred Maelickeb, Richard J. Lewisa; aInstitute for Molecular Bioscience, University of Queensland, Brisbane, Qld. 4072, Australia bInstitute for Physiological Chemistry and Pathobiochemistry, University of Mainz, D-55099 Mainz, Germany First published online 24 December 2003

ChemistryBiophysicsSubtype selectivityCell BiologyPharmacologyBiochemistrylaw.inventionNicotinic agonistGanglion type nicotinic receptorStructural BiologylawPhysiological chemistryGeneticsRecombinant DNAAlpha-4 beta-2 nicotinic receptorMolecular BiologyAcetylcholine receptorα conotoxinFEBS Letters
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Synthesis and in vitro evaluation of galanthamine derivatives for examination of nicotinic acetylcholine receptor system

2001

ISunmrary: The syntheses and radioactive labeling of several galanthamine derivatives, 6-O-demethyl-6-O-fluoroethylgalanthamine, 10-N-demethyl-lO-Nfluoroethylgalanthamine and N-methylgalanthaminium are reported. First ill vitro evaluations were carried out to determine their properties as allosterically potentiating ligands of nicotinic receptors. N-methylgalanthaminium was found to be a promising candidate for further investigations. The most commonly applied therapeutic approach to balance nicotinic cholinergic deficits in Alzheimer’s disease (AD) patients is the administration of acetylcholinesterase inhibitors (AChE-I) although they have been proven to be of limited therapeutic value [ …

ChemistryOrganic ChemistryPharmacologyBiochemistryAnalytical ChemistryNicotinic acetylcholine receptorGanglion type nicotinic receptorNicotinic agonistBiochemistryDrug DiscoveryMuscarinic acetylcholine receptormedicineCholinergicRadiology Nuclear Medicine and imagingAlpha-4 beta-2 nicotinic receptorSpectroscopyAcetylcholineAcetylcholine receptormedicine.drugJournal of Labelled Compounds and Radiopharmaceuticals
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Determination of sialic acid and gangliosides in biological samples and dairy products: A review

2009

Gangliosides are sphingolipids containing one or more moieties of sialic acid in their structure. Both gangliosides and sialic acid are bioactive compounds related to animal physiology. Due to their biological relevance, analytical methods adapted to each type of matrix have been developed over time. The present study reviews the main methods applied to the analysis of sialic acid and gangliosides in biological samples and dairy products.

ChromatographyGangliosideChromatographySpectrum AnalysisClinical BiochemistryPharmaceutical ScienceSphingolipidN-Acetylneuraminic AcidAnalytical ChemistrySialic acidcarbohydrates (lipids)chemistry.chemical_compoundGlycolipidBiochemistrychemistryMilk productsGangliosidesDrug DiscoveryAnimalsDairy ProductsQuantitative analysis (chemistry)SpectroscopyJournal of Pharmaceutical and Biomedical Analysis
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A Measure of Concurrent Neural Firing Activity Based on Mutual Information

2021

Multiple methods have been developed in an attempt to quantify stimulus-induced neural coordination and to understand internal coordination of neuronal responses by examining the synchronization phenomena in neural discharge patterns. In this work we propose a novel approach to estimate the degree of concomitant firing between two neural units, based on a modified form of mutual information (MI) applied to a two-state representation of the firing activity. The binary profile of each single unit unfolds its discharge activity in time by decomposition into the state of neural quiescence/low activity and state of moderate firing/bursting. Then, the MI computed between the two binary streams is…

Computer scienceModels NeurologicalAction PotentialsBinary numberRetinal ganglionMeasure (mathematics)050105 experimental psychologySynchronizationSurrogate data03 medical and health sciencesBursting0302 clinical medicineComputer Simulation0501 psychology and cognitive sciencesRepresentation (mathematics)Neuronsbusiness.industryGeneral Neuroscience05 social sciencesFiring patternsPattern recognitionMutual informationCorrelationConcurrent activityMutual informationArtificial intelligencebusinessNeural synchrony030217 neurology & neurosurgerySoftwareInformation Systems
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Stimulation of the sphenopalatine ganglion in intractable cluster headache: expert consensus on patient selection and standards of care.

2014

Context and overview Chronic cluster headache (CCH) is a debilitating headache disorder with a significant impairment of the patients' lives. Within the past decade, various invasive neuromodulatory approaches have been proposed for the treatment of CCH refractory to standard preventive drug, but only very few randomized controlled studies exist in the field of neuromodulation for the treatment of drug-refractory headaches. Based on the prominent role of the cranial parasympathetic system in acute cluster headache attacks, high-frequency sphenopalatine ganglion (SPG) stimulation has been shown to abort ongoing attacks in some patients in a first small study. As preventive effects of SPG-sti…

Consensusbusiness.industryCluster headachePatient SelectionExpert consensusContext (language use)StimulationCluster HeadacheElectric Stimulation TherapyGanglia ParasympatheticStandard of CareGeneral MedicineControlled studiesmedicine.diseaseNeuromodulation (medicine)Ganglionmedicine.anatomical_structureAnesthesiamedicineHumansNeurology (clinical)Headachesmedicine.symptombusinessCephalalgia : an international journal of headache
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Biopsia selectiva del ganglio centinela en pacientes con cáncer de mama. Efecto de la quimioterapia neoadyuvante y grado de respuesta clínica y patol…

2015

El cáncer de mama es, globalmente, la neoplasia más frecuente en mujeres. En 2012 se calcularon 1.7 millones de nuevos casos en el mundo, representando el 12% de todos los cánceres y el 25% de los cánceres en mujeres. el diagnóstico y tratamiento del cáncer de mama se sustenta en un conjunto de especialistas que forman parte de equipos multidisciplinares que incluyen principalmente a oncólogos, radiólogos, médicos nucleares, patólogos y cirujanos. Durante muchos años los ganglios axilares en los niveles I/II eran extirpados de forma rutinaria, procedimiento que se asociaba con una morbilidad significativa, que incluía hasta un 20% de riesgo de linfedema, dolor y disfunción en hombro y brazo…

Cáncer de mama:CIENCIAS MÉDICAS ::Medicina del trabajo::Medicina nuclear [UNESCO]UNESCO::CIENCIAS MÉDICAS ::Medicina del trabajo::Medicina nuclearGanglio centinelaQuimioterapia neoadyuvante
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Divergent Distribution in Vascular and Avascular Mammalian Retinae Links Neuroglobin to Cellular Respiration

2005

The visual function of the vertebrate retina relies on sufficient supply with oxygen. Neuroglobin is a respiratory protein thought to play an essential role in oxygen homeostasis of neuronal cells. For further understanding of its function, we compared the distribution of neuroglobin and mitochondria in both vascular and avascular mammalian retinae. In the vascular retinae of mouse and rat, oxygen is supplied by the outer choroidal, deep retinal, and inner capillaries. We show that in this type of retina, mitochondria are concentrated in the inner segments of photoreceptor cells, the outer and the inner plexiform layers, and the ganglion cell layer. These are the same regions in which oxyge…

DNA Complementarygenetic structuresGuinea PigsMolecular Sequence DataRespiratory chainNeuroglobinNerve Tissue ProteinsMitochondrionBiologyBiochemistryRetinaMicechemistry.chemical_compoundOxygen ConsumptionOxygen homeostasismedicineAnimalsPhotoreceptor CellsTissue DistributionAmino Acid SequenceCloning MolecularMolecular BiologyGanglion cell layerMice Inbred BALB CRetinaChoroidAntibodies MonoclonalCytochromes cRetinal VesselsRetinalCell BiologyAnatomyImmunohistochemistryeye diseasesCapillariesGlobinsMitochondriaRatsCell biologyRespiratory proteinmedicine.anatomical_structurechemistryNeuroglobinsense organsSequence AlignmentJournal of Biological Chemistry
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Novel σ1 antagonists designed for tumor therapy: Structure – activity relationships of aminoethyl substituted cyclohexanes

2021

Abstract Depending on the substitution pattern and stereochemistry, 1,3-dioxanes 1 with an aminoethyl moiety in 4-position represent potent σ1 receptor antagonists. In order to increase the stability, a cyclohexane ring first replaced the acetalic 1, 3-dioxane ring of 1. A large set of aminoethyl substituted cyclohexane derivatives was prepared in a six-step synthesis. All enantiomers and diastereomers were separated by chiral HPLC at the stage of the primary alcohol 7, and their absolute configuration was determined by CD spectroscopy. Neither the relative nor the absolute configuration had a large impact on the σ1 affinity. The highest σ1 affinity was found for cis-configured benzylamines…

DU145 tumor cellsCachannelPrimary alcohol01 natural sciencesAminoethylcyclohexanes; Antagonistic activity; Biotransformation; Ca; 2+; influx assay; Calculated free energy of binding; CD spectroscopy; Chiral HPLC; DU145 tumor cells; Inhibition of human prostate tumor cell growth; Lipophilicity; Molecular dynamics simulations; Molecular interactions; per-residue binding free energy; Selectivity; Stereochemistry; Structure affinity relationships; Voltage gated Ca; 2+; channel; σ receptors; σ; 1; receptor affinityInhibition of human prostate tumor cell growthStereochemistryDrug DiscoveryMoietySelectivityBiotransformationσ receptor0303 health sciencesChemistryAminoethylcyclohexanesCD spectroscopyAbsolute configurationAminoethylcyclohexaneMolecular interactionGeneral MedicineAntagonistic activityper-residue binding free energyreceptor affinityLipophilicityVoltage gated CaStereochemistry12+Calculated free energy of bindingRetinal ganglion03 medical and health sciencesσMolecular dynamics simulationChiral HPLCLipophilicityMolecular interactionsStructure affinity relationship030304 developmental biologyPharmacologyDU145 tumor cellinflux assayMolecular dynamics simulations010405 organic chemistryOrganic ChemistryDiastereomer0104 chemical sciencesChiral column chromatographyσ receptorsStructure affinity relationshipsEnantiomerEuropean Journal of Medicinal Chemistry
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An update to Hippocampome.org by integrating single-cell phenotypes with circuit function in vivo.

2021

Understanding brain operation demands linking basic behavioral traits to cell-type specific dynamics of different brain-wide subcircuits. This requires a system to classify the basic operational modes of neurons and circuits. Single-cell phenotyping of firing behavior during ongoing oscillations in vivo has provided a large body of evidence on entorhinal–hippocampal function, but data are dispersed and diverse. Here, we mined literature to search for information regarding the phase-timing dynamics of over 100 hippocampal/entorhinal neuron types defined in Hippocampome.org. We identified missing and unresolved pieces of knowledge (e.g., the preferred theta phase for a specific neuron type) a…

DYNAMICSGABAERGIC INTERNEURONPhysiologyAction PotentialsSocial SciencesHippocampal formationHippocampusNeuron typesBehavioral traitsMice0302 clinical medicineAnimal CellsMedicine and Health SciencesEntorhinal CortexPsychologyNETWORKBiology (General)Function (engineering)media_commonNeurons0303 health sciencesPHYSIOLOGICAL-PROPERTIESGeneral NeurosciencePyramidal CellsMethods and ResourcesBrainPhenotypeMOSSY CELLS3. Good healthElectrophysiologyPhenotypeAnatomyCellular TypesGeneral Agricultural and Biological SciencesGanglion CellsHeuristic (computer science)QH301-705.5media_common.quotation_subjectNeurophysiologyBiologyMembrane PotentialGeneral Biochemistry Genetics and Molecular Biology03 medical and health sciencesAnimalsin vivo -menetelmähippokampus030304 developmental biologyBehaviorNeuron typeGeneral Immunology and MicrobiologyGranule CellsTHETA OSCILLATIONShermoverkot (biologia)Biology and Life SciencesCell BiologyNeuronal DendritesSILICON PROBESRatshermosolutBrain stateCellular Neuroscience1182 Biochemistry cell and molecular biologyfenotyyppi3111 BiomedicineNeuroscience030217 neurology & neurosurgeryNeurosciencePLoS biology
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Agreement among 3 optical imaging methods for the assessment of optic disc topography.

2005

Purpose To assess the agreement of disc topography measurements between the Heidelberg Retina Tomograph (HRT II), Retinal Thickness Analyzer (RTA), and Optical Coherence Tomograph (StratusOCT). Design Observational cross-sectional study. Participants Forty-two randomly chosen eyes of 42 subjects. Methods Each subject underwent HRT II, RTA, and StratusOCT examination. Two experienced examiners drew the contour lines for the HRT II and RTA. Bland and Altman plots were used to evaluate agreement for each topographic parameter among the instruments. The Spearman coefficient of rank correlation was evaluated for each topographic parameter. Main Outcome Measures Agreement in the measurement of op…

Diagnostic ImagingMaleRetinal Ganglion Cellsmedicine.medical_specialtygenetic structuresOptic DiskGlaucomaSpearman's rank correlation coefficientRetinal thickness analyzerOptical imagingNerve FibersOphthalmologyLinear regressionOptic Nerve DiseasesMedicineHumansIntraocular PressureRank correlationAgedRetrospective Studiesbusiness.industryReproducibility of ResultsMiddle Agedmedicine.diseaseeye diseasesOphthalmologymedicine.anatomical_structureCross-Sectional StudiesFemalesense organsTomographybusinessGlaucoma Open-AngleOptic discOphthalmology
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