Search results for "lino"

showing 10 items of 1310 documents

Pyrrolo[2,3-h]quinolinones: A new ring system with potent photoantiproliferative activity

2006

A new class of compounds, the pyrrolo[2,3-h]quinolin-2-ones, nitrogen isosters of the angular furocoumarin Angelicin, was synthesized with the aim of obtaining new photochemotherapeutic agents with increased antiproliferative activity and lower undesired toxic effects than the lead compound. Two synthetic pathways were approached to allow the isolation both of the dihydroderivatives 10-17 and of the aromatic ring system 23. Compounds 10-17 showed a remarkable phototoxicity and a great UVA dose dependence reaching IC(50) values at submicromolar level. Intracellular localization of these compounds has been evaluated by means of fluorescence microscopy using tetramethylrhodamine methyl ester a…

Ultraviolet RaysStereochemistryFibrosarcomaClinical BiochemistryPharmaceutical ScienceHL-60 CellsAdenocarcinomaQuinolonesBiochemistryChemical synthesisMass Spectrometrychemistry.chemical_compoundAngelicinangelicinDrug DiscoverymedicineHumansMolecular BiologyChromatography High Pressure LiquidCell ProliferationFluorescent DyesPhotosensitizing AgentsRhodaminesChemistryFurocoumarinErythrocyte MembraneOrganic ChemistryAcridine orangeProteinsDNAAcridine OrangeIntercalating AgentsMitochondriapyrroloquinolinoneCross-Linking ReagentsMicroscopy FluorescencePhotochemotherapyMechanism of actionMolecular MedicineLipid Peroxidationmedicine.symptomantitumour activityLysosomesPhototoxicityLead compoundDNA DamageMacromolecule
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Thermal Induction of 9t12t Linoleic Acid: a New Pathway for the Formation of Conjugated Linoleic Acids

2009

Accepted version of an article published in the journal: International Journal of Engineering and Technology Published version available at: http://www.ijetch.org/papers/066.pdf Thermal induction of 9t12t fatty acid leading to the formation of Conjugated Linoleic Acids (CLA) has been demonstrated by subjecting glyceride, and methyl ester of the acid to heat treatment. Fifteen micro liter portions of the glyceride sample containing 9t12t fatty acid (trilinoelaidin) were placed in micro glass ampoules and sealed under nitrogen and then subjected to thermal treatment at 250oC. The glass ampoules were taken out at regular time intervals, and the contents were subjected to composition analysis b…

VDP::Mathematics and natural science: 400::Basic biosciences: 470::Biochemistry: 476chemistry.chemical_compoundChemistryLinoleic acidOrganic chemistryConjugated systemGeneralLiterature_REFERENCE(e.g.dictionariesencyclopediasglossaries)International Journal of Engineering and Technology
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Integrin-dependent and -independent functions of astrocytic fibronectin in retinal angiogenesis

2011

Fibronectin (FN) is a major component of the extracellular matrix and functions in cell adhesion, cell spreading and cell migration. In the retina, FN is transiently expressed and assembled on astrocytes (ACs), which guide sprouting tip cells and deposit a provisional matrix for sprouting angiogenesis. The precise function of FN in retinal angiogenesis is largely unknown. Using genetic tools, we show that astrocytes are the major source of cellular FN during angiogenesis in the mouse retina. Deletion of astrocytic FN reduces radial endothelial migration during vascular plexus formation in a gene dose-dependent manner. This effect correlates with reduced VEGF receptor 2 and PI3K/AKT signalli…

Vascular Endothelial Growth Factor AIntegrinsAngiogenesisIntegrinNeovascularization PhysiologicMice TransgenicExtracellular matrixMicePhosphatidylinositol 3-KinasesCell MovementAnimalsProtein Interaction Domains and MotifsMolecular BiologyResearch ArticlesMice KnockoutSprouting angiogenesisbiologyRetinal VesselsCell migrationKinase insert domain receptorVascular Endothelial Growth Factor Receptor-2Extracellular MatrixFibronectinsCell biologyMice Inbred C57BLFibronectinVascular endothelial growth factor AAstrocytesbiology.proteinHeparitin SulfateOligopeptidesProto-Oncogene Proteins c-aktIntegrin alpha5beta1Signal TransductionDevelopmental BiologyDevelopment
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Let it flow: Morpholino knockdown in zebrafish embryos reveals a pro-angiogenic effect of the metalloprotease meprin alpha2.

2010

BACKGROUND: Meprin metalloproteases are thought to be involved in basic physiological functions such as cell proliferation and tissue differentiation. However, the specific functions of these enzymes are still ambiguous, although a variety of growth factors and structural proteins have been identified as meprin substrates. The discovery of meprins alpha(1), alpha(2) and beta in teleost fish provided the basis for uncovering their physiological functions by gene silencing in vivo. METHODOLOGY/PRINCIPAL FINDINGS: A Morpholino knockdown in zebrafish embryos targeting meprin alpha(1) and beta mRNA caused defects in general tissue differentiation. But meprin alpha(2) morphants were affected more…

Vascular Endothelial Growth Factor AMorpholinoAngiogenesisMorpholinesCellular differentiationlcsh:MedicineCell Biology/Cell SignalingBiochemistry/Protein ChemistryAnimalsGene silencingCardiovascular Disorders/Vascular Biologylcsh:ScienceZebrafishZebrafishMultidisciplinarybiologyCell growthPhysiology/Cardiovascular Physiology and Circulationlcsh:RMetalloendopeptidasesMorphantCardiovascular Disorders/Cardiovascular Imagingbiology.organism_classificationMolecular biologyCell biologyVascular endothelial growth factor AGene Knockdown TechniquesAngiogenesis Inducing Agentslcsh:QResearch ArticlePLoS ONE
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Su alcune piante nuove delle Isole Pelagie

2013

On some new plants to Pelagic islands (Straits of Sicily) – Fifteen vascular plants belonging to the families Aizoaceae, Amaryllidaceae, Asteraceae, Brassicaceae, Euphorbiaceae, Myoporaceae, Orobanchaceae, Oxalidaceae, Portulacaceae and Solanaceae are reported as new to one or both the major Pelagic islands. With the exception of Narcissus serotinus and Orobanche minor, they are non-native plants, probably of recent human introduction, mostly in areas heavily modified by man. Myoporum insulare, widely used for reforestation and for ornament, occurs also in sub and semi-natural environments.

Vascular flora Lampedusa Linosa BiogeographySettore BIO/02 - Botanica SistematicaSettore BIO/03 - Botanica Ambientale E Applicata
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Phosphatidylinositol phosphate kinase type I gamma regulates dynamics of large dense-core vesicle fusion.

2005

Phosphatidylinositol-4,5-bisphosphate was proposed to be an important regulator of large dense-core vesicle exocytosis from neuroendocrine tissues. Here, we have examined the kinetics of secretion in chromaffin cells from mice lacking phosphatidylinositol phosphate kinase type Iγ, the major neuronal phosphatidylinositol-4-phosphate 5-kinase. Absence of this enzyme caused a reduction of the readily releasable vesicle pool and its refilling rate, with a small increase in morphologically docked vesicles, indicating a defect in vesicle priming. Furthermore, amperometry revealed a delay in fusion pore expansion. These results provide direct genetic evidence for a key role of phosphatidylinositol…

Vesicle fusionChromaffin CellsBiologyIn Vitro TechniquesMembrane FusionExocytosisExocytosischemistry.chemical_compoundMiceAnimalsPhosphatidylinositolCells CulturedMultidisciplinaryVesicleSecretory VesiclesSNAP25Munc-18Kiss-and-run fusionBiological SciencesSecretory VesicleCell biologyKineticsMicroscopy ElectronPhosphotransferases (Alcohol Group Acceptor)chemistryCalciumProceedings of the National Academy of Sciences of the United States of America
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Calcium-dependent conformational changes of membrane-bound Ebola fusion peptide drive vesicle fusion

2003

AbstractThe fusogenic subdomain of the Ebola virus envelope glycoprotein is an internal sequence located ca. 20 residues downstream the N-terminus of the glycoprotein transmembrane subunit. Partitioning of the Ebola fusion peptide into membranes containing phosphatidylinositol in the absence of Ca2+ stabilizes an α-helical conformation, and gives rise to vesicle efflux but not vesicle fusion. In the presence of millimolar Ca2+ the membrane-bound peptide adopts an extended β-structure, and induces inter-vesicle mixing of lipids. The peptide conformational polymorphism may be related to the flexibility of the virus–cell intermembrane fusogenic complex.

Vesicle fusionEbola glycoproteinSpectrophotometry InfraredProtein ConformationvirusesBiophysicsPeptideBiologymedicine.disease_causePhosphatidylinositolsBiochemistryMembrane FusionProtein Structure Secondarychemistry.chemical_compoundProtein structureFusion peptideMembranes (Biologia)Structural BiologyGeneticsmedicinePhosphatidylinositolMolecular Biologychemistry.chemical_classificationEbola virusVesicleCircular DichroismLipid bilayer fusionViral fusionWaterMembranes ArtificialCell BiologyEbolavirusLipidsTransmembrane proteinPeptide FragmentsBiochemistrychemistryLiposomesBiophysicsCalciumPèptidsPeptide–lipid interactionViral Fusion Proteins
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Differential involvement of mussel hemocyte sub-populations in the clearance of bacteria.

2008

Abstract Mussels are filter-feeders living in a bacteria-rich environment. We have previously found that numerous bacterial species are naturally present within the cell-free hemolymph, including several of the Vibrio genus, whereas the intra-cellular content of hemocytes was sterile. When bacteria were injected into the circulation of the mussel, the number of living intra-hemocyte bacteria dramatically increased in less than an hour, suggesting intense phagocytosis, then gradually decreased, with no viable bacteria remaining 12 h post-injection for Micrococcus lysodeikticus, 24 h for Vibrio splendidus and more than 48 h for V ibrio anguillarum. The total hemocyte count (THC) was dramatica…

Vibrio anguillarumHemocytesPhagocytosisAntimicrobial peptidesColony Count MicrobialMytiluAquatic ScienceFlow cytometryMicrobiologyMicrococcusHemolymphHemolymphHyalinocytemedicineEnvironmental ChemistryAnimalsVibrio anguillarumGram-Positive Bacterial InfectionsVibrioMytilusVibrio splendidubiologymedicine.diagnostic_testGranulocyteGeneral MedicineMusselMolluscsbiology.organism_classificationFlow CytometryMicrococcus lysodeikticuVibrioVibrio InfectionsClearanceBacteriaFishshellfish immunology
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Comparison of three activity monitors for estimating sedentary time among children

2016

Background: Time spent sedentary appears to be associated with several health outcomes in adults, but findings are inconsistent in children. Further, the assessment of sedentary time represents a major challenge. The objectives of the present study were to determine whether 1) ActiGraph GT3X+, ActivPAL and SenseWear Armband Pro3 (SWA) provide comparable estimates of sedentary time in 9–12-year-old children, 2) these devices are valid compared with direct observation, and 3) ActivPAL discriminates between sitting and standing behavior. Methods: The sample was 67 children. Data were collected during three consecutive days in November 2012. To test the activity monitors in contexts related to …

Video gamingmedicine.medical_specialtySports medicinePhysical Therapy Sports Therapy and RehabilitationIndirect calorimetryHealth outcomesSitting03 medical and health sciences0302 clinical medicinePhysical medicine and rehabilitationActivPALmedicineOrthopedics and Sports MedicineSenseWear030212 general & internal medicineSedentary timebusiness.industryRehabilitationDirect observation030229 sport sciencesActiGraphSitting timeConfidence intervalAccelerometerInclinometerPhysical therapybusinesshuman activitiesResearch Article
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Villino Basile a Palermo. La casa-studio come opera manifesto per una variabile latna della nuova cultura dell'abitare modernista

2016

Ricordata, ancora all’inizio degli anni Ottanta del XX secolo, da Giuseppe Spatrisano come “architettura dalla modernità esemplare” che negli anni Venti si imponeva ancora per la sua semplice raffinatezza, in una scena urbana oramai affetta da una variegata patologia tradizionalista, la casa-studio palermitana di Ernesto Basile non poteva però assumere in toto il ruolo di modello declinabile per l’architettura modernista siciliana. Detta anche “villino Ida” in omaggio alla consorte, la casa di Ernesto Basile, ad onta della volumetria discreta e della calligrafica strumentazione formale dal nitido tenore astilo, si distingueva rispetto alla pur elegante compagine edilizia circostante, costru…

Villino Basile Ernesto Basile abitare modernistaSettore ICAR/18 - Storia Dell'Architettura
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