Search results for "medicinal"

showing 10 items of 2966 documents

Formation of meso-1,2-Bis(dimethylamino)-1,2-diphenylethane by Oxidative C-C Coupling Reaction

2005

The title compound was obtained from the reaction of N,N-dimethylbenzylamine with n-butyl lithium and sulfur in tetrahydrofuran at room temperature. Its molecular structure was investigated by means of single crystal X-ray diffraction and quantum chemical DFT methods. The formation of meso-1,2-bis(dimethylamino)-1,2-diphenylethane is likely to be due to an unusual α-deprotonation of N,N-dimethylbenzylamine, instead of the well known ortho-lithiation, with a subsequent oxidative C-C coupling of the anions. Ab initio calculations of the corresponding α- and o-deprotonated anions of N,N-dimethylbenzylamine showed the former to be more stable than the latter, due to delocalisation of the negati…

chemistry.chemical_elementGeneral ChemistryCrystal structureRing (chemistry)Medicinal chemistrySolventchemistry.chemical_compoundchemistryAb initio quantum chemistry methodsComputational chemistryMoleculeLithiumSingle crystalTetrahydrofuranZeitschrift für Naturforschung B
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ChemInform Abstract: Polycondensed Nitrogen Heterocycles. Part 17. Isoxazolo(4,3-d)pyrazolo-(3,4-f)(1,2,3)triazepine. A New Ring System.

1988

The title compounds were prepared by nitration of compounds 2, reduction of the dinitro derivatives 4 and diazotization of the diamino derivatives 6 followed by an intramolecular coupling reaction. Compound 4a showed good activity against Salmonella cholerasuis and Clostridium perfringens bacteria.

chemistry.chemical_elementGeneral MedicineClostridium perfringensRing (chemistry)medicine.disease_causeNitrogenMedicinal chemistryCoupling reactionSalmonella cholerasuischemistry.chemical_compoundchemistryIntramolecular forceNitrationmedicineChemInform
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Base-assisted synthesis of 4-pyridinate gold(I) metallaligands: a study of their use in self-assembly reactions

2021

Made available in DSpace on 2021-06-25T12:16:58Z (GMT). No. of bitstreams: 0 Previous issue date: 2021-05-06 Ministerio de Economia y Competitividad (MINECO/FEDER) of Spain Conselho Nacional de Desenvolvimento Científico e Tecnológico (CNPq) Coordenação de Aperfeiçoamento de Pessoal de Nível Superior (CAPES) The synthesis of di- and tritopic gold(I) metallaligands of the type [(Au4-py)(2)(mu(2)-diphosphane)] (diphosphane = bis(diphenylphosphanyl)isopropane or dppip (1), 1,2-bis(diphenylphosphanyl)ethane or dppe (2), 1,3-bis(diphenylphosphanyl)propane or dppp (3) and 1,4-bis(diphenylphosphanyl)butane or dppb (4)) and [(Au4-py)(3)(mu(3)-triphosphane)] (triphosphane = 1,1,1-tris(diphenylphosph…

chemistry.chemical_elementOrNuclear magnetic resonance spectroscopyLigandsMedicinal chemistryAcceptorComplexos metàl·licsTriphosInorganic ChemistryTrigonal bipyramidal molecular geometrychemistry.chemical_compoundTriphosphaneLligandschemistryMetal complexesDiphosphaneGoldPlatinumPalladium
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Homoleptic Pnictogen-Chalcogen Coordination Complexes

2012

The synthesis and structural characterization of dicationic selenium and tellurium analogues of the carbodiphosphorane and triphosphenium families of compounds are reported. These complexes, [Ch(dppe)][OTf](2) [Ch = Se, Te; dppe = 1,2-bis(diphenylphosphino)ethane; OTf = trifluoromethanesulfonate], are formed using [Ch](2+) reagents via a ligand-exchange protocol and represent extremely rare examples of homoleptic pnictogen → chalcogen coordination complexes. The corresponding arsenic compounds were also prepared, [Ch(dpAse)][OTf](2) [Ch = Se, Te; dpAse = 1,2-bis(diphenylarsino)ethane], exhibiting the first instance of an arsenic → chalcogen dative bond. The electronic structures of these un…

chemistry.chemical_elementPhotochemistryMedicinal chemistryInorganic Chemistrychemistry.chemical_compoundChalcogenchemistryReagentPhysical and Theoretical ChemistryHomolepticTelluriumPnictogenTrifluoromethanesulfonateta116SeleniumArsenicInorganic Chemistry
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(+)-(E)-Chrysanthenyl Acetate: A Molecule with Interesting Biological Properties Contained in the Anthemis secundiramea (Asteraceae) Flowers

2020

Anthemis secundiramea is a perennial herb native widespread throughout the Mediterranean basin. The oil obtained from the flowers of this plant has antimicrobial properties against gram-positive and -negative bacteria, and inhibits the biofilm formation. The extract of A. secundiramea also has antioxidant activity&mdash

chrysanthenyl acetateAntibacterial and antioxidant activitieAntioxidantmedicine.medical_treatmentAnthemis secundiramea01 natural scienceslcsh:Technologyessential oillcsh:ChemistryNutraceuticalBotanymedicineGeneral Materials Scienceantibacterial and antioxidant activitiesInstrumentationessential oilslcsh:QH301-705.5Fluid Flow and Transfer Processes<i>Anthemis secundiramea</i>Anthemis secundirameabiology010405 organic chemistryChemistrylcsh:TProcess Chemistry and TechnologyfungiGeneral EngineeringBiofilmfood and beveragesAsteraceaeAntimicrobialbiology.organism_classificationChrysanthenyl acetatelcsh:QC1-9990104 chemical sciencesComputer Science Applications010404 medicinal & biomolecular chemistrylcsh:Biology (General)lcsh:QD1-999lcsh:TA1-2040lcsh:Engineering (General). Civil engineering (General)Bacterialcsh:PhysicsApplied Sciences
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In vivo discovery of a peptide that prevents CUG-RNA hairpin formation and reverses RNA toxicity in myotonic dystrophy models

2011

6 pages, 5 figures. PMID:21730182[PubMed] PMCID: PMC3141925[Available on 2012/1/19]

congenital hereditary and neonatal diseases and abnormalitiesProtein ConformationRNA-binding proteinProtein Serine-Threonine KinasesBiologyMyotonic dystrophyMyotonin-Protein Kinasedrug discoveryMicechemistry.chemical_compoundnon-coding RNA diseasePeptide Librarymedicinal chemistryDrug DiscoveryGene expressionmedicineAnimalsMyotonic DystrophyMBNL1MultidisciplinaryMusclesdisease modelAlternative splicingRNA-Binding ProteinsRNADystrophyBiological Sciencesmedicine.diseaseRNA secondary structureMolecular biologyDNA-Binding ProteinschemistryRNA splicingDrosophilaTrinucleotide Repeat ExpansionOligopeptides
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4-Chloronaphthalen-1-yl 4-methylbenzenesulfonate

2018

In the title compound, C17H13ClO3S, the naphthalene ring system and the benzene ring of the tosylate substituent are inclined to one another by 55.32 (5)°. The crystal structure features weak intermolecular C—H...O hydrogen bonds, one of which forms inversion dimers. Additional C—H...O hydrogen bonds and weak Cl...Cl halogen bonds stack the molecules along the b-axis direction.

crystal structure010405 organic chemistryChemistryHydrogen bondSubstituentGeneral MedicineCrystal structure010402 general chemistryRing (chemistry)01 natural sciencesMedicinal chemistryCoupling reactioncrosscoupling reactions0104 chemical scienceschemistry.chemical_compoundSulfonatecross-coupling reactionsHalogenlcsh:QD901-999lcsh:CrystallographyPhysics::Chemical PhysicsBenzenetosylatesIUCrData
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Catena-poly[[di-n-butyltin(IV)]-mu-trifluoromethanesulfonato-[[di-n-butyl(trifluoromethanesulfonato)tin(IV)]-di-mu-hydroxo]]

2006

International audience

crystal structure010405 organic chemistryChemistrycatena complexGeneral Chemistry[CHIM.INOR]Chemical Sciences/Inorganic chemistry010402 general chemistryCondensed Matter Physics01 natural sciencesMedicinal chemistry0104 chemical sciences3. Good healthtinGeneral Materials ScienceComputingMilieux_MISCELLANEOUS
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3,5-Dimethoxyphenyl 4-methylbenzenesulfonate

2017

Molecules of the title compound, C15H16O5S, are composed of a 3,5-dimethoxyphenyl moiety substituted with a toluene-4-sulfonate group. The dihedral angle between two aromatic rings is 57.23 (4)°. In the crystal, molecules are connected by weak C—H...O hydrogen bonds and S...O van der Waals interactions.

crystal structure010405 organic chemistryHydrogen bondStereochemistryChemistryAromaticityCrystal structuretosyl­atesDihedral angle010403 inorganic & nuclear chemistry01 natural sciencesMedicinal chemistryCoupling reaction0104 chemical sciencessymbols.namesakechemistry.chemical_compoundSulfonatecross-coupling reactionssymbolsMoietyvan der Waals forceIUCrData
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catena-Poly[[diaquabis[1,4-bis(pyridin-4-yl)buta-1,3-diyne-κN]iron(II)]-μ-cyanido-κ2N:C-[dicyanido-κ2C-platinum(II)]-μ-cyanido-κ2C:N]

2017

The molecular structure of the title compound, [FePt(CN)4(C14H8N2)2(H2O)2]n, consists of one-dimensional polymeric [–Fe–NC–Pt(CN)2–CN–]∞chains. Two water molecules and two monodentate 1,4-bis(pyridin-4-yl)buta-1,3-diyne (bpb) ligand molecules complete the octahedral coordination sphere of the FeIIatoms. The Fe—N(py) bond length (py is pyridine) is 2.2700 (15) Å, Fe—N(cyanide) is 2.1185 (16) Å and the Fe—O distance is 2.1275 (14) Å. The water molecules are hydrogen bonded to either bpb ligands or cyanide groups of the planar [Pt(CN)4]2−anion of adjacent polymeric chains. These O—H...N hydrogen bonds, in conjunction with offset and tilted π–π stacking interactions between bpb ligands and cyan…

crystal structureCoordination sphereDenticityLigandHydrogen bondStereochemistryCyanideCrystal structurebitopic bpb ligandhydrogen bonding010402 general chemistry010403 inorganic & nuclear chemistry01 natural sciencesMedicinal chemistry0104 chemical sciencesBond lengthchemistry.chemical_compoundchemistryπ–π stacking interactionsPyridinelcsh:QD901-999lcsh:CrystallographyIUCrData
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