Search results for "mrm"

showing 6 items of 6 documents

Antiepileptogenic Effect of Subchronic Palmitoylethanolamide Treatment in a Mouse Model of Acute Epilepsy

2018

Research on the antiepileptic effects of (endo-)cannabinoids has remarkably progressed in the years following the discovery of fundamental role of the endocannabinoid (eCB) system in controlling neural excitability. Moreover, an increasing number of well-documented cases of epilepsy patients exhibiting multi-drug resistance report beneficial effects of cannabis use. Pre-clinical and clinical research has increasingly focused on the antiepileptic effectiveness of exogenous administration of cannabinoids and/or pharmacologically induced increase of eCBs such as anandamide (also known as arachidonoylethanolamide [AEA]). Concomitant research has uncovered the contribution of neuroinflammatory p…

0301 basic medicinemedicine.medical_treatmentFAAH inhibitorsPharmacologyeicosanoidslcsh:RC321-57103 medical and health scienceschemistry.chemical_compoundEpilepsyCellular and Molecular Neuroscience0302 clinical medicineFatty acid amide hydrolaseMedicineantiepileptic drugsPentylenetetrazolendocannabinoidsMolecular Biologypalmitoylethanolamidelcsh:Neurosciences. Biological psychiatry. NeuropsychiatryOriginal ResearchPalmitoylethanolamidebusiness.industryAnandamidemedicine.diseaseEndocannabinoid system030104 developmental biologyAnticonvulsantchemistryLC-MRMSystemic administrationlipidomicsepilepsybusiness030217 neurology & neurosurgerymedicine.drugNeuroscienceFrontiers in Molecular Neuroscience
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In vitro evaluation of poloxamer in situ forming gels for bedaquiline fumarate salt and pharmacokinetics following intramuscular injection in rats

2019

Graphical abstract

In situPO Propylene oxideIV IntravenousP338 Poloxamer 338lcsh:RS1-441Pharmaceutical Sciencechemistry.chemical_compoundn Sample sizeSD Standard deviationIM Intramuscularchemistry.chemical_classificationC0 Analyte plasma concentration at time zeroDoE Design of experimentsUV UltravioletPharmacology. TherapyK2.EDTA Potassium ethylenediaminetetraacetic acidLC–MS/MS Liquid chromatography-tandem mass spectrometryH&E Hematoxylin and eosintmax Sampling time to reach the maximum observed analyte plasma concentrationIn situ forming gelsCMC Critical micellar concentrationCmax Maximum observed analyte plasma concentrationIntramuscular injectionDN Dose normalizedGPT Gel point temperaturePLGA Poly-(DL-lactic-co-glycolic acid)TFA Trifluoroacetic acidCAN AcetonitrileATP Adenosine 5′ triphosphateSalt (chemistry)Polyethylene glycolPoloxamerArticlelcsh:Pharmacy and materia medicaPharmacokineticsIn vivoUHPLC Ultra-high performance liquid chromatographyPharmacokineticsAUClast Area under the analyte concentration versus time curve from time zero to the time of the last measurable (non-below quantification level) concentrationEO Ethylene oxideNMP N-methyl-2-pyrrolidoneComputingMethodologies_COMPUTERGRAPHICSAUC∞ Area under the analyte concentration vs time curve from time zero to infinite timeP407 Poloxamer 407In vitro releasePoloxamerCMT Critical micellar temperatureGel erosionIn vitrot1/2 Apparent terminal elimination half-lifechemistryMDR-TB Multi-drug resistant tuberculosisAUC80h Area under the analyte concentration versus time curve from time zero to 80 htlast Sampling time until the last measurable (non-below quantification level) analyte plasma concentrationMRM Multiple reaction monitoringNuclear chemistrySustained releaseInternational Journal of Pharmaceutics: X
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Lipidomic profiling identifies signatures of metabolic risk

2020

Background: Metabolic syndrome (MetS), the clustering of metabolic risk factors, is associated with cardiovascular disease risk. We sought to determine if dysregulation of the lipidome may contribute to metabolic risk factors. Methods: We measured 154 circulating lipid species in 658 participants from the Framingham Heart Study (FHS) using liquid chromatography-tandem mass spectrometry and tested for associations with obesity, dysglycemia, and dyslipidemia. Independent external validation was sought in three independent cohorts. Follow-up data from the FHS were used to test for lipid metabolites associated with longitudinal changes in metabolic risk factors. Results: Thirty-nine lipids were…

Male0301 basic medicineResearch paperdhSL dihydrosphingolipidBMI body mass indexlcsh:MedicineATHEROGENIC LIPOPROTEINSBioinformaticsFHS Framingham Heart StudyPC phosphatidylcholinePESA Progression of Early Subclinical Atherosclerosis0302 clinical medicineFramingham Heart StudyRisk FactorsSAFHS San Antonio Family Heart StudyLC-MS/MS liquid chromatography-tandem mass spectrometryMedicineLongitudinal StudiesMetabolic riskPLASMA SPHINGOLIPID METABOLISMPOPULATIONlcsh:R5-920education.field_of_studySPHINGOMYELINCE cholesteryl esterDysglycemiaGeneral MedicineMiddle AgedLipidomePS phosphatidylserineCardiovascular diseaseLipidsMetabolic syndrome3. Good healthCARDIOVASCULAR-DISEASE030220 oncology & carcinogenesisHEARTMetS metabolic syndromeFemaleDisease SusceptibilityLGPL lysoglycerophospholipidSL sphingolipidlcsh:Medicine (General)LPE lysophosphatidylethanolamineAdultFDR false discovery rateTAG triacylglycerolPopulationCer ceramideCVD cardiovascular diseasePE phosphatidylethanolamineDENSITY-LIPOPROTEINRisk AssessmentGeneral Biochemistry Genetics and Molecular Biology03 medical and health sciencesAnimalsHumanseducationT2DM type II diabetes mellitusAgedLPC lysophosphatidylcholineSM sphingomyelinbusiness.industryCERAMIDElcsh:RHDL-C High density lipoprotein cholesterolBiomarkerLipid Metabolismmedicine.diseaseObesitySphingolipidCross-Sectional Studies030104 developmental biologyDyslipidemiaERF Erasmus Family StudyLipidomicsMetabolic syndromeINDUCED INSULIN-RESISTANCEbusinessDAG diacylglycerolBody mass indexBiomarkersDyslipidemiaMRM multiple reaction monitoringFASTING GLUCOSE
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Detección de nuevos marcadores asociados a daño por reperfusión y fibrosis en infarto de miocardio validados histopatológicamente mediante análisis m…

2022

La resonancia magnética cardiovascular (RMC) con realce tardío es la técnica de referencia para la evaluación no invasiva del daño cardíaco después de un infarto de miocardio (IM). Sin embargo, la interpretación de estas imágenes en términos de daño tisular es aún complicado y el uso de agentes de contraste en esta técnica está contraindicado en un amplio sector de la población con insuficiencia renal crónica. La microscopía de resonancia magnética (MRM) proporciona un nivel de detalle comparable al objetivo macroscópico de la microscopía óptica. Por ello, podría ser una herramienta muy útil en la interpretación de la imagen de RMC y en la identificación de nuevos marcadores de imagen de re…

plsdapca:CIENCIAS MÉDICAS ::Patología::Patología cardiovascular [UNESCO]análisis multivariableUNESCO::CIENCIAS MÉDICAS ::Patología::Patología cardiovascular:FÍSICA::Física atómica y nuclear ::Resonancia magnética nuclear [UNESCO]fase agudareperfusióncorrelación histopatológicamicroimagenrmnUNESCO::FÍSICA::Física atómica y nuclear ::Resonancia magnética nuclearmapas paramétricosfase crónicamrmmodelo porcino de IM por hinchado de balónirminfarto de miocardio
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An Endemic Plant of the Mediterranean Area: Phytochemical Characterization of Strawberry Tree (Arbutus unedo L.) Fruits Extracts at Different Ripenin…

2022

This work focused on the extraction, quantification, and characterization of bioactive compounds of Arbutus unedo L. fruits, comparing the results obtained from the different ripening states. Extractions were performed by different methods (such as maceration extraction and ultrasonic extraction) and food grade solvents (aqueous and hydroalcoholic solvents) in each of the all ripening states (four states considered, associated with four different colors, i.e., green, yellow, orange, and red). The presence of (poly)phenols was quantified and characterized, and scavenging activity was determined by the Folin–Ciocâlteu reagent and the DPPH method, respectively. The content of bioactive compoun…

radical scavenging activitiesSettore BIO/01 - Botanica GeneraleMRM mass spectrometryNutrition and DieteticsSettore BIO/02 - Botanica SistematicaEndocrinology Diabetes and Metabolismtotal phenolic compoundsSettore BIO/03 - Botanica Ambientale E Applicataripening processArbutus unedo LFood ScienceFrontiers in Nutrition
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Latvijas zemes izmantošanas un zemes izmantošanas maiņas matricas izveidošana, izmantojot meža resursu monitoringa ģeotelpisko informāciju

2020

Zemes izmantošanas un zemes izmantošanas maiņas aprēķina matrica ir viena no svarīgākajām valsts siltumnīcefekta gāzu (SEG) inventarizācijas sastāvdaļām zemes izmantošanas, zemes izmantošanas maiņas un mežsaimniecības (ZIZIMM) sektorā, kas sniedz kopsavilkumu par izmaiņām zemes izmantošanā valstī kopš 1990. gada. Informāciju par zemes izmantošanu un zemes izmantošanas maiņu izmanto, lai aprēķinātu pārējos parametrus, kuri ir svarīgi SEG emisiju un oglekļa krājumu izmaiņu noteikšanai dzīvajā un nedzīvajā biomasā, augsnē un zemsegā, kā arī tā sniedz informāciju par pielietoto klimata pārmaiņu mazināšanas pasākumu ietekmi uz SEG emisijām. Zemes izmantošanas maiņas aprēķinus var veikt daļēji au…

ĢeogrāfijaZemes izmantošana un zemes izmantošanas maiņaMRMZemes izmantošanas matricaSEG inventarizācija
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