Search results for "pine"

showing 10 items of 2022 documents

Effects of cimetidine, atropine and prostaglandin E2 on rat mucosal erosions produced by intragastric distension

1980

Abstract The effects of three typical antisecretory agents: cimetidine, atrophine and prostaglandin E2 were compared on an acute rat gastric ulcer model which consisted of perfusing the stomach continuously, at a high intraluminal pressure (120 mm H2O), with a simulated gastric juice (0.1 M HCl plus 600 mg pepsin/1). As the acid and pepsin are given exogenously the inhibitory action of the antisecretory drugs is obviated in this model. Cimetidine and atropine failed to reduce gastric erosions, whereas prostaglandin E2 markedly reduced the severity of the mucosal lesions with respect to control values. Long-term treatment with cimetidine also failed to increase the resistance of the gastric …

AtropineMalemedicine.medical_treatmentPharmacologyGuanidinesPepsinmedicineGastric mucosaAnimalsStomach UlcerProstaglandin E2CimetidinePharmacologyGastric Juicebiologybusiness.industryProstaglandins EGastric distensionStomachdigestive oral and skin physiologyRatsDisease Models AnimalAtropinemedicine.anatomical_structureAnesthesiabiology.proteinmedicine.symptomCimetidinebusinessProstaglandin Emedicine.drugEuropean Journal of Pharmacology
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Uveal effusion syndrome complicated by anterior ischemic optic neuropathy

1995

We report on a case of idiopathic uveal effusion syndrome complicated by AION. To our knowledge such an association hasn't been previously described. We suggest that scleral thickening caused obstruction of vortex veins followed by uveal effusion and compression of posterior ciliary arteries within their intrascleral tract, leading to AION. Nevertheless it can't be excluded that AION was the result of mechanical compression on ciliary vessels of optic disc by choroidal detachment. © 1996, Kluwer Academic Publishers. All rights reserved.

AtropineMydriaticsmedicine.medical_specialtyFundus OculiAnti-Inflammatory AgentsVisual AcuityIdiopathic uveal effusion syndromeDexamethasoneOptic neuropathyPregnenedionesPhysiology (medical)Ophthalmologymedicine.arteryHumansMedicineOptic Neuropathy IschemicFluorescein Angiographymedicine.diagnostic_testbusiness.industrySettore MED/30 - Malattie Apparato VisivoCiliary BodyRetinal DetachmentChoroid DiseasesSyndromeUveal DiseasesMiddle AgedFluorescein angiographymedicine.diseaseeye diseasesSensory SystemsScleral thickeningCiliary arteriesSurgeryOphthalmologyAnterior ischemic optic neuropathymedicine.anatomical_structureEffusionOptic nerveAnterior ischemic optic neuropathyFemalesense organsOphthalmic SolutionsbusinessOptic disc
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Electrical stimulation of glossopharyngeal nerve and oesophageal EMG response in the pigeon

1985

The effects of the efferent glossopharyngeal nerve stimulation, on EMG activity of the pigeon cervical oesophagus, were studied. In control animals, stimulation caused a biphasic response characterized by an intra-stimulus excitatory component followed by a post-stimulus inhibitory one. The EMG response to glossopharyngeal stimulation appeared simultaneously throughout the cervical oesophagus. A bell-shaped mechanical wave was detected relating to the electrical excitatory component. Atropine administration antagonized the excitatory component, while the inhibitory one persisted. It occurs intra-stimulus, and its duration is increased, compared to control ones. A reduction in the oesophagea…

AtropinePhysiologyEfferentStimulationHexamethonium CompoundsElectromyographyIn Vitro TechniquesInhibitory postsynaptic potentialBiochemistrychemistry.chemical_compoundEsophagusmedicineAnimalsColumbidaeGlossopharyngeal Nervemedicine.diagnostic_testElectromyographybusiness.industryElectric Stimulationmedicine.anatomical_structurechemistryPeripheral nervous systemAnesthesiaGlossopharyngeal nerveExcitatory postsynaptic potentialHexamethoniumbusinessArchives Internationales de Physiologie et de Biochimie
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Primary peristalsis in pigeon cervical oesophagus: two EMG patterns.

1984

Swallowing elicits two propagated EMG peristaltic patterns in pigeon cervical oesophagus: i) "simple" peristaltic pattern and ii) "complex" peristaltic pattern. "Simple" peristaltic pattern is characterized by an intense, long-lasting burst of spikes, high in amplitude with an aboral increasing delay in onset. "Complex" peristaltic pattern presents an early short period of reduction in spontaneous electrical activity, followed by an excitatory period similar to that of "simple" pattern. The early inhibitory component has a very short delay in onset increasing aborally. Atropine abolishes the EMG excitatory component of both patterns, while the inhibitory period persists, showing increased d…

AtropinePhysiologyElectromyographyCholinergic NervesAnatomyBiologyInhibitory postsynaptic potentialBiochemistryElectrophysiologyCervical oesophagusEsophagusMuscarinic acetylcholine receptorExcitatory postsynaptic potentialCholinergicAnimalsPeristalsisColumbidaeGastrointestinal MotilityPeristalsisArchives internationales de physiologie et de biochimie
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Cholinesterase activity and exposure time to acetylcholine as factors influencing the muscarinic inhibition of [3H]-noradrenaline overflow from guine…

1985

Guinea-pig isolated atria were incubated and loaded with [3H]-noradrenaline. The release of 3H and of [3H]-noradrenaline was induced by field stimulation (6-9 trains of 150 pulses at 5 Hz). The stimulation-evoked overflows of 3H and of [3H]-noradrenaline were determined. In the absence of an inhibitor of acetylcholinesterase, acetylcholine (12 min preincubation before nerve stimulation, up to 10 microM) failed to inhibit the evoked [3H]-noradrenaline overflow. In the presence of atropine, an increase by acetylcholine of evoked release was observed in the same atria. In contrast, the selective muscarinic agonist methacholine significantly decreased the evoked overflow. The inhibition was ant…

AtropinePhysostigminemedicine.medical_specialtyTime FactorsPhysostigmineGuinea PigsHexamethonium CompoundsIn Vitro TechniquesHexamethoniumMuscarinic agonistNorepinephrinechemistry.chemical_compoundCocaineInternal medicineMuscarinic acetylcholine receptormedicineAnimalsMethacholine CompoundsDrug InteractionsHeart AtriaPhentolamineMethacholine ChlorideCholinesterasePharmacologybiologyHeartPropranololReceptors MuscarinicAcetylcholineAtropineEndocrinologychemistryAcetylcholinesterasebiology.proteinMethacholineHexamethoniumCorticosteroneAcetylcholineResearch Articlemedicine.drugBritish Journal of Pharmacology
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Acetylcholine via Muscarinic Receptors Inhibits Histamine Release from Human Isolated Bronchi

1997

Human bronchi were incubated in organ baths to measure histamine release. The calcium ionophore A23187 (10 mumol/L; 1 min) stimulated histamine release by 148 +/- 28% (n = 11) above the prestimulation level but was ineffective in epithelium-denuded bronchi. Neither bradykinin (0.1 mumol/L) nor compound 48/80 (10 micrograms/ml) triggered the release of histamine from epithelium-intact bronchi. Acetylcholine did not affect spontaneous histamine release (about 2 nmol/g x 5 min) but inhibited A23187-evoked histamine release in an atropine-sensitive manner. Already a concentration as low as 0.1 nmol/L acetylcholine was effective, the maximal inhibition (by 89%) occurred at 100 nmol/L, whereas a …

AtropinePulmonary and Respiratory MedicineAgonistPhysostigminemedicine.medical_specialtyTime Factorsmedicine.drug_classPhysostigmineBradykininBronchiMuscarinic AntagonistsMuscarinic AgonistsCritical Care and Intensive Care MedicineHistamine Releasechemistry.chemical_compoundCulture TechniquesInternal medicineMuscarinic acetylcholine receptormedicineOxotremorineHumansDrug InteractionsCalcimycinDose-Response Relationship DrugIonophoresbusiness.industryOxotremorineImmunoglobulin EReceptors MuscarinicAcetylcholineEndocrinologychemistryAcetylcholinesterase inhibitorDepression ChemicalCholinesterase InhibitorsbusinessAcetylcholineHistaminemedicine.drugAmerican Journal of Respiratory and Critical Care Medicine
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Release of [3H]Acetylcholine in Human Isolated Bronchi: Effect of Indomethacin on Muscarinic Autoinhibition

1995

Receptor-mediated regulation of acetylcholine release in the airways, particularly in humans, remains unclear. In the present study, the tissue content of acetylcholine and release of [3H]acetylcholine were measured in freshly dissected human bronchi obtained at thoracotomy. Large (main and lobar bronchi) and small (segmental and subsegmental bronchi) airways contained considerable amounts of endogenous acetylcholine (300 +/- 50 pmol/100 mg wet weight), whereas significantly less was found in lung parenchyma (60 +/- 30 pmol/100 mg). Isolated small bronchi incubated in an organ bath with the precursor [3H]choline synthesized significant amounts of [3H]acetylcholine (26,000 +/- 4,000 dpm/100 …

AtropinePulmonary and Respiratory Medicinemedicine.medical_specialtyIndomethacinStimulationBronchiIn Vitro TechniquesCritical Care and Intensive Care Medicinechemistry.chemical_compoundInternal medicineMuscarinic acetylcholine receptormedicineOxotremorineCholineHumansbusiness.industryOxotremorinerespiratory systemReceptors MuscarinicAcetylcholineElectric StimulationAtropineEndocrinologychemistryTetrodotoxinCholinergicbusinessAcetylcholinemedicine.drugAmerican Journal of Respiratory and Critical Care Medicine
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Electrophysiological and microiontophoretic analysis of the habenulo-hippocampal circuit.

1991

In the cat, the effects of lateral habenula stimulation, at different ranges of frequency, on hippocampal units were studied. Habenular stimulation at low frequency excited, while at high frequency inhibited the greater part of hippocampal units. Moreover, in order to clarify the possible pathway involved in the habenulo-hippocampal circuit, the effects of iontophoretic acetylcholine and serotonin on hippocampal units were compared with those of habenular stimulation. Iontophoretic acetylcholine induced both excitatory and inhibitory responses while serotonin induced only inhibitory responses. Iontophoretic atropine blocked the effects of acetylcholine ejection but did not antagonize stimul…

AtropineSerotoninMethysergideStimulationHippocampal formationInhibitory postsynaptic potentialHippocampusThalamusNeural PathwaysmedicineAnimalsNeuronsChemistryMethysergideGeneral MedicineIontophoresisAcetylcholineElectric StimulationElectrophysiologyElectrophysiologyExcitatory postsynaptic potentialCatsSerotoninNeuroscienceAcetylcholinemedicine.drugArchives internationales de physiologie, de biochimie et de biophysique
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Use of atropine-treated Daphnia magna survival for detection of environmental contamination by acetylcholinesterase inhibitors.

2003

The toxicity of cholinesterase-inhibiting compounds (e.g., carbamates and organophosphates) is due to a decrease in acetylcholine metabolism, which results in a continuous stimulation of cholinergic receptors (muscarinic and nicotinic) that can be fatal. The goal of this study was to evaluate the protective effect of atropine (muscarinic receptor antagonist) against paraoxon-induced toxicity to Daphnia magna using its survival rate for the detection of environmental contamination by cholinesterase-inhibiting compounds. As expected, paraoxon was lethal to D. magna in a concentration-dependent manner. Noteworthy, the pretreatment of these organisms with atropine dramatically increased their s…

AtropineSurvivalHealth Toxicology and MutagenesisDaphnia magnaMuscarinic AntagonistsBiologyPharmacologyParaoxonToxicologychemistry.chemical_compoundMuscarinic acetylcholine receptormedicineAnimalsreproductive and urinary physiologyParaoxonfungiPublic Health Environmental and Occupational HealthGeneral Medicinebiology.organism_classificationPollutionAcetylcholinesteraseAtropineNicotinic agonistchemistryDaphniaToxicityCholinergicCholinesterase InhibitorsBiomarkersWater Pollutants Chemicalmedicine.drugEcotoxicology and environmental safety
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Delivering Inorganic and Organic Reagents and Enzymes from Zein and Developing Optical Sensors.

2018

Nowadays, interest in using environmentally friendly materials is increasing in many fields. However, the rational design of sensors with biodegradable materials is a challenge. The main aim of this work is to show the possibility of using zein, a protein from corn, as a biodegradable and low-cost material for immobilizing, stabilizing, and delivering different kind of reagents for developing optical sensors. Enzymes, metallic salts, and aromatic and small organic compounds were tested. In addition, different techniques of immobilization, entrapment and adsorption, were used, and different formats, such as solid devices and also multiwell platforms, were proposed. The capacity of zein for i…

AtropineZein02 engineering and technologyBiosensing Techniques01 natural sciencesZea maysAnalytical ChemistryPhosphatesAdsorptionHumanschemistry.chemical_classificationFerric hydroxamateChemistry010401 analytical chemistryRational designA proteinSubstrate (chemistry)021001 nanoscience & nanotechnologyEnzymes ImmobilizedCombinatorial chemistryEnvironmentally friendly0104 chemical sciencesEnzymeSpectrometry FluorescencePharmaceutical PreparationsReagentColorimetryIndicators and Reagents0210 nano-technologyAnalytical chemistry
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