Search results for "porter"

showing 10 items of 920 documents

Evidence of oxidative stress in very long chain fatty acid--treated oligodendrocytes and potentialization of ROS production using RNA interference-di…

2011

X-linked adrenoleukodystrophy (X-ALD) and pseudo neonatal adrenoleukodystrophy (P-NALD) are neurodegenerative demyelinating diseases resulting from the functional loss of the peroxisomal ATP-binding cassette transporter D (ABCD1) and from single peroxisomal enzyme deficiency (Acyl-CoA oxidase1: ACOX1), respectively. As these proteins are involved in the catabolism of very long chain fatty acids (VLCFA: C24:0, C26:0), X-ALD and P-NALD patients are characterized by the accumulation of VLCFA in plasma and tissues. Since peroxisomes are involved in the metabolism of reactive oxygen species (ROS) and nitrogen species (RNS), we examined the impact of VLCFA on the oxidative status of 158N murine o…

congenital hereditary and neonatal diseases and abnormalitiesendocrine systemendocrine system diseasesVery long chain fatty acidBlotting Westernmedicine.disease_causeReal-Time Polymerase Chain ReactionTransfectionATP Binding Cassette Transporter Subfamily D Member 1Gas Chromatography-Mass SpectrometrySuperoxide dismutaseLipid peroxidationchemistry.chemical_compoundMicemedicinePeroxisomesAnimalsAdrenoleukodystrophyCells Culturedchemistry.chemical_classificationReactive oxygen speciesbiologyReverse Transcriptase Polymerase Chain ReactionGeneral NeuroscienceFatty Acidsnutritional and metabolic diseasesPeroxisomemedicine.diseaseFlow CytometryOligodendrogliaOxidative StressBiochemistrychemistryGene Knockdown Techniquesbiology.proteinACOX1AdrenoleukodystrophyATP-Binding Cassette TransportersRNA InterferenceAcyl-CoA OxidaseReactive Oxygen SpeciesOxidation-ReductionOxidative stressNeuroscience
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Study of the aryl hydrocarbon receptor mediated effects through in silico modeling and in vitro bioassays

2020

The aryl hydrocarbon receptor (AhR) is a cytoplasmatic sensor of diverse endogenous and exogenous substances. In a toxicological context, the former known as “dioxin receptor” has been investigated as a xenobiotic chemoreceptor and due to its roles in mediating carcinogenesis, endocrine disruption, among other immunological, hepatic, cardiovascular, and dermal toxicity mechanisms. The deep physiological implications of AhR in cellular proliferation, adhesion, division, differentiation, as well as in the reproductive, immunological and cardiovascular homeostasis have opened a new field of research in order to harness AhR’s pharmacological potential. Hence, AhR has become a therapeutic target…

endocrine disruptoraryl hydrocarbon receptorQSARUNESCO::QUÍMICAtoxicophoremolecular dockingrespiratory system:QUÍMICA [UNESCO]:CIENCIAS DE LA VIDA [UNESCO]UNESCO::CIENCIAS DE LA VIDAantimicrobialluciferase reporter gene assaytranscription factor
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L‐Aspartate as a high‐quality nitrogen source in Escherichia coli : Regulation of L‐aspartase by the nitrogen regulatory system and interaction of L‐…

2020

Escherichia coli uses the C4-dicarboxylate transporter DcuA for L-aspartate/fumarate antiport, which results in the exploitation of L-aspartate for fumarate respiration under anaerobic conditions and for nitrogen assimilation under aerobic and anaerobic conditions. L-Aspartate represents a high-quality nitrogen source for assimilation. Nitrogen assimilation from L-aspartate required DcuA, and aspartase AspA to release ammonia. Ammonia is able to provide by established pathways the complete set of intracellular precursors (ammonia, L-aspartate, L-glutamate, and L-glutamine) for synthesizing amino acids, nucleotides, and amino sugars. AspA was regulated by a central regulator of nitrogen meta…

endocrine system diseasesNitrogenGlutaminePII Nitrogen Regulatory ProteinsNitrogen assimilationDeaminationGlutamic AcidBiologymedicine.disease_causeAspartate Ammonia-LyaseMicrobiology03 medical and health sciencesBacterial ProteinsAmmoniaEscherichia colimedicineProtein Interaction Domains and MotifsNucleotideMolecular BiologyEscherichia coliNitrogen cycle030304 developmental biologyDicarboxylic Acid Transporterschemistry.chemical_classificationAspartic Acid0303 health sciences030306 microbiologyEscherichia coli ProteinsAssimilation (biology)Gene Expression Regulation BacterialAmino acidEnzymechemistryBiochemistryMutationKetoglutaric AcidsMetabolic Networks and PathwaysMolecular Microbiology
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In vitro evaluation of glycol chitosan based formulations as oral delivery systems for efflux pump inhibition.

2017

Recently, we have reported that glycol chitosan (GCS) was able to reverse the P- glycoprotein (P-gp) efflux pump. The objective of the present study was to evaluate the potential of two GCS-based dosage forms (aqueous solution or nanoparticle suspension) for oral administration of the P-gp substrate Rho-123. A further aim of the present study was to assess the effect of the glycol chitosan-4-thiobutylamidine thiomer (GCS-TBA) on P-gp activity considering that the corresponding thiomer of chitosan series is a well-known P-gp inhibitor. Pre-treatment of Caco-2 cell monolayer with a GCS solution or GCS-based nanoparticles increased the absorptive transport of Rho-123 across the monolayer of 1.…

endocrine systemATP Binding Cassette Transporter Subfamily BPolymers and Plastics02 engineering and technologyPharmacologyDosage formChitosan03 medical and health scienceschemistry.chemical_compoundGlycols0302 clinical medicineDrug Delivery SystemsOral administrationhealth services administrationpolycyclic compoundsMaterials ChemistryHumansGlycol chitosan-based formulations P-gp inhibition properties Rhodamine 123 Glycol chitosan-4-thiobutylamidine thiomer Caco-2 cells Oral bioavailabilityChitosanChemistryThiomerOrganic ChemistryGlycol chitosan-based formulations P-gp inhibition properties Rhodamine 123 Glycol chitosan-4-thiobutylamidine thiomer Caco-2 cells Oral bioavailability021001 nanoscience & nanotechnologyBioavailabilityCaco-2Settore CHIM/09 - Farmaceutico Tecnologico Applicativo030220 oncology & carcinogenesisNanoparticlessense organsEffluxCaco-2 Cells0210 nano-technologyhormones hormone substitutes and hormone antagonistsConjugateCarbohydrate polymers
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Multipotential nestin and Isl-1 positive mesenchymal stem cells isolated from human pancreatic islets.

2006

Mesenchymal cells in the developing pancreas express the neural stem cell marker nestin and the transcription factor islet-1 (Isl-1). Using defined culture conditions we isolated on a single cell basis nestin producing cells from human pancreatic islets. These cells were immortalized with lentiviral vectors coding for telomerase and mBmi. They are positive for Isl-1 and nestin and have the potential to adopt a pancreatic endocrine phenotype with expression of critical transcription factors including Ipf-1, Isl-1, Ngn-3, Pax4, Pax6, Nkx2.2, and Nkx6.1 as well as the islet hormones insulin, glucagon, and somatostatin. In addition, they can be differentiated into human albumin producing cells …

endocrine systemLIM-Homeodomain ProteinsBiophysicsCell Culture TechniquesNerve Tissue ProteinsBiologyBiochemistryNestinIslets of LangerhansIntermediate Filament ProteinsNeurosphereAlbuminsmedicineAdipocytesATP Binding Cassette Transporter Subfamily G Member 2HumansMolecular BiologyStem cell transplantation for articular cartilage repairHomeodomain ProteinsNeuronsOsteoblastsPancreatic isletsMesenchymal stem cellLentivirusNuclear ProteinsCell DifferentiationMesenchymal Stem CellsCell BiologyNestinNeural stem cellNeoplasm Proteinsmedicine.anatomical_structureHomeobox Protein Nkx-2.2Cancer researchPAX4ATP-Binding Cassette TransportersPancreasTranscription FactorsBiochemical and biophysical research communications
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Glial Chloride Homeostasis Under Transient Ischemic Stress

2021

High water permeabilities permit rapid adjustments of glial volume upon changes in external and internal osmolarity, and pathologically altered intracellular chloride concentrations ([Cl–]int) and glial cell swelling are often assumed to represent early events in ischemia, infections, or traumatic brain injury. Experimental data for glial [Cl–]int are lacking for most brain regions, under normal as well as under pathological conditions. We measured [Cl–]int in hippocampal and neocortical astrocytes and in hippocampal radial glia-like (RGL) cells in acute murine brain slices using fluorescence lifetime imaging microscopy with the chloride-sensitive dye MQAE at room temperature. We observed s…

excitatory amino acid transportersOsmotic concentrationchemical stress mimicking ischemiaChemistryDentate gyrusINTintracellular chloride concentrationsNeurosciences. Biological psychiatry. NeuropsychiatryHippocampal formationChlorideCellular and Molecular NeuroscienceNa-K-2Cl cotransporterBiophysicsmedicineddc:610K-Cl cotransportersCotransporterHomeostasisIntracellularRC321-571NeuroscienceOriginal Researchfluorescence lifetime imaging microscopymedicine.drugFrontiers in Cellular Neuroscience
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Reflecting on the PRET A Rapporter Framework Via a Field Study of Adolescents’ Perceptions of Technology and Exercise

2013

PRET A Rapporter (PRETAR) was developed to explicitly structure user-centered evaluation studies to ensure all necessary elements are individually and independently considered. Its creators see its benefit as twofold: for study design and in retrospective evaluations. We evaluate PRETAR’s potential by applying it retrospectively to one of our eHealth field studies in which we investigated the design requirements for mobile technologies that would support and motivate adolescents to exercise opportunistically. We also use PRETAR to evaluate the key literature for this eHealth study. This shows that typically the research methodology is under-reported. Then we document the study in terms of i…

field studyopportunistic exerciseadolescent participantstechnology probePRET A Rapporterreflection
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Analisi tecnica di cantieri meccanizzati nelle operazioni di utilizzazioni forestali in Sicilia

2005

The authors describe the results of a research performed in a wood of the Western Sicily, covered with Pinus halepensis Mill. and Cupressus sempervirens L. Felling, delimbing, cross-cutting and extraction of the logs were carried out. The wood obtained was used as firewood. Two different methods of logs extraction were carried out: with transporters and with polyethylene timber chutes. The working time and the labour productivity recorded during each operations are reported. The results show that in the forest utilization performed in Sicily the mean labour productivity per operator is 2.4 t of firewood per day. This value fits well the mean value recorded in Italy (2-3 t of firewood per da…

forest utilization transporters timber chutes
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Enhanced transport through binding cooperativity in a circulating system

1991

Abstract Allosteric cooperativity in a multiphase circulating system is shown to enhance ion transport when long contact times are involved.

genetic structuresChemistryOrganic ChemistryClinical BiochemistryAllosteric regulationPharmaceutical ScienceCooperativityBiochemistryBiochemistryDrug DiscoveryBiophysicsMolecular MedicineMolecular BiologyIon transporterBioorganic & Medicinal Chemistry Letters
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Interaction of glutamic-acid-rich proteins with the cGMP signalling pathway in rod photoreceptors.

1999

The assembly of signalling molecules into macromolecular complexes (transducisomes) provides specificity, sensitivity and speed in intracellular signalling pathways. Rod photoreceptors in the eye contain an unusual set of glutamic-acid-rich proteins (GARPs) of unknown function. GARPs exist as two soluble forms, GARP1 and GARP2, and as a large cytoplasmic domain (GARP' part) of the beta-subunit of the cyclic GMP-gated channel. Here we identify GARPs as multivalent proteins that interact with the key players of cGMP signalling, phosphodiesterase and guanylate cyclase, and with a retina-specific ATP-binding cassette transporter (ABCR), through four, short, repetitive sequences. In electron mic…

genetic structuresPhosphodiesterase InhibitorsMolecular Sequence DataCyclic Nucleotide-Gated Cation ChannelsGlutamic AcidNerve Tissue ProteinsPlasma protein bindingBiologyIn Vitro TechniquesRetinal Rod Photoreceptor CellsAnimalsAmino Acid SequenceTransducinEye ProteinsPeptide sequenceCyclic GMPMultidisciplinaryPhosphoric Diester HydrolasesPhosphodiesteraseProteinsTransporterGlutamic acidRod Cell Outer SegmentRecombinant ProteinsCell biologyBiochemistryCytoplasmGuanylate CyclaseATP-Binding Cassette TransportersCattleTransducinSignal transductionProtein BindingSignal TransductionNature
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