Search results for "relation"

showing 10 items of 10542 documents

Effects of Nandrolone Stimulation on Testosterone Biosynthesis in Leydig Cells

2016

Anabolic androgenic steroids (AAS) are among the drugs most used by athletes for improving physical performance, as well as for aesthetic purposes. A number of papers have showed the side effects of AAS in different organs and tissues. For example, AAS are known to suppress gonadotropin‐releasing hormone, luteinizing hormone, and follicle‐stimulating hormone. This study investigates the effects of nandrolone on testosterone biosynthesis in Leydig cells using various methods, including mass spectrometry, western blotting, confocal microscopy and quantitative real‐time PCR. The results obtained show that testosterone levels increase at a 3.9 μM concentration of nandrolone and return to the ba…

0301 basic medicineEnzymologicMalePhysiologyClinical BiochemistryAndrogenAnabolic Agents; Androgens; Animals; Cell Line; Cell Survival; Dose-Response Relationship Drug; Gene Expression Regulation Enzymologic; Leydig Cells; Male; Nandrolone; Phosphoproteins; Rats; Steroid 17-alpha-Hydroxylase; Testosterone; Physiology; Clinical Biochemistry; Cell BiologyAnabolic AgentsOriginal Research ArticlesNandroloneTestosteroneOriginal Research ArticleTestosteroneAnabolic Agents; Androgens; Animals; Cell Line; Cell Survival; Dose-Response Relationship Drug; Gene Expression Regulation Enzymologic; Leydig Cells; Male; Nandrolone; Phosphoproteins; Rats; Steroid 17-alpha-Hydroxylase; Testosterone; Clinical Biochemistry; Cell Biology; Physiology; Medicine (all)Steroidogenic acute regulatory proteinMedicine (all)Leydig CellsSteroid 17-alpha-HydroxylaseCYP17A1PhosphoproteinAndrogensDrugLuteinizing hormonemedicine.drugAnabolic Agents; Androgens; Animals; Cell Line; Cell Survival; Dose-Response Relationship Drug; Gene Expression Regulation Enzymologic; Leydig Cells; Male; Nandrolone; Phosphoproteins; Rats; Steroid 17-alpha-Hydroxylase; TestosteroneLeydig Cellendocrine systemmedicine.medical_specialtyCell SurvivalBiologyGene Expression Regulation EnzymologicCell LineDose-Response Relationship03 medical and health sciencesDownregulation and upregulationIn vivoInternal medicinemedicineAnimalsDose-Response Relationship DrugAnimalCell BiologyPhosphoproteinsRats030104 developmental biologyEndocrinologyGene Expression RegulationNandroloneAnabolic AgentRatHormone
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Lawsone derivatives target the Wnt/β-catenin signaling pathway in multidrug-resistant acute lymphoblastic leukemia cells.

2017

Abstract Multidrug resistance (MDR) represents a serious problem in cancer treatment. One strategy to overcome this obstacle is to identify agents that are selectively lethal to MDR cells. The aim of this study was to discover novel compounds against MDR leukemia and to determine the molecular mechanisms behind collateral sensitivity. A library of 1162 compounds was tested against parental, drug-sensitive CCRF-CEM cells using the resazurin assay. A total of 302 compounds showed reasonable activity (less than 50% cell viability). Eleven out of 30 lawsone derivatives revealed considerable collateral sensitivity in MDR P-glycoprotein (Pgp)-overexpressing CEM/ADR5000 cells. They reduced β-caten…

0301 basic medicineFrizzledAntineoplastic AgentsPharmacologyBiologyBiochemistryLawsone03 medical and health scienceschemistry.chemical_compound0302 clinical medicineCell Line TumormedicineHumansViability assaybeta CateninPharmacologyDose-Response Relationship DrugMolecular StructureWnt signaling pathwayResazurinPrecursor Cell Lymphoblastic Leukemia-Lymphomamedicine.diseaseMultiple drug resistanceWnt ProteinsLeukemia030104 developmental biologychemistryCell cultureDrug Resistance Neoplasm030220 oncology & carcinogenesisCancer researchReactive Oxygen SpeciesNaphthoquinonesSignal TransductionBiochemical pharmacology
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Lost Strings in Genomes: What Sense Do They Make?

2017

We studied the sets of avoided strings to be observed over a family of genomes. It was found that the length of the minimal avoided string rarely exceeds 9 nucleotides, with neither respect to a phylogeny of a genome under consideration. The lists of the avoided strings observed over the sets of (related) genomes have been analyzed. Very low correlation between the phylogeny, and the set of those strings has been found.

0301 basic medicineGeneticsanimal structuresgenetic structuresinformation scienceString (physics)GenomeCombinatoricsSet (abstract data type)03 medical and health sciences030104 developmental biology0302 clinical medicinePhylogeneticscardiovascular systemLow correlation030217 neurology & neurosurgerySelection (genetic algorithm)Mathematics
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Clinical and molecular characterization of 112 single-center patients with Neurofibromatosis type 1.

2018

Abstract Background The aim of this retrospective study was to define clinical and molecular characteristics of a large sample of neurofibromatosis type 1 (NF1) patients, as well as to evaluate mutational spectrum and genotype-phenotype correlation. NF1 is a relatively common neurogenetic disorder (1:2500–1:3000 individuals). It is caused by mutations of the NF1 gene on chromosome 17ql1.2, with autosomal dominant pattern of inheritance and wide phenotypical variability. Café-au-lait spots (CALs), cutaneous and/or subcutaneous neurofibromas (CNFs/SCNFs), skinfold freckling, skeletal abnormalities, Lisch nodules of the iris and increased risk of learning and intellectual disabilities, as well…

0301 basic medicineGenotype-phenotype correlation; New mutation; NF1 gene; NF1 microdeletion syndrome; Adolescent; Adult; Age Factors; Child; Child Preschool; Cohort Studies; DNA Mutational Analysis; Female; Genes Neurofibromatosis 1; Genetic Association Studies; Genetic Predisposition to Disease; Humans; Italy; Male; Middle Aged; Neurofibromatosis 1; Prevalence; Prognosis; Retrospective Studies; Risk Assessment; Sex Factors; Young Adult; Mutation MissenseMaleGenotype-phenotype correlationDNA Mutational AnalysisDiseaseCohort Studies0302 clinical medicineDNA Mutational AnalysisGenotypePrevalenceMedicineYoung adultChildNew mutationlcsh:RJ1-570Age FactorsMiddle AgedPrognosisItalyNF1 geneChild PreschoolCohortFemaleNF1 microdeletion syndromeCohort studyAdultmedicine.medical_specialtycongenital hereditary and neonatal diseases and abnormalitiesNeurofibromatosis 1AdolescentMutation MissenseRisk Assessment03 medical and health sciencesYoung AdultSex FactorsGenes Neurofibromatosis 1HumansGenetic Predisposition to DiseaseNeurofibromatosisPreschoolGenetic Association StudiesRetrospective Studiesbusiness.industryResearchRetrospective cohort studylcsh:Pediatricsmedicine.diseaseDermatology030104 developmental biologyGenesPediatrics Perinatology and Child HealthMutationMissensebusiness030217 neurology & neurosurgeryItalian journal of pediatrics
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Structure-Activity Relationships of Cytotoxic Lactones as Inhibitors and Mechanisms of Action.

2020

Background: Some lactones prevent protein Myb-dependent gene expression. Objective: The object is to calculate inhibitors of Myb-brought genetic manifestation. Methods: Linear quantitative structure–potency relations result expanded, among sesquiterpene lactones of a variety of macrocycles (pseudoguaianolides, guaianolides, eudesmanolides and germacranolides), to establish which part of the molecule constitutes their pharmacophore, and predict their inhibitory potency on Myb-reliant genetic manifestation, which may result helpful as leads for antileukaemic therapies with a new mechanism of action. Results: Several count indices are connected with structure–activity. The α-methylene-γ-lacto…

0301 basic medicineGermacranolidePaclitaxelStereochemistrySesquiterpeneRing (chemistry)Ligands030226 pharmacology & pharmacy03 medical and health scienceschemistry.chemical_compoundLactonesStructure-Activity Relationship0302 clinical medicineTubulinNeoplasmsDrug DiscoverymedicinePotencyMoleculeHumansEtoposidechemistry.chemical_classification030102 biochemistry & molecular biologyAntineoplastic Agents PhytogenicTubulin ModulatorsMolecular Docking SimulationMechanism of actionchemistryStructural Homology ProteinDrug DesignPharmacophoremedicine.symptomTopotecanSesquiterpenesLactoneCurrent drug discovery technologies
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Using the Intervention Mapping protocol to develop a family-based intervention for improving lifestyle habits among overweight and obese children: st…

2016

Abstract Background In light of the high prevalence of childhood overweight and obesity, there is a need of developing effective prevention programs to address the rising prevalence and the concomitant health consequences. The main aim of the present study is to systematically develop and implement a tailored family-based intervention for improving lifestyle habits among overweight and obese children, aged 6–10 years old, enhancing parental self-efficacy, family engagement and parent-child interaction. A subsidiary aim of the intervention study is to reduce the prevalence of overweight and obesity among those participating in the intervention study. Methods/design The Intervention Mapping p…

0301 basic medicineGerontologyCounselingParentsmedicine.medical_specialtyPediatric ObesityPilot ProjectsHealth PromotionOverweightChildhood obesity03 medical and health sciencesIntervention mappingStudy Protocol0302 clinical medicineIntervention (counseling)Health caremedicineHumansParental involvement030212 general & internal medicineChildhood obesityParent-Child RelationsChildExerciseLife Style030109 nutrition & dieteticsEnergy balance related behaviorbusiness.industryNorwayPublic healthlcsh:Public aspects of medicinePublic Health Environmental and Occupational Healthlcsh:RA1-1270Feeding Behaviormedicine.diseaseFamily lifeIntervention Mapping protocolResearch DesignChild PreschoolPhysical therapyFamily TherapyFemaleBiostatisticsmedicine.symptombusinessBMC Public Health
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Determinants of diet and physical Activity (DEDIPAC): a summary of findings

2017

The establishment of the Determinants of Diet and Physical Activity (DEDIPAC) Knowledge Hub, 2013 – 2016, was the first action taken by the ‘ Healthy Diet for a Healthy Life ’ European Joint Programming Initiative. DEDIPAC aimed to provide better insight into the determinants of diet, physical activity and sedentary behaviour across the life course, i.e. insight into the causes of the causes of important, non-commu nicable diseases across Europe and beyond. DEDIPAC was launched in late 2013, and delivered its final report in late 2016. In this paper we give an overview of what was achieved in terms of furthering measurement and monitoring, providing overviews of the state-of-the-art in the …

0301 basic medicineGerontologyDebateHealth BehaviorPsychological interventionMedicine (miscellaneous)Diseasedeterminants of health behaviours; dietary behaviour; Europe; interventions; physical activity; policy evaluation; sedentary behaviour[SHS]Humanities and Social SciencesCohort Studies0302 clinical medicineddc:150Medizinische FakultätMedicine030212 general & internal medicinelcsh:RC620-627InterventionsNutrition and Dieteticslcsh:Public aspects of medicineBenchmarkingPublic relationsPeer reviewDietary behaviour ; Interventions ; Physical activity ; Sedentary behaviour ; Europe ; Determinants of health behaviours ; Policy evaluationEuropelcsh:Nutritional diseases. Deficiency diseasesWork (electrical)Life course approachDeterminants of health behavioursDiet HealthyBehavioural sciencesInterventionPhysical Therapy Sports Therapy and RehabilitationDietary behaviour-Determinants of health behaviours;Dietary behaviour;Europe;Physical activity;Policy evaluation;Sedentary behaviour;InterventionsPolicy evaluation03 medical and health sciencesHumansddc:610Exercise030109 nutrition & dieteticsbusiness.industryPhysical activityResearchlcsh:RA1-1270Sedentary behaviourDietAction (philosophy)Determinants of health behaviourSedentary BehaviorbusinessDEDIPAC consortium
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Predictive ability of the Mini Nutritional Assessment Short Form (MNA-SF) in a free-living elderly population: a cross-sectional study

2017

Background Various scales have been used to perform a quick and first level nutritional assessment, and the MNA is one of the most used and recommended by experts in the elderly in all areas. This scale has a short form, the MNA-SF, revised and validated in 2009, which has two versions: the BMI-MNA-SF contains the first six items of the full scale including Body Mass Index while the CC-MNA-SF includes Calf Circumference instead of BMI. Objective To evaluate the predictive ability for nutritional status of the two versions of the MNA-SF against the MNA in free-living elderly in the province of Valencia. Methods Cross-sectional study of 660 free-living elderly in the province of Valencia sel…

0301 basic medicineGerontologyFree-living elderlyCross-sectional studyESTADISTICA E INVESTIGACION OPERATIVAPopulationlcsh:MedicineNursingGeneral Biochemistry Genetics and Molecular Biology03 medical and health sciences0302 clinical medicineMedicine030212 general & internal medicineeducationNutritionRank correlationeducation.field_of_study030109 nutrition & dieteticsReceiver operating characteristicbusiness.industryGeneral Neurosciencelcsh:RGeneral MedicineGold standard (test)Nutritional assessmentMNA-SFmedicine.diseaseMalnutritionGeriatricsEnfermeríaGeneral Agricultural and Biological SciencesbusinessBody mass indexKappaDemographyPeerJ
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An assessment of the test-retest reliability of the New Nordic Diet score

2015

Background : There is a growing interest in the New Nordic Diet (NND) as a potentially health promoting, environmentally friendly, and palatable regional diet. Also, dietary scores are gaining ground as a complementary approach for examining relations between dietary patterns and various health outcomes. A score assessing adherence to the NND has earlier been published, yet not tested for reliability. Objective : To assess the test–retest reliability of the NND score in a sample of parents of toddlers, residing in Southern Norway. Design : A questionnaire survey was completed on two occasions, approximately 14 days apart, by 67 parents of toddlers [85% females, mean age 34 years (SD=5.3 yea…

0301 basic medicineGerontologyNew Nordic Dietlcsh:TX341-64103 medical and health sciences0302 clinical medicinetest–retest reliabilityMedicine030212 general & internal medicineadherencePublic Health NutritionReliability (statistics)Rank correlationContingency table030109 nutrition & dieteticsNutrition and DieteticsHuman nutrition; Food composition; Nutrition epidemiologybusiness.industryPublic Health Environmental and Occupational HealthMean agehealthdiet scoreDietary patternTest (assessment)Original ArticleNutrition researchdietary patternbusinesslcsh:Nutrition. Foods and food supplyKappaFood ScienceClinical psychology
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BDE-47 exposure modulates cellular responses, oxidative stress and biotransformation related-genes in Mytilus galloprovincialis.

2020

Abstract Polybrominated diphenyl ethers (PBDEs) are flame retardants, characterized by elevated stability in the marine environment, where are accumulated by organisms, inducing a wide panel of negative effects. In this study, some biochemical patterns related to toxicity, biotransformation and oxidative stress, were studied in the marine model system, Mytilus galloprovincialis, exposed to BDE-47. Mussels were fed with microalgae, previously treated with increasing concentrations of PBDEs (maximum dose 100 ng L-1 of BDE-47 per day). After 15 days of treatment, mussels were fed with the same diet without BDE-47, for additional 15 days. Gills and digestive glands were analyzed at T 0, at 15 a…

0301 basic medicineGillanimal structuresTime FactorsGene ExpressionAquatic SciencePBDEmedicine.disease_causeAndrology03 medical and health sciencesRandom AllocationPolybrominated diphenyl ethersBiotransformationSettore AGR/20 - ZoocoltureDetoxificationGene expressionmedicineHalogenated Diphenyl EthersEnvironmental ChemistryMusselsAnimalsTissue DistributionSettore BIO/06 - Anatomia Comparata E CitologiaBiotransformationMytilusbiologyDose-Response Relationship DrugfungiCell Cycle04 agricultural and veterinary sciencesGeneral Medicinebiology.organism_classificationBioaccumulationMytilusDrug Resistance MultipleOxidative Stress030104 developmental biologyToxicityInactivation Metabolic040102 fisheries0401 agriculture forestry and fisheriesOxidative stressWater Pollutants ChemicalFishshellfish immunology
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