Search results for "urea"

showing 10 items of 888 documents

I laureati triennali

2009

profilo post-laurea placementSettore SECS-S/05 - Statistica Sociale
researchProduct

I laureati a ciclo unico

2009

profilo post-laurea placementSettore SECS-S/05 - Statistica Sociale
researchProduct

I laureati specialistici

2009

profilo post-laurea placementSettore SECS-S/05 - Statistica Sociale
researchProduct

I laureati dell'Università degli studi di Palermo

2009

profilo post-laurea placementSettore SECS-S/05 - Statistica Sociale
researchProduct

Synthesis and Antitumor Evaluation of Menthone-Derived Pyrimidine-Urea Compounds as Potential PI3K/Akt/mTOR Signaling Pathway Inhibitor.

2022

A series of novel menthone derivatives bearing pyrimidine and urea moieties was designed and synthesized to explore more potent natural product-derived antitumor agents. The structures of the target compounds were confirmed by FTIR, NMR, and HRMS. The in vitro antitumor activity was tested by standard methyl thiazolytetrazolium assay and showed that 4i, 4g, 4s, and 4m are the best compounds with IC50 values of 6.04 ± 0.62µM, 3.21 ± 0.67µM, 19.09 ± 0.49µM, and 18.68 ± 1.53µM, against Hela, MGC-803, MCF-7, and A549, respectively. The results of the preliminary action mechanism studies showed that compound 4i, the representative compound, could induce cell apoptosis in Hela cells in a dose-dep…

pyrimidineChemistrysynthesisnervous systemgenetic structuresPI3K/AKT/mTORantitumor activitymenthoneureaGeneral ChemistryQD1-999behavioral disciplines and activitiespsychological phenomena and processesFrontiers in chemistry
researchProduct

Sulfonilurea preparātu farmakoģenētika cukura diabēta ārstēšanā

2015

Darba aktualitāte: Otrā tipa cukura diabēta (2TCD) prevalence pieaug gan Latvijas, gan pasaules mērogā. Pacientiem ir nepieciešama personalizēta pieeja, kas labāk ļautu sasniegt terapijas mērķi un izvairīties no komplikācijām. Sulfonilurea (SU) preparāti ir viena no visbiežāk izmantotajām perorālo antidiabētisko preparātu klasēm, tāpēc ir būtiski apzināt šo preparātu individuālos efektus. Pētījuma mērķis: Noskaidrot, vai SU preparātu farmakoģenētika ietekmē 2TCD pacientu ārstēšanas rezultātu. Metodes un materiāli: Longitudinālā prospektīvā pētījumā tika iesaistīti 315 2TCD pacienti, retrospektīvi tika iesaistīti 162, no kuriem kopumā sulfonilurea preparātus bija lietojuši 162, atlases kritē…

rs2237895otrā tipa cukura diabētsfarmakoģenētikasulfonilureaMedicīna
researchProduct

I laureati triennali

2010

sbocchi occupazionali post-laureaSettore SECS-S/05 - Statistica Sociale
researchProduct

I laureati specialistici

2010

sbocchi occupazionali post-laureaSettore SECS-S/05 - Statistica Sociale
researchProduct

I laureati a ciclo unico

2010

sbocchi occupazionali post-laureaSettore SECS-S/05 - Statistica Sociale
researchProduct

Analisi per Ateneo. L'Università degli studi di Palermo.

2011

Il capitolo mette in evidenza le caratteristiche salienti dei profili post-laurea dei laureati dell'ateneo di Palermo elaborati attraverso un'indagine campionaria. Il capitolo tratta anche un approfondimento dei laureati delle principali caratteristiche socio demografiche.

sbocchi occupazionalianalisi descrittiva occupazione dei laureatiindagine post-laureaSettore SECS-S/05 - Statistica Sociale
researchProduct