0000000000640131

AUTHOR

Alexandre Bouillon

showing 2 related works from this author

Novel oxybispyridylboronic acids: synthesis and study of their reactivity in Suzuki-type cross-coupling reactions

2007

Abstract This paper sets forth the synthesis of novel oxybispyridylboronic acids, which are prepared from the corresponding halo-oxybispyridines via halogen–metal exchange using n-butyllithium and treatment with triisopropylborate. A range of efficient cross-coupling reactions of these novel boronic acids with selected aryl halides is described. This strategy produces novel pyridylethers of interest in cholinergic medicinal chemistry.

inorganic chemicalschemistry.chemical_compoundchemistryArylOrganic ChemistryDrug DiscoveryOrganic chemistryHalideReactivity (chemistry)General MedicineBiochemistryCombinatorial chemistryCoupling reactionTetrahedron
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Synthesis of Novel Triazolopyridylboronic Acids and Esters. Study of Potential Application to Suzuki-Type Reactions.

2004

This paper describes a general method for the synthesis of novel [1,2,3]triazolo[1,5-a]pyridylboronic acids and esters, and the first results on Suzuki cross-coupling reactions with these new compounds and [1,2,3]triazolo[5,1-a]isoquinolylboronic acid, reacting with a variety of aryl halides as a route to 7-aryltriazolopyridines and 5-aryltriazoloisoquinolines.

chemistry.chemical_compoundGeneral methodSuzuki reactionChemistryArylOrganic ChemistryDrug DiscoveryOrganic chemistryHalideGeneral MedicineBiochemistryCombinatorial chemistryChemInform
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