6533b854fe1ef96bd12aea8e
RESEARCH PRODUCT
Synthesis of Novel Triazolopyridylboronic Acids and Esters. Study of Potential Application to Suzuki-Type Reactions.
José-reynaldo Domı́nguezAlexandre BouillonJean-charles LancelotValérie CollotSylvain RaultRafael BallesterosBelén AbarcaFernando Blancosubject
chemistry.chemical_compoundGeneral methodSuzuki reactionChemistryArylOrganic ChemistryDrug DiscoveryOrganic chemistryHalideGeneral MedicineBiochemistryCombinatorial chemistrydescription
This paper describes a general method for the synthesis of novel [1,2,3]triazolo[1,5-a]pyridylboronic acids and esters, and the first results on Suzuki cross-coupling reactions with these new compounds and [1,2,3]triazolo[5,1-a]isoquinolylboronic acid, reacting with a variety of aryl halides as a route to 7-aryltriazolopyridines and 5-aryltriazoloisoquinolines.
| year | journal | country | edition | language |
|---|---|---|---|---|
| 2004-09-21 | ChemInform |