Fluorinated Heterocyclic Compounds. A Photochemical Approach to a Synthesis of Polyfluoroaryl-1,2,4-triazoles.

6533b7d2fe1ef96bd125f543

RESEARCH PRODUCT

Fluorinated Heterocyclic Compounds. A Photochemical Approach to a Synthesis of Polyfluoroaryl-1,2,4-triazoles.

Nicolò Vivona Ivana Pibiri Silvestre Buscemi Antonio Palumbo Piccionello Andrea Pace

subject

Pharmacology FLUORO HETEROCYCLES Methylamine Organic Chemistry QUINAZOLIN-4-ONES 1 2 4-Triazole 1 2 4-OXADIAZOLES Propylamine Settore CHIM/06 - Chimica Organica General Medicine EXPEDIENT ROUTE Photochemistry Medicinal chemistry Analytical Chemistry chemistry.chemical_compound 1 2 4-TRIAZOLES chemistry Triazole derivatives Organic chemistry 5-MEMBERED HETEROCYCLES Irradiation Methanol Acetonitrile PHOTOINDUCED MOLECULAR-REARRANGEMENTS

description

The reaction of some fluorinated 1,2,4-oxadiazoles in the presence of methylamine or propylamine has been investigated. The irradiation in methanol or acetonitrile leads with acceptable yields to the corresponding fluorinated 1- methyl- or 1-propyl-1,2,4-triazole.

year	journal	country	edition	language
2005-06-14	ChemInform

https://doi.org/10.1002/chin.200524123

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