Antimykotische wirkstoffe. XX . Fluorierte 2-(4-toluidino)pyrimidine

6533b821fe1ef96bd127b729

RESEARCH PRODUCT

Antimykotische wirkstoffe. XX . Fluorierte 2-(4-toluidino)pyrimidine

subject

Diketone chemistry.chemical_compound Pyrimidine chemistry Stereochemistry Organic Chemistry Condensation Biological activity

description

Aus der Kondensation von 4-Tolylguanidin (1) mit den β-Diketonen 2a-f gehen die fluorierten 2-(4-Toluidino)pyrimidine 3a-f hervor. Strukturtyp 3 zeichnet sich durch antimykotische Wirkung aus. Condensation of 4-tolylguanidine (1) with the β-diketones 2a-f yields the fluorinated 2-(4-toluidino)pyrimidines 3a-f. Structures of type 3 exhibit antimycotic activity.

year	journal	country	edition	language
1985-01-01	Journal of Heterocyclic Chemistry

https://doi.org/10.1002/jhet.5570220126

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