Search results for " Competitive"

showing 10 items of 237 documents

Distribution of chlorpromazine in a simplified blood influenced by various drugs

1973

The binding of chlorpromazine to erythrocytes and to albumin as influenced by other drugs was studied in a simplified blood (31.5±0.3% bovine erythrocytes, 4 g-% bovine serum albumin in 0.02 M phosphate buffer solution containing 0.15 M NaCl). the total concentration of chlorpromazine in the simplified blood was 10−4 M, the concentration of the displacing drugs was 10−3 M. After an incubation period of 3 h at 22° C the chlorpromazine concentration was determined in the albumin solution after centrifugation of the blood at 3000×g and in the aqueous phase after ultracentrifugation at 150000×g. Under control conditions 68.1±0.9% of chlorpromazine was bound to the erythrocytes, 28.5±0.9% was bo…

ErythrocytesChlorpromazineIndomethacinSuraminBenzoatesBinding CompetitiveIncubation periodCoumarinsmedicineAnimalsDistribution (pharmacology)CentrifugationThiopentalBovine serum albuminChlorpromazinePharmacologySulfonamidesBinding SitesChromatographyQuininebiologyProbenecidChemistryFatty AcidsAqueous two-phase systemAlbuminSerum Albumin BovineGeneral MedicineChlorothiazideTetracyclineAntidepressive AgentsSalicylatesAcetazolamidePhenylbutazoneSolubilityPhenytoinbiology.proteinCattleUltracentrifugeDeoxycholic AcidProtein Bindingmedicine.drugNaunyn-Schmiedeberg's Archives of Pharmacology
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The atractiveness and competitiveness of tourist destinations: A study on Southern Italian regions

2009

The present paper aims to assess the relative attractiveness of competing tourist destinations on the basis of individual visitors' perceptions regarding a holiday destination. Using the feeling of tourist well-being achieved by individual tourists we evaluate indirectly the competitive ability of the tourist area to offer a compound tourist site attractiveness. The methodology employed here uses individual survey questionnaires on the tourists' evaluation of the quality of tourist facilities and attributes in a given area (the 'regional tourist profile') as the basis for constructing an aggregate expression for the relative attractiveness of that area. Using various multidimensional statis…

EstimationAttractivenessTourist competitiveneStrategy and Managementmedia_common.quotation_subjectPrincipal component analysisTransportationResource based view Multi-attribute utilityDevelopmentTourist attractiveneGeographyTourism Leisure and Hospitality ManagementSettore SECS-S/03 - Statistica EconomicaResource-based viewRegional scienceMulti-attribute utilityTourist destinationsQuality (business)MarketingTourismmedia_commonTourism Management
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The economic impact of the EFF on the competitiveness of Sicilian fish companies

2017

The measure 2.3 of the European Fisheries Fund, in Sicily, claimed investments of fish companies in production capacity expansion and modernization of fish processing. Have these investments been effective in supporting the competitiveness of these companies and have they influenced the economic sustainability of the regional seafood chain? Proposed analysis contributes to this assessment through an exploratory survey and a review of the changes in their business performance.

European Fisheries Fund fish companies innovation investments competitivenessSettore SECS-P/06 - Economia Applicata
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Faktori, kas ietekmē Latvijas loģistikas uzņēmumu konkurētspēju ES

2019

Promocijas darbā tiek pētīta Latvijas loģistikas uzņēmumu konkurētspēja. Loģistika ir viena no galvenajām Latvijas nozarēm. Tāpēc ir svarīgi pievērsties galvenās nozares uzlabošanai. Tomēr konkurence nav balstīta uz vienu faktoru; būs vairāki faktori, kas ietekmē konkurētspēju. Promocijas darbā tiek pētīti Latvijas loģistikas uzņēmumu konkurētspēju ietekmējošie faktori. Konkurence Eiropas Savienībā ir tik spēcīga, tāpēc ir svarīgi koncentrēties uz Latvijas loģistikas uzņēmumu konkurētspēju, lai uzlabotu produktivitāti un peļņu. Loģistikas nozares sarežģītība arī padara to par būtisku to izpētei. Tā kā loģistikas nozare ir atkarīga no vairākiem faktoriem, promocijas darbā tiek analizēti četr…

Factors of competitivenessEuro UnionEkonomikaLogisticsLatviaCompetitiveness
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Sicilian floriculture companies and the role of transport in increasing their competitiveness

2008

The aim of this study is to provide a deeper understanding of the Sicilian floriculture sector, which has recently become one of the most important on a regional and national scale. By analysing production, sales and logistical aspects of its production companies and specifically looking at aspects regarding transport logistics, this study highlights the sector operators. preference for road transport that offers better guarantees in terms of delivery speed with respect to other means of transport, an essential requirement for the transport of flowers and plants. However, operators are increasingly showing interest in alternative means of transport that may reduce transport time and, especi…

Flower and ornamental plant sector sicily competitiveness logistics and transportSettore AGR/01 - Economia Ed Estimo Rurale
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SYNTHESIS AND IN VITRO AFFINITIES OF VARIOUS MDL 100907 DERIVATIVES AS POTENTIAL 18F-RADIOLIGANDS FOR 5-HT2A RECEPTOR IMAGING WITH PET

2008

Radiolabelled piperidine derivatives such as [(11)C]MDL 100907 and [(18)F]altanserin have played an important role in diagnosing malfunction in the serotonergic neurotransmission. A variety of novel piperidine MDL 100907 derivatives, possible to label with (18)F-fluorine, were synthesized to improve molecular imaging properties of [(11)C]MDL 100907. Their in vitro affinities to a broad spectrum of neuroreceptors and their lipophilicities were determined and compared to the clinically used reference compounds MDL 100907 and altanserin. The novel compounds MA-1 (53) and (R)-MH.MZ (56) show K(i)-values in the nanomolar range towards the 5-HT(2A) receptor and insignificant binding to other 5-HT…

Fluorine RadioisotopesReceptor StatusStereochemistryClinical BiochemistryPharmaceutical ScienceLigandsBinding CompetitiveBiochemistryChemical synthesisMiceRadioligand AssayStructure-Activity Relationshipchemistry.chemical_compoundPiperidinesDrug DiscoveryRadioligandAnimalsHumansReceptor Serotonin 5-HT2AReceptorMolecular Biology5-HT receptorOrganic ChemistryLigand (biochemistry)AffinitiesRatsFluorobenzenesKineticschemistryPositron-Emission TomographyAltanserinNIH 3T3 CellsMolecular MedicineRadiopharmaceuticals
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Total synthesis and evaluation of [18F]MHMZ.

2007

Radiochemical labeling of MDL 105725 using the secondary labeling precursor 2-[(18)F]fluoroethyltosylate ([(18)F]FETos) was carried out in yields of approximately 90% synthesizing [(18)F]MHMZ in a specific activity of approximately 50MBq/nmol with a starting activity of approximately 3GBq. Overall radiochemical yield including [(18)F]FETos synthon synthesis, [(18)F]fluoroalkylation and preparing the injectable [(18)F]MHMZ solution was 42% within a synthesis time of approximately 100 min. The novel compound showed excellent specific binding to the 5-HT(2A) receptor (K(i)=9.0 nM) in vitro and promising in vivo characteristics.

Fluorine RadioisotopesStereochemistryClinical BiochemistryPharmaceutical ScienceBiochemistryBinding CompetitiveRadioligand AssayPiperidinesIn vivoDrug DiscoveryAnimalsRadionuclide imagingReceptor Serotonin 5-HT2ARadionuclide ImagingMolecular BiologyChemistryOrganic ChemistrySynthonTotal synthesisBrainBiological activityRadioligand AssayRatsFluorobenzenesKineticsYield (chemistry)Isotope LabelingSerotonin 5-HT2 Receptor AntagonistsMolecular MedicineSpecific activityKetanserinSerotonin AntagonistsRadiopharmaceuticalsNuclear chemistryBioorganicmedicinal chemistry letters
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RNA-binding activity of the rat calmodulin-binding PEP-19 protein and of the long PEP-19 isoform

2012

Synthesis of H1˚ histone protein, in the developing rat brain, seems to be regulated mainly at the post-transcriptional level. Since regulation of RNA metabolism depends on a series of RNA-binding proteins, we have been searching for RNA-binding proteins involved in the post-transcriptional regulation of the H1˚ gene. We recently reported isolation, from a cDNA expression library, of an insert encoding a novel protein, the C-terminal half of which is identical to that of PEP-19, a brain-specific protein involved in calcium metabolism. The novel protein was called long PEP-19 isoform (LPI). Herein we show that LPI, as well as PEP-19, can bind H1˚ RNA. Moreover, in order to improve production…

Gene isoformCalmodulinCalmodulin binding domainNerve Tissue ProteinsRNA-binding proteinRNA-binding proteins histone variants H1˚ PEP-19 long PEP-19 isoform calmodulinBiologyBinding CompetitiveRats Sprague-DawleyCalmodulinGeneticsAnimalsProtein IsoformsE2F1RNA Processing Post-TranscriptionalGeneHistidineRNA-Binding ProteinsRNAGeneral MedicineMolecular biologyRatsBiochemistrybiology.proteinRNACalmodulin-Binding ProteinsProtein BindingInternational Journal of Molecular Medicine
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Emerging Economies’ Institutional Quality and International Competitiveness: A PLS-SEM Approach

2021

The home country’s institutional framework determines the capacity to compete in the global arena. This paper discusses the linkage between institutional quality (IQ) and international competitiveness (IC). We measured institutions’ quality in emerging economies through the use of selected indicators between 2007–2017. To evaluate the proposed IQ constructs and their relationship with IC, we applied partial least squares – structural equation modeling (PLS-SEM) analysis. The model outcomes suggest that political and lack of systemic conditions have a significant and negative effect on international competitiveness, while science, technology, engineering and mathematics (STEM) resource condi…

General Mathematicsmedia_common.quotation_subjectLinkage (mechanical)Structural equation modelinglaw.inventionResource (project management)lawinternational competitiveness0502 economics and businessPartial least squares regressionQA1-939institutional qualityComputer Science (miscellaneous)Quality (business)Emerging marketsemerging economieEngineering (miscellaneous)pls-semIndustrial organizationmedia_common05 social sciencesinternational competitivene050211 marketingMathematicsemerging economies050203 business & managementInstitutional qualityMathematics
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Zebrafish Reveals Different and Conserved Features of Vertebrate Neuroglobin Gene Structure, Expression Pattern, and Ligand Binding

2004

Neuroglobin has been identified as a respiratory protein that is primarily expressed in the mammalian nervous system. Here we present the first detailed analysis of neuroglobin from a non-mammalian vertebrate, the zebrafish Danio rerio. The zebrafish neuroglobin gene reveals a mammalian-type exon-intron pattern in the coding region (B12.2, E11.0, and G7.0), plus an additional 5'-non-coding exon. Similar to the mammalian neuroglobin, the zebrafish protein displays a hexacoordinate deoxy-binding scheme. Flash photolysis kinetics show the competitive binding on the millisecond timescale of external ligands and the distal histidine, resulting in an oxygen affinity of 1 torr. Western blotting, i…

GillsDNA Complementaryanimal structuresBlotting WesternDanioNeuroglobinNerve Tissue ProteinsIn situ hybridizationBiologyLigandsBinding CompetitiveBiochemistryRetinaDiffusionExonChloridesAnimalsCoding regionHistidineRNA MessengerCloning MolecularMolecular BiologyZebrafishConserved SequenceIn Situ HybridizationZebrafishMessenger RNAModels GeneticExonsOlfactory PathwaysCell Biologybiology.organism_classificationMolecular biologyIntronsRecombinant ProteinsGlobinsMitochondriaCell biologyOxygenRespiratory proteinKineticsGene Expression RegulationMicroscopy FluorescenceSpectrophotometryNeuroglobinJournal of Biological Chemistry
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