Search results for "62"

showing 10 items of 970 documents

Identification of Biphenyl-Based Hybrid Molecules Able To Decrease the Intracellular Level of Bcl-2 Protein in Bcl-2 Overexpressing Leukemia Cells

2009

With the aim of enhancing the structural complexity and diversity of an existing collection of bi- and terphenyl compounds, we synthesized hybrid molecules comprising of spirocyclic ketones (a complexity-bearing core) and bi/terphenyls (privileged fragments). Compounds 1, 3, 4, and 6 showed well-defined activity on apoptosis and differentiation, making them potential leads for development as new anticancer agents and chemical probes to study signaling networks in neoplastic cells.

Antineoplastic AgentsApoptosisHL-60 CellsChemical synthesisStructure-Activity RelationshipLeukemia Myelogenous Chronic BCR-ABL PositiveTerphenyl CompoundsDrug DiscoverymedicineHumansSpiro CompoundsChemistryBiphenyl CompoundsCell DifferentiationBiological activityKetonesmedicine.diseaseIn vitroLeukemiaProto-Oncogene Proteins c-bcl-2BiochemistryApoptosisCell cultureMolecular MedicineTerphenyl CompoundsK562 CellsIntracellularJournal of Medicinal Chemistry
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Antimicrobial and antiproliferative activity of Peucedanum nebrodense (Guss.) Strohl.

2003

Abstract Acetone extract of Peucedanum nebrodense (Guss.) Strohl., a rare endemic species from the Madonie mountains (Sicily), was tested in vitro for its antimicrobial activity against bacterial reference strains and antiproliferative activity against K562 (human chronic myelogenous leukemia), HL-60 (human leukemia) and L1210 (murine leukemia) cell lines. The acetone extract showed antiproliferative IC 50 values in the range of 14–0.27 μg/ml.

Antineoplastic AgentsHL-60 CellsBiologyPlant RootsAcetoneMiceAnti-Infective Agentshemic and lymphatic diseasesDrug DiscoverymedicinePeucedanum nebrodenseCoumarins Antimicrobial Antiproliferative activityAnimalsHumansLeukemia L1210PharmacologyTraditional medicinePlant ExtractsBiological activityPlant Components AerialAntimicrobialmedicine.diseaseIn vitroLeukemiaCell cultureK562 CellsPeucedanum nebrodenseCell DivisionChronic myelogenous leukemiaK562 cellsApiaceaeJournal of ethnopharmacology
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ChemInform Abstract: (a)-Anellated Carbazoles with Antitumor Activity: Synthesis and Cytotoxicity.

2010

The cycloadducts3,5, and7, readily available from methoxy-substituted 3-vinylindoles1 and2, were dehydrogenated withDDQ to the coplanar [a]-anellated carbazoles4,6, and8. Compound4a, also characterized by X-ray structural analysis, shows significant cytotoxicity against K562 und RXF393 human tumor cell lines.

Antitumor activityHuman tumorStereochemistryCell cultureChemistryGeneral MedicineCytotoxicityK562 cellsChemInform
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Stress concentration for closely located inclusions in nonlinear perfect conductivity problems

2019

We study the stress concentration, which is the gradient of the solution, when two smooth inclusions are closely located in a possibly anisotropic medium. The governing equation may be degenerate of $p-$Laplace type, with $1<p \leq N$. We prove optimal $L^\infty$ estimates for the blow-up of the gradient of the solution as the distance between the inclusions tends to zero.

Applied Mathematics010102 general mathematicsMathematical analysisDegenerate energy levelsZero (complex analysis)Perfect conductorAnalysiGradient blow-upType (model theory)Conductivity01 natural sciences010101 applied mathematicsNonlinear systemMathematics - Analysis of PDEsFOS: MathematicsFinsler p-Laplacian0101 mathematicsPerfect conductorAnisotropy35J25 35B44 35B50 (Primary) 35J62 78A48 58J60 (Secondary)AnalysisAnalysis of PDEs (math.AP)MathematicsStress concentration
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La factoría de la Empresa Nacional Elcano en Manises : una valoración patrimonial

2010

La factoría de la Empresa Nacional Elcano de Manises (Valencia) fue construida entre 1946 y 1953 dentro de los planes estatales de reconstrucción industrial de la postguerra. Sus arquitecturas plantean una dualidad entre la modernidad y racionalidad de los espacios productivos y la tradición historicista de los edificios representativos, directamente relacionada con los programas ideológicos del Régimen. De su valoración a partir de los criterios establecidos por el Ministerio de Cultura para el Plan Nacional de Patrimonio Industrial, se desprende el extraordinario valor de la factoría como conjunto, el cual se sitúa por encima de la ya alta calidad de sus edificios a nivel individual, por …

Art i indústriaUNESCO::CIENCIAS DE LAS ARTES Y LAS LETRASAdrià 269 288:CIENCIAS DE LAS ARTES Y LAS LETRAS [UNESCO]0211-5808 9678 Archivo de arte valenciano 277874 2010 91 3629817 La factoría de la Empresa Nacional Elcano en Manises una valoración patrimonial Besó RosArquitectura
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Juan II de Aragón y las artes suntuarias

2015

Producción Científica

Artes decorativas - España6203.03 Artes decorativasJuan II Rey de AragónArtículos de lujoUNESCO::HISTORIA::Historia por especialidades::Historia del arte5506.02 Historia del ArteArtículo:HISTORIA::Historia por especialidades::Historia del arte [UNESCO]
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The role of contact chemoreception in the host location process of an egg parasitoid

2016

Taste allows insects to detect palatable or toxic foods, identify a mate, and select appropriate oviposition sites. The gustatory system strongly contributes to the survival and reproductive success of many species, yet it is rarely studied in insect parasitoids. In order to locate and assess a host in which they will lay their eggs, female wasps actively search for chemical cues using their sensory organs present mainly on the antennae. In this paper, we studied the role of antennal taste sensilla chaetica in the perception of contact semiochemicals in Trissolcus brochymenae (Hymenoptera: Platygastridae), an egg parasitoid of the brassicaceae pest Murgantia histrionica (Heteroptera: Pentat…

Arthropod AntennaeMale0106 biological sciencesTastePhysiologyOvipositionmedia_common.quotation_subject[SDV]Life Sciences [q-bio]WaspsZoologySensilla chaeticaHymenopteraInsect010603 evolutionary biology01 natural sciencesGas Chromatography-Mass SpectrometryHost-Parasite InteractionsParasitoidHeteroptera016-3962PlatygastridaeAnimalsBehaviourLaboratory of Entomologymedia_commonAppetitive BehaviorReproductive successbiologyAnimalEcologyHost (biology)Behaviour Electrophysiology Gustation Kairomone Platygastridae Sensilla chaeticafungiHost-Parasite InteractionTaste PerceptionWaspPentatomidaebiology.organism_classificationLaboratorium voor EntomologieElectrophysiological PhenomenaElectrophysiology010602 entomologySettore AGR/11 - Entomologia Generale E ApplicataInsect ScienceKairomoneKairomoneFemaleGustation
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The Polarized Image of a Synchrotron-emitting Ring of Gas Orbiting a Black Hole

2021

Full list of authors: Narayan, Ramesh; Palumbo, Daniel C. M.; Johnson, Michael D.; Gelles, Zachary; Himwich, Elizabeth; Chang, Dominic O.; Ricarte, Angelo; Dexter, Jason; Gammie, Charles F.; Chael, Andrew A.; Event Horizon Telescope Collaboration; Akiyama, Kazunori; Alberdi, Antxon; Alef, Walter; Algaba, Juan Carlos; Anantua, Richard; Asada, Keiichi; Azulay, Rebecca; Baczko, Anne-Kathrin; Ball, David Baloković, Mislav; Barrett, John; Benson, Bradford A.; Bintley, Dan; Blackburn, Lindy; Blundell, Raymond; Boland, Wilfred; Bouman, Katherine L.; Bower, Geoffrey C.; Boyce, Hope; Bremer, Michael; Brinkerink, Christiaan D.; Brissenden, Roger; Britzen, Silke; Broderick, Avery E.; Broguiere, Domini…

AstrofísicaCamps magnèticsAccretion010504 meteorology & atmospheric sciencesAstronomyAstrophysics::High Energy Astrophysical PhenomenaStrong gravitational lensingSynchrotron radiationFOS: Physical sciencesF50001 natural sciencesAstrophysics - high energy astrophysical phenomena994General Relativity and Quantum Cosmology0103 physical sciencesPolarimetrySchwarzschild metric010303 astronomy & astrophysics0105 earth and related environmental sciences162astro-ph.HEEvent Horizon TelescopePhysicsHigh Energy Astrophysical Phenomena (astro-ph.HE)1278Accretion (meteorology)Black holes14Astronomy and AstrophysicsPolarization (waves)Computational physicsMagnetic fieldBlack holeSpace and Planetary ScienceMagnetic fields14 162 1278 994
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EVIDENCE OF NON-THERMAL X-RAY EMISSION FROM HH 80

2013

Protostellar jets appear at all stages of star formation when the accretion process is still at work. Jets travel at velocities of hundreds of km s -1, creating strong shocks when interacting with the interstellar medium. Several cases of jets have been detected in X-rays, typically showing soft emission. For the first time, we report evidence of hard X-ray emission possibly related to non-thermal processes not explained by previous models of the post-shock emission predicted in the jet/ambient interaction scenario. HH 80 is located at the south head of the jet associated with the massive protostar IRAS 18162-2048. It shows soft and hard X-ray emission in regions that are spatially separate…

AstrofísicaCiencias AstronómicasCiencias FísicasAstrophysics::High Energy Astrophysical PhenomenaFOS: Physical sciencesSynchrotron radiationAstrophysics::Cosmology and Extragalactic AstrophysicsAstrophysicsIndividual: Iras 18162-2048 [Stars]//purl.org/becyt/ford/1 [https]Herbig-Haro objects ISM: jets and outflows radiation mechanisms: non-thermal stars: individual: IRAS 18162-2048 stars: pre-main sequence X-rays: generalHigh Energy Physics - Phenomenology (hep-ph)Herbig-Haro objectsGeneral [X-Rays]jets and outflows radiation mechanisms: non-thermal stars: individual: IRAS 18162-2048 stars: pre-main sequence X-rays: general [Herbig-Haro objects ISM]Jets And Outflows [Ism]ThermalProtostarstars: individualAstrophysics::Galaxy AstrophysicsHigh Energy Astrophysical Phenomena (astro-ph.HE)PhysicsStar formationX-rayAstronomy and Astrophysics//purl.org/becyt/ford/1.3 [https]radiation mechanisms: non-thermalHerbig-Haro ObjectsAstrophysics - Astrophysics of GalaxiesAccretion (astrophysics)Non-Thermal [Radiation Mechanisms]AstronomíaInterstellar mediumHigh Energy Physics - PhenomenologyISM: jets and outflowsSpace and Planetary ScienceAstrophysics of Galaxies (astro-ph.GA)Astrophysics - High Energy Astrophysical PhenomenaCIENCIAS NATURALES Y EXACTASThe Astrophysical Journal
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Search for heavy neutral lepton production in K+ decays to positrons

2020

A search for heavy neutral lepton ($N$) production in $K^+\to e^+N$ decays using the data sample collected by the NA62 experiment at CERN in 2017--2018 is reported. Upper limits of the extended neutrino mixing matrix element $|U_{e4}|^2$ are established at the level of $10^{-9}$ over most of the accessible heavy neutral lepton mass range 144--462 MeV/$c^2$, with the assumption that the lifetime exceeds 50 ns. These limits improve significantly upon those of previous production and decay searches. The $|U_{e4}|^2$ range favoured by Big Bang Nucleosynthesis is excluded up to a mass of about 340 MeV/$c^2$.

AstrofísicaNuclear and High Energy PhysicsHeavy neutral lepton kaon meson kaon decay positronPontecorvo–Maki–Nakagawa–Sakata matrixSocio-culturaleFOS: Physical sciencesNA62 experiment7. Clean energy01 natural sciencesNA62High Energy Physics - ExperimentNuclear physicsHigh Energy Physics - Experiment (hep-ex)Positronkaon decays heavy neutral lepton SM extensionsPE2_2Big Bang nucleosynthesisSM extensionskaon physics0103 physical sciences[PHYS.HEXP]Physics [physics]/High Energy Physics - Experiment [hep-ex]010306 general physicsComputingMilieux_MISCELLANEOUSPhysicsRange (particle radiation)Large Hadron Colliderkaon decays010308 nuclear & particles physicshep-exSettore FIS/04Heavy neutral leptonlepton flavour violationFísicalcsh:QC1-999kaon mesonkaon decaykaon physics; lepton flavour violation; NA62positronProduction (computer science)High Energy Physics::Experimentkaonlcsh:PhysicsParticle Physics - ExperimentLepton
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