Search results for "ALPHA"

showing 10 items of 3228 documents

CCDC 934572: Experimental Crystal Structure Determination

2013

Related Article: A.Brzuszkiewicz,M.Makowski,M.Lisowski,E.Lis,M.Otreba,T.Lis|2013|Acta Crystallogr.,Sect.C:Cryst.Struct.Commun.|69|277|doi:10.1107/S0108270113002539

Space GroupCrystallographycdelta-methyl (3-([t-butoxycarbonylglycyl-alphabeta-(Z)-dehydrophenylalanyl]amino)propyl)phosphonateCrystal SystemCrystal StructureCell ParametersExperimental 3D Coordinates
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CCDC 178153: Experimental Crystal Structure Determination

2002

Related Article: M.Zaidlewicz, W.Sokol, A.Wojtczak, P.Neumann, M.Nissinen|2002|Tetrahedron Lett.|43|3525|doi:10.1016/S0040-4039(02)00587-7

Space GroupCrystallographysyn-6-(alpha-Hydroxybenzyl)-3455-tetramethylcyclohex-2-enoneCrystal SystemCrystal StructureCell ParametersExperimental 3D Coordinates
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CCDC 248542: Experimental Crystal Structure Determination

2004

Related Article: C.Boskovic, A.Sieber, G.Chaboussant, H.U.Gudel, J.Ensling, W.Wernsdorfer, A.Neels, G.Labat, H.Stoeckli-Evans, S.Janssen|2004|Inorg.Chem.|43|5053|doi:10.1021/ic049600f

Space GroupCrystallographytris((mu~2~-2-(alpha-phenylsalicylidenealdiminato)ethanolato)-(mu~2~-acetato)-iron(iii)) dichloromethane solvateCrystal SystemCrystal StructureCell ParametersExperimental 3D Coordinates
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Psoriatic arthritis and COVID ‐19 pandemic: Consequences in medical treatment?

2020

The COVID‐19 pandemic has a strong negative impact on human society world‐wide. Patients with immune‐mediated disease may be prone to an increased risk of infection and/ or more severe course. We review the available data for patients with psoriatic arthritis (PSA) and systemic treatments. Current treatment options are summarized. Based upon the experience with COVID‐19 the following problems are addressed: (a) Can systemic treatment reduce comorbidities of PsA that are also comorbidities for COVID‐19? Does systemic medical treatment pose an increased risk of infection with SARS‐CoV‐2? Does systemic drug therapy have an impact on the risk of pulmonary fibrosis ‐ a factor with strong negativ…

Special Issue Articlesmedicine.medical_specialtyDiseaseComorbidityDermatologyPlacebo030207 dermatology & venereal diseases03 medical and health sciencesPsoriatic arthritisPsoriatic arthritis; systemic medical treatment0302 clinical medicinePharmacotherapyCOVID‐19Internal medicinePandemicmedicineHumansJanus Kinase InhibitorsbiologicsBiological Productsbusiness.industrySARS-CoV-2Tumor Necrosis Factor-alphaArthritis PsoriaticInterleukinSpecial Issue ArticleCOVID-19General Medicinemedicine.diseaseComorbiditysmall molecules030220 oncology & carcinogenesisAirwaybusinessDermatologic Therapy
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Molecular mechanism of T-cell protein tyrosine phosphatase (TCPTP) activation by mitoxantrone.

2013

T-cell protein tyrosine phosphatase (TCPTP) is a ubiquitously expressed non-receptor protein tyrosine phosphatase. It is involved in the negative regulation of many cellular signaling pathways. Thus, activation of TCPTP could have important therapeutic applications in diseases such as cancer and inflammation. We have previously shown that the α-cytoplasmic tail of integrin α1β1 directly binds and activates TCPTP. In addition, we have identified in a large-scale high-throughput screen six small molecules that activate TCPTP. These small molecule activators include mitoxantrone and spermidine. In this study, we have investigated the molecular mechanism behind agonist-induced TCPTP activation.…

SpermidineProtein tyrosine phosphataseBiochemistryAnalytical Chemistry0302 clinical medicinePhosphorylationDatabases Protein0303 health sciencesProtein Tyrosine Phosphatase Non-Receptor Type 2biologyChemistrySmall molecule3. Good healthCell biologyisothermal titration calorimetryMolecular Docking Simulationmolecular dynamics simulation030220 oncology & carcinogenesis/dk/atira/pure/sustainabledevelopmentgoals/good_health_and_well_beingThermodynamicsHydrophobic and Hydrophilic InteractionsProtein BindingSignal TransductionCell signalingintegrinIntegrinPhosphataseStatic ElectricityBiophysicsAntineoplastic AgentsMolecular Dynamics Simulationta3111mitoxantroneIntegrin alpha1beta1Small Molecule Libraries03 medical and health sciencesSDG 3 - Good Health and Well-beingdifferential scanning fluorimetryHumansBinding siteMolecular Biology030304 developmental biologyT-cell protein tyrosine phosphataseta1182ta3122In vitroProtein Structure TertiaryKineticsCytoplasmbiology.proteinMitoxantronePeptidesBiochimica et Biophysica Acta: Proteins and Proteomics
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Light-induced proton slip and proton leak at the thylakoid membrane

2005

A treatment of leaves of Spinacia oleracea L. with light or with the thiol reagent dithiothreitol in the dark led to partly uncoupled thylakoids. After induction in intact leaves, the partial uncoupling was irreversible at the level of isolated thylakoids. We distinguish between uncoupling by proton slip, which means a decrease of the H+/e(-) -ratio due to less efficient proton pumping, and proton leak as defined by enhanced kinetics of proton efflux. Proton slip and proton leak made about equal contributions to the total uncoupling. The enhanced proton efflux kinetics corresponded to reduction of subunit CF1-gamma of the ATP synthase as shown by fluorescence labeling of thylakoid proteins …

SpinaciaLightProtonPhysiologyKineticsAnalytical chemistryPlant ScienceThylakoidsDithiothreitolElectron Transportchemistry.chemical_compoundSpinacia oleraceaChloroplast Proton-Translocating ATPasesPhotosynthesisATP synthasebiologybiology.organism_classificationPlant LeavesDithiothreitolchemistryPhotophosphorylationThylakoidbiology.proteinBiophysicsProtonsThioredoxinAgronomy and Crop ScienceATP synthase alpha/beta subunitsJournal of Plant Physiology
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NineTeen Complex-subunit Salsa is required for efficient splicing of a subset of introns and dorsal-ventral patterning

2020

© 2020 Rathore et al. This article is distributed exclusively by the RNASociety for the first 12 months after the full-issue publication date (see http://rnajournal.cshlp.org/site/misc/terms.xhtml). After 12 months, it is available under a Creative Commons License (Attribution-NonCommercial 4.0 International), as described at http://creativecommons.org/licenses/by-nc/4.0/.

SpliceosomeBiochemistry & Molecular BiologyRNA SplicingBiologySplicingGermlineArticleMidblastulaDorsal-ventral patterning03 medical and health sciencesAnimalsDrosophila ProteinsFemale fertilityGurkenMolecular BiologyGene030304 developmental biologyBody Patterning0303 health sciencesMessenger RNA030302 biochemistry & molecular biologyfungiIntronGene Expression Regulation DevelopmentalTransforming Growth Factor alphaRNA Helicase AIntronsCell biologyDorsal-ventral patterning; Drosophila; Female fertility; Gurken; Splicing; dorsal–ventral patterning; female fertility; splicingDNA-Binding ProteinsDrosophila melanogasterRNA splicingSpliceosomesFemaleDrosophilaInfertility Female
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Prognostic importance of DNA from human papillomavirus in patients with oral squamous cell carcinoma.

2021

Survival of patients with oral squamous cell carcinoma (OSCC) is generally low, with the likelihood of locoregional recurrence or disease progression (LR/DP). Knowledge of prognostic factors for survival is key to achieving an understanding and increased survival. The present study aimed to identify prognostic factors for patients with OSCC, especially the presence of DNA from human papillomavirus (HPV). Retrospective cohort study including 119 patients with OSCC treated at the National Cancer Institute in Mexico City (2009-2013). Clinical information was obtained from patient records including LR/DP. Formalin-fixed, paraffin-embedded tissues were obtained and used for detecting DNA from di…

Squamous Cell Carcinoma of Head and NeckPapillomavirus InfectionsAlphapapillomavirusPrognosisOropharyngeal NeoplasmsOtorhinolaryngologyramal asymmetryHead and Neck NeoplasmsDNA ViralCarcinoma Squamous CellHumansSurgeryodontogenic cystsMouth Neoplasmscondylar asymmetryNeoplasm Recurrence LocalGeneral DentistryPapillomaviridaeUNESCO:CIENCIAS MÉDICASRetrospective StudiesMedicina oral, patologia oral y cirugia bucal
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Stable expression in HEK-293 cells of the rat alpha3/beta4 subtype of neuronal nicotinic acetylcholine receptor.

1996

The alpha3/beta4 subtype of neuronal nicotinic acetylcholine receptor (nAChR) was stably expressed in human embryonic kidney (HEK) 293 cells that co-expressed a voltage-gated Ca2+ channel. alpha3/beta4-nAChR-expressing clones were identified using the fura-2 Ca2+ imaging technique, and were further characterised by single-cell and whole-cell patch-clamp studies. Acetylcholine (ACh) induced fast activating currents which showed desensitisation and inward rectification. The conductance of the ACh-activated channel was 29 pS. The order of potency of the nicotinic agonists tested was cytisine approximately = nicotine > acetylcholine. The EC50 value for ACh was 145 microM; the Hill coefficient w…

Stable expressionPatch-Clamp Techniquesα3/β4 nAChRBiophysicsNicotinic AntagonistsPharmacologyReceptors NicotinicTransfectionBiochemistryCell LineGanglionic nAChRCa2+ imagingGanglion type nicotinic receptorStructural BiologyMuscarinic acetylcholine receptorGeneticsmedicineAnimalsHumansNicotinic AgonistsNicotinic AntagonistHEK cellMolecular BiologyNeuronsurogenital systemChemistryMuscarinic acetylcholine receptor M3Cell BiologyAcetylcholineRecombinant ProteinsRatsNicotinic acetylcholine receptorNicotinic agonistCalciumCalcium ChannelsAlpha-4 beta-2 nicotinic receptorAcetylcholinemedicine.drugFEBS letters
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Alpha-toxin of Staphylococcus aureus

1991

Alpha-toxin, the major cytotoxic agent elaborated by Staphylococcus aureus, was the first bacterial exotoxin to be identified as a pore former. The protein is secreted as a single-chain, water-soluble molecule of Mr 33,000. At low concentrations (less than 100 nM), the toxin binds to as yet unidentified, high-affinity acceptor sites that have been detected on a variety of cells including rabbit erythrocytes, human platelets, monocytes and endothelial cells. At high concentrations, the toxin additionally binds via nonspecific absorption to lipid bilayers; it can thus damage both cells lacking significant numbers of the acceptor and protein-free artificial lipid bilayers. Membrane damage occu…

Staphylococcus aureusCell Membrane PermeabilityToxinBacterial ToxinsCell MembraneBiologymedicine.disease_causeHemolysin ProteinsApplied Microbiology and BiotechnologyTransmembrane proteinExocytosisCell membraneHemolysin ProteinsStructure-Activity Relationshipmedicine.anatomical_structureBiochemistrymedicineBiophysicsAnimalsHumansLipid bilayerStaphylococcus aureus alpha toxinExotoxinResearch ArticleMicrobiological Reviews
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