Search results for "Anus"

showing 10 items of 841 documents

Self-assembly of janus dendrimers into uniform dendrimersomes and other complex architectures

2010

Janus Drug Delivery Vehicle Efficient drug delivery vehicles need to be produced in a limited size range and with uniform size distribution. The self-assembly of traditional small-molecule and polymeric amphiphiles has led to the production of micelles, liposomes, polymeric micelles, and polymersomes for use in drug delivery applications. Now, Percec et al. (p. 1009 ) describe the self-assembly of Janus-type (i.e., two-headed) dendrimers to produce monodisperse supramolecular constructs, termed “dendrimersomes,” and other complex architectures. The structures, which showed long-term stability as well as very narrow size distributions, were easily produced by the injection of an ethanolic so…

Models MolecularDendrimersMaterials scienceSurface Propertiesta221Complex ArchitecturesNanotechnologyMolecular Dynamics SimulationSurface-Active AgentsBiomimetic MaterialsDendrimerAmphiphileJanusta218LiposomeDrug Carriersta214MultidisciplinaryAntibiotics Antineoplasticta114Molecular StructureVesicleCryoelectron MicroscopyWaterMembranes ArtificialNanostructuresJanus DendrimersSelf-AssemblyMembraneUniform DendrimersomesDoxorubicinPolymersomeSelf-assemblyHydrophobic and Hydrophilic InteractionsScience
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Pharmacology and safety of tofacitinib in ulcerative colitis.

2020

The use of Janus kinase (JAK) inhibitors is a new approach in the therapy of inflammatory diseases with immune base. Tofacitinib is one of these inhibitors targeting JAK1 and JAK3, and its efficacy has been demonstrated in the treatment of moderate to severe ulcerative colitis (UC). It is a small synthetic molecule administered orally, with a fast bioavailability and elimination rate, predictable pharmacokinetics and lack of immunogenicity, which are convenient characteristics for both efficacy and safety. This article reviews the pharmacological characteristics of tofacitinib and its safety profile.

Moderate to severePharmacologyHerpes ZosterArthritis Rheumatoid03 medical and health sciences0302 clinical medicineImmune systemPharmacokineticsPiperidinesNeoplasmsMedicineHerpes Zoster VaccineHumansJanus Kinase InhibitorsDrug InteractionsTofacitinibbusiness.industryImmunogenicityJanus Kinase 3Janus Kinase 1Venous Thromboembolismmedicine.diseaseUlcerative colitisBioavailabilityPyrimidines030220 oncology & carcinogenesis030211 gastroenterology & hepatologyColitis UlcerativeJanus kinasebusinessGastroenterologia y hepatologia
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Matheus Molanus, in G. C. SCIOLLA (a cura di), Cielo terra e acque: il paesaggio nella pittura fiamminga e olandese tra Cinquecento e Seicento, Torin…

2006

Matheus Molanus, in G. C. SCIOLLA (a cura di), Cielo terra e acque: il paesaggio nella pittura fiamminga e olandese tra Cinquecento e Seicento, Torino, Elede, 2006 p. 35-133

Molanus pittura fiamminga pittura olandese paesaggio cinquecento seicento cielo terra acqueSettore L-ART/02 - Storia Dell'Arte Moderna
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Synthetic antitumor vaccines containing MUC1 glycopeptides with two immunodominant domains-induction of a strong immune response against breast tumor…

2011

A shot in the arm for cancer treatment: two MUC1 tetanus toxoid vaccines were synthesized and induced a strong immune response in mice. The antibodies elicited by the vaccines show a high selectivity for the tumor cells in mammary carcinoma tissues and also distinguish between tumor tissues at different stages.

Molecular ConformationAntineoplastic AgentsBreast Neoplasmscomplex mixturesCancer VaccinesCatalysisBreast tumorMiceImmune systemmedicineAnimalsMUC1Mice Inbred BALB CVaccines SyntheticbiologyTetanusChemistryMucin-1ToxoidGlycopeptidesMammary Neoplasms ExperimentalGeneral Chemistrymedicine.diseaseGlycopeptideCancer researchbiology.proteinMCF-7 CellsExperimental pathologyFemaleAntibodyDrug Screening Assays AntitumorAngewandte Chemie (International ed. in English)
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Enzyme-accelerated and structure-guided crystallization of calcium carbonate: Role of the carbonic anhydrase in the homologous system

2014

Abstract The calcareous spicules from sponges, e.g. from Sycon raphanus, are composed of almost pure calcium carbonate. In order to elucidate the formation of those structural skeletal elements, the function of the enzyme carbonic anhydrase (CA), isolated from this species, during the in vitro calcium carbonate-based spicule formation, was investigated. It is shown that the recombinant sponge CA substantially accelerates calcium carbonate formation in the in vitro diffusion assay. A stoichiometric calculation revealed that the turnover rate of the sponge CA during the calcification process amounts to 25 CO2 s−1 × molecule CA−1. During this enzymatically driven process, initially pat-like pa…

Molecular Sequence DataInorganic chemistryBiomedical Engineeringchemistry.chemical_elementCalciumBiochemistryCalcium Carbonatelaw.inventionBiomaterialschemistry.chemical_compoundSponge spiculelawSpectroscopy Fourier Transform InfraredAnimalsAmino Acid SequenceSycon raphanusCrystallizationMolecular BiologyCarbonic AnhydrasesMineralsbiologyGeneral MedicineElementsbiology.organism_classificationPoriferaCrystallographySpongeCalcium carbonatechemistryCrystallizationCalcareousBiotechnologyBiomineralizationActa Biomaterialia
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Liquid methane at extreme temperature and pressure: Implications for models of Uranus and Neptune

2012

We present large scale electronic structure based molecular dynamics simulations of liquid methane at planetary conditions. In particular, we address the controversy of whether or not the interior of Uranus and Neptune consists of diamond. In our simulations we find no evidence for the formation of diamond, but rather sp2-bonded polymeric carbon. Furthermore, we predict that at high tem- perature hydrogen may exist in its monoatomic and metallic state. The implications of our finding for the planetary models of Uranus and Neptune are in detail discussed.

Monatomic gasMaterials sciencePhysics and Astronomy (miscellaneous)HydrogenUranusDiamondchemistry.chemical_elementElectronic structureengineering.materialAstrobiologyMolecular dynamicschemistryNeptunePhysics - Chemical PhysicsengineeringCarbonPhysics - Computational PhysicsCondensed Matter - Statistical MechanicsAstrophysics - Earth and Planetary Astrophysics
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The Antigerminative Activity of Twenty-Seven Monoterpenes

2010

Made available in DSpace on 2013-08-28T14:11:28Z (GMT). No. of bitstreams: 1 WOS000282221100055.pdf: 183420 bytes, checksum: 31d5a1904cd2424113da7989e2e65f14 (MD5) Made available in DSpace on 2013-09-30T18:36:29Z (GMT). No. of bitstreams: 2 WOS000282221100055.pdf: 183420 bytes, checksum: 31d5a1904cd2424113da7989e2e65f14 (MD5) WOS000282221100055.pdf.txt: 26866 bytes, checksum: 653cedb4f682463998ef7f37cae8dd63 (MD5) Previous issue date: 2010-09-01 Submitted by Vitor Silverio Rodrigues (vitorsrodrigues@reitoria.unesp.br) on 2014-05-20T13:48:46Z No. of bitstreams: 2 WOS000282221100055.pdf: 183420 bytes, checksum: 31d5a1904cd2424113da7989e2e65f14 (MD5) WOS000282221100055.pdf.txt: 26866 bytes, ch…

MonoterpenePharmaceutical ScienceRaphanusphytotoxicityBiologyradicle elongationArticleLepidium sativumRaphanusAnalytical ChemistryBorneollcsh:QD241-441Structure-Activity Relationshipchemistry.chemical_compoundlcsh:Organic chemistryDrug DiscoveryBotanyRadiclePhysical and Theoretical ChemistryCarvoneDose-Response Relationship DrugOrganic Chemistrymonoterpenesfood and beveragesbiology.organism_classificationHorticultureEucalyptolgerminationchemistryChemistry (miscellaneous)GerminationAlcoholsSeedsMonoterpenesMolecular Medicinemonoterpenes; germination; radicle elongation; phytotoxicityGeraniolMolecules
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Los motivos caballerescos del manuscrito encontrado y el falso cronista en El Señor de los Anillos

2013

El manuscrito encontrado es uno de los motivos presentes en la mayoría de los libros de caballerías y, si bien se trata de un elemento de origen remoto, su frecuente aparición en estas obras, ha hecho que se convierta en uno de sus rasgos característicos. En este artículo se pone de manifiesto la forma en que se plasma este mismo motivo en El Señor de los Anillos de J.R.R. Tolkien, autor que tenía una especial vinculación con la literatura medieval y con lo hispánico.

Motivos caballerescos; manuscrito encontrado; falsa traducción; cronista; Tolkien; El Señor de los Anillos.TolkienMotivos caballerescosEl Señor de los Anillos.cronistamanuscrito encontradofalsa traducción
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: Noeud visuel, site monastique, production d'image

2018

Le manuscrit 1 conservé à la Bibliothèque municipale de Semur est l’un des plus anciens manuscrits conservés en Bourgogne, sinon le plus ancien, pour les uns à dater autour de l’an mil, pour les autres à rattacher, vers la même époque, au grand mouvement des « abbés réformateurs » et aux livrets hagio-liturgiques de prestige. C’est un recueil composite, de 260 mm par 207, comprenant 78 feuillets réunis en cahiers, et provenant de l’abbaye de Saint-Jean de Réôme (Moutiers-Saint-Jean), en Côte-d’Or. Les différentes pièces qui le composent furent probablement réalisées entre le Xe et le XVe siècle ; la reliure en carton date de 1834.Au fil de son histoire, au cours des différentes étapes de sa…

Moutiers Saint-Jeanmanuscrit hagiographique et liturgiquemoyen âge[SHS.HIST] Humanities and Social Sciences/HistorylettrinesBourgogne-Franche-ComtéSemur-en-Auxois[SHS.ART] Humanities and Social Sciences/Art and art history[SHS.ART]Humanities and Social Sciences/Art and art history[SHS.HIST]Humanities and Social Sciences/HistoryCôte d’OrAbbaye de Saint-Jean de Réôme
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Hagiographie et diplomatique dans le monachisme réformé en Bourgogne au miroir du manuscrit 1 de Semur-en-Auxois

2014

International audience; Le propos de cet article est, à partir de l'exemple du manuscrit 1 de la Bibliothèque municipale de Semur-en-Auxois, de penser la question de la transtextualité, en empruntant cette notion à la théorie littéraire, tout en la restituant non seulement en fonction du texte de l'énoncé, mais également en relation aux signes visuels et matériels de la mise par écrit, « la raison graphique », sur la longue durée. Il s'agit aussi d'interroger le rôle des différents chantiers scripturaires propres à la "renovatio" monastique au tournant des X e et XI e siècles, comme l'un des moyens de « mise en norme » dans le cadre d'une redéfinition plus large de la place occupée par les …

Moutiers-Saint-JeanmonachismeMoyen Âge[ SHS.HIST ] Humanities and Social Sciences/Historyhagiographie[SHS.HIST] Humanities and Social Sciences/Historymanuscritdiplômes royaux[SHS.HIST]Humanities and Social Sciences/History16. Peace & justiceSaint-Jean de Réôme
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