Search results for "Contraction"

showing 10 items of 1092 documents

Different muscarine receptors mediate the prejunctional inhibition of [3H]-noradrenaline release in rat or guinea-pig iris and the contraction of the…

1989

To investigate the muscarine receptor type mediating inhibition of [3H]-noradrenaline release from the isolated rat and guinea-pig iris we have determined the potency of antimuscarinic drugs to antagonize the methacholine-induced inhibition of [3H]-noradrenaline overflow evoked by field stimulation (3 Hz, 2 min). The prejunctional apparent affinities were compared with those obtained for postjunctional muscarine receptors mediating the methacholine-induced contraction of the isolated rabbit iris sphincter muscle. Prejunctional apparent affinity constants of pirenzepine (6.67), himbacine (8.51), methoctramine (7.92), 4-diphenylacetoxy-N-methylpiperidine methiodide (4-DAMP, 8.00), hexahydro-d…

medicine.medical_specialtyContraction (grammar)Iris sphincter muscleIrisIn Vitro TechniquesBiologyGuinea pigNorepinephrinechemistry.chemical_compoundPiperidinesInternal medicineMuscarinic acetylcholine receptormedicineAnimalsMethacholine CompoundsNeurotransmitterReceptorPharmacologyMuscarineMuscle SmoothRats Inbred StrainsGeneral MedicineReceptors MuscarinicElectric StimulationRatsKineticsmedicine.anatomical_structureEndocrinologychemistrySphincterRabbitsMuscle ContractionNaunyn-Schmiedebergs Archives of Pharmacology
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Analysis of Rabbit Vascular Responses to DBI, an Ingol Derivative Isolated from Euphorbia canariensis

1997

Abstract We have analysed the effects of 7,12-O-diacetyl-8-O-benzoil-2,3-diepiingol (DBI), an ingol derivative isolated from E. canariensis, on isometric tension developed by isolated rabbit basilar and carotid arteries. Concentration-response curves to DBI (10−8 - 3 × 10−5 m) were obtained cumulatively in both arteries at resting tension and active tone (KC1, 50 mm). At resting tension, DBI induced a concentration-dependent contraction, which was not inhibited in Ca2+-free medium. H7 (1-(5-isoquinoline sulphonyl)-2-methylpiperazine dichloride) (10−4 m) inhibited the DBI-induced contraction both in basilar and in carotid arteries. Calmidazolium (10−4 m) inhibited the maximum contraction of …

medicine.medical_specialtyContraction (grammar)LatexCarotid Artery CommonMuscle RelaxationPharmaceutical ScienceProstacyclinNitric OxideNitroarginineMuscle Smooth VascularEuphorbia canariensisCalmodulin1-(5-Isoquinolinesulfonyl)-2-MethylpiperazineInternal medicinemedicine.arterymedicineBasilar arteryAnimalsEnzyme InhibitorsProtein Kinase CPharmacologyPlants MedicinalLagomorphabiologyPlant Extractsbiology.organism_classificationEpoprostenolEndocrinologymedicine.anatomical_structureBasilar ArteryCirculatory systemcardiovascular systemCalciumRabbitsDiterpenesMuscle Contractionmedicine.drugBlood vesselArteryJournal of Pharmacy and Pharmacology
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Changes in motor unit characteristics after eccentric elbow flexor exercise

2010

Morphological evidence suggests that fast-twitch fibers are prone to disruption of their membrane structures by eccentric exercise. However, it is unclear how this is reflected in the discharge rate and action potential propagation of individual motor units, especially at high contraction levels. High-density surface electromyograms were recorded from biceps brachii muscle and decomposed to individual motor unit action potentials at isometric contraction levels between 10% and 75% of maximal voluntary contraction (MVC) before intermittent maximal elbow flexor eccentric exercise, and two hours (2H), two days (2D) and four days (4D) post-exercise. Maximal voluntary force decreased by 21.3±5.6…

medicine.medical_specialtyContraction (grammar)Motor unit characteristicsElbow flexorAction potentialBiceps brachii musclebusiness.industry030209 endocrinology & metabolismPhysical Therapy Sports Therapy and Rehabilitation030229 sport sciencesIsometric exerciseMotor unit03 medical and health sciences0302 clinical medicineInternal medicineCardiologyMedicineEccentricOrthopedics and Sports MedicinebusinessJapanese Journal of Physical Fitness and Sports Medicine
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Effects of inhibitors of cGMP-dependent protein kinase in atrial heart and aortic smooth muscle from rats

1995

Several activators of cGMP-dependent protein kinase (protein kinase G) such as 8-Br-cGMP reduced force of contraction in rat left atria. Inhibitors of protein kinase G antagonized the negative inotropic effect of 8-Br-cGMP but not of acetylcholine in atria. However, the acetylcholine-induced relaxation in aortic rings was significantly inhibited by protein kinase G inhibition. It is concluded that the reduction by 8-Br-cGMP of force of contraction in atria is related to activation of protein kinase G. In response to acetylcholine, activation of protein kinase G is probably a major step in smooth muscle relaxation but is not involved in the reduction of force of contraction in atria.

medicine.medical_specialtyContraction (grammar)Muscle RelaxationAorta ThoracicIn Vitro TechniquesMuscle Smooth VascularIsometric ContractionInternal medicineCyclic GMP-Dependent Protein KinasesmedicineAnimalsHeart AtriaProtein kinase ACyclic GMPRho-associated protein kinasePharmacologybiologyHeartMyocardial ContractionAcetylcholineRatsEnzyme ActivationEndocrinologyEnzyme inhibitorSecond messenger systemcardiovascular systembiology.proteinmedicine.symptomcGMP-dependent protein kinaseAcetylcholineMuscle Contractionmedicine.drugMuscle contractionEuropean Journal of Pharmacology
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Neuromuscular fatigue differs following unilateral vs bilateral sustained submaximal contractions

2011

The purpose of the present study was to compare the mechanisms of fatigue induced by a unilateral vs a bilateral submaximal isometric knee extension. Ten physically active men completed two experimental sessions, randomly presented. They were asked to maintain an isometric knee extension force corresponding to 20% of the maximal voluntary contraction (MVC) until task failure with one leg (unilateral) vs two legs (bilateral). MVCs were performed before and after the sustained contraction. Transcutaneous electrical stimuli were used to examine central (voluntary activation) and peripheral (peak doublet force at rest) fatigue on the exercised leg. Time to task failure was significantly shorter…

medicine.medical_specialtyContraction (grammar)Muscle fatiguemedicine.diagnostic_testbusiness.industryPhysical Therapy Sports Therapy and Rehabilitation030229 sport sciencesIsometric exerciseElectromyographybehavioral disciplines and activitiesPeripheral03 medical and health sciences0302 clinical medicineVoluntary contractionPhysical medicine and rehabilitationFemoral nerveNeuromuscular fatiguemedicinePhysical therapyOrthopedics and Sports Medicinebusinesspsychological phenomena and processes030217 neurology & neurosurgeryScandinavian Journal of Medicine & Science in Sports
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The Sources of Ca2+ for Muscarinic Receptor-induced Contraction in the Rat Ileum

1996

Abstract The contractile responses obtained by activation of different muscarinic receptor subtypes in the longitudinal muscle of the rat ileum and especially the responses of this muscle to acetylcholine in a Ca2+-free medium have been investigated. In Ca2+-containing solution, acetylcholine elicited similar concentration-dependent contractile responses in the duodenum, jejunum and ileum strips of the rat intestine. The response to a maximal concentration of the agonist (1 μM) consisted of a rapid phasic response followed by a slower tonic one. Nifedipine completely relaxes or inhibits the sustained response and only partially diminishes the phasic one, which suggests that the phasic contr…

medicine.medical_specialtyContraction (grammar)NifedipinePharmaceutical ScienceIn Vitro TechniquesMuscarinic AgonistsBiologyTonic (physiology)chemistry.chemical_compoundIleumInternal medicineMuscarinic acetylcholine receptormedicineMethoctramineAnimalsRats WistarPharmacologyMuscle SmoothPirenzepineCalcium Channel BlockersReceptors MuscarinicPirenzepineAcetylcholineRatsAtropineEndocrinologychemistryCalciumFemalemedicine.symptomAcetylcholineMuscle Contractionmedicine.drugMuscle contractionJournal of Pharmacy and Pharmacology
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Soleus and lateral gastrocnemius H-reflexes during standing with unstable footwear

2015

Introduction: Unstable footwear has been shown to increase lower extremity muscle activity, but the reflex response to perturbations induced by this intervention is unknown. Methods: Twenty healthy subjects stood in stable and unstable footwear conditions (presented randomly) while H-reflex amplitude and background muscle activity were measured in the soleus and lateral gastrocnemius (LG) muscles. Results: Wearing unstable footwear resulted in larger H-reflexes (normalized to the maximal M-wave) for the LG (+12%; P = 0.025), but not for the soleus (+4%; P > 0.05). Background activity of both muscles was significantly higher in the unstable condition. Conclusions: The H-reflex facilitation o…

medicine.medical_specialtyContraction (grammar)Physiologybusiness.industryHealthy subjectsAnatomyGaitReflex responseCellular and Molecular NeurosciencePhysiology (medical)Internal medicineMotor unit recruitmentCardiologymedicineReflexNeurology (clinical)H-reflexbusinessLateral gastrocnemiusMuscle & Nerve
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Isolated human chorionic vascular reactivity: Technical considerations for fresh preparations

1998

1. 1. Sixty chorionic vascular rings from normal term placentas were immersed in an organ bath for isometric tension recording to study (A) the contractile response to 120 mM of potassium chloride (KCI) after adjustment and equilibration to 1–5 g of passive tension; and (B) the concentration-response curve to KCI after adjustment and equilibration to the optimal passive tension. 2. 2. Adjustment to 4 g of passive tension elicited the maximal (P<0.007) and the latest (P<0.006) KCl-induced contraction among arterial rings. Venous rings showed the greatest contraction when adjusted to 3 g, but the differences were not significant except when compared to 1 g of passive tension (P<0.03). 3. 3. T…

medicine.medical_specialtyContraction (grammar)PlacentaPotassiumchemistry.chemical_elementIsometric exerciseIn Vitro TechniquesMuscle Smooth VascularPotassium ChlorideVeinsPregnancyIsometric ContractionPlacentaInternal medicinemedicineHumansPharmacologyArteriesChorionKineticsmedicine.anatomical_structureEndocrinologychemistryCirculatory systemFemalemedicine.symptomVasoconstrictionBlood vesselArteryGeneral Pharmacology: The Vascular System
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Sonographische Darstellbarkeit der Gallenwege und Beurteilbarkeit der Gallenblasenkinetik bei gesunden Neugeborenen

2008

The gallbladder and the biliary tract of 85 neonates were sonographically examined, in the fasting state. The gallbladder was detectable in all neonates and showed a measurable contraction. Two types of biliary contraction could be observed: a concentric contraction of length, depth and width (concentric type) or a contraction of depth and width (collapse type). The grade of postprandial contraction was independent of the level of serum bilirubin. Furthermore, sonographic criteria were established allowing the differentiation of the bile ducts and their discrimination from hepatic arteries.

medicine.medical_specialtyContraction (grammar)business.industryGallbladderGastroenterologySerum bilirubinmedicine.anatomical_structurePostprandialBiliary tractInternal medicinemedicineUltrasound imagingRadiology Nuclear Medicine and imagingbusinessFasting stateUltraschall in der Medizin
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Alteration of Esophageal Peristalsis by Pentagastrin in Patients with Diffuse Esophageal Spasm

1975

Although it has been shown that gastrin and gastric alkalinization affect the lower esophageal sphincter, in vivo studies have not demonstrated a measurable effect of pentagastrin on esophageal peristalsis. In 9 patients with diffuse esophageal spam and in 10 control subjects esophageal peristalsis was recorded before and after pentagastrin infections. Subcutaneous pentagastrin increased peak amplitude significantly more in patients, 31.2 +/- 8.1 mm Hg (mean +/- S.E.M.), than in controls, 12.1 +/- 5.1 mm Hg (P less than 0.02). Max. duration of contraction waves in patients showed a rise of 11.3 +/- 2.7 sec as compared to controls, 1.9 +/- 0.9 sec (P less than 0.01). The effect of pentagastr…

medicine.medical_specialtyContraction (grammar)business.industrydigestive oral and skin physiologyGastroenterologyGastroenterologyDenervation supersensitivityPentagastrinIn vivoInternal medicinemedicineIn patientEsophageal spasmEsophageal peristalsisbusinessGastrinmedicine.drugScandinavian Journal of Gastroenterology
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