Search results for "D2"

showing 10 items of 2418 documents

D2R striatopallidal neurons inhibit both locomotor and drug reward processes.

2009

The specific functions of dopamine D(2) receptor-positive (D(2)R) striatopallidal neurons remain poorly understood. Using a genetic mouse model, we found that ablation of D(2)R neurons in the entire striatum induced hyperlocomotion, whereas ablation in the ventral striatum increased amphetamine conditioned place preference. Thus D(2)R striatopallidal neurons limit both locomotion and, unexpectedly, drug reinforcement.

Time FactorsstriatumParkinson's diseaseStriatumNeurons -- drug effectsEnkephalins -- metabolism10263 Institute of Experimental ImmunologyMiceDopamine Uptake InhibitorsTyrosine 3-Monooxygenase -- geneticsCorpus Striatum -- cytologyDiphtheria ToxinGlutamate Decarboxylase -- metabolismstriatum; indirect opathway; A2A receptors; D2 receptors; locomotion; amphetamine addiction; Parkinson's diseaseNeuronsamphetamine addictionGlutamate DecarboxylaseGeneral NeuroscienceAmphetamine -- pharmacologyNeurodegeneration2800 General NeuroscienceEnkephalinsSciences bio-médicales et agricoleslocomotionmedicine.anatomical_structureA2A receptorsIntercellular Signaling Peptides and ProteinsReceptors Dopamine D2 -- metabolismPsychologyLocomotionmedicine.drugHeparin-binding EGF-like Growth FactorProtein BindingGlobus Pallidus -- cytologyReceptors Dopamine D2 -- deficiencyReinforcement ScheduleTyrosine 3-MonooxygenaseGlutamate Decarboxylase -- geneticsLocomotion -- geneticsIntercellular Signaling Peptides and Proteins -- genetics610 Medicine & healthMice TransgenicNerve Tissue ProteinsDiphtheria Toxin -- pharmacologyGlobus PallidusNeurons -- physiologyLocomotion -- drug effectsRewardDopamineDopamine receptor D2medicineNerve Tissue Proteins -- metabolismAnimalsGene Expression Regulation -- geneticsAmphetamineD2 receptorsReceptors Adenosine A2Receptors Dopamine D2indirect opathwayVentral striatumReceptors Adenosine A2 -- geneticsDopamine Uptake Inhibitors -- pharmacologymedicine.diseaseConditioned place preferenceCorpus StriatumMice Inbred C57BLGene Expression Regulation -- drug effectsAmphetaminenervous systemGene Expression RegulationProtein Binding -- drug effectsTyrosine 3-Monooxygenase -- metabolism570 Life sciences; biologyAutoradiographyConditioning OperantNeuronConditioning Operant -- physiologyNeuroscienceEnkephalins -- geneticsNature neuroscience
researchProduct

The Effect of Calcium on the Cohesive Strength and Flexural Properties of Low-Methoxyl Pectin Biopolymers.

2019

Abstract: Pectin binds the mesothelial glycocalyx of visceral organs, suggesting its potential role as a mesothelial sealant. To assess the mechanical properties of pectin films, we compared pectin films with a less than 50% degree of methyl esterification (low-methoxyl pectin, LMP) to films with greater than 50% methyl esterification (high-methoxyl pectin, HMP). LMP and HMP polymers were prepared by step-wise dissolution and high-shear mixing. Both LMP and HMP films demonstrated a comparable clear appearance. Fracture mechanics demonstrated that the LMP films had a lower burst strength than HMP films at a variety of calcium concentrations and hydration states. The water content also influe…

Toughnessfood.ingredientanimal structuresPectin0206 medical engineeringpolysaccharidesPharmaceutical Sciencechemistry.chemical_element02 engineering and technologyCalciumPolysaccharideArticleAnalytical Chemistrylcsh:QD241-441Medicinal and Biomolecular Chemistryfoodlcsh:Organic chemistryFlexural strengthTheoretical and Computational ChemistryDrug DiscoveryFlexural Strengthotorhinolaryngologic diseasesPhysical and Theoretical ChemistryDissolutionchemistry.chemical_classificationOrganic ChemistryWaterPolymer021001 nanoscience & nanotechnology020601 biomedical engineeringstomatognathic diseasesChemical engineeringchemistryfracture mechanicsChemistry (miscellaneous)Molecular MedicinePectinsTitrationCalcium0210 nano-technologymaterial propertiesmethoxylationhydrationMolecules (Basel, Switzerland)
researchProduct

Da poeta a poeta, da traduttore a traduttore: il carteggio tra Umberto Saba e Tomàs Garcés

2015

Riassunto: Il rapporto personale tra Umberto Saba e Tomàs Garcés cominciò agli inizi degli anni  Trenta e si interruppe poco prima della guerra civile spagnola. Quest’articolo analizza  ed edita per la prima volta tutte le lettere scritte da Saba al poeta catalano che sono  state conservate presso l’archivio della famiglia Garcés.   Parole chiave: poesia, traduzione, Umberto Saba, Tomàs Garcés   Abstract: The personal relationship between Umberto Saba and Tomàs Garcés began in the early  thirties and stopped just before the Spanish Civil War. This article analyses and edits for  the first time all the letters written by Saba to the Catalan poet that have been preserved  in the archives of f…

Traducció literàriaHistoryLiterature and Literary TheoryFilologíasmedia_common.quotation_subjectlcsh:Literature (General)lcsh:D111-203Poesialcsh:Medieval historyLanguage and LinguisticspoesiaTomàs Garcésmedia_commonUNESCO::CIENCIAS DE LAS ARTES Y LAS LETRAStraduzionePoetryPersonal relationshipFilologías. GeneralidadesArtlcsh:PN1-6790language.human_languageLiterary translationSpanish Civil Warlcsh:D204-475:CIENCIAS DE LAS ARTES Y LAS LETRAS [UNESCO]languagePoetryCatalanUmberto SabaHumanitieslcsh:Modern history 1453-Scripta: Revista Internacional de Literatura i Cultura Medieval i Moderna
researchProduct

Stability of phospholipase D in primary astrocytes.

2002

Induction of expression and proteolytic breakdown of phospholipase D (PLD) isoforms in primary astrocyte cultures have been investigated. Astrocytes express both PLD1 and 2 and are dependent on PLD activity for cell proliferation [K. Kotter, J. Klein, J. Neurochem. 73 (1999) 2517]. Competitive RT-PCR analysis demonstrated a higher level of PLD1 mRNA than PLD2 mRNA (8.9 vs. 0.9amol/microg RNA, respectively). Treatment of astroglial cultures with the phorbol ester, 4beta-phorbol-12beta,13alpha-dibutyrate (0.1 microM), for 24-48h selectively induced PLD1b but not PLD1a or 2 expression as shown by PCR and Western blot; the effect was sensitive to Go 6976. In cells transiently permeabilized with…

Transcription GeneticBiophysicsCycloheximideBiologyBiochemistryGene Expression Regulation EnzymologicOligodeoxyribonucleotides Antisensechemistry.chemical_compoundWestern blotmedicinePhospholipase DAnimalsCycloheximideMolecular BiologyProtein kinase CCells CulturedPhorbol 1213-DibutyrateProtein Synthesis InhibitorsMessenger RNAmedicine.diagnostic_testPhospholipase DReverse Transcriptase Polymerase Chain ReactionPLD2BrainCell BiologyMolecular biologyCell biologyRatsIsoenzymesKineticsmedicine.anatomical_structurechemistryAnimals NewbornCytoplasmAstrocytesCell DivisionAstrocyteBiochemical and biophysical research communications
researchProduct

Generation and characterization of tTS-H4: a novel transcriptional repressor that is compatible with the reverse tetracycline-controlled TET-ON system

2007

Background Conditional gene regulatory systems ensuring tight and adjustable expression of therapeutic genes are central for developing future gene therapy strategies. Among various regulatory systems, tetracycline-controlled gene expression has emerged as a safe and reliable option. Moreover, the tightness of tetracycline-regulated gene switches can be substantially improved by complementing transcriptional activators with antagonizing repressors. Methods To develop novel tetracycline-responsive transcriptional repressors, we fused various transcriptional silencing domains to the TetR (B/E) DNA-binding and dimerization domain of the Tn10-encoded tetracycline resistance operon (TetR (B/E)).…

Transcription GeneticOperonRepressorBiologyHistone DeacetylasesHistonesMicechemistry.chemical_compoundGenes ReporterDrug DiscoveryGeneticsAnimalsHumansGene silencingTetRPromoter Regions GeneticMolecular BiologyGenetics (clinical)Regulation of gene expressionYY1Genetic TherapyTetracyclineMolecular biologyHDAC4Repressor ProteinsGene Expression RegulationchemistryGATAD2BNIH 3T3 CellsMolecular Medicine
researchProduct

Robust existence of nonhyperbolic ergodic measures with positive entropy and full support

2021

We prove that for some manifolds $M$ the set of robustly transitive partially hyperbolic diffeomorphisms of $M$ with one-dimensional nonhyperbolic centre direction contains a $C^1$-open and dense subset of diffeomorphisms with nonhyperbolic measures which are ergodic, fully supported and have positive entropy. To do so, we formulate abstract conditions sufficient for the construction of an ergodic, fully supported measure $\mu$ which has positive entropy and is such that for a continuous function $\phi\colon X\to\mathbb{R}$ the integral $\int\phi\,d\mu$ vanishes. The criterion is an extended version of the control at any scale with a long and sparse tail technique coming from the previous w…

Transitive relationPure mathematicsHyperbolicityMathematics::Dynamical SystemsDense setContinuous function (set theory)[MATH.MATH-DS]Mathematics [math]/Dynamical Systems [math.DS][MATH.MATH-DS] Mathematics [math]/Dynamical Systems [math.DS]Scale (descriptive set theory)Dynamical Systems (math.DS)Measure (mathematics)Theoretical Computer SciencePositive entropyMathematics (miscellaneous)FOS: MathematicsErgodic theory37D25 37D35 37D30 28D99Mathematics - Dynamical SystemsMathematicsCriterion
researchProduct

Tributyltin(Iv) butyrate: A novel epigenetic modifier with er stress-and apoptosis-inducing properties in colon cancer cells

2021

Organotin(IV) compounds are a class of non-platinum metallo-conjugates exhibiting antitumor activity. The effects of different organotin types has been related to several mechanisms, including their ability to modify acetylation protein status and to promote apoptosis. Here, we focus on triorganotin(IV) complexes of butyric acid, a well-known HDAC inhibitor with antitumor properties. The conjugated compounds were synthesized and characterised by FTIR spectroscopy, multi-nuclear (1H, 13C and 119Sn) NMR, and mass spectrometry (ESI-MS). In the triorganotin(IV) complexes, an anionic monodentate butyrate ligand was observed, which coordinated the tin atom on a tetra-coordinated, monomeric enviro…

Triorganotin(IV) butyratesPharmaceutical ScienceOrganic chemistryApoptosisButyrateArticleHistone DeacetylasesAnalytical ChemistryEpigenesis GeneticButyric acidchemistry.chemical_compoundQD241-441HDAC inhibitorsCell Line TumorSettore BIO/10 - BiochimicaDrug DiscoveryHumansPhysical and Theoretical ChemistrybiologyAcetylationLigand (biochemistry)Endoplasmic Reticulum StressColon cancerHistonechemistryBiochemistryHistone acetylationChemistry (miscellaneous)ApoptosisAcetylationSettore CHIM/03 - Chimica Generale E InorganicaColonic NeoplasmsTributyltinbiology.proteinUnfolded protein responseMolecular MedicineButyric AcidTrialkyltin CompoundsER stressProtein Processing Post-Translational
researchProduct

Competence Utilization for Innovation Capabilities - A Question of Trust?

2015

The purpose of this paper is to show how trust as an organizational value contributes to employee competence utilization in the case of innovation capability. Thus, it is the objective of this paper to analyze the positive impacts, but also potential limits of trust in business management. The research paper uses two different quantitative empirical studies drawn from German and Austrian mid-sized companies to empirically test this interrelation. As a result, the paper determines particular aspects of trust such as accountability, shared norms and the ability to take responsibility to be interrelated with the usage of employee competences and underlines a positive connection between product…

Trust employee competence utilization innovation creativityjel:D83jel:D23lcsh:BusinessTrustemployee competence utilizationinnovationjel:L22jel:O31jel:M11jel:O30jel:L20jel:M14jel:O34jel:L25jel:O32lcsh:HF5001-6182creativityExpert Journal of Business and Management
researchProduct

Mycobacterium tuberculosis Immune Response in Patients With Immune-Mediated Inflammatory Disease

2021

Subjects with immune-mediated inflammatory diseases (IMID), such as rheumatoid arthritis (RA), have an intrinsic higher probability to develop active-tuberculosis (TB) compared to the general population. The risk ranges from 2.0 to 8.9 in RA patients not receiving therapies. According to the WHO, the RA prevalence varies between 0.3% and 1% and is more common in women and in developed countries. Therefore, the identification and treatment of TB infection (TBI) in this fragile population is important to propose the TB preventive therapy. We aimed to study the M. tuberculosis (Mtb) specific T-cell response to find immune biomarkers of Mtb burden or Mtb clearance in patients with different TB …

TuberculosisImmunologyPopulationchemical and pharmacologic phenomenaDiseaseMycobacterium tuberculosisImmune systemmedicineM. tuberculosisImmunology and AllergyCytotoxic T celleducationIFN-γCD27Original Researcheducation.field_of_studybiologybusiness.industryRC581-607bacterial infections and mycosesmedicine.diseasebiology.organism_classificationtuberculosisRheumatoid arthritisImmunologyTumor necrosis factor alphaImmunologic diseases. Allergybusinessimmune-mediated inflammatory disease
researchProduct

Mycobacterium tuberculosis secretory proteins downregulate T cell activation by interfering with proximal and downstream T cell signalling events

2015

Background Mycobacterium tuberculosis (M. tuberculosis) modulates host immune response, mainly T cell responses for its own survival leading to disease or latent infection. The molecules and mechanisms utilized to accomplish immune subversion by M. tuberculosis are not fully understood. Understanding the molecular mechanism of T cell response to M. tuberculosis is important for development of efficacious vaccine against TB. Methods Here, we investigated effect of M. tuberculosis antigens Ag85A and ESAT-6 on T cell signalling events in CD3/CD28 induced Peripheral blood mononuclear cells (PBMCs) of PPD+ve healthy individuals and pulmonary TB patients. We studied CD3 induced intracellular calc…

TuberculosisT-LymphocytesT cellCD3Upstream and downstream (transduction)ImmunologyIntracellular SpaceReceptors Antigen T-CellLymphocyte ActivationMycobacterium tuberculosisBacterial ProteinsCD28 AntigensmedicineHumansAntigens BacterialNFATC Transcription FactorsbiologyT-cell receptorNF-kappa BCD28hemic and immune systemsNFATMycobacterium tuberculosismedicine.diseasebiology.organism_classificationmedicine.anatomical_structureImmunologyLeukocytes Mononuclearbiology.proteinCalciumMitogen-Activated Protein KinasesAcyltransferasesResearch ArticleSignal TransductionBMC Immunology
researchProduct