Search results for "FATE"

showing 10 items of 765 documents

A Combination of Celecoxib and Glucosamine Sulfate Has Anti-Inflammatory and Chondroprotective Effects: Results from an In Vitro Study on Human Osteo…

2021

This study investigated the possible anti-inflammatory and chondroprotective effects of a combination of celecoxib and prescription-grade glucosamine sulfate (GS) in human osteoarthritic (OA) chondrocytes and their possible mechanism of action. Chondrocytes were treated with celecoxib (1.85 µM) and GS (9 µM), alone or in combination with IL-1β (10 ng/mL) and a specific nuclear factor (NF)-κB inhibitor (BAY-11-7082, 1 µM). Gene expression and release of some pro-inflammatory mediators, metalloproteinases (MMPs), and type II collagen (Col2a1) were evaluated by qRT-PCR and ELISA

Interleukin-1betachondrocytesAnti-Inflammatory AgentsApoptosisPharmacologymedicine.disease_causeNF-κBchemistry.chemical_compoundchondroprotectionoxidative stressSulfonesBiology (General)SpectroscopyCells CulturedGlucosamineglucosamine sulfatebiologycelecoxibChemistrySuperoxideNF-kappa BGeneral MedicineComputer Science ApplicationsChemistrychondrocyteosteoarthritiDrug Therapy Combinationmedicine.symptomInflammation Mediatorsmedicine.drugSignal TransductionNF-BQH301-705.5Cell SurvivalGlucosamine SulfateCatalysisArticleInorganic ChemistrySuperoxide dismutaseNitrilesOsteoarthritismedicineHumansPhysical and Theoretical ChemistryQD1-999Molecular Biologyoxidative streOrganic ChemistryMechanism of actionApoptosisinflammationbiology.proteinCelecoxibCyclooxygenaseOxidative stressInternational Journal of Molecular Sciences
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Soft Nanoonions: A Dynamic Overview onto Catanionic Vesicles Temperature-Driven Transition.

2020

Catanionic vesicles are emerging interesting structures for bioapplications. They self-generate by a pairing of oppositely charged ionic surfactants that assemble into hollow structures. Specifically, the anionic-cationic surfactant pair assumes a double-tailed zwitterionic behavior. In this work, the multilamellar-to-unilamellar thermal transition of several mixed aqueous systems, with a slight excess of the anionic one, were investigated. Interestingly, it was found that the anionic counterion underwent a dissociation as a consequence of a temperature increase, leading to the mentioned thermal transition. The present work proposed the spectroscopic techniques, specifically multinuclear NM…

Ionic bonding02 engineering and technology01 natural sciencesDissociation (chemistry)nanoreservoirslcsh:ChemistryDiffusionPulmonary surfactantNanoreservoirlcsh:QH301-705.5SpectroscopyMicelleschemistry.chemical_classificationMicroscopyAqueous solutionMicroscopy ConfocalVesiclediffusionTemperatureSodium Dodecyl SulfateGeneral Medicine021001 nanoscience & nanotechnologyComputer Science ApplicationsChemical physicsDrug deliveryCetrimonium Compoundsmicroscopy0210 nano-technologyAnionsMaterials science010402 general chemistryCatanionic vesicles; Diffusion; Microscopy; Nanoreservoirs; NMRCatalysisPhase TransitionArticleInorganic ChemistrySurface-Active AgentsCationsPhysical and Theoretical ChemistryMolecular BiologyNuclear Magnetic Resonance BiomolecularNanotubes CarbonOrganic ChemistryCatanionic vesicleNMR0104 chemical scienceslcsh:Biology (General)lcsh:QD1-999chemistrySettore CHIM/09 - Farmaceutico Tecnologico ApplicativoPairingcatanionic vesiclesCounterionInternational journal of molecular sciences
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Portrait of inflammatory response to ionizing radiation treatment

2015

Ionizing radiation (IR) activates both pro-and anti-proliferative signal pathways producing an imbalance in cell fate decision. IR is able to regulate several genes and factors involved in cell-cycle progression, survival and/or cell death, DNA repair and inflammation modulating an intracellular radiation-dependent response. Radiation therapy can modulate anti-tumour immune responses, modifying tumour and its microenvironment. In this review, we report how IR could stimulate inflammatory factors to affect cell fate via multiple pathways, describing their roles on gene expression regulation, fibrosis and invasive processes. Understanding the complex relationship between IR, inflammation and …

Ionizing radiationDNA repairFibrosimedicine.medical_treatmentClinical BiochemistryInflammationReviewCell fate determinationBioinformaticsImmune systemMedicineCytokineRegulation of gene expressionInflammationInvasivenebusiness.industryCancerIonizing radiation Inflammation Cytokine Fibrosis InvasivenessCell Biologymedicine.diseaseFibrosisInvasivenessRadiation therapyCytokineCancer researchmedicine.symptombusinessJournal of Inflammation
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Early C3A hydration in the presence of different kinds of calcium sulfate.

2009

International audience; Hydration reactions of C3A with various amounts of calcium sulfate hemihydrate, gypsum or a mixture of two, were investigated by isothermal microcalorimetry, and a monitoring of the ionic concentrations of diluted suspensions. This study shows that sulfate type used modifies the early C3A-CaSO4 hydration products and the rate of this hydration. The fast initial AFm formation observed before ettringite precipitation in the C3A-gypsum system is avoided as soon as hemihydrate is present in the suspension. This was attributed to.higher super saturation degrees and then higher nucleation frequency with regard to the ettringite obtained in the presence of hemihydrate. More…

Isothermal microcalorimetryEttringiteGypsumInorganic chemistry0211 other engineering and technologiesNucleationHydrationchemical and pharmacologic phenomena02 engineering and technologyengineering.materialEttringitechemistry.chemical_compound021105 building & constructionGeneral Materials ScienceTricalcium aluminateSulfateSupersaturationPrecipitation (chemistry)Chemistry[CHIM.MATE]Chemical Sciences/Material chemistryBuilding and ConstructionCa3Al2O6021001 nanoscience & nanotechnologyKinetics[ CHIM.MATE ] Chemical Sciences/Material chemistryengineering0210 nano-technology
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Proteoglycan occurrence in gastrolith of the crayfish Cherax quadricarinatus (Malacostraca: Decapoda).

2012

14 pages; International audience; Biomineralized structures are hybrid composites formed and stabilized by the close interaction of the organic and the inorganic phases. Crayfish are good models for studying biomineralization because they develop, in a molting-mineralization cycle, semi-spherical mineralized structures referred to as gastroliths. The organic matrix of these structures consists of proteins, polysaccharides, and lipids. Chitin is the main polysaccharide and is concentrically arranged as fibrous chitin-protein lamellar structures. Although several proteins and low-molecular weight phosphorylated components have been reported to be involved in gastrolith mineralization, the occ…

Keratan sulfateCheraxAnatomyAquatic ScienceBiologyMatrix (biology)biology.organism_classificationbiomineralization[ SDV.IB.BIO ] Life Sciences [q-bio]/Bioengineering/BiomaterialsMolting cycleAmorphous calcium carbonatecarbohydrates (lipids)chemistry.chemical_compoundBiochemistrychemistryGastrolithProteoglycanglycosaminoglycansCherax quadricarinatusamorphous calcium carbonategastrolithbiology.proteinproteoglycanscalcium storageBiomineralization
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Enhanced expression of IL-8 in normal human keratinocytes and human keratinocyte cell line HaCaT in vitro after stimulation with contact sensitizers,…

1994

Abstract To investigate the interleukin-8 production of keratinocytes after stimulation in vitro we have used various agents: (i) contact sensi-tizer (2,4-dinitrofiuorobenzene, 3-n-penladecylcatechol); (ii) tolerogen (5-methyl-3-n-pentadecylcatechol); (iii) irritant (sodium lauryl sulfate). Interleukin-8 gene expression was assessed by northern blot hybridization of the total cytoplasmic RNA extracted from subconfluent normal human keratinocyte cultures and the keratinocyte cell line HaCaT using a radiolabeled DNA probe specific for human interleukin-8. Intcrleukin-8 gene expression was markedly increased upon in vitro stimulation after 1-6 h with contact sensitizers, tolerogen and the irri…

KeratinocytesCatecholsStimulationDermatologyDermatitis ContactBiochemistryGene expressionmedicineImmune ToleranceHumansInterleukin 8Northern blotRNA MessengerMolecular BiologyCells CulturedCell Line TransformedChemistryInterleukin-8Sodium Dodecyl SulfateMolecular biologyIn vitroHaCaTmedicine.anatomical_structureGene Expression RegulationCell cultureImmunologyIrritantsDinitrofluorobenzeneKeratinocyteExperimental dermatology
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Potential antipsoriatic effect of chondroitin sulfate through inhibition of NF-κB and STAT3 in human keratinocytes

2012

Abstract Chondroitin sulfate (CS) is a natural glycosaminoglycan, formed by the 1–3 linkage of d -glucuronic acid to N-acetylgalactosamine, present in the extracellular matrix. It is used as a slow acting disease modifying agent in the treatment of osteoarthritis, and part of its beneficial effects are due to its antiinflammatory properties that result from an inhibitory effect on NF-κB signaling pathway. This ability raises the hypothesis that CS might be effective in other chronic inflammatory processes such as psoriasis, in which a deregulation of NF-κB is a key feature. In addition, psoriasis is characterized by an upregulation of STAT3 signaling pathway that is related to the epidermal…

KeratinocytesSTAT3 Transcription FactorBlotting WesternPrimary Cell CultureAnti-Inflammatory AgentsDermoscopyElectrophoretic Mobility Shift AssayPharmacologyStat3 Signaling Pathwaychemistry.chemical_compoundDownregulation and upregulationPsoriasismedicineHumansPsoriasisChondroitin sulfateCells CulturedPharmacologyChemistryChondroitin SulfatesNF-kappa BNF-κBmedicine.diseaseMicroscopy FluorescenceImmunologyPhosphorylationTumor necrosis factor alphaSignal transductionProtein BindingPharmacological Research
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Preclinical Effect of Absorption Modifying Excipients on Rat Intestinal Transport of Model Compounds and the Mucosal Barrier Marker 51Cr-EDTA

2017

There is a renewed interest from the pharmaceutical field to develop oral formulations of compounds, such as peptides, oligonucleotides, and polar drugs. However, these often suffer from insufficient absorption across the intestinal mucosal barrier. One approach to circumvent this problem is the use of absorption modifying excipient(s) (AME). This study determined the absorption enhancing effect of four AMEs (sodium dodecyl sulfate, caprate, chitosan, N-acetylcysteine) on five model compounds in a rat jejunal perfusion model. The aim was to correlate the model compound absorption to the blood-to-lumen clearance of the mucosal marker for barrier integrity, 51Cr-EDTA. Sodium dodecyl sulfate a…

KetoprofenFysiologiPhysiologyabsorption modifiersPharmaceutical ScienceExcipient51cr edtaPharmacology and Toxicology02 engineering and technologyAbsorption (skin)030226 pharmacology & pharmacyChitosan03 medical and health scienceschemistry.chemical_compound0302 clinical medicineintestinal perfusionDrug DiscoverymedicineIntestinal transportSodium dodecyl sulfatebioequivalenceChromatographypermeation enhancersPermeationFarmakologi och toxikologi021001 nanoscience & nanotechnologypharmaceutical developmentchemistryMolecular Medicine0210 nano-technologymedicine.drugMolecular Pharmaceutics
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Comparison between sodium dodecylsulphate and cetyltrimethylammonium bromide as mobile phases in the micellar liquid chromatography determination of …

2004

The retention behaviour of non-steroidal anti-inflammatory drugs (NSAIDs) using micellar mobile phases of sodium dodecylsulphate (SDS) is studied and compared with that observed with micellar mobile phases of cetyltrimethylammonium bromide (CTAB). A liquid chromatographic procedure for the determination of acemetacin, diclofenac, indomethacin, ketoprofen, naproxen and tolmetin in pharmaceutical preparations is described. The proposed system uses a Kromasil C18 analytical column and a solution of 0.15 M SDS at pH 3 with 10% 1-propanol as mobile phase. Under these conditions, the studied NSAIDs elute between 6 and 10 min at a 1 mL min(-1) flow rate. Limits of detection (LOD) are lower than 0.…

KetoprofenNaproxenSodiumClinical BiochemistryAcemetacinPharmaceutical Sciencechemistry.chemical_elementAnalytical Chemistrychemistry.chemical_compoundBromideDrug DiscoverymedicineSpectroscopyChromatography Micellar Electrokinetic CapillaryDetection limitChromatographyElutionCetrimoniumAnti-Inflammatory Agents Non-SteroidalSodium Dodecyl SulfateReference StandardsSolutionschemistryMicellar liquid chromatographyCalibrationCetrimonium CompoundsIndicators and ReagentsSpectrophotometry Ultravioletmedicine.drugJournal of pharmaceutical and biomedical analysis
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Mannoproteins from the cell wall ofKluyveromyces lactis

1986

Wall mannoproteins from Kluyveromyces lactis have been solubilised by treatment of cell walls with sodium dodecyl sulphate (SDS) or zymolyase. While the former reagent liberates a large number of molecular species, zymolyase preferentially releases a high-molecular-weight material that is sensitive to endo-β-N-acetylglucosaminidase H, and a 29-kDa molecule that reacts with the antiserum raised against a similar species from walls of Saccharomyces cerevisiae. In contrast with observations on isolated walls of S. cerevisiae, dithiothreitol pretreatment of K. lactis walls does not enhance the effect of zymolyase upon mannoprotein release. However, the action of thiol agents is still necessary …

Kluyveromyces lactisAntiserumbiologySaccharomyces cerevisiaebiology.organism_classificationMicrobiologyYeastDithiothreitolCell wallchemistry.chemical_compoundchemistryBiochemistryKluyveromycesGeneticsSodium dodecyl sulfateMolecular BiologyFEMS Microbiology Letters
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