Search results for "H30"

showing 10 items of 1587 documents

Metal complexes of oxadiazole ligands: An overview

2019

Oxadizoles are heterocyclic ring systems that find application in different scientific disciplines, from medicinal chemistry to optoelectronics. Coordination with metals (especially the transition ones) proved to enhance the intrinsic characteristics of these organic ligands and many metal complexes of oxadiazoles showed attractive characteristics for different research fields. In this review, we provide a general overview on different metal complexes and polymers containing oxadiazole moieties, reporting the principal synthetic approaches adopted for their preparation and showing the variety of applications they found in the last 40 years.

OxadizoleAnti-Inflammatory AgentsOxadiazoleAntineoplastic AgentsReviewmetal complexes010402 general chemistryRing (chemistry)01 natural sciencesCatalysisInorganic ChemistryMetallcsh:ChemistryAntineoplastic Agentchemistry.chemical_compoundOrganometallic CompoundsPhysical and Theoretical ChemistryMolecular Biologylcsh:QH301-705.5SpectroscopyScientific disciplinesGroup 2 organometallic chemistryOrganometallic CompoundOxadiazoles010405 organic chemistryChemistryMetalOrganic ChemistryGeneral MedicineCombinatorial chemistry0104 chemical sciencesComputer Science ApplicationsAnti-Inflammatory Agent124-oxadizolelcsh:Biology (General)lcsh:QD1-999MetalsSettore CHIM/03 - Chimica Generale E Inorganicavisual_artvisual_art.visual_art_mediumMetal complexe134-oxadizole
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Water Extract of Cryphaea heteromalla (Hedw.) D. Mohr Bryophyte as a Natural Powerful Source of Biologically Active Compounds

2019

Bryophytes comprise of the mosses, liverworts, and hornworts. Cryphaea heteromalla, (Hedw.) D. Mohr, is a non-vascular lower plant belonging to mosses group. To the date, the most chemically characterized species belong to the liverworts, while only 3.2% and 8.8% of the species belonging to the mosses and hornworts, respectively, have been investigated. In this work, we present Folin–Ciocalteu and oxygen radical absorbance capacity (ORAC) data related to crude extracts of C. heteromalla obtained by three di erent extraction solvents: pure water (WT), methanol:water (80:20 v/v) (MET), and ethanol:water (80:20 v/v) (ETH). The water extract proved to be the best solvent showing the highest con…

Oxygen radical absorbance capacityBryophytaCoumaric acidMass spectrometryCatalysisArticleInorganic ChemistryExtract HPLC-ESI-TOF-MS analysilcsh:Chemistrychemistry.chemical_compoundCryphaea heteromalla; bryophytes; extract HPLC-ESI-TOF-MS analysis; oxidative stress evaluationMiceCryphaea heteromallabryophytesAnimalsPhysical and Theoretical ChemistryMolecular Biologylcsh:QH301-705.5SpectroscopyExtract HPLC-ESI-TOF-MS analysisChromatographyEthanolChemistryPlant ExtractsOxidative stress evaluationOrganic ChemistryExtraction (chemistry)Bryophytesoxidative stress evaluationGeneral MedicineFree Radical Scavengersextract hplc-esi-tof-ms analysisComputer Science ApplicationsSolventOxidative Stresslcsh:Biology (General)lcsh:QD1-999<i>cryphaea heteromalla</i>BryophyteSettore BIO/03 - Botanica Ambientale E ApplicataNIH 3T3 CellsBryophyteMethanolReactive Oxygen SpeciesInternational Journal of Molecular Sciences
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Differential Expression of the Demosponge (Suberites domuncula) Carotenoid Oxygenases in Response to Light: Protection Mechanism Against the Self-Pro…

2012

The demosponge Suberites domuncula has been described to contain high levels of a proteinaceous toxin, Suberitine, that displays haemolytic activityIn the present study this 7–8 kDa polypeptide has been isolated and was shown to exhibit also cytotoxic effects on cells of the same species. Addition of retinal, a recently identified metabolite of β-carotene that is abundantly present in S. domuncula was found to reduce both the haemolytic and the cell toxic activity of Suberitine at a molar ratio of 1:1. Spectroscopic analyses revealed that the interaction between β-carotene and Suberitine can be ascribed to a reversible energy transfer reaction. The enzyme that synthesises retinal in the spo…

OxygenaseLightMolecular Sequence DataPharmaceutical Sciencemedicine.disease_causeretinalArticle03 medical and health sciencesSuberitineDioxygenaseβ-caroteneDrug DiscoverymedicineAnimalsAmino Acid SequenceCloning Molecularlcsh:QH301-705.5Pharmacology Toxicology and Pharmaceutics (miscellaneous)Carotenoidsponges030304 developmental biologyβ-carotene dioxygenasechemistry.chemical_classification0303 health sciencesbiologyBacteriaToxinCarotenoid oxygenase030302 biochemistry & molecular biologyProteinsSuberitine; β-carotene; retinal; β-carotene dioxygenase; sponges; <em>Suberites domuncula</em>biology.organism_classificationSuberites domunculaSuberites domunculaEnzymelcsh:Biology (General)Biochemistrychemistrybiology.proteinOxygenasesRetinaldehydeSuberitesSuberitesMarine Drugs
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The Eureka! by Kary Mullis

2019

Not available.

PCRNobelKary Mullilcsh:Biology (General)Biochemistry (medical)Plant ScienceSettore MED/49 - Scienze Tecniche Dietetiche Applicatelcsh:QH301-705.5General Biochemistry Genetics and Molecular BiologyJournal of Biological Research
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Cellular Uptake of siRNA-Loaded Nanocarriers to Knockdown PD-L1: Strategies to Improve T-cell Functions

2020

T-cells are a type of lymphocyte (a subtype of white blood cells) that play a central role in cell-mediated immunity. Currently, adoptive T-cell immunotherapy is being developed to destroy cancer cells. In this therapy, T-cells are harvested from a patient&rsquo

PD-L1Small interfering RNAT-LymphocytesLymphocytemedicine.medical_treatmentT cellImmunotherapy AdoptiveB7-H1 AntigenArticlemedicineHumansNanotechnologyRNA Small Interferinglcsh:QH301-705.5Gene knockdownnanocarriersChemistryT-cellsCancercellular uptakeGeneral MedicineImmunotherapymedicine.diseasemedicine.anatomical_structurelcsh:Biology (General)siRNACancer cellCancer researchNanocarriersadoptive immunotherapyCells
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Repeatability and Reliability of the Rheumatoid Arthritis Foot Disease Activity Index in Spanish Patients: A Transcultural Adaptation

2021

Simple Summary The Rheumatoid Arthritis Foot Disease Activity Index (RADAI-F5) is the first questionnaire designed to check the level of involvement in the feet of patients with rheumatoid arthritis. It is a validated and reliable five-question questionnaire in English. It is also considered suitable for clinical use. We aim was to translate and validate the Spanish version. The findings of this research suggest that is a valid, strong and trustworthy clinimetric tool that appropriately applies to the Spanish community and can be managed as a whole or in terms of its respective dimensions, such as arthritis activity in the foot, joint tenderness and swelling, and foot arthritis pain sub-sca…

Pain measurementArtritisGeneral Immunology and MicrobiologyQH301-705.5QuestionnaireFootquestionnairePiequestionnaire; arthritis chronic pain; pain measurement; footarthritis chronic painpain measurementArticleGeneral Biochemistry Genetics and Molecular BiologyMedida de dolorExtremitatsArthritis chronic painfootEnfermeríaArtritis crónicaPacientsBiology (General)General Agricultural and Biological SciencesCuestionario
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Speleogenesis of the Hermannshöhle cave system (Austria): Constraints from 230Th/U-dating and palaeomagnetic analysis

2015

Hermannshöhle is a show cave located near Kirchberg/Wechsel in Lower Austria. Together with three nearby and genetically connected caves, it forms the Hermannshöhlen cave system (HHS). With a length of 5 km, the HHS is the longest cave in the Lower Austroalpine unit. It is arranged as an extreme three-dimensional maze on a ground area of 200 x 200 x 82 m. Speleothems are abundant in this cave and represent the focus of this study. Low carbon isotope values indicate the presence of a soil-covered catchment above the HHS during times of speleothem deposition. 28 samples were dated by the 230Th/U-method and, in combination with palaeomagnetic data from a 5 m-high sediment profile, indicate mul…

PaleontologygeographyQE1-996.5geography.geographical_feature_categoryCaveQH301-705.5GeologySpeleogenesisParagenesisBiology (General)GeologyEarth-Surface ProcessesInternational Journal of Speleology
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Modelling the spatial and temporal constrains of the GABAergic influence on neuronal excitability

2021

GABA (γ-amino butyric acid) is an inhibitory neurotransmitter in the adult brain that can mediate depolarizing responses during development or after neuropathological insults. Under which conditions GABAergic membrane depolarizations are sufficient to impose excitatory effects is hard to predict, as shunting inhibition and GABAergic effects on spatiotemporal filtering of excitatory inputs must be considered. To evaluate at which reversal potential a net excitatory effect was imposed by GABA (EGABAThr), we performed a detailed in-silico study using simple neuronal topologies and distinct spatiotemporal relations between GABAergic and glutamatergic inputs. These simulations revealed for GABAe…

Patch-Clamp TechniquesAction potentialPhysiologyAction PotentialsSynaptic TransmissionNervous SystemBiochemistryMiceNerve FibersAnimal CellsMedicine and Health SciencesGABAergic NeuronsBiology (General)gamma-Aminobutyric AcidNeuronsMembrane potentialEcologyChemistryPyramidal CellsDepolarizationNeurochemistryNeurotransmittersCA3 Region HippocampalElectrophysiologyReceptors GlutamateComputational Theory and MathematicsModeling and SimulationExcitatory postsynaptic potentialGABAergicAnatomyCellular TypesShunting inhibitionResearch Articlemedicine.drugQH301-705.5Models NeurologicalNeurophysiologyAMPA receptorMembrane Potentialgamma-Aminobutyric acidCellular and Molecular NeuroscienceGlutamatergicSpatio-Temporal AnalysisGeneticsmedicineAnimalsComputer SimulationReceptors AMPAReversal potentialMolecular BiologyEcology Evolution Behavior and SystematicsComputational BiologyBiology and Life SciencesNeural InhibitionDendritesCell BiologyNeuronal DendritesAxonsMice Inbred C57BLAnimals Newbornnervous systemCellular NeuroscienceSynapsesDepolarizationNeuroscienceNeurosciencePLOS Computational Biology
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Unmasking epithelial-mesenchymal transition in a breast cancer primary culture: a study report

2012

Abstract Background Immortalized cancer cell lines are now well-established procedures in biomedicine for a more complete understanding of cellular processes in cancer. However, they are more useful in preparation of fresh tumour tissue, in order to obtain cancer cells with highly preserved individual tumour properties. In the present study we report an analytical investigation on a breast cancer primary cell culture isolated from a surgical specimen obtained from a patient with an infiltrating ductal carcinoma. The objective of the research was to reveal unrecognized aspects of neoplastic cells, typical of the tumour from where the cells were derived, but masked in fixed tissue sections, i…

Pathologymedicine.medical_specialtyEpithelial-Mesenchymal TransitionImmunocytochemistryShort Reportlcsh:MedicineBreast NeoplasmsBiologyGeneral Biochemistry Genetics and Molecular BiologyCell LineBreast cancerBreast cancerCarcinomamedicineBiomarkers TumorTumor Cells CulturedHumansVimentinMicroscopy Phase-ContrastEpithelial–mesenchymal transitionPrimary cell culturelcsh:Science (General)lcsh:QH301-705.5Medicine(all)Biochemistry Genetics and Molecular Biology(all)Reverse Transcriptase Polymerase Chain Reactionlcsh:RMesenchymal stem cellCarcinoma Ductal BreastCancerMuscle SmoothBreast cancer Primary cell culture Epithelial-mesenchymal transition (EMT)General Medicinemedicine.diseaseCadherinsImmunohistochemistryActinsGene Expression Regulation NeoplasticEpithelial-mesenchymal transition (EMT)lcsh:Biology (General)Cell cultureCancer cellKeratinsFemalelcsh:Q1-390
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Current Experience in Testing Mitochondrial Nutrients in Disorders Featuring Oxidative Stress and Mitochondrial Dysfunction: Rational Design of Chemo…

2014

An extensive number of pathologies are associated with mitochondrial dysfunction (MDF) and oxidative stress (OS). Thus, mitochondrial cofactors termed "mitochondrial nutrients" (MN), such as alpha-lipoic acid (ALA), Coenzyme Q10 (CoQ10), and L-carnitine (CARN) (or its derivatives) have been tested in a number of clinical trials, and this review is focused on the use of MN-based clinical trials. The papers reporting on MN-based clinical trials were retrieved in MedLine up to July 2014, and evaluated for the following endpoints: (a) treated diseases; (b) dosages, number of enrolled patients and duration of treatment; (c) trial success for each MN or MN combinations as reported by authors. The…

Pathologymedicine.medical_specialtyMitochondrial Diseasesmitochondrial nutrientsCoenzymesoxidative phosphorylationReviewPharmacologyMitochondrionBiologyControlled studiesmedicine.disease_causeChemopreventionCatalysislcsh:ChemistryInorganic Chemistrychemistry.chemical_compoundmitochondrial dysfunctionmedicineAnimalsHumansPhysical and Theoretical Chemistrylcsh:QH301-705.5Molecular BiologySpectroscopyCoenzyme Q10Clinical Trials as TopicOrganic ChemistryGeneral Medicine3. Good healthComputer Science ApplicationsMitochondriaClinical trialOxidative Stresslcsh:Biology (General)lcsh:QD1-999chemistrymitochondrial dysfunction and oxidative streKrebs cycleOxidative stressmitochondrial nutrient
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