Search results for "HILIC"

showing 10 items of 745 documents

Unusual Regioselectivity in the Opening of Epoxides by Carboxylic Acid Enediolates

2008

Addition of carboxylic acid dianions appears to be a potential alternative to the use of aluminium enolates for nucleophilic ring opening of epoxides. These conditions require the use of a sub-stoichiometric amount of amine (10% mol) for dianion generation and the previous activation of the epoxide with LiCl. Yields are good, with high regioselectivity, but the use of styrene oxide led, unexpectedly, to a mixture resulting from the attack on both the primary and secondary carbon atoms. Generally, a low diastereoselectivity is seen on attack at the primary center, however only one diastereoisomer was obtained from attack to the secondary carbon of the styrene oxide.

diastereoselectivity.Carboxylic acidCarboxylic AcidsPharmaceutical ScienceEpoxideMedicinal chemistryAnalytical Chemistrylcsh:QD241-441chemistry.chemical_compoundLactoneslcsh:Organic chemistryNucleophileStyrene oxideDrug DiscoveryOrganic chemistryPhysical and Theoretical Chemistrylithium chloridechemistry.chemical_classificationNucleophilic additionCommunicationOrganic ChemistryDiastereomerRegioselectivitydiastereoselectivitynucleophilic additionchemistryChemistry (miscellaneous)regioselectivityMolecular MedicineEpoxy CompoundsAmine gas treatingMolecules
researchProduct

Late Breaking Abstract - Dose-ranging study of mepolizumab in eosinophilic COPD

2018

Background: Patients with eosinophilic COPD & frequent exacerbations may benefit from mepolizumab (MEP) treatment. Objective: Assess efficacy & safety of 2 MEP doses vs placebo (PBO) in COPD with blood eosinophils ≥150 cells/µL [screening] or ≥300 cells/µL [prior yr], history of ≥2 moderate/≥1 severe exacerbations & ICS+≥2 bronchodilator maintenance therapies (ICS+MT). Methods: Phase III, randomised, PBO-controlled, double-blind, parallel-group trial (METREO); patients received SC MEP 100mg, MEP 300mg or PBO plus ICS+MT, every 4 wks for 52 wks. Primary endpoint: rate/yr of moderate (systemic corticosteroids/antibiotics)/severe(hospitalisation or death) exacerbations. Secondary endpoints inc…

education.field_of_studymedicine.medical_specialtyCOPDmedicine.drug_classbusiness.industryPopulationPlaceboDose-ranging studymedicine.diseaseGastroenterology03 medical and health sciences0302 clinical medicineBronchodilatorInternal medicineEosinophilicClinical endpointmedicine030212 general & internal medicineeducationbusinessMepolizumab030217 neurology & neurosurgerymedicine.drugClinical Problems
researchProduct

A histological study of eosinophilic granuloma in mice following infestation with Anisakis larvae

2014

eosinophilic granuloma Anisakis
researchProduct

Retention/release equilibrium of aroma compounds in fat-free dairy gels

2010

BACKGROUND: The replacement of fat by thickeners in fat-free yoghurts leads to an important modification of aroma compound partitioning, with an impact on aroma perception. Investigation of retention/release equilibria allows a good understanding of aroma compound behaviour depending on food composition. RESULTS: Vapour/liquid equilibria of ten aroma compounds (two esters, two ketones, three aldehydes and three alcohols) in several media were studied to investigate the influence of pectin addition to fat-free dairy gel on the retention/release equilibrium. The partition coefficient of each aroma compound was measured by headspace analysis at equilibrium in six media (pure water, low-methoxy…

food.ingredientPectinPolysaccharide01 natural sciencesPhase TransitionDAIRY GELchemistry.chemical_compound0404 agricultural biotechnologyfoodPECTINAROMA RELEASE[SDV.IDA]Life Sciences [q-bio]/Food engineeringAroma compoundFood scienceAromaHYDROPHOBICITYchemistry.chemical_classificationVolatile Organic CompoundsNutrition and DieteticsChromatographyAqueous mediumbiologyFood additive010401 analytical chemistryfood and beveragesFood composition data04 agricultural and veterinary sciencesbiology.organism_classificationDietary Fats040401 food science0104 chemical sciencesPartition coefficientKineticschemistryPectinsDairy ProductsGelsHydrophobic and Hydrophilic InteractionsAgronomy and Crop ScienceFood ScienceBiotechnologyJournal of the Science of Food and Agriculture
researchProduct

Primo ricerche sulla ultrastruttura dell'uovo delle Ascidie

1959

Summary The cytoplasmic constituents of the unfertilized eggs of Ciona intestinalis were separated by centrifugation and studied at the electron microscope, with the following results. Lipid droplets collect at the centripetal pole; they are boundered by a thin membrane. The yolk granules are homogeneous in appearance; a few have a granular structure. Mitochondria contain numerous cristae; they accumulate in two different layers centripetally and centrifugally to the yolk granules layer respectively. Basophilic material collects at both poles of the egg in two hyaline caps: a centripetal one constituted by small Vesicles and a centrifugal represented by dense clumps. The latter, as well as …

food.ingredientVesicleAnatomyBiologybiology.organism_classificationlaw.inventionBasophilicfoodlawLipid dropletYolkembryonic structuresBiophysicsAnimal Science and ZoologyCentrifugationCiona intestinalisElectron microscopeHyalineBolletino di zoologia
researchProduct

Estimation of the mechanical properties of the eye through the study of its vibrational modes.

2017

Measuring the eye's mechanical properties in vivo and with minimally invasive techniques can be the key for individualized solutions to a number of eye pathologies. The development of such techniques largely relies on a computational modelling of the eyeball and, it optimally requires the synergic interplay between experimentation and numerical simulation. In Astrophysics and Geophysics the remote measurement of structural properties of the systems of their realm is performed on the basis of (helio-)seismic techniques. As a biomechanical system, the eyeball possesses normal vibrational modes encompassing rich information about its structure and mechanical properties. However, the integral a…

genetic structureslcsh:MedicineEyeCornea0302 clinical medicineNormal modeMedicine and Health Scienceslcsh:ScienceLens (Anatomy)PhysicsMultidisciplinaryPhysicsClassical MechanicsEye MusclesInverse problemContact Lenses Hydrophilicmedicine.anatomical_structureBiological Physics (physics.bio-ph)Physical SciencessymbolsAnatomyResearch ArticleAcousticsOcular AnatomyMaterials ScienceMaterial PropertiesFOS: Physical sciencesCondensed Matter - Soft Condensed MatterModels BiologicalVibrationResonance03 medical and health sciencessymbols.namesakeOcular SystemElastic ModulusmedicineHumansMechanical PropertiesComputer SimulationPhysics - Biological PhysicsEigenvalues and eigenvectorsComputer simulationlcsh:RFinite difference methodBiology and Life SciencesEigenvaluesPhysics - Medical PhysicsPoisson's ratioeye diseasesResonance FrequencyVibrationAlgebraLinear Algebra030221 ophthalmology & optometryEyesSoft Condensed Matter (cond-mat.soft)Human eyelcsh:QMedical Physics (physics.med-ph)sense organsHead030217 neurology & neurosurgeryMathematicsPLoS ONE
researchProduct

Diagnosis and treatment of chronic synovitis in patients with haemophilia: consensus statements from the Italian Association of Haemophilia Centres

2022

Although synovitis is recognized as a marker of joint disease activity, its periodic assessment is not included in routine clinical surveillance of patients with haemophilia (PwH). In order to evaluate the current knowledge and to identify controversial issues, a preliminary literature search by the Musculoskeletal Committee of the Italian Association of Haemophilia Centres (AICE) has been conducted. Statements have been established and sent to the Italian AICE members to collect their level of agreement or disagreement by a Delphi process. Thirty-seven consensus recommendations have been drafted. We found a general agreement on the indication to consider the presence of synovitis as a mark…

haemophilia; haemophilic arthropathy; synovitis; Chronic Disease; Consensus; Hemophilia A; Humans; Italy; Synovitishaemophilia haemophilic arthropathy synovitisConsensusSynovitisItalyChronic Diseasehaemophilic arthropathyhaemophiliaHumansHematologyHemophilia ABritish Journal of Haematology
researchProduct

Effect of long-term salinity increase on nitritation and denitritation kinetics in activated sludge and granular sludge reactors

2017

The aim of this work was to investigate the effects of moderate and drastic long-termincrease of salinity.Particularly, the study was aimed at assessing the shock effecton nitritationand denitritation kineticsof halophilic biomass inboth forms:flocculent activated sludge and granular sludge.

halophilic biomass industrial wastewater salinity shocks sequencing batch reactorsSettore ICAR/03 - Ingegneria Sanitaria-Ambientale
researchProduct

An Off-On-Off Fluorescent Sensor for pH Windows Based on the 13aneN4-Zn 2+ System

2016

International audience; The new ligand L was prepared and features a 13-membered tetraaza macrocyclic ring with a 1,8-naphthalimide fluorophore appended to a C atom of its backbone. The protonation constants of L as well as its complexation constants with Zn2+ ions were determined in 1:1 water/methanol solutions by potentiometric titrations. Fluorimetric pH titrations were performed with L alone and L in the presence of Zn2+ ions (1:1), and the species distributions (%) versus pH were compared. A window-shaped fluorescence trend was observed with pH for the L/Zn2+ system, which behaves as an off-on-off pH sensor. The on window is centred in the 6.5-7.5 pH range, in correspondence with the f…

inorganic chemicalsFluorophorePotentiometric titrationInorganic chemistryProtonationYeast cellsSensors; Fluorescence; Zinc; Yeast cells; Macrocyclic ligands010402 general chemistry01 natural sciencesMicelleFluorescenceInorganic Chemistrychemistry.chemical_compoundMacrocyclic ligandsCyclamLipophilicity[SDV.IDA]Life Sciences [q-bio]/Food engineeringEquilibriaMicellesIonsChemosensors010405 organic chemistryLigandSensorsChelation-enhanced fluorescencezinc[ SDV.IDA ] Life Sciences [q-bio]/Food engineeringMetal-complexesFluorescence0104 chemical scienceschemistryCyclamTitrationMacrocycles
researchProduct

Reaction of 2-acetyltetralone with some esters of benzoic acid

1986

In order to investigate the pharmacological screening of a number of pyran-4-ones their synthesis by cyclization with sulphuric acid of the corresponding 1,3,5-triketones has been carried out with high yields. In the course of preparation of the latter the reaction of 2-acetyltetralone with some esters of benzoic acid derivatives has been studied and in particular, for a number of them, an interesting nucleophilic substitution of a chlorine atom with an alkoxy group on a benzenic nucleus has been evidenced.

inorganic chemicalschemistry.chemical_compoundBicyclic moleculechemistryOrganic ChemistryChlorine atomAlkoxy groupNucleophilic substitutionTriketoneOrganic chemistryAcid hydrolysisSulfuric acidBenzoic acidJournal of Heterocyclic Chemistry
researchProduct