Search results for "INTERACTION"

showing 10 items of 5710 documents

Docking and synthesis of pyrrolopyrimidodiazepinone derivatives (PPDs) and their precursors: New scaffolds for DNA-interacting agents

2007

New classes of pyrrolopyrimidodiazepinone derivatives (PPDs) and their precursors were studied in silico for their ability to form stable complex with DNA fragment. In the docking studies two binding modes can be envisaged: groove mode and intercalating mode. In the case of the best ligands the docking studies revealed a common binding mode with the chromophore intercalated between GC base pairs whereas the side chain lies close to the minor groove. Synthetic approach to the PPD ring systems is discussed.

ChemistryStereochemistryBase pairIn silicoIntercalation (chemistry)ChromophoreCondensed Matter PhysicsBiochemistryCombinatorial chemistrychemistry.chemical_compoundDocking (molecular)Side chainDockingDNA interactionPPDIntercalating modeMinor groove modePhysical and Theoretical ChemistryDNAMinor grooveJournal of Molecular Structure: THEOCHEM
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Interaction effects of enniatin B, deoxinivalenol and alternariol in Caco-2 cells.

2015

Enniatin B (ENN B), deoxinivalenol (DON) and alternariol (AOH) are secondary metabolites of filamentous fungi. These mycotoxins are contaminants of vegetables and cereals. They are cytotoxic and their effects are enhanced by their mixtures. The objectives of this study were to compare the cytotoxicity of ENN B, DON and AOH alone or in combination in human adenocarcinoma (Caco-2) cells and to evaluate the type of interactions of mycotoxin mixtures by the isobologram analysis. Cells were treated with concentrations ranging from 1.85 to 90μM (AOH) and from 0.312 to 10μM (for ENN B and DON), individually and in combination of two and three mycotoxins (from 1.85 to 30μM for AOH and from 0.312 to…

ChemistryStereochemistryCell SurvivalAlternariolFood Contamination04 agricultural and veterinary sciencesGeneral MedicineMycotoxinsToxicology040401 food scienceCellular viabilitychemistry.chemical_compoundLactones0404 agricultural biotechnologyCaco-2DepsipeptidesIc50 valuesHumansDrug InteractionsFood scienceCaco-2 CellsMycotoxinTrichothecenesCell survivalEnniatin BToxicology letters
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Modelling of the cation motions in complex system: case of Na-mordenites

2002

Abstract Semi-empirical inter-atomic potentials and Monte Carlo algorithms are proposed to predict the evolution of the interaction energy between sodium ions and a mordenite type aluminosilicate network as a function of Si/Al ratio. This result is favourably compared with the activation energy barriers for Na + `jumps' responsible for the polarization change, measured by thermally stimulated current (TSC) spectroscopy, for Na-mordenites characterized by Si/Al ratios ranged from 5.5 to 12. Finally, we propose a possible mechanism for the cation motions, which involves activation barriers within the same order of magnitude than those measured by TSC.

ChemistryThermodynamicsInteratomic potentialActivation energyInteraction energyCondensed Matter PhysicsMordeniteElectronic Optical and Magnetic MaterialsIonComputational chemistryAluminosilicateMaterials ChemistryCeramics and CompositesSpectroscopyOrder of magnitudeJournal of Non-Crystalline Solids
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Anharmonic vibrational frequency calculations for solvated molecules in the B3LYP Kohn–Sham basis set limit

2012

Abstract The solvent dependence of harmonic and anharmonic vibrational wavenumbers of water, formaldehyde and formamide was studied using the B3LYP method. The results obtained with the hierarchy of Jensen's polarization-consistent basis sets were fitted with two-parameter formula toward the B3LYP Kohn–Sham complete basis set (CBS) limit. Anharmonic corrections have been obtained by a second order perturbation treatment (VPT2) and vibrational configuration interaction (VCI) method. The solvent environment was treated according to the self-consistent reaction field polarizable continuum model (SCRF PCM) approach.

ChemistryVibrational partition functionMolecular vibrationAnharmonicityPhysics::Atomic and Molecular ClustersKohn–Sham equationsPhysics::Chemical PhysicsSolvent effectsConfiguration interactionAtomic physicsPolarizable continuum modelSpectroscopyBasis setVibrational Spectroscopy
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Validation of the Tetracycline Regulatable Gene Expression System for the Study of the Pathogenesis of Infectious Disease

2011

Understanding the pathogenesis of infectious disease requires the examination and successful integration of parameters related to both microbial virulence and host responses. As a practical and powerful method to control microbial gene expression, including in vivo, the tetracycline-regulatable system has recently gained the favor of many investigative groups. However, some immunomodulatory effects of the tetracyclines, including doxycycline, could potentially limit its use to evaluate host responses during infection. Here we have used a well-established murine model of disseminated candidiasis, which is highly dependent on both the virulence displayed by the fungal cells and on the host im…

ChemokineScienceImmunologyVirulenceMycologyPathogenesisKidneyResponse ElementsMicrobiologyMicrobiologyPathogenesisMiceGene Expression Regulation FungalCandida albicansGene expressionmedicineAnimalsPromoter Regions GeneticCandida albicansBiologyImmunity to InfectionsProtein Synthesis InhibitorsDoxycyclineMultidisciplinaryVirulencebiologyQCandidiasisImmunityRTetracyclinebiology.organism_classificationDisseminated CandidiasisDisease Models AnimalInfectious DiseasesMedical MicrobiologyInfectious disease (medical specialty)DoxycyclineHost-Pathogen InteractionsMutationImmunologybiology.proteinCytokinesMedicineChemokinesSpleenResearch Articlemedicine.drug
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Sequential analyses in coercive mother-child interaction: the predictability hypothesis in abusive versus nonabusive dyads.

1999

Abstract Objective: A two-fold purpose guided the present study: 1) To test the sequential relationship between the child’s aversive behavior and both the predictability and the compliance episodes, as well as the sequential relationship between these two mothering episodes proposed by the new predictability hypothesis (Wahler, Williams, & Cerezo, 1990) ; 2) to explore whether or not these patterns are specific to these dysfunctional dyads by using a nonabusive comparison group. Method: Fifty mother-child dyads, 25 abusive and 25 nonabusive, participated in this study. Lag sequential analyses were carried out on 302 hours of direct observation, 178 hours in the abusive group, and 124 in the…

Child abuseAdultMaleAdolescentCoercionVictimologyPoison controlDysfunctional familyChild Behavior DisordersDevelopmental psychologyDevelopmental and Educational PsychologymedicineHumansPredictabilityChildMaternal Behaviormedicine.diseaseSocial relationMother-Child RelationsPsychiatry and Mental healthSocioeconomic FactorsConduct disorderResearch DesignMother child interactionChild PreschoolPediatrics Perinatology and Child HealthFemalePsychologyChild abuseneglect
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Childhood adversity and psychosis: a systematic review of bio-psycho-social mediators and moderators.

2020

AbstractThe association between childhood adversity (CA) and psychosis has been extensively investigated in recent years. An increasing body of research has also focused on the mediating or moderating role of biological and psychological mechanisms, as well as other risk factors that might account for the link between CA and psychosis. We conducted a systematic search of the PsychINFO, Embase, Ovid, and Web of Science databases for original articles investigating the role of genetic vulnerabilities, environmental factors, psychological and psychopathological mechanisms in the association between CA and psychosis up to August 2019. We included studies with individuals at different stages of …

Child abuseBiopsychosocial modelMediation (statistics)Psychosisgene-environment correlationchild abuseEffect Modifier Epidemiologic03 medical and health sciences0302 clinical medicineAdverse Childhood ExperiencesmedicineHumanspsychotic experiencesSettore MED/25 - PsichiatriaApplied Psychologymechanismschildhood traumaGene-environment correlationmedicine.diseaseModeration030227 psychiatryPsychiatry and Mental healthMoodAdult Survivors of Child Adverse EventsPsychotic DisordersGene-Environment InteractionmaltreatmentPsychology030217 neurology & neurosurgeryClinical psychologyPsychopathologyPsychological medicine
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Form factors of the isovector scalar current and the ηπ scattering phase shifts

2015

33 pages.- 14 figures.- v2: Some clarifications and corrections of typos

Chiral perturbation theoryFinal state interactionPhysics and Astronomy (miscellaneous)Scalar (mathematics)01 natural sciencesMatrix (mathematics)Quantum mechanicsChiral perturbation theory0103 physical sciencesComputer Science::General LiteratureOrder (group theory)010306 general physicsNuclear ExperimentEngineering (miscellaneous)ComputingMilieux_MISCELLANEOUSMathematical physicsPhysicsIsovectorUnitarity010308 nuclear & particles physicsComputer Science::Information RetrievalAstrophysics::Instrumentation and Methods for AstrophysicsForm factor (quantum field theory)Computer Science::Computation and Language (Computational Linguistics and Natural Language and Speech Processing)Scattering amplitudeTheoryofComputation_MATHEMATICALLOGICANDFORMALLANGUAGES[PHYS.HPHE]Physics [physics]/High Energy Physics - Phenomenology [hep-ph]ComputingMethodologies_DOCUMENTANDTEXTPROCESSINGHigh Energy Physics::Experiment
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Implementation of local chiral interactions in the hyperspherical harmonics formalism

2021

With the goal of using chiral interactions at various orders to explore properties of the few-body nuclear systems, we write the recently developed local chiral interactions as spherical irreducible tensors and implement them in the hyperspherical harmonics expansion method. We devote particular attention to three-body forces at next-to-next-to leading order, which play an important role in reproducing experimental data. We check our implementation by benchmarking the ground-state properties of $^3$H, $^3$He and $^4$He against the available Monte Carlo calculations. We then confirm their order-by-order truncation error estimates and further investigate uncertainties in the charge radii obta…

Chiral perturbation theoryNuclear TheoryTruncation error (numerical integration)Formalism (philosophy)Materials Science (miscellaneous)QC1-999Monte Carlo methodBiophysicsGeneral Physics and AstronomyFOS: Physical sciences01 natural scienceschiral effective field theoryNuclear Theory (nucl-th)Theoretical physics0103 physical sciencesPhysical and Theoretical Chemistry010306 general physicsMathematical PhysicsExotic atomPhysics010308 nuclear & particles physicsPhysicsOrder (ring theory)light nucleiCharge (physics)Harmonicshyperspherical harmonicsnuclear interactionsab-initio theory
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Réponses des cellules de Nicotiana tabacum à des molécules microbiennes : évènements de signalisation précoce, influence de la dynamique membranaire …

2018

In their natural environment plants are in close interaction with beneficial, neutral, or pathogenic microbes, which are highly dependent on carbon resources exuded by plant roots. Sugar transport, which is a key process of plant physiology, is essential to support the fate of plant-microbe interactions. During evolution, plants have acquired the ability to perceive microbial molecules, initiating specific signal transduction cascades and leading to adapted response for microbe lifestyles (avirulent, virulent, or benefic). Plant survival will depend on the nature of the induced mechanisms. My PhD work, carried out on a simplified experimental system, contributes to the understanding of mech…

Chitotetrasacchraides[SDV.SA]Life Sciences [q-bio]/Agricultural sciences[SDV.SA] Life Sciences [q-bio]/Agricultural sciencesInteractions plantes-MicroorganismesCryptogéineChitotétrasacchraidesNicotiana tabacum[SDV.EE.IEO] Life Sciences [q-bio]/Ecology environment/SymbiosisTrafic membranaireTransport de sucresSugar transportPlant-Microbe interactions[SDV.BV]Life Sciences [q-bio]/Vegetal Biology[SDV.BV] Life Sciences [q-bio]/Vegetal BiologyCryptogeinMembrane dynamics[SDV.EE.IEO]Life Sciences [q-bio]/Ecology environment/Symbiosis
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