Search results for "Intestin"

showing 10 items of 2215 documents

Cre-mediated cell ablation contests mast cell contribution in models of antibody- and T cell-mediated autoimmunity.

2011

SummaryImmunological functions of mast cells remain poorly understood. Studies in Kit mutant mice suggest key roles for mast cells in certain antibody- and T cell-mediated autoimmune diseases. However, Kit mutations affect multiple cell types of both immune and nonimmune origin. Here, we show that targeted insertion of Cre-recombinase into the mast cell carboxypeptidase A3 locus deleted mast cells in connective and mucosal tissues by a genotoxic Trp53-dependent mechanism. Cre-mediated mast cell eradication (Cre-Master) mice had, with the exception of a lack of mast cells and reduced basophils, a normal immune system. Cre-Master mice were refractory to IgE-mediated anaphylaxis, and this defe…

Cell typeEncephalomyelitis Autoimmune ExperimentalCarboxypeptidases AT cellT-LymphocytesImmunologyAutoimmunityImmunoglobulin E03 medical and health sciencesMice0302 clinical medicineImmune systemTh2 CellsmedicineImmunology and AllergyAnimalsGenetic Predisposition to DiseaseMast CellsIntestinal MucosaInterleukin 5Anaphylaxis030304 developmental biologyAutoantibodiesMice Knockout0303 health sciencesStem Cell FactorbiologyIntegrasesGene Expression ProfilingImmunoglobulin EMast cellArthritis Experimental3. Good healthInterleukin 33Mice Inbred C57BLDisease Models Animalmedicine.anatomical_structureInfectious DiseasesImmunologyGene Targetingbiology.proteinAntibodyTumor Suppressor Protein p53030215 immunologyImmunity
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Mast cells control the expansion and differentiation of IL-10-competent B cells

2014

Abstract The discovery of B cell subsets with regulatory properties, dependent on IL-10 production, has expanded our view on the mechanisms that control inflammation. Regulatory B cells acquire the ability to produce IL-10 in a stepwise process: first, they become IL-10 competent, a poised state in which B cells are sensitive to trigger signals but do not actually express the Il-10 gene; then, when exposed to appropriate stimuli, they start producing IL-10. Even if the existence of IL-10–competent B cells is now well established, it is not yet known how different immune cell types cross talk with B cells and affect IL-10–competent B cell differentiation and expansion. Mast cells (MCs) contr…

Cell typeRegulatory B cellsCellular differentiationImmunologyCD40 LigandB-Lymphocyte SubsetsRegulatory B cellsB-cellBiologyExosomesLymphocyte ActivationImmunophenotypingMast cellMiceImmunophenotypingImmune systemmedicineImmunology and AllergyAnimalsMast CellsB cell differentiationCD40 AntigensB cellmast cell; IL-10; B-cellMice KnockoutCD40Cell DifferentiationCell biologyInterleukin-10Gastrointestinal TractInterleukin 10medicine.anatomical_structurePhenotypeMast cell; Regulatory B cells; IL-10; B cell differentiationImmunologyIL-10biology.proteinFemaleJournal of immunology (Baltimore, Md.
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Nitrergic modulation of gastrointestinal function during early endotoxemia.

2006

After bacterial infection, the host reacts by signalling to the central nervous system where a cascade of physiologic, neuroendocrine and behavioural processes is orchestrated, collectively termed the acute phase response. Endotoxemia following Gram-negative bacterial infection induces a wide array of effects, including fever, loss of appetite and changes in gastrointestinal function that attempt to eliminate the challenge and restore homeostasis. Systemic administration of low doses of endotoxin (5-40 microg/kg) to rats is associated with changes in gastrointestinal motor function, inhibition of gastric acid secretion and increase in the gastric mucosal resistance to damage. These changes …

Central Nervous Systemmedicine.medical_specialtyCentral nervous systemMyenteric PlexusNitric OxideNitric oxideGastric Acidchemistry.chemical_compoundInternal medicineNitrergic NeuronsDrug DiscoverymedicineAnimalsHumansPharmacologyGastrointestinal tractbiologyStomachVagus NerveEndotoxemiaRatsNitric oxide synthaseGastrointestinal Tractmedicine.anatomical_structureEndocrinologychemistryGastric MucosaRegional Blood Flowbiology.proteinGastric acidNitric Oxide SynthaseGastrointestinal functionGastrointestinal MotilityHomeostasisCurrent pharmaceutical design
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Identification of Patulin from Penicillium coprobium as a Toxin for Enteric Neurons

2019

The identification and characterization of fungal commensals of the human gut (the mycobiota) is ongoing, and the effects of their various secondary metabolites on the health and disease of the host is a matter of current research. While the neurons of the central nervous system might be affected indirectly by compounds from gut microorganisms, the largest peripheral neuronal network (the enteric nervous system) is located within the gut and is exposed directly to such metabolites. We analyzed 320 fungal extracts and their effect on the viability of a human neuronal cell line (SH-SY5Y), as well as their effects on the viability and functionality of the most effective compound on primary ent…

Central nervous systemPharmaceutical SciencemicrobiomeBiologymedicine.disease_causeAnalytical ChemistryMicrobiologyPatulinlcsh:QD241-44103 medical and health sciencesPolyketidechemistry.chemical_compound0404 agricultural biotechnologyenteric nervous systemlcsh:Organic chemistrymycotoxinsDrug DiscoverymedicineMicrobiomePhysical and Theoretical Chemistryfusarium030304 developmental biologyCalcium signaling0303 health sciencesToxinOrganic Chemistry04 agricultural and veterinary sciences040401 food science<i>Penicillium</i>medicine.anatomical_structurechemistryChemistry (miscellaneous)Cell cultureMolecular Medicinegastrointestinal systemEnteric nervous systemfungiMolecules
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DNA barcoding reveals different cestode helminth species in northern European marine and freshwater ringed seals

2021

Three subspecies of the ringed seal (Pusa hispida) are found in northeastern Europe: P. h. botnica in the Baltic Sea, P. h saimensis in Lake Saimaa in Finland, and P. h. ladogensis in Lake Ladoga in Russia. We investigated the poorly-known cestode helminth communities of these closely related but ecologically divergent subspecies using COI barcode data. Our results show that, while cestodes from the Baltic Sea represent Schistocephalus solidus, all worms from the two lakes are identified as Ligula intestinalis, a species that has previously not been reported from seals. The observed shift in cestode communities appears to be driven by differential availability of intermediate fish host spec…

CestodaZoologyschistocephalus solidusBiologySubspeciesDNA barcodingPusa hispidasaimaannorppaloisetparasitic diseasesligula intestinalisCOI barcodingHelminthslaatokannorppaLigula intestinaliscestodaFreshwater sealspusa hispidaHost (biology)norppaRegular Articlebiology.organism_classificationheisimadotPusa hispidaInfectious DiseasesQL1-991DNA-viivakooditSchistocephalus solidusSchistocephalus soliduslajinmääritysCestodaAnimal Science and ZoologyParasitologyfreshwater sealsLigula intestinalisitämerennorppaZoologyInternational Journal for Parasitology: Parasites and Wildlife
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Toward Biopredictive Dissolution for Enteric Coated Dosage Forms

2016

The aim of this work was to develop a phosphate buffer based dissolution method for enteric-coated formulations with improved biopredictivity for fasted conditions. Two commercially available enteric-coated aspirin products were used as model formulations (Aspirin Protect 300 mg, and Walgreens Aspirin 325 mg). The disintegration performance of these products in a physiological 8 mM pH 6.5 bicarbonate buffer (representing the conditions in the proximal small intestine) was used as a standard to optimize the employed phosphate buffer molarity. To account for the fact that a pH and buffer molarity gradient exists along the small intestine, the introduction of such a gradient was proposed for p…

Chemistry PharmaceuticalCmaxBiological AvailabilityPharmaceutical Science02 engineering and technologyBuffers030226 pharmacology & pharmacyDosage form03 medical and health sciencesFirst pass effect0302 clinical medicineIVIVCCoated Materials BiocompatibleIntestine SmallDrug DiscoverymedicineHumansSolubilityDissolutionDosage FormsChromatographyAspirinGastric emptyingChemistryHydrogen-Ion Concentration021001 nanoscience & nanotechnologyEnteric coatingBicarbonatesDrug LiberationKineticsGastric EmptyingSolubilityArea Under CurveMolecular Medicine0210 nano-technologymedicine.drugMolecular Pharmaceutics
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Activity–Bioavailability balance in Oral Drug Development for a Selected Group of 6‐Fluoroquinolones

2002

Abstract A nomogram is proposed to select the best candidate in drug development studies with quinolones and is intended to substitute other possible models. The nomogram is referred to as an activity–bioavailability balance (ABB) because it includes the following two criteria: ABB= 1 / gm MIC ( drug candidate ) 1 /gm MIC ( ciprofloxacin ) · F calc \( drug candidate \) F calc ( ciproflaxacin ) . The in vitro activity of a group of 4′ N ‐alkyl‐ciprofloxacin derivatives was determined together with that of ciprofloxacin, initially against some reference strains and subsequently against 159 clinical isolates of eight selected species. The inverse of the geometric mean of the lowest concentrati…

ChemistryAdministration OralBiological AvailabilityPharmaceutical ScienceBiological activityMicrobial Sensitivity TestsPharmacologyAntimicrobialIntestinal absorptionRatsBioavailabilityCiprofloxacinStructure-Activity RelationshipMinimum inhibitory concentrationAnti-Infective AgentsDrug developmentmedicineAnimalsTechnology PharmaceuticalFluoroquinolonesAntibacterial agentmedicine.drugJournal of Pharmaceutical Sciences
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Does the addition of caseinophosphopeptides or milk improve zinc in vitro bioavailability in fruit beverages?

2009

Abstract The influence of caseinophosphopeptides (CPPs) added to fruit beverage versus milk based fruit beverage upon zinc retention, transport, and uptake, as well as the influence of Fe supplementation, were studied using a combined simulated gastrointestinal digestion/Caco-2 cell system. Zinc retention, transport, and uptake of milk based fruit beverage was 4- to 5-fold greater than that of fruit beverages with or without CPPs – no statistically significant differences being observed in relation to the presence or absence of CPPs. Possibly, a slow release of CPPs throughout the digestive tract, as can be expected to take place during the digestion of casein, has a more beneficial effect …

ChemistryCaseinfood and beverageschemistry.chemical_elementDigestive tractZincFood scienceDigestionIn vitroFood ScienceGastrointestinal digestionCell systemBioavailabilityFood Research International
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Beeinflussung der Darmmotorik durch Xylit

1963

Mit Hilfe der Tuschetransportmethode wurde an Mausen die Darmwirksamkeit von Xylit gepruft. Durch perorale Xylitgaben in Mengen von 0,5–1,0 g/kg Korpergewicht wurde die Darmtatigkeit deutlich angeregt. Kleinere Xylit-Dosen hatten demgegenuber keinen Einflus auf die Darmperistaltik. Die Anregung der Darmmotorik durch hohe Xylitgaben wird als osmotischer Effekt gedeutet.

ChemistryDrug DiscoveryMolecular MedicineSweetening agentsGeneral MedicineBody weightMolecular biologyGenetics (clinical)Intestinal motilityKlinische Wochenschrift
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Zur Frage der Resorption von Polyphosphaten

1965

Zur Klarung der Frage nach der Resorption von Polyphosphaten wurden Losungen von32P-markiertem Diphosphat, Triphosphat und einem Natriumpolyphosphat mit 64% P2O5 Ratten mit der Schlundsonde appliziert. Nach einer Verweildauer von 1, 2, 4, 8 und 16 Std dieser Polyphosphate im Magen-Darmtrakt wurden die Ratten dekapitiert und das erhaltene Frischblut radiometrisch und papierchromatographisch untersucht. Im enteiweisten Vollblut konnten nur Monophosphat und AMP nachgewiesen werden, d. h. es wird ausschlieslich anorganisches Monophosphat resorbiert, das durch enzymatische Aufspaltung der Polyphosphate gebildet wird. Dieses Monophosphat wird dann in die organische Bindung der AMP ubergefuhrt und…

ChemistryMedicine (miscellaneous)General MedicineBiochemistryMolecular biologyIntestinal absorptionResorptionPaper chromatographyDrug DiscoveryMolecular MedicineDigestive tractAbsorption (chemistry)Genetics (clinical)Food ScienceNuclear chemistryKlinische Wochenschrift
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