Search results for "Lymph"

showing 10 items of 4590 documents

Aaptamine Derivatives from the Indonesian Sponge Aaptos suberitoides

2013

Four new aaptamine derivatives (1-4) along with aaptamine (5) and three related compounds (6-8) were isolated from the ethanol extract of the sponge Aaptos suberitoides collected in Indonesia. The structures of the new compounds were unambiguously determined by one- and two-dimensional NMR and by HRESIMS measurements. Compounds 3, 5, and 6 showed cytotoxic activity against the murine lymphoma L5178Y cell line, with IC(50) values ranging from 0.9 to 8.3 μM.

PharmacologyMolecular StructurebiologyMurine lymphomaStereochemistryOrganic ChemistryPharmaceutical ScienceAntineoplastic AgentsAaptos suberitoidesbiology.organism_classificationPoriferaAnalytical ChemistryInhibitory Concentration 50MiceSpongeComplementary and alternative medicineIndonesiaDrug DiscoveryAnimalsHumansMolecular MedicineInhibitory concentration 50Drug Screening Assays AntitumorNaphthyridinesNuclear Magnetic Resonance BiomolecularJournal of Natural Products
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Ircinal E, a New Manzamine Derivative from the Indonesian Marine Sponge Acanthostrongylophora ingens

2015

Chemical investigation of the MeOH extract of the sponge Acanthostrongylophora ingens afforded the new manzamine derivative ircinal E (1), in addition to six known metabolites (2–7). The structure of the new compound was unequivocally elucidated using one- and two-dimensional NMR spectroscopy, as well as high-resolution mass spectrometry. Compounds 1–6 exhibited strong to moderate cytotoxicity against the murine lymphoma L5178Y cell line with IC50 values ranging from 2.8 to 21.7 μM.

PharmacologyMurine lymphomabiologyStereochemistryAcanthostrongylophora ingensPlant ScienceGeneral MedicineNuclear magnetic resonance spectroscopybiology.organism_classificationMass spectrometrySpongechemistry.chemical_compoundComplementary and alternative medicinechemistryDrug DiscoveryBotanyMoleculeCytotoxicityDerivative (chemistry)Natural Product Communications
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The many faces of erythropoietin: from erythropoiesis to a rational neuroprotective strategy

2008

It has been more than 10 years since the discovery that erythropoietin (EPO) and its receptor are expressed by the nervous system. In that brief time, a remarkable acceleration in understanding the...

PharmacologyNervous systembusiness.industrySettore MED/27 - NeurochirurgiaGeneral MedicineNeuroprotectionRecombinant ProteinsNeuroprotective Agentsmedicine.anatomical_structureErythropoietinhemic and lymphatic diseasesReceptors ErythropoietinmedicineAnimalsHumansErythropoiesisErythropoietin neuroprotectionPharmacology (medical)ReceptorbusinessErythropoietinNeurosciencemedicine.drug
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Crystal cell pattern modification in a melanotic tumor strain of Drosophila melanogaster.

1988

3rd instar larvae of the melanotic tumor tu-pb strain of Drosophila melanogaster hold a lower number of free-circulating crystal cells in their hemolymph than the wild type ones. This pattern could result from an abnormal retention of mature crystal cells in the hematopoietic organs, as the strong hemocyte melanization inside the lymph glands of heat-treated tu-pb larvae seems to demonstrate. Melanotic tumor formation and modification of the crystal cell pattern may be related.

Pharmacologyanimal structuresStrain (chemistry)biologyfungiWild typeTemperatureCell Biologybiology.organism_classificationCell biologyCellular and Molecular NeuroscienceHaematopoiesisDrosophila melanogasterGenesHemolymphImmunologyHemolymphMelanogasterMolecular MedicineInstarAnimalsLymphDrosophila melanogasterMolecular BiologyMelanomaExperientia
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Metabolites from Combretum dolichopetalum and its associated endophytic fungus Nigrospora oryzae--Evidence for a metabolic partnership.

2015

Abstract A new altersolanol derivative, 4-dehydroxyaltersolanol A ( 9 ), along with two known sesquiterpenoids, ( S )-7′-hydroxyabscisic acid ( 7 ) and ( S )-abscisic acid ( 8 ) were obtained from the endophytic fungus, Nigrospora oryzae , isolated from leaves of Combretum dolichopetalum . The host plant yielded six known compounds including ellagic acid ( 1 ), 3, 3′, 4-tri-O-methylellagic acid ( 2 ), arjunolic acid ( 3 ), 4′-dihydrophaseic acid ( 4 ), echinulin ( 5 ) and arestrictin B ( 6 ). Close structural similarities with regard to compounds 4 , 7 and 8 were observed between the metabolites from the host plant and those of the endophytic fungus. Furthermore compounds 5 and 6 are relate…

PharmacologybiologyMolecular StructureStereochemistryMouse LymphomaCombretumAnthraquinonesGeneral MedicineEndophytic fungusbiology.organism_classificationPlant Leaveschemistry.chemical_compoundMicechemistryAscomycotaCell Line TumorDrug DiscoveryEndophytesAnimalsCombretumArestrictin BNigrospora oryzaeCytotoxicityTwo-dimensional nuclear magnetic resonance spectroscopyEllagic acidFitoterapia
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Demethylnobiletin inhibits delayed-type hypersensitivity reactions, human lymphocyte proliferation and cytokine production

2007

Background and purpose: Our aim was to examine the effect of demethylnobiletin on various experimental models of delayed-type hypersensitivity (DTH) reactions and to determine its influence on the mediators and enzymes involved in these reactions. Experimental approach: DTH was induced in mice by oxazolone, dinitrofluorobenzene (DNFB) and sheep red blood cells (SRBC). The effect of demethylnobiletin on the ensuing DTH was studied, especially in relation to oedema formation, cell infiltration and tissue damage. Its activity on different mediators implicated in DTH reactions was also determined and its effect on nitric oxide synthase (NOS)-2 analysed. Finally, its influence on T lymphocyte pr…

Pharmacologybiologymedicine.medical_treatmentLymphocyteLymphocyte proliferationPharmacologyNitric oxideOxazoloneNitric oxide synthasechemistry.chemical_compoundCytokinemedicine.anatomical_structurechemistryApoptosisDelayed hypersensitivityImmunologymedicinebiology.proteinBritish Journal of Pharmacology
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Aminobisphosphonates as New Weapons for γ δ T Cell-Based Immunotherapy of Cancer

2008

Several observations in mice and in humans have collectively laid the foundation for examining the potential of γ δ T cells to exert tumor immunotherapy. Human γ δ T cells can be activated in a non-MHC dependent fashion either by low molecular mass phosphoantigens, or by agents that provoke the accumulation of endogenous pyrophosphates such as isopentenylpyrophosphate. Among the latter, aminobisphosphonates are well-established in the clinic, and extensive data are available on the compounds antiangiogenic, antiosteolytic and pro-apoptotic properties. In this review we discuss on the possibility that the intentional activation of γ δ T cells in vivo by aminobisphosphonates may represent a p…

Pharmacologybusiness.industrymedicine.medical_treatmentT cellOrganic ChemistryCancerEndogenyImmunotherapyT lymphocytemedicine.diseaseBiochemistrymedicine.anatomical_structureMechanism of actionAntigenIn vivoDrug DiscoveryImmunologymedicineMolecular Medicinemedicine.symptombusinessCurrent Medicinal Chemistry
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Profiling the diversity of innate lymphoid cells

2015

Genome-wide transcriptional profiling of tissue-resident innate lymphoid cells (ILCs) has provided important insight not only into their developmental relationships and phenotypic plasticity but also into previously unknown functions.

Phenotypic plasticityImmunologyInnate lymphoid cellImmunology and AllergyProfiling (information science)BiologyCell biologyNature Immunology
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Standard versus personalized schedule of regorafenib in metastatic gastrointestinal stromal tumors: a retrospective, multicenter, real-world study

2021

Background Despite its proven activity as third-line treatment in gastrointestinal stromal tumors (GIST), regorafenib can present a poor tolerability profile which often leads to treatment modifications and transient or permanent discontinuation; thus, in clinical practice physicians usually adopt various dosing and interval schedules to counteract regorafenib-related adverse events and avoid treatment interruption. The aim of this real-world study was to investigate the efficacy and safety of personalized schedules of regorafenib in patients with metastatic GIST, in comparison with the standard schedule (160 mg daily, 3-weeks-on, 1-week-off). Patients and methods Institutional registries a…

Phenylurea CompoundOncologyCancer Researchmedicine.medical_specialtyScheduleStromal cellPyridinesGastrointestinal Stromal TumorsPyridinePersonalized treatmentchemical and pharmacologic phenomenaMultikinase inhibitorchemistry.chemical_compoundQuality of lifeRetrospective Studieimmune system diseaseshemic and lymphatic diseasesInternal medicineRegorafenibmedicineHumansOriginal ResearchRetrospective StudiesGiSTbusiness.industryPhenylurea Compoundstoxicityhemic and immune systemspersonalized treatmentdigestive system diseasesquality of lifeOncologychemistryregorafenibGIST; personalized treatment; quality of life; regorafenib; toxicity; Humans; Phenylurea Compounds; Pyridines; Retrospective Studies; Gastrointestinal Stromal TumorsbusinessHumanGISTESMO Open
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Evaluation of thrombin generation in classical Philadelphianegative myeloproliferative neoplasms / Evaluarea generării trombinei în neoplasmele mielo…

2016

Abstract Introduction: Patients with Philadelphia-negative chronic myeloproliferative neoplasms (Ph-MPN), polycytemia vera (PV), essential thrombocythaemia (ET) and primary myelofibrosis (PMF), are prone to develop thrombotic events. We aimed to investigate the coagulation status in their plasma using thrombin generation assay (TGA), a functional global assay, on Ceveron® Alpha. Materials and methods: The samples were collected from 89 consecutive Ph-negative MPN patients and from 78 controls into K2EDTA and CTAD tubes for blood cell counts, TGA and coagulation screening tests. Thrombin generation was analysed in platelet-poor plasma using Technothrombin® TGA assay kit. Results: We found a …

Philadelphia negativeessential thrombocythemiaidiopatic myelofibrosisbusiness.industryR030204 cardiovascular system & hematologyThrombin generation03 medical and health sciences0302 clinical medicinepolycythemia verahemic and lymphatic diseasesthrombin generationCancer researchMedicineMedicinebusinessthrombosis030215 immunologyRomanian Journal of Laboratory Medicine
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