Search results for "NOE"

showing 10 items of 825 documents

Tarantula Hemocyanin Shows Phenoloxidase Activity

1998

An enzyme generally catalyzes one well defined reaction with high specificity and efficiency. We report here in contrast that the copper protein hemocyanin of the tarantula Eurypelma californicum exhibits two different functions. These occur at the same active site. While hemocyanin usually is an oxygen carrier, its function can be transformed totally to monophenoloxidase and o-diphenoloxidase activity after limited proteolysis with trypsin or chymotrypsin. N-acetyldopamine (NADA) is more effectively oxidized than L-dopa or dopamine. This irreversible functional switch of tarantula hemocyanin function is limited to the two subunits b and c of its seven subunit types. A conserved phenylalani…

Models MolecularStereochemistryCopper proteinDopamineProtein subunitmedicine.medical_treatmentPhenylalanineBiochemistrySubstrate SpecificityLevodopaMetalloproteinsMetalloproteinmedicineAnimalsChymotrypsinTrypsinImmunoelectrophoresisMolecular Biologychemistry.chemical_classificationBinding SitesbiologyMonophenol MonooxygenaseActive siteSpidersHemocyaninCell BiologyTrypsinOxygenEnzymeBiochemistrychemistrySpectrophotometryHemocyaninsbiology.proteinElectrophoresis Polyacrylamide GelCoppermedicine.drugJournal of Biological Chemistry
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Annular Tautomerism of 3(5)-Disubstituted-1H-pyrazoles with Ester and Amide Groups

2019

A series of disubstituted 1H-pyrazoles with methyl (1), amino (2), and nitro (3) groups, as well as ester (a) or amide (b) groups in positions 3 and 5 was synthesized, and annular tautomerism was investigated using X-ray, theoretical calculations, NMR, and FT-IR methods. The X-ray experiment in the crystal state showed for the compounds with methyl (1a, 1b) and amino (2b) groups the tautomer with ester or amide groups at position 3 (tautomer 3), but for those with a nitro group (3b, 4), tautomer 5. Similar results were obtained in solution by NMR NOE experiments in CDCl3, DMSO-d6, and CD3OD solvents. However, tautomer equilibrium was observed for 2b in DMSO. The FT-IR spectra in chloroform …

Models MolecularconformationNICSMolecular ConformationSubstituentPharmaceutical SciencePyrazoleCrystallography X-RayDFTMedicinal chemistryArticleAnalytical ChemistryX-raylcsh:QD241-441chemistry.chemical_compoundtautomerlcsh:Organic chemistryAmideDrug DiscoveryPhysical and Theoretical ChemistryAcetonitrileNOEMolecular StructureHydrogen bondSpectrum AnalysisOrganic ChemistryEstersHydrogen BondingAromaticityModels TheoreticalAmidesTautomerpyrazoleFT-IRchemistryChemistry (miscellaneous)NitroPyrazolesMolecular MedicineMolecules
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Subunit organization of the abalone Haliotis tuberculata hemocyanin type 2 (HtH2), and the cDNA sequence encoding its functional units d, e, f, g and…

1999

We have developed a HPLC procedure to isolate the two different hemocyanin types (HtH1 and HtH2) of the European abalone Haliotis tuberculata. On the basis of limited proteolytic cleavage, two-dimensional immunoelectrophoresis, PAGE, N-terminal protein sequencing and cDNA sequencing, we have identified eight different 40-60-kDa functional units (FUs) in HtH2, termed HtH2-a to HtH2-h, and determined their linear arrangement within the elongated 400-kDa subunit. From a Haliotis cDNA library, we have isolated and sequenced a cDNA clone which encodes the five C-terminal FUs d, e, f, g and h of HtH2. As shown by multiple sequence alignments, defg of HtH2 correspond structurally to defg from Octo…

Models Molecularfood.ingredientDNA ComplementarySequence analysismedicine.medical_treatmentMolecular Sequence DataOctopodiformesMegathura crenulataBiochemistryEvolution MolecularfoodSequence Analysis ProteinComplementary DNAmedicineAnimalsHaliotisAmino Acid SequenceCloning MolecularProtein Structure QuaternaryPeptide sequenceImmunoelectrophoresisbiologySequence Homology Amino AcidcDNA libraryHelix SnailsProtein primary structureHemocyaninAnatomySequence Analysis DNAbiology.organism_classificationPeptide FragmentsBiochemistryMolluscaHemocyaninsEuropean journal of biochemistry
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Immunohistochemical investigation on the pattern of vimentin expression in regenerated and intact monkey and human periodontal ligament.

2003

The expression of vimentin is well documented in the intact animal and human periodontal ligament (PDL), but there is limited information on the pattern of vimentin expression in the regenerated PDL. The aim of the present study was to investigate the pattern of vimentin expression in the regenerated and intact monkey and human PDL. A total of 12 chronic recession-type defects were created in three monkeys (Macaca fascicularis) and treated either with guided tissue regeneration (GTR), or with an enamel matrix protein derivative (EMD). After 5 months, the animals were sacrificed and specimens containing the defects and surrounding tissues were dissected free, decalcified in EDTA and embedded…

MolarMalePathologymedicine.medical_specialtyPeriodontal LigamentVimentinImmunoenzyme Techniquesstomatognathic systemDental Enamel ProteinsmedicinePeriodontal fiberAnimalsHumansVimentinCementumPeriodontitisGeneral DentistryPeriodontitisEnamel paintbiologyChemistryMesenchymal stem cellCell BiologyGeneral Medicinemedicine.diseaseMacaca fascicularismedicine.anatomical_structureOtorhinolaryngologyvisual_artChronic Diseasevisual_art.visual_art_mediumbiology.proteinGuided Tissue Regeneration PeriodontalImmunohistochemistryFollow-Up StudiesArchives of oral biology
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Inhibition of tumor lactate oxidation: consequences for the tumor microenvironment.

2011

Abstract Background and purpose Tumor cells are recognized as being highly glycolytic. However, recently it was suggested that lactate produced in hypoxic tumor areas may be taken up by the monocarboxylate transporter MCT1 and oxidized in well-oxygenated tumor parts. Furthermore, it was shown that inhibition of lactate oxidation using the MCT1 inhibitor α-cyano-hydroxycinnamate (CHC) can radio-sensitize tumors possibly by forcing a switch from lactate oxidization to glycolysis in oxygenated cells, which in turn improves tumor oxygenation and indirectly kills radio-resistant hypoxic tumor cells from glucose starvation. Material and methods To provide direct evidence for the existence of a ta…

Monocarboxylic Acid TransportersPasteur effectMice NudeUterine Cervical NeoplasmsImmunoenzyme Techniques03 medical and health sciencesMice0302 clinical medicineLactate oxidationFluorodeoxyglucose F18Cell Line TumorTumor MicroenvironmentPimonidazoleAnimalsRadiology Nuclear Medicine and imaging030304 developmental biologyMonocarboxylate transporter0303 health sciencesTumor microenvironmentbiologySymportersChemistryGlucose analogHematologyTumor OxygenationWarburg effectCell Hypoxia3. Good healthGlucoseOncologyCinnamatesHead and Neck NeoplasmsNitroimidazoles030220 oncology & carcinogenesisImmunologyLuminescent Measurementsbiology.proteinCancer researchCarcinoma Squamous CellLactatesLinear ModelsAutoradiographyFemaleGlycolysisOxidation-ReductionRadiotherapy and oncology : journal of the European Society for Therapeutic Radiology and Oncology
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The phylogeny of the Papaveraceae sensu lato: morphological, geographical and ecological implications

1995

On the background of the phylogeny of the Papaveraceae s.l., the evolution of the androecium and gynoecium, the geographical distribution, and the ecological differentiation of the family is discussed. An effort is made to homologize the diverse androecia of Pteridophyllum, Hypecoum, Fumariaceae and Papaveraceae s.str., and it is concluded that both the polyandrous androecium as found in the Papaveraceae s.str. and the polycarpellate gynoecium as found in Papaveraceae s. str. subfam. Papaveroideae incl. Platystemonoideae are secondary and derived from whorled oligomerous androecia and bicarpellate gynoecia, respectively. The comparative consideration of the geographical distribution, ecolog…

MonophylyGynoeciumSensuAridificationPhylogeneticsEcologyPapaveraceaePapaveroideaeBiologyPteridophyllumbiology.organism_classification
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PHENOLOGICAL AND MORPHOLOGICAL STUDIES OF PISTACIA TEREBINTHUS L. GENOTYPES NATIVE OF BULGARIA WITH DIFFERENT ASSET OF TREE SEXUALITY

2009

The genus Pistacia is a dioecious species staminate and pistillate inflorescences born on different trees and are wind pollinated. In pistachio orchards, female and male flowering periods are often not synchronized. In fact, male trees spread their pollen before the flowers of female trees become receptive. Pollination is commonly devoted to spontaneous males of P. terebinthus. In this research authors refer to the results obtained observing the phenology of the blooming period of monoicous genotypes of P. terebinthus discovered in the Rhodope Mountains (Bulgaria). In some selected trees phenological stages have been observed in situ. The blooming date is influenced by local environmental c…

MorphologybiologyPhenologyMonoeciouDioeciouFlower biologyHorticulturebiology.organism_classificationPistacia terebinthusSettore AGR/03 - Arboricoltura Generale E Coltivazioni ArboreeHorticulturePhenologyInflorescencePlant morphologyBotanyPlant reproductive morphologyP. terebinthuActa Horticulturae
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The monocyte-macrophage system is affected in lysosomal storage diseases: an immunoelectron microscopic study

1997

Studying peripheral blood mononuclear cells (PBMCs) has become an important diagnostic tool in lysosomal storage diseases. Previous studies revealed that B and subclasses of T lymphocytes participate in the storage process, whereas the role of circulating monocytes was not clear. In this study, the involvement of CD14+ monocytes in lysosomal diseases was investigated. Blood samples from six patients with different lysosomal storage disorders were studied, including one with late--infantile and three with juvenile neuronal ceroid--lipofuscinoses, and two with mucopolysaccharidosis type VI. CD14+ cells were separated immunomagnetically from PBMCs and studied by light and electron microscopy. …

Mucopolysaccharidosis VIMacrophagesMucopolysaccharidosisCD14MonocyteMucopolysaccharidosis type VILipopolysaccharide ReceptorsBiologymedicine.diseasePeripheral blood mononuclear cellMonocytesPathology and Forensic MedicineLysosomal Storage DiseasesCellular and Molecular Neurosciencemedicine.anatomical_structureNeuronal Ceroid-LipofuscinosesImmunologyLysosomal storage diseasemedicineHumansMacrophageNeuronal ceroid lipofuscinosisNeurology (clinical)Microscopy ImmunoelectronActa Neuropathologica
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Ferrocenyl glycopeptides as electrochemical probes to detect autoantibodies in multiple sclerosis patients' será

2008

Abstract Glycopeptide analogues of CSF114(Glc), modified at N-terminus with new ferrocenyl carboxylic acid and a new ferrocenyl-thiphosphino amino acid, were used to implement a new electrochemical biosensor for autoantibody detection in multiple sclerosis. The ferrocenyl moiety of these "electrochemical probes" did not affect autoantibody recognition both in SP-ELISA and in inhibition experiments. By electrochemical monitoring the interactions of the modified peptides Fc-CSF114(Glc) and 4-FcPhP(S)Abu-CSF114(Glc) with the autoantibodies, we demonstrated that autoantibodies could be detected with a sensitivity comparable to ELISA method. The new electrochemical probes can be proposed to char…

Multiple SclerosisMetallocenesCarboxylic acidBiophysics010402 general chemistry01 natural sciencesBiochemistryBiomaterialsImmunoenzyme Techniques[ CHIM.CATA ] Chemical Sciences/CatalysismedicineElectroanalytical methodElectrochemistryMoietyHumansFerrous CompoundsAntigensComputingMilieux_MISCELLANEOUSAutoantibodieschemistry.chemical_classification010405 organic chemistryChemistryMultiple sclerosisOrganic ChemistryAutoantibodyGlycopeptidesGeneral Medicine[CHIM.CATA]Chemical Sciences/Catalysismedicine.diseaseGlycopeptide0104 chemical sciences3. Good healthAmino acidSolutionsBiochemistryMolecular ProbesGoldCyclic voltammetryChromatography Liquid
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The phosphorylated pathway of serine biosynthesis is essential both for male gametophyte and embryo development and for root growth in Arabidopsis.

2013

This study characterizes the phosphorylated pathway of Ser biosynthesis (PPSB) in Arabidopsis thaliana by targeting phosphoserine phosphatase (PSP1), the last enzyme of the pathway. Lack of PSP1 activity delayed embryo development, leading to aborted embryos that could be classified as early curled cotyledons. The embryo-lethal phenotype of psp1 mutants could be complemented with PSP1 cDNA under the control of Pro35S (Pro35S:PSP1). However, this construct, which was poorly expressed in the anther tapetum, did not complement mutant fertility. Microspore development in psp1.1/psp1.1 Pro35S:PSP1 arrested at the polarized stage. The tapetum from these lines displayed delayed and irregular devel…

MutantCitric Acid CycleGreen Fluorescent ProteinsImmunoblottingArabidopsisPlant ScienceBiologyPlant RootsSerineMicrosporeMicroscopy Electron TransmissionGene Expression Regulation PlantArabidopsisSerineArabidopsis thalianaAmino AcidsPhosphorylationResearch ArticlesTapetumArabidopsis ProteinsReverse Transcriptase Polymerase Chain ReactionGene Expression Regulation DevelopmentalEmbryoPhosphoserine phosphataseCell Biologybiology.organism_classificationPlants Genetically ModifiedPhosphoric Monoester HydrolasesBiosynthetic PathwaysBiochemistryMicroscopy FluorescenceMutationSeedsPollenGlycolysisThe Plant cell
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