Search results for "Nandrolone"

showing 10 items of 12 documents

Effects of Nandrolone Stimulation on Testosterone Biosynthesis in Leydig Cells

2016

Anabolic androgenic steroids (AAS) are among the drugs most used by athletes for improving physical performance, as well as for aesthetic purposes. A number of papers have showed the side effects of AAS in different organs and tissues. For example, AAS are known to suppress gonadotropin‐releasing hormone, luteinizing hormone, and follicle‐stimulating hormone. This study investigates the effects of nandrolone on testosterone biosynthesis in Leydig cells using various methods, including mass spectrometry, western blotting, confocal microscopy and quantitative real‐time PCR. The results obtained show that testosterone levels increase at a 3.9 μM concentration of nandrolone and return to the ba…

0301 basic medicineEnzymologicMalePhysiologyClinical BiochemistryAndrogenAnabolic Agents; Androgens; Animals; Cell Line; Cell Survival; Dose-Response Relationship Drug; Gene Expression Regulation Enzymologic; Leydig Cells; Male; Nandrolone; Phosphoproteins; Rats; Steroid 17-alpha-Hydroxylase; Testosterone; Physiology; Clinical Biochemistry; Cell BiologyAnabolic AgentsOriginal Research ArticlesNandroloneTestosteroneOriginal Research ArticleTestosteroneAnabolic Agents; Androgens; Animals; Cell Line; Cell Survival; Dose-Response Relationship Drug; Gene Expression Regulation Enzymologic; Leydig Cells; Male; Nandrolone; Phosphoproteins; Rats; Steroid 17-alpha-Hydroxylase; Testosterone; Clinical Biochemistry; Cell Biology; Physiology; Medicine (all)Steroidogenic acute regulatory proteinMedicine (all)Leydig CellsSteroid 17-alpha-HydroxylaseCYP17A1PhosphoproteinAndrogensDrugLuteinizing hormonemedicine.drugAnabolic Agents; Androgens; Animals; Cell Line; Cell Survival; Dose-Response Relationship Drug; Gene Expression Regulation Enzymologic; Leydig Cells; Male; Nandrolone; Phosphoproteins; Rats; Steroid 17-alpha-Hydroxylase; TestosteroneLeydig Cellendocrine systemmedicine.medical_specialtyCell SurvivalBiologyGene Expression Regulation EnzymologicCell LineDose-Response Relationship03 medical and health sciencesDownregulation and upregulationIn vivoInternal medicinemedicineAnimalsDose-Response Relationship DrugAnimalCell BiologyPhosphoproteinsRats030104 developmental biologyEndocrinologyGene Expression RegulationNandroloneAnabolic AgentRatHormone
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Changes in neuromuscular performance and muscle fiber characteristics of elite power athletes self-administering androgenic and anabolic steroids

1984

The influence of androgenic-anabolic steroid-induced changes in measures of body composition, muscle fiber characteristics and various aspects of the neuromuscular performance of the leg extensor muscles was investigated in five experimental and six control power athletes during the 24-week programmed strength training followed by the additional six week training without hormone drugs. The mean values of the dosages of self-administration during the 24-week period were 31.0 +/- 14.3 mg/day for anabolic steroids (methandienone, stanozolol, nandrolone) and 178.4 +/- 82.7 mg/week for testosterone. During the 24-week hormone period the experimental group gained in fat-free weight (p less than 0…

AdultMalemedicine.medical_specialtyAnabolismPhysiologyVastus lateralis muscleStrength trainingMuscle RelaxationNeuromuscular JunctionSquatIsometric exercisemedicine.disease_causeAnabolic AgentsJumpingIsometric ContractionInternal medicinemedicineHumansNandroloneTestosteroneTestosteroneDoping in Sportsbusiness.industryMusclesEndocrinologyNandroloneAndrogensbusinessStanozololMuscle Contractionmedicine.drugActa Physiologica Scandinavica
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Gonadotrophin-releasing hormone analogue or dienogest plus estradiol valerate to prevent pain recurrence after laparoscopic surgery for endometriosis…

2015

Objectives To evaluate the efficacy of dienogest + estradiol valerate (E2V) and gonadotrophin-releasing hormone analogue (GnRH-a) in reducing recurrence of pain in patients with chronic pelvic pain due to laparoscopically diagnosed and treated endometriosis. Design Multi-center, prospective, randomized study. Setting Three university departments of obstetrics and gynecology in Italy. Population Seventy-eight women who underwent laparoscopic surgery for endometriosis combined with chronic pelvic pain. Methods Post-operative administration of dienogest + E2V for 9 months (group 1) or GnRH-a monthly for 6 months (group 2). Main outcome measures A visual analogue scale was used to test intensit…

Laparoscopic surgerymedicine.medical_treatmentEndometriosischronic pelvic painlaw.inventionGonadotropin-Releasing Hormonechemistry.chemical_compoundEndometriosis;dienogest;GnRH-analogue;pain recurrence;chronic pelvic painRandomized controlled triallawRecurrenceSurveys and QuestionnairesMedicineNandroloneSurveys and QuestionnaireProspective StudiesEndometriosiPain Measurementeducation.field_of_studyEstradiolMedicine (all)Estradiol valerateObstetrics and GynecologyGeneral MedicineMiddle Agedpain recurrenceDrug CombinationsDienogestItalyFemalemedicine.symptommedicine.drugHumanAdultmedicine.medical_specialtyAdolescentVisual analogue scalePopulationEndometriosisPelvic PainHumansPain ManagementEndometriosis GnRH-analogue chronic pelvic pain dienogest pain recurrence.educationGnRH-analoguebusiness.industryPelvic painmedicine.diseaseSettore MED/40 - Ginecologia E OstetriciaSurgeryProspective StudiechemistrydienogestQuality of LifeLaparoscopybusiness
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Nandrolone decanoate interferes with testosterone biosynthesis altering blood-testis barrier components

2017

Abstract The aim of this study was to investigate whether nandrolone decanoate (ND) use affects testosterone production and testicular morphology in a model of trained and sedentary mice. A group of mice underwent endurance training while another set led a sedentary lifestyle and were freely mobile within cages. All experimental groups were treated with either ND or peanut oil at different doses for 6 weeks. Testosterone serum levels were measured via liquid chromatography–mass spectrometry. Western blot analysis and quantitative real‐time PCR were utilized to determine gene and protein expression levels of the primary enzymes implicated in testosterone biosynthesis and gene expression leve…

Male0301 basic medicinemedicine.medical_specialtyNandrolone decanoateStimulationEndogenyMUC1BiologyMale infertilityMice03 medical and health sciencesAnabolic AgentsWestern blotPhysical Conditioning AnimalInternal medicineTestisGene expressionmedicineAnimalsNandroloneBlood-testis barrier; MMP-2; MMP-9; MUC1; Nandrolone decanoate; Testosterone; TJP1; Molecular Medicine; Cell Biologyblood–testis barrierInducerTestosteroneTJP1TestosteroneBlood-testis barrierBlood–testis barrierMMP‐9medicine.diagnostic_testMMP-2Mucin-1Tissue Inhibitor of MetalloproteinasesOriginal ArticlesCell Biologymedicine.diseaseProtein Transport030104 developmental biologyEndocrinologyGene Expression RegulationMatrix Metalloproteinase 9Zonula Occludens-1 ProteinMatrix Metalloproteinase 2Molecular MedicineOriginal ArticleMMP‐2Sedentary BehaviorMMP-9Signal Transduction
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Nandrolone decanoate interferes on testosterone biosynthesis and alters blood-testis barrier.

2018

Nandrolone decanoate (ND) is a synthetic testosterone analogue considered one of the most commonly abused anabolic androgenic steroids by adolescents and athletes. ND is alleged to promote an increase in muscle mass and improves both physical appearance and sporting performance, but ND abuse is often associated with serious adverse effects, interfering with the endocrine system and the reproductive system. In a previous study, we demonstrated that ND treatment of Leydig cells interferes with the biosynthesis of testosterone in a dose increase-dependent fashion (1). As a consequence of the results obtained in vitro, in this study an animal model was utilized to better understand the side eff…

Nandrolone decanoatetestosteroneblood–testis barrier
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Retention-structure relationship studies for some steroidal hormones in micellar liquid chromatography

2000

The retention behavior in a C18 column of fourteen steroidal hormones (clostebol acetate, dehydrotestosterone, dydrogesterone, medroxyprogesterone, medroxyprogesterone acetate, methandienone, methyltestosterone, nandrolone, nandrolone decanoate, progesterone, testosterone, testosterone enanthate, testosterone propionate and, stanozolol) with pure micellar mobile phases prepared from sodium dodecyl sulfate (SDS), and hybrid mobile phases comprising SDS-acetonitrile and SDS-pentanol, was correlated with their octanol-water partition coefficients. Similar correlations were found with retention data obtained by other authors in gas chromatography, conventional reversed-phase liquid chromatograp…

Testosterone propionateChromatographyChemistrymedicine.medical_treatmentMedroxyprogesteroneOrganic ChemistryClinical BiochemistryBiochemistryMicellar electrokinetic chromatographyAnalytical ChemistrySteroidchemistry.chemical_compoundMicellar liquid chromatographyNandroloneCLOSTEBOL ACETATEmedicineMethyltestosteronemedicine.drug
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DETERMINATION OF STEROIDAL HORMONES IN URINE SAMPLES BY MICELLAR LIQUID CHROMATOGRAPHY FOLLOWING SOLID-PHASE EXTRACTION

2001

Steroidal hormones were determined in spiked urine samples using micellar mobile phases of sodium dodecyl sulphate (SDS)-pentanol, solid-phase extraction (SPE), and detection in the UV region. In the optimized procedure, a 10 mL aliquot of urine sample is loaded into a C18 cartridge and washed with 2 mL of 50:50 (v/v) methanol-water, followed by 200 μL of 70:30 (v/v) methanol-water. The retained steroids are eluted with 2 mL of methanol and the eluate evaporated to dryness under nitrogen at 50°C. The residue is redissolved with 200 μL of the micellar mobile phase used in the chromatographic separation and injected into the chromatograph. The performance of the procedure was checked for 13 s…

Testosterone propionateChromatographyElutionMedroxyprogesteroneClinical BiochemistryPharmaceutical ScienceBiochemistryMicellar electrokinetic chromatographyAnalytical Chemistrychemistry.chemical_compoundchemistryNandroloneMicellar liquid chromatographymedicineSolid phase extractionMethyltestosteronemedicine.drugJournal of Liquid Chromatography & Related Technologies
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SENSITIZED LANTHANIDE FLUORESCENCE DETECTION OF STEROIDAL HORMONES

2000

Several steroidal hormones with an α,β-unsaturated carbonyl group sensitized the fluorescence of terbium(III) ions: medroxyprogesterone, medroxyprogesterone acetate, methyltestosterone, nandrolone, nandrolone decanoate, progesterone, testosterone, testosterone enanthate, and testosterone propionate, but other steroids which have this chromophore did not give any signal: clostebol acetate, dehydrotestosterone, dydrogesterone, methandienone, and methenolone enanthate. Sensitized fluorescence was used to detect the steroids when eluted with micellar mobile phases of sodium dodecyl sulphate (SDS)-acetonitrile and SDS-pentanol containing 0.01 M Tb(III), with 245 nm and 545 nm as excitation and e…

Testosterone propionateChromatographyMedroxyprogesteroneClinical BiochemistryMetandienoneClostebolPharmaceutical ScienceBiochemistryAnalytical Chemistrychemistry.chemical_compoundchemistryNandroloneCLOSTEBOL ACETATEmedicineMethyltestosteroneMetenolonemedicine.drugJournal of Liquid Chromatography & Related Technologies
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Lack of effects of anabolic-androgenic steroids on locomotor activity in intact male mice.

1999

Anabolic-androgenic steroid abusers have reported hyperactivity euphoria, and decreased fatigue, among other behavioral effects. It has been suggested that the effects of these substances on the central nervous system are similar to those of psychostimulants; however, the influence of steroids on general locomotor activity in laboratory animals is not well understood, especially how noncastrated male rodents are affected. In this study, spontaneous locomotor activity displayed by gonadally intact male mice submitted to several experimental conditions was analyzed. Different housing conditions (individual or cohabiting with a female), diverse steroids (testosterone propionate, nandrolone de…

Testosterone propionateMalemedicine.medical_specialtymedicine.drug_classPeriod (gene)medicine.medical_treatmentCentral nervous systemExperimental and Cognitive PsychologyEndogenyMotor ActivityEuphoriantSteroid03 medical and health scienceschemistry.chemical_compoundMiceRandom Allocation0302 clinical medicineAnabolic AgentsInternal medicineTestismedicineAnimalsNandroloneTestosteroneIntact male030222 orthopedicsBehavior Animalbusiness.industry030229 sport sciencesAndrogenHousing AnimalSensory Systemsmedicine.anatomical_structureEndocrinologychemistryNandrolone DecanoateFemalebusinessLocomotionPerceptual and motor skills
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Ver�nderungen an Proteinen der Leber und des Blutes bei experimenteller Lebercirrhose und nach Behandlung mit Decortin und einem anabolen Steroid

1963

medicine.medical_specialtyCirrhosisbiologyChemistrymedicine.medical_treatmentGeneral MedicineMitochondrionmedicine.diseaseFibrinogenMolecular medicineBlood proteinsEndocrinologyNandroloneInternal medicineDrug Discoverymedicinebiology.proteinMolecular MedicineCeruloplasminGenetics (clinical)Anabolic steroidmedicine.drugKlinische Wochenschrift
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