Search results for "Nuclear magnetic resonance spectroscopy"

showing 10 items of 843 documents

A New Aromatic Compound from the Stem Bark of Terminalia catappa

2015

A new aromatic compound 3,4,5-trimethoxyphenyl-1- O-(4-sulfo)-β-D-glucopyranoside (1), in addition to two triterpenoid saponins (chebuloside II, arjunoglucoside II), two triterpenes (arjunolic acid and 3-betulinic acid) and sitosterol-3- O-β-D-glucopyranoside have been isolated from the barks of Terminalia catappa. Their structures have been established on the basis of spectroscopic techniques (1D/2D NMR) and MS. Their cytotoxicity and anti-inflammatory activity, together with the antioxidant capacity of compound 1 were also evaluated.

PharmacologyStem barkMagnetic Resonance SpectroscopyCombretaceaeMolecular StructurePlant StemsbiologyPlant ExtractsChemistryArjunolic acidTerminaliaPlant ScienceGeneral Medicinebiology.organism_classificationTerpeneAntioxidant capacityComplementary and alternative medicineDrug DiscoveryPlant BarkTerminaliaOrganic chemistryCytotoxicityTwo-dimensional nuclear magnetic resonance spectroscopyNatural Product Communications
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Cytotoxic Bufadienolides from the Leaves of Melianthus major

2020

Melianthus major is a medicinal plant endemic to South Africa. Its leaf extract led to the isolation of five new bufadienolides, 2β-acetoxy-3,5-di-O-acetylhellebrigenin (1), 2β-acetoxy-3-O-acetylhellebrigenin (2), 2β-acetoxy-14-deoxy-15β,16β-epoxymelianthugenin (4), 2β-acetoxy-14-deoxy-15β,16β-epoxymelianthusigenin (5), and 2β-hydroxymelianthusigenin (6), and four known analogues. The structures of the compounds were elucidated using NMR and HRESIMS data analyses. The relative configurations were defined by single-crystal X-ray crystallography and NOESY correlations. The isolated compounds exhibited strong cytotoxicity against MCF-7 breast cancer cells and sensitive CCRF-CEM and multidrug-r…

Pharmacologybiology010405 organic chemistryChemistryCcrf cemOrganic ChemistryPharmaceutical Sciencemedicine.diseasebiology.organism_classification01 natural sciencesMolecular biologyMelianthus major0104 chemical sciencesAnalytical Chemistry010404 medicinal & biomolecular chemistryLeukemiaComplementary and alternative medicineDrug DiscoverymedicineIc50 valuesMolecular MedicineCytotoxic T cellBreast cancer cellsCytotoxicityTwo-dimensional nuclear magnetic resonance spectroscopyJournal of Natural Products
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Metabolites from Combretum dolichopetalum and its associated endophytic fungus Nigrospora oryzae--Evidence for a metabolic partnership.

2015

Abstract A new altersolanol derivative, 4-dehydroxyaltersolanol A ( 9 ), along with two known sesquiterpenoids, ( S )-7′-hydroxyabscisic acid ( 7 ) and ( S )-abscisic acid ( 8 ) were obtained from the endophytic fungus, Nigrospora oryzae , isolated from leaves of Combretum dolichopetalum . The host plant yielded six known compounds including ellagic acid ( 1 ), 3, 3′, 4-tri-O-methylellagic acid ( 2 ), arjunolic acid ( 3 ), 4′-dihydrophaseic acid ( 4 ), echinulin ( 5 ) and arestrictin B ( 6 ). Close structural similarities with regard to compounds 4 , 7 and 8 were observed between the metabolites from the host plant and those of the endophytic fungus. Furthermore compounds 5 and 6 are relate…

PharmacologybiologyMolecular StructureStereochemistryMouse LymphomaCombretumAnthraquinonesGeneral MedicineEndophytic fungusbiology.organism_classificationPlant Leaveschemistry.chemical_compoundMicechemistryAscomycotaCell Line TumorDrug DiscoveryEndophytesAnimalsCombretumArestrictin BNigrospora oryzaeCytotoxicityTwo-dimensional nuclear magnetic resonance spectroscopyEllagic acidFitoterapia
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Steroidal Saponins from the Fruits of Cestrum ruizteranianum

2011

Seven spirostane and furostane-type glycosides were isolated from the aqueous methanolic extract of the fruits of Cestrum ruizteranianum and characterized mainly by 2D NMR spectroscopy and mass spectrometry. These known saponins belong to the Δ5-spirostene and Δ5-furostene series and are reported in this species for the first time.

Pharmacologychemistry.chemical_classificationChromatographybiologyChemistryCestrumGlycosidePlant ScienceGeneral MedicineNuclear magnetic resonance spectroscopyMass spectrometrybiology.organism_classificationComplementary and alternative medicineDrug DiscoverySpectroscopyTwo-dimensional nuclear magnetic resonance spectroscopyNatural Product Communications
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Phytochemistry of Weigela x “kosteriana variegata” (Caprifoliaceae)

2018

One new triterpene glycoside 3- O-β-D-xylopyranosyl-(1→4)-[β-D-glucopyranosyl-(1→3)]-β-D-xylopyranosyl-(1→4)-β-D-xylopyranosyl-(1→3)-α-L-rhamnopyranosyl-(1→2)-α-L-arabinopyranosyloleanolic acid, was isolated from Weigela x “kosteriana variegata” (Caprifoliaceae), with three known ones. Their structures were characterized by a combination of mass spectrometry and 1D and 2D NMR spectrocopic techniques including 1H- and 13C NMR, COSY, TOCSY, NOESY, HSQC, and HMBC experiments. The toxicological properties of some glycosides were determined with a zebrafish-based assay. The results show that the most active compounds were toxic to the larvae in the range of 1 μM.

Pharmacologychemistry.chemical_classificationWeigelaPhytochemistrybiology010405 organic chemistryStereochemistryGlycosidePlant ScienceGeneral MedicineCarbon-13 NMRbiology.organism_classification01 natural sciences0104 chemical sciences010404 medicinal & biomolecular chemistryComplementary and alternative medicineTriterpenechemistryDrug DiscoveryCaprifoliaceaeTwo-dimensional nuclear magnetic resonance spectroscopyHeteronuclear single quantum coherence spectroscopyNatural Product Communications
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Steroidal saponins from Chlorophytum deistelianum

2016

Abstract Phytochemical investigation of the aerial parts of Chlorophytum deistelianum led to the isolation of four previously undescribed steroidal saponins called chlorodeistelianosides A–D with five known ones. Their structures were established mainly by extensive 1D and 2D NMR spectroscopic techniques and mass spectrometry as (25R)-3β-[(β- d -glucopyranosyl-(1 → 3)-[α- l -rhamnopyranosyl-(1 → 4)]-β- d -xylopyranosyl-(1 → 3)-[β- d -glucopyranosyl-(1 → 2)]-β- d -glucopyranosyl-(1 → 4)-β- d -galactopyranosyl)oxy]-5α-spirostan-12-one, (24S,25S)-24-[(β- d -glucopyranosyl)oxy]-3β-[(β- d -glucopyranosyl-(1 → 2)-[β- d -xylopyranosyl-(1 → 3)]-β- d -glucopyranosyl-(1 → 4)-β- d -galactopyranosyl)ox…

Pharmacologychemistry.chemical_classificationbiologyChemistryStereochemistryOrganic ChemistryPharmaceutical ScienceGlycosidebiology.organism_classificationAnalytical ChemistryComplementary and alternative medicineDrug DiscoveryMolecular MedicineChlorophytumCytotoxicityTwo-dimensional nuclear magnetic resonance spectroscopyHuman cancerPlanta Medica
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Antiproliferative oleanane saponins from Polyscias guilfoylei

2008

Three new oleanane saponins (1–3), together with four known ones (4–7), were isolated from the aerial parts of Polyscias guilfoylei. Their structures were elucidated by 1D and 2D NMR experiments, including 1D TOCSY, DQF-COSY, ROESY, HSQC, and HMBC spectroscopy, as well as ESIMS analysis. The antiproliferative activity of all compounds was evaluated using three murine and human cancer cell lines; J774.A1, HEK-293, and WEHI-164. All the compounds were inactive except for 3β- O-[β-D-glucopyranosyl-(1→2)-α-L-arabinopyranosyl]-echinocystic acid 28-[ O-β-D-glucopyranosyl-(1→6) O-β-D-glucopyranosyl] ester (3), which was active against all the cell lines.

Pharmacologychemistry.chemical_classificationbiologyStereochemistryGlycosidePlant ScienceGeneral Medicinebiology.organism_classificationPolyscias guilfoyleiSettore CHIM/08 - Chimica FarmaceuticaOleanane Saponins Antiproliferative effectsTerpenechemistry.chemical_compoundComplementary and alternative medicinechemistryDrug DiscoverySettore BIO/14 - FarmacologiaTwo-dimensional nuclear magnetic resonance spectroscopyOleanane
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Preparation and Structure of Bicycloalkane-Condensed Aryldiaziridines Accompanied by Pyrimidines

2007

Di-exo- and di-endo-2-aminonorbomane/enemethanamines 1-3, di-exo-oxanorbomene derivative 4 and cis-cyclohexane and trans-4-cyclohexene analogues 5, 6 were reacted with p-chlorobenzaldehyde in the presence of N-bromosuccinimide in dichloromethane. Via the reactions of 1-6, condensed diaziridines 7-12 accompanied by pyrimidine derivatives 13-16 were prepared after isolation with column chromatography. The mechanisms proposed for alternative transformations were supported by DFT calculations. The structures of the new compounds were proved by IR and NMR spectroscopy and, for 7, 9 and 12, also by means of X-ray crystallography.

Pharmacologychemistry.chemical_compoundColumn chromatographyDiaziridinechemistryPyrimidineComputational chemistryOrganic ChemistryOrganic chemistryGeneral MedicineNuclear magnetic resonance spectroscopyAnalytical ChemistryDichloromethaneHETEROCYCLES
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Stimulated 7^Li echo NMR spectroscopy of slow ionic motions in a solid electrolyte

2000

Abstract Lithium spin-alignment spectroscopy is presented as an NMR technique for studying slow translational motions in solid and solid-like ionic conductors. We employ phase cycling that allows to measure two-time translational correlation functions via the generation of a pure quadrupolar ordered state. Correlation functions of the crystalline electrolyte Li 3 Sc 2 (PO 4 ) 3 were recorded for times ranging from about 0.1 ms to more than 10 s, implying that translational diffusion coefficients smaller than 10 −20 m 2 /s become accessible.

Phase cyclingChemistryDiffusionAnalytical chemistryGeneral Physics and AstronomyIonic bondingchemistry.chemical_elementElectrolyteNuclear magnetic resonance spectroscopy530LithiumPhysical and Theoretical ChemistrySpectroscopyElectrical conductor
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Static and MAS 35CI NMR and Molecular Motions of ClO −4 Ions in the Various Phases of Multimethylammonium Perchlorates

1986

Static and MAS*) 35CI NMR data of CIO−4 ions in the low-, intermediate- and high-temperature phases of trimethylammonium, dimethylammonium and monomethylammonium perchlorates are reported. The observed solid-solid phase transitions are interrelated with the motional state of the perchlorate ions. In the low-temperature phase III of trimethylammonium perchlorate there is an anisotropic motion of the ClO−4 ions with a constant quadrupole frequency of 185 kHz and an increasing value of the asymmetry parameter when approaching phase transition III-II. The activation energy for this motion is found to be 44.3 kj/mol. At the transition III-II the ClO−4 ions gain orientational degrees of freedom m…

Phase transitionPerchloratechemistry.chemical_compoundMagic angleNuclear magnetic resonanceChemistryGeneral Chemical EngineeringPhase (matter)QuadrupolePhysical chemistryNuclear magnetic resonance spectroscopyActivation energyIonBerichte der Bunsengesellschaft für physikalische Chemie
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