Search results for "PREP"

showing 10 items of 1334 documents

Effects of controlled-release on the pharmacokinetics and absorption characteristics of a compound undergoing intestinal efflux in humans

2006

Abstract Objective The number of active pharmaceutical ingredients (API) undergoing inhibitable and saturable intestinal efflux is considerable. As a consequence, absorption and bioavailability may depend on the intestinal concentration profile of the drug and may vary as a function of dose and release rate of the drug from the dosage form. The impact of controlled versus immediate-release on the absorption of P-glycoprotein substrates is currently unknown. Thus, the main focus of the present study was a comparison of the pharmacokinetics of the P-gp model substrate talinolol following administration of immediate-release (IR) and controlled-release (CR) tablets to healthy human volunteers w…

AdultMaleActive ingredientChemistryPharmaceutical ScienceAbsorption (skin)PharmacologyCrossover studyControlled releaseDosage formBioavailabilityPropanolamineschemistry.chemical_compoundIntestinal AbsorptionSolubilityPharmacokineticsDelayed-Action PreparationsHumansFemaleATP Binding Cassette Transporter Subfamily B Member 1TabletsTalinololEuropean Journal of Pharmaceutical Sciences
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An assessment of prime‐boost vaccination schedules with AS03A‐adjuvanted prepandemic H5N1 vaccines: a randomized study in European adults

2012

Please cite this paper as: Gillard et al. (2012) An assessment of prime‐boost vaccination schedules with AS03A‐adjuvanted prepandemic H5N1 vaccines: a randomized study in European adults. Influenza and Other Respiratory Viruses DOI: 10.1111/j.1750‐2659.2012.00349.x. Background  Long‐term persistence of immune response and safety of an H5N1 prepandemic influenza vaccine adjuvanted with AS03 (an α‐tocopherol oil‐in‐water emulsion‐based adjuvant system) was evaluated using various prime‐boost schedules that mimicked potential pandemic scenarios (NCT00430521). Methods  Five hundred and twelve healthy adults aged 18–60 years received primary vaccination with one or two doses (0, 21 days schedule…

AdultMaleAdolescentalpha-TocopherolImmunization SecondaryAntibodies ViralAS03Young Adultprime‐boostAdjuvants ImmunologicInfluenza HumanHumansAdjuvantImmunization ScheduleInfluenza A Virus H5N1 SubtypeVaccinationOriginal ArticlesH5N1Hemagglutination Inhibition TestsMiddle AgedAntibodies NeutralizingTreatment OutcomeInfluenza VaccinesOriginal ArticleFemaleinfluenzaprepandemicInfluenza and Other Respiratory Viruses
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Application of headspace solid phase dynamic extraction gas chromatography/mass spectrometry (HS-SPDE-GC/MS) for biomonitoring of n-heptane and its m…

2011

Abstract Solid phase dynamic extraction (SPDE) is an innovative sample preparation and enrichment technique in connection with gas chromatography (GC). Using SPDE, we developed a method for simultaneous determination of n-heptane and its mono-oxygenated metabolites heptane-4-one, 3-one, 2-one, 4-ol, 3-ol, 2-ol, and 1-ol in blood. After adjustment of various extraction and desorption parameters, method validation resulted in limits of detection (LOD) between 0.006 (heptane-4-one) and 0.021 mg/L (heptane-1-ol). Intra-assay coefficients of variation ranged between 4.8% and 20.8% while relative recovery ranged between 100% and 117% (spiked concentration 0.128 mg/L, n  = 8). The method was appli…

AdultMaleAnalyteAnalytical chemistryToxicologySensitivity and SpecificityGas Chromatography-Mass SpectrometryHeptaneschemistry.chemical_compoundYoung AdultBiomonitoringHumansSample preparationDetection limitHeptaneInhalation ExposureChromatographyDose-Response Relationship DrugMolecular StructureChemistryExtraction (chemistry)Reproducibility of ResultsGeneral MedicineEnvironmental ExposureGas chromatographyGas chromatography–mass spectrometryBiomarkersEnvironmental MonitoringToxicology letters
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The Use of Hall's Technique Preformed Metal Crown (HTPMC) by Pediatric Dentists in Malaysia

2021

Introduction. Hall’s technique preformed metal crown (HTPMC) has been used widely by pediatric dentists in developed countries as a new approach for managing decayed primary molars without local anesthesia, caries removal, and tooth preparation. Currently, inadequate information is available regarding the implementation of this technique (HTPMC) in Malaysia. This study is aimed at evaluating the implementation of HTPMC by Malaysia’s pediatric dentists and identify the co-occurrence frequencies of the HTPMC implementation with the respondents’ demographic profile. Materials and Methods. A cross-sectional questionnaire-based research was conducted among 65 pediatric dentists in Malaysia. Onli…

AdultMaleArticle SubjectDentistsDental CariesGeneral Biochemistry Genetics and Molecular BiologySettore MED/28 - Malattie OdontostomatologicheSurveys and QuestionnairesHumansTooth DeciduousDental Restoration PermanentPractice Patterns Dentists'preformed metal crownGeneral Immunology and MicrobiologyCrownsRMalaysiaGeneral MedicineMiddle AgedMolarCross-Sectional StudiesMedicineFemaleDental Cavity PreparationHall’s TechniqueResearch ArticleBioMed Research International
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Analyzing the teeth next to the alveolar cleft: Examination and treatment proposal prior to bone grafting based on three-dimensional versus two-dimen…

2016

Abstract Purpose The objective was to evaluate the diagnostic and prognostic value of three-dimensional (3D) cone beam computed tomography (CBCT) on information about the cleft and alignment of cleft neighboring teeth. Materials and methods Panoramic X-rays, small-volume CBCTs, and study casts of 20 patients with a total of 22 alveolar clefts were analyzed prior to secondary bone grafting. Six maxillofacial surgeons and 6 orthodontists rated the following parameters: visibility of alveolar cleft expansion, position and probability of alignment of cleft neighbored teeth. Two-dimensional (2D) X-rays and casts were rated first; CBCT and casts followed at least 4 weeks later. Radiologic bone he…

AdultMaleCone beam computed tomographyDental radiographyAdolescentmedicine.medical_treatmentTreatment outcomeDentistryBone graftingCohort StudiesYoung Adult03 medical and health sciencesImaging Three-Dimensional0302 clinical medicinePreoperative CareRadiography PanoramicHumansMedicineSurgical preparationBone heightChild030223 otorhinolaryngologyRetrospective StudiesOrthodonticsMaxillofacial surgeonsmedicine.diagnostic_testAlveolar Bone Graftingbusiness.industry030206 dentistryCone-Beam Computed TomographyCleft PalateOtorhinolaryngologyFemaleSurgeryOral SurgeryAlveolar bone graftingbusinessToothJournal of Cranio-Maxillofacial Surgery
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Fixed dental prostheses with vertical tooth preparations without finish lines: A report of two patients

2016

Tooth abutments can be prepared to receive fixed dental prostheses with different types of finish lines. The literature reports different complications arising from tooth preparation techniques, including gingival recession. Vertical preparation without a finish line is a technique whereby the abutments are prepared by introducing a diamond rotary instrument into the sulcus to eliminate the cementoenamel junction and to create a new prosthetic cementoenamel junction determined by the prosthetic margin. This article describes 2 patients whose dental abutments were prepared to receive ceramic restorations using vertical preparation without a finish line.

AdultMaleEngineeringDentistryDental Abutments02 engineering and technology03 medical and health sciences0302 clinical medicinestomatognathic systemDental AbutmentsmedicineHumansGingival recessionCrownsbusiness.industryA diamond030206 dentistryFinish lineMiddle Aged021001 nanoscience & nanotechnologyIncisorstomatognathic diseasesCementoenamel junctionDental Prosthesis DesignFemaleDental Prosthesis Implant-SupportedTooth PreparationsOral Surgerymedicine.symptom0210 nano-technologybusinessThe Journal of Prosthetic Dentistry
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Exposure to toxic agents alters organic elemental composition in human fingernails.

2008

Abstract Background and objective: The human fingernail plate is highly keratinized. The keratin structure is held together by disulfide bonds. The organic elements sulfur and nitrogen occur almost exclusively in amino acids of the nail plate. This study analyzed whether occupational exposure to harmful chemical agents alters the organic elemental composition in fingernails. Subjects and methods: Participants were 71 occupationally exposed workers (49 hairdressers, 22 painters) and 49 unexposed controls. Aspects of exposure were assessed by questionnaire. Nail clippings of index and little fingers were analyzed for sulfur (S), nitrogen (N), carbon (C), and hydrogen (H) contents, using an au…

AdultMaleEnvironmental EngineeringChemical compoundStereochemistryNitrogenHair Preparationschemistry.chemical_elementchemistry.chemical_compoundSex FactorsOccupational ExposurePaintmedicineEnvironmental ChemistryHumansWaste Management and DisposalDiminutionElemental compositionintegumentary systemChemistryNail plateMiddle AgedPollutionNitrogenSulfurCarbonmedicine.anatomical_structureNailsEnvironmental chemistryNail (anatomy)FemaleOccupational exposureSulfurHydrogenThe Science of the total environment
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Urinary levels of enniatin B and its phase I metabolites: First human pilot biomonitoring study

2018

Abstract Enniatins (Enns) are mycotoxins produced by Fusarium spp. and are widely distributed contaminants of cereals and derivate products. Among the different identified enniatins, Enn B is the most relevant analogue in cereals in Europe. Therefore, the aim of this study was to investigate for the first time the occurrence of Enn B and Enn B phase I metabolites in 300 human urine samples throughout an ultrahigh-performance liquid chromatography-high resolution mass spectrometry (UHPLC-Q-Orbitrap HRMS) methodology. Three different sample preparation procedures were evaluated and salting-out liquid-liquid extraction showed satisfactory validation results. Enn B was quantified in 83.7% of sa…

AdultMaleFusariumEnniatin B Metabolites Urine Human Biomonitoring OrbitrapPilot ProjectsUrineToxicologyOrbitrap01 natural sciencesMass Spectrometrylaw.inventionchemistry.chemical_compound0404 agricultural biotechnologyUrinary levelslawDepsipeptidesBiomonitoringHumansSample preparationMycotoxinChromatography High Pressure LiquidEnniatin BChromatographybiology010401 analytical chemistryReproducibility of Results04 agricultural and veterinary sciencesGeneral MedicineMiddle Agedbiology.organism_classification040401 food science0104 chemical sciencesItalychemistryMicrosomes LiverFemaleEnvironmental MonitoringFood Science
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In vivo evaluation of periodontal microcirculatory changes associated with endodontic treatment.

2014

The purpose of this study was to investigate in vivo the gingival microcirculatory changes associated with endodontic treatment using the continuous wave of condensation technique. MATERIALS AND METHODS: Twenty necrotic one canal roots of 20 cooperative patients of both sexes, aged between 20 and 43 years, were selected. All patients were examined by capillaroscopy before, immediately after endodontic treatment, and after 7 days. The last examination was carried out by the same operator, and repeated twice for each examined area: masticatory, buccal and labial mucosa corresponding to the endodontically treated root. All canals were prepared using a simultaneous technique with Ni-Ti files (M…

AdultMaleHot TemperatureGingivaVideo RecordingHemorrhageCAPILLAROSCOPYBody TemperatureMicroscopic AngioscopyYoung AdultSettore MED/28 - Malattie OdontostomatologicheNickelRoot Canal ObturationDental Pulp NecrosisHumansPERIODONTAL MICROCIRCULATIONCAPILLAROSCOPY; ENDODONTIC TREATMENT; PERIODONTAL MICROCIRCULATIONTitaniumWound HealingMouth MucosaCapillariesRoot Canal TherapyENDODONTIC TREATMENTFemaleRoot Canal PreparationDental AlloysFollow-Up StudiesEuropean journal of paediatric dentistry
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Safety and tolerability of slow-release oral morphine versus methadone in the treatment of opioid dependence

2014

Opioid substitution treatment (OST) for opioid dependence may be limited by adverse events (AEs). Increasing the range of therapeutic options optimizes outcomes and facilitates patient management. An international, multi-center, two-phase study investigated the efficacy and safety of slow-release oral morphine (SROM) versus methadone in patients receiving methadone therapy for opioid dependence. In phase 1 (two way cross-over, 11 weeks each period) patients were randomized to SROM or methadone oral solution. In phase 2 (25 weeks), patients continued treatment with SROM (group A) or switched from methadone to SROM (group B). In total, 211 out of 276 completed phase 1 and 198 entered phase 2 …

AdultMaleInternational CooperationAdministration OralMedicine (miscellaneous)QT intervalHeroinOpiate Substitution TreatmentHumansMedicineIn patientOral morphineAdverse effectCross-Over StudiesMorphinebusiness.industryOpioid-Related DisordersEuropePsychiatry and Mental healthClinical PsychologyTreatment OutcomeOpioidTolerabilityDelayed-Action PreparationsAnesthesiaFemalePshychiatric Mental HealthbusinessMethadonemedicine.drugMethadoneJournal of Substance Abuse Treatment
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