Search results for "PRODUCTS"

showing 10 items of 980 documents

Bioactive polyketides and alkaloids from Penicillium citrinum , a fungal endophyte isolated from Ocimum tenuiflorum

2013

Chemical investigation of the endophytic fungus Penicillium citrinum cultured on white beans or on rice led to the isolation of two new alkaloids (1 and 2), along with fourteen known polyketides (6-12, 14-20) and four known alkaloids (3-5, and 13). The structures of the isolated compounds were determined by extensive analysis of the 1D, 2D NMR, and MS data, and by comparison with the literature. Compound 13, which had been previously obtained only by chemical synthesis, was isolated as a natural product for the first time, while compound 6 was firstly reported as a fungal metabolite. A re-isolation of sclerotinin A (14) revealed it to be a diastereoisomeric mixture (14a and 14b), whose ster…

Staphylococcus aureusLymphomaStereochemistryAntineoplastic Agentsmedicine.disease_causeChemical synthesisEndophyteInhibitory Concentration 50Micechemistry.chemical_compoundAlkaloidsCell Line TumorDrug DiscoveryEndophytesmedicineAnimalsPenicillium citrinumCytotoxicityPharmacologyBiological ProductsNatural productMolecular StructurebiologyPenicilliumGeneral Medicinebiology.organism_classificationOcimumAnti-Bacterial AgentsOcimumchemistryStaphylococcus aureusPolyketidesAntibacterial activityFitoterapia
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Genericity of dimension drop on self-affine sets

2017

We prove that generically, for a self-affine set in $\mathbb{R}^d$, removing one of the affine maps which defines the set results in a strict reduction of the Hausdorff dimension. This gives a partial positive answer to a folklore open question.

Statistics and ProbabilityPure mathematicsthermodynamic formalismDynamical Systems (math.DS)01 natural sciencesself-affine setsingular value functionAffine combinationAffine hullClassical Analysis and ODEs (math.CA)FOS: MathematicsMathematics - Dynamical Systems0101 mathematicsMathematicsDiscrete mathematicsta111010102 general mathematicsMinkowski–Bouligand dimensionproducts of matricesEffective dimension010101 applied mathematicsAffine coordinate systemMathematics - Classical Analysis and ODEsHausdorff dimensionAffine transformationStatistics Probability and UncertaintyStatistics & Probability Letters
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Acylated oleanane-type saponins from Ganophyllum giganteum

2014

Abstract Five oleanane-type saponins , 3- O -β- D -glucuronopyranosylzanhic acid 28- O -β- D -xylopyranosyl-(1→3)-[α- L -rhamnopyranosyl-(1→2)]-(4- O -acetyl)-β- D -fucopyranosyl ester ( 1 ), 3- O -β- D -glucopyranosylzanhic acid 28- O -β- D -xylopyranosyl-(1→3)-[α- L -rhamnopyranosyl-(1→2)]-(4- O -acetyl)-β- D -fucopyranosyl ester ( 2 ), zanhic acid 28- O -β- D -xylopyranosyl-(1→3)-[α- L -rhamnopyranosyl-(1→2)]-(4- O -acetyl)-β- D -fucopyranosyl ester ( 3 ), zanhic acid 28- O -α- L -rhamnopyranosyl-(1→2)-4- O -[(3′-hydroxy-2′-methyl-butyroyloxy)-3-hydroxy-2-methyl-butyroyloxy]-β- D -fucopyranosyl ester ( 4 ), medicagenic acid 28- O -α- L -rhamnopyranosyl-(1→2)-4- O -[(3′-hydroxy-2′-methyl-…

StereochemistryAcylationMolecular ConformationPlant ScienceHorticulturePlant RootsBiochemistryMiceStructure-Activity Relationshipchemistry.chemical_compoundSapindaceaeCell Line TumorAnimalsHumansOrganic chemistryMoietyOleanolic AcidMolecular BiologyOleananeCell ProliferationInflammationBiological ProductsDose-Response Relationship DrugChemistryHydrolysisAnti-Inflammatory Agents Non-SteroidalGeneral MedicineSaponinsAntineoplastic Agents PhytogenicMedicagenic acidDoratoxyleaeDrug Screening Assays AntitumorPhytochemistry
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Beyond Pseudo‐natural Products: Sequential Ugi/Pictet‐Spengler Reactions Leading to Steroidal Pyrazinoisoquinolines That Trigger Caspase‐Independent …

2021

In this work, we describe how stereochemically complex polycyclic compounds can be generated by applying a synthetic sequence comprising an intramolecular Ugi reaction followed by a Pictet-Spengler cyclization on steroid-derived scaffolds. The resulting compounds, which combine a fragment derived from a natural product and a scaffold not found in nature. are both structurally distinct and globally similar to natural products at the same time, and interrogate an alternative region of the chemical space. One of the new compounds showed significant antiproliferative activity on HepG2 cells through a caspase-independent cell-death mechanism, an appealing feature when new antitumor compounds are…

StereochemistryAntineoplastic AgentsSequence (biology)01 natural sciencesBiochemistryPiperazineschemistry.chemical_compoundDrug DiscoveryHumansGeneral Pharmacology Toxicology and PharmaceuticsCell ProliferationPharmacologyBiological ProductsNatural productPictet–Spengler reactionCell DeathMolecular Structure010405 organic chemistryOrganic ChemistryCaspase independentStereoisomerismHep G2 CellsIsoquinolinesChemical space0104 chemical sciences010404 medicinal & biomolecular chemistrychemistryCaspasesIntramolecular forceHepg2 cellsMolecular MedicineUgi reactionSteroidsDrug Screening Assays AntitumorChemMedChem
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Cytotoxic activity of some natural and syntetic sesquiterpene lactones

2006

Several natural and synthetic sesquiterpene lactones with different skeletons were tested and found to be active against nine cancer cell lines. Elemane (4), heliangolane (5) and their hydroxy analogues 9 and 10, all containing an α,β-unsaturated aldehyde substituent, were the most potent compounds.

StereochemistrySubstituentPharmaceutical ScienceCentaureaPharmacognosySesquiterpeneAldehydeANTITUMOR AGENTSAnalytical Chemistrychemistry.chemical_compoundInhibitory Concentration 50LactonesStructure-Activity RelationshipCell Line TumorDrug DiscoveryStructure–activity relationshipOrganic chemistryCytotoxic T cellHumansCENTAUREA-PAUICytotoxicityPharmacologychemistry.chemical_classificationBiological ProductsMolecular StructureDERIVATIVESOrganic ChemistryCNICINSettore CHIM/06 - Chimica OrganicaAntineoplastic Agents PhytogenicComplementary and alternative medicinechemistryMolecular MedicineSesquiterpenesLactone
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Explaining the relationship between socially responsible products and the operations of the firm: The case of equine assisted therapy

2018

Abstract Although there is a growing interest in social responsibility in research as well as in practice, the majority of studies on corporate social responsibility do not explicitly investigate operations management issues when adopting socially responsible practices under the “people” pillar of sustainability. This paper, dealing with the theme of social responsibility in operations management, aims at clarifying the complex relationship between socially responsible product/service and the operations of the company. The empirical context of the study is the sport industry, where the attention to social issues is well established. We used a mixed theoretical-empirical approach to develop …

Strategy and ManagementContext (language use)Social issuesIndustrial and Manufacturing EngineeringProduct innovation0502 economics and businessOperations management in sportProduct (category theory)Operational performanceMarketing0505 lawGeneral Environmental ScienceService (business)2300Renewable Energy Sustainability and the Environment05 social sciencesSettore ING-IND/35 - Ingegneria Economico-GestionaleVirtuous circle and vicious circleEquine assisted therapyStrategy and Management1409 Tourism Leisure and Hospitality Management050501 criminologyCorporate social responsibilityPortfolioBusinessSocially responsible products/serviceSocial responsibility050203 business & management
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Use of gases to improve survival of Bifidobacterium bifidum by modifying redox potential in fermented milk

2011

The aim of this work was to study the effect of the oxidoreduction potential, modified using gas, on the growth and survival of a probiotic strain, Bifidobacterium bifidum, and 2 yogurt strains, Streptococcus thermophilus and Lactobacillus delbrueckii ssp. bulgaricus. Three fermented milks were manufactured with an initial oxidoreduction potential value adjusted to +440 mV (control milk), +350 mV (milk gassed with N(2)), and -300 mV [milk gassed with N(2) plus 4% (vol/vol) H(2) (N(2)-H(2))]. Acidification profiles, growth during milk fermentation and survival during storage at 4 °C for 28 d were determined. This study showed that fermented probiotic dairy products made from milk gassed with…

Streptococcus thermophilusCultured Milk ProductsFood HandlingNitrogenved/biology.organism_classification_rank.specieslaw.inventionProbioticfluids and secretionslawFood PreservationLactobacillusGeneticsAnimalsStreptococcus thermophilusFood microbiologyFood scienceLactobacillus delbrueckiiBifidobacterium bifidumbiologyved/biologyFood preservationfood and beveragesActinomycetaceaeHydrogen-Ion Concentrationbiology.organism_classificationFermentationFood MicrobiologyAnimal Science and ZoologyFermentationBifidobacteriumOxidation-ReductionHydrogenFood ScienceJournal of Dairy Science
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Is the Eco-label EU Decision for hard coverings really capable of capturing the environmental performances of the marble productive chain? A field ve…

2014

Purpose This work intends to show whether the Eco-label EU Decision for hard coverings, in which marble is contemplated among hard coverings as a natural product, is really capable of capturing the environmental performances of the marble productive chain, in other words whether it is actually viable for the natural products, like marble. Methods After a preliminary critical analysis of the suitability formarble of the current EU Decision (2009/607/EC), a classical life cycle assessment (LCA) methodology has been applied on the field to the marble “Perlato di Sicilia.” More specifically, the whole productive chain of a couple of firms treating the “Perlato di Sicilia” marble has been examin…

Structure (mathematical logic)EngineeringEU Eco-label DecisionNatural productsSettore ING-IND/11 - Fisica Tecnica AmbientaleNatural stonebusiness.industryLCAEnvironmental economicsCivil engineeringChain (unit)Field (computer science)Set (abstract data type)Hard coveringWork (electrical)Order (exchange)Marble productive chainbusinessLife-cycle assessmentGeneral Environmental Science
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Trihalomethanes in swimming pool water in four areas of Spain participating in the INMA project

2010

ResumenObjetivoLa natación es uno de los deportes más practicados en España, por personas de todas las edades y condiciones físicas. También es una vía de exposición a subproductos de la desinfección, compuestos potencialmente tóxicos. Su concentración en el agua de las piscinas no está legislada y es poco conocida. El objetivo de este trabajo es describir la concentración de trihalometanos en el agua de piscinas de los municipios de cuatro cohortes del estudio INMA.MétodosEn julio de 2009 se analizaron los trihalometanos en el agua de piscinas (n=27) de Asturias, Granada, Valencia y Sabadell.ResultadosLa concentración media de trihalometanos totales fue de 42,7μg/l (desviación estándar [DE…

Subproductos de la desinfecciónPublic Health Environmental and Occupational HealthWaterAguaSwimming pool waterExposureSwimming poolTrihalomethanechemistry.chemical_compoundDisinfection by-productschemistryTrihalometanosExposiciónEnvironmental healthEnvironmental sciencehuman activitiesPiscinaTrihalomethanesGaceta Sanitaria
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Acid- and Base-Catalysis in the Mononuclear Rearrangement of Some (Z)-arylhydrazones of 5-Amino-3-benzoyl-1,2,4-oxadiazole in Toluene: Effect of Subs…

2011

The reaction rates for the rearrangement of eleven (Z)-arylhydrazones of 5-amino-3-benzoyl-1,2,4-oxadiazole 3a-k into the relevant (2-aryl-5-phenyl-2H-1, 2,3-triazol-4-yl)ureas 4a-k in the presence of trichloroacetic acid or of piperidine have been determined in toluene at 313.1 K. The results have been related to the effect of the aryl substituent by using Hammett and/or Ingold-Yukawa-Tsuno correlations and have been compared with those previously collected in a protic polar solvent (dioxane/water) as well as with those on the analogous rearrangement of the corresponding (Z)-arylhydrazones of 3-benzoyl-5-phenyl-1,2,4-oxadiazole 1a-k in benzene. Some light can thus be shed on the general di…

SubstituentOxadiazoleAlkaliesMedicinal chemistryCatalysisDioxanesStructure-Activity RelationshipAcid catalysischemistry.chemical_compoundPiperidinesUreaOrganic chemistryAminesTrichloroacetic AcidBenzeneBiological ProductsOxadiazolesMolecular StructureArylMRH acid- and base-catalysis kinetic measurementsOrganic ChemistryHydrazonesTemperatureWaterSettore CHIM/06 - Chimica OrganicaTolueneSolventKineticschemistryMononuclear rearrangements of heterocycles; (Z)-Arylhydrazones; acid catalysis; base catalysis.PiperidineHydrophobic and Hydrophilic InteractionsToluene
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