Search results for "Pyridine"

showing 10 items of 2516 documents

Antihyperalgesic and analgesic properties of the N-methyl-d-aspartate (NMDA) receptor antagonist neramexane in a human surrogate model of neurogenic …

2006

Abstract NMDA-receptors are a major target in the prevention and treatment of hyperalgesic pain states in neuropathic pain. However, previous studies revealed equivocal results depending on study design and efficacy parameters. We tested the analgesic (generalized reduction of generation and processing of nociceptive signalling) and anti-hyperalgesic (prevention of central sensitization) properties of the NMDA-receptor antagonist neramexane and the potassium channel opener flupirtine in the intradermal capsaicin injection model. Furthermore, we tested the effect on pain summation (wind up). Eighteen healthy subjects received either a single dose of neramexane (40 mg p.o.), flupirtine (100 m…

Injections IntradermalAnalgesicAminopyridinesPainCyclopentanesPharmacologyPlaceboReceptors N-Methyl-D-AspartateDouble-Blind MethodPhysical StimulationHumansMedicineAnalgesicsCross-Over StudiesDose-Response Relationship Drugbusiness.industryNeramexaneTreatment OutcomeAnesthesiology and Pain MedicineAllodyniaNociceptionHyperalgesiaAnesthesiaNeuropathic painHyperalgesiaCapsaicinNervous System Diseasesmedicine.symptomFlupirtinebusinessmedicine.drugEuropean Journal of Pain
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Tuning the spin crossover above room temperature: iron(II) complexes of substituted and deprotonated 2,6-bis(benzimidazol-2-yl)pyridine

2005

Abstract The complex [Fe(tzimpy)2](ClO4)2 · 2H2O (tzimpy = 2,4,6-tris-(benzimidazol-2-yl)pyridine) shows an abrupt spin crossover (S = 0–2 transition) above room temperature centered at Tc = 323 K with a hysteresis width of ΔT = 35 K. The neutral iron(II) complex with deprotonated bzimpy ligands (bzimpy = 2,6-bis(benzimidazol-2-yl)pyridine) exhibits a gradual spin transition on the first heating with Tc = 424 K. There are irreversible changes between T = 503 and 523 K: the liberation of the crystal water, the color change (blue–green) followed by a structure change. Next thermal cycles are reproducible though, heating/cooling paths are different from the first heating.

Inorganic ChemistryCrystalCrystallographyHysteresischemistry.chemical_compoundDeprotonationNuclear magnetic resonancechemistrySpin crossoverPyridineMaterials ChemistrySpin transitionPhysical and Theoretical ChemistryInorganic Chemistry Communications
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Magneto-structural studies on heterobimetallic malonate-bridged M(II)Re(IV) complexes (M = Mn, Co, Ni and Cu).

2010

The mononuclear Re(IV) compound of formula (PPh(4))(2)[ReBr(4)(mal)] (1) was used as a ligand to obtain the heterobimetallic species [ReBr(4)(μ-mal)Co(dmphen)(2)]· MeCN (2), [ReBr(4)(μ-mal)Ni(dmphen)(2)] (3), [ReBr(4)(μ-mal)Mn(dmphen)(2)] (4a), [ReBr(4)(μ-mal)Mn(dmphen)(H(2)O)(2)]·dmphen·MeCN·H(2)O (4b), [ReBr(4)(μ-mal)Cu(phen)(2)]·1/4H(2)O (5) and [ReBr(4)(μ-mal)Cu(bipy)(2)] (6) (mal = malonate dianion, dmphen = 2,9-dimethyl-1,10-phenanthroline, phen = 1,10-phenanthroline and bipy = 2,2'-bipyridine). The structures of 2 and 5 (single-crystal X-ray diffraction) are made up of neutral [ReBr(4)(μ-mal)M(AA)] dinuclear units [AA = dmphen with M = Co (2) and AA = phen with M = Cu (5)] where the …

Inorganic ChemistryCrystallographyBipyridinechemistry.chemical_compoundDenticityMalonateChemistryFerrimagnetismLigandIntramolecular forceMetal ions in aqueous solutionAntiferromagnetismDalton transactions (Cambridge, England : 2003)
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Increasing the Ordering Temperatures in Oxalate-Based 3D Chiral Magnets:  the Series [Ir(ppy)2(bpy)][MIIMIII(ox)3]·0.5H2O (MIIMIII = MnCr, FeCr, CoCr…

2006

The synthesis, structure, and physical properties of a novel series of oxalate-based bimetallic magnets obtained by using the Ir(ppy)2(bpy)]+ cation as a template of the bimetallic [MIIMIII(ox)3]- ...

Inorganic ChemistryCrystallographychemistry.chemical_compoundchemistryMagnetInorganic chemistry2-PhenylpyridinePhysical and Theoretical ChemistryNichromeBimetallic stripOxalate22'-BipyridineInorganic Chemistry
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Stability and kinetics of the acid-promoted decomposition of Cu(II) complexes with hexaazacyclophanes: kinetic studies as a probe to detect changes i…

2004

The synthesis, protonation and Cu(II) coordination features of the novel azacyclophane type receptors 2,6,10,13,17,21-hexaza[22]-(2,6)-pyridinophane (L2), 2,6,9,12,15,19-hexaza[20]-(2,6)-pyridinophane (L5) and 2,6,9,12,15,19-hexaza[20]metacyclophane (L6) are presented. The protonation and Cu(II) constants are analysed and compared with the previously reported open-chain polyamines 4,8,11,15-tetrazaoctadecane-1,18-diamine (L1) and 4,7,10,13-tetraazahexadecane-1,16-diamine (L4) and of the cyclophane 2,6,10,13,17,21-hexaaza[22]paracyclophane (L3). All the systems form mono- and dinuclear complexes whose stability and pH range of existence depend on the type of hydrocarbon chains and molecular …

Inorganic ChemistryCrystallographychemistry.chemical_compoundchemistryStereochemistryLigandMetal ions in aqueous solutionKineticsPyridineProtonationDecompositionCyclophaneIonDalton transactions (Cambridge, England : 2003)
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The [1,2,3]triazolo[1,5-a]pyridine ring: a sensitive sensor for the electronic profile of phosphorus substituents.

2009

The unique nature of the [1,2,3]triazolo[1,5-a]pyridine reveals without any external perturbation the electronic contribution of various substituents to the phosphorus atom in phosphines, based on the equilibrium of two possible ring-chain isomers.

Inorganic ChemistryCrystallographychemistry.chemical_compoundchemistryStereochemistryPhosphorus atomPyridineDalton transactions (Cambridge, England : 2003)
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A Bis(tridentate)cobalt Polypyridine Complex as Mediator in Dye‐Sensitized Solar Cells

2015

Dye-sensitized solar cells equipped with cationic and neutral RuII-based sensitizers [Ru(ddpd){tpy(COOH)3}]2+ [12+; ddpd = N,N′-dimethyl-N,N′-di(pyridin-2-yl)pyridin-2,6-diamine, tpy(COOH)3 = 2,2″6′,2″-terpyridine-4,4′,4″-tricarboxylic acid] and [Ru(ddpd){tpy(COOH)(COO)2}] (2) with and without the coadsorbent chenodeoxycholic acid were constructed with I3–/I– or the CoIII/II-based redox mediators [Co(bpy)3]3+/2+ (33+/2+; bpy = 2,2′-bipyridine) and [Co(ddpd)2]3+/2+ (43+/2+) in the presence of LiClO4 and 4-tert-butylpyridine. The best photovoltaic performance was achieved by using the 43+/2+ shuttle and the neutral sensitizer 2 without coadsorbent. The higher short-circuit photocurrent densit…

Inorganic ChemistryElectron transferDye-sensitized solar cellCrystallographyPolypyridine complexChemistryKineticsCationic polymerizationchemistry.chemical_elementPhotochemistryRedoxCobaltRutheniumEuropean Journal of Inorganic Chemistry
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Enhancing Performance of a Bis(arylimino)pyridine‐Iron Precatalyst for Ethylene Polymerization by Substitution with a 2,4‐Bis(4,4′‐dimethoxybenzhydry…

2021

A series of unsymmetrical 2-(2,4-bis(bis(4-methoxyphenyl)methyl)-6-MeC6H2N)-6-(1-(arylimino)ethyl)pyridine-iron halides has been synthesized and characterized. The molecular structure of two representative species was determined by the single-crystal X-ray diffraction. Activated with either MAO or MMAO, the precatalysts displayed high activity, reaching 2.19×107 g PE (mol Fe)−1 h−1 at 60 °C in ethylene polymerization. The microstructural analysis of the polymers obtained indicates highly linear polyethylene containing a vinyl chain end.

Inorganic ChemistryEthylene polymerizationchemistry.chemical_compoundPrecatalystsEthylene polymerizationChemistryGroup (periodic table)Substitution (logic)PyridineVinyl polyethyleneHigh activityIron(II)Medicinal chemistryEuropean Journal of Inorganic Chemistry
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In situ generation of Ph3PO in cyanido-bridged heterometallic {FeIIILnIII}2 molecular squares (Ln = Eu, Sm)

2019

Two new examples of cyanido-bridged {FeIIILnIII}2 molecular squares, with pyim and PPh3O as capping ligands at the LnIII sites, exhibit weak antiferromagnetic interactions [Ln = Eu (1), Sm (2), pyim = 2-(1H-imidazol-2-yl)pyridine, PPh3PO = triphenylphosphine oxide].

Inorganic ChemistryIn situCrystallographychemistry.chemical_compound010405 organic chemistryChemistryPyridineAntiferromagnetism010402 general chemistry01 natural sciencesTriphenylphosphine oxide0104 chemical sciencesDalton Transactions
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Further synthetic investigation of the general lanthanoid(iii) [Ln(iii)]/copper(ii)/pyridine-2,6-dimethanol/carboxylate reaction system: {CuII5LnIII4…

2021

In addition to previously studied {CuII3Gd6}, {CuII8Gd4}, {CuII15Ln7} and {CuII4Ln8} coordination clusters (Ln = trivalent lanthanide) containing pdm2− or Hpdm− ligands (H2pdm = pyridine-2,6-dimethanol) and ancillary carboxylate groups (RCO2−), the present work reports the synthesis and study of three new members of a fifth family of such complexes. Compounds [Cu5Ln4O2(OMe)4(NO3)4(O2CCH2But)2(pdm)4(MeOH)2] (Ln = Dy, 1; Ln = Tb, 2; Ln = Ho, 3) were prepared from the reaction of Ln(NO3)3·xH2O (x = 5, 6), CuX2·yH2O (X = ClO4, Cl, NO3; y = 6, 2 and 3, respectively), H2pdm, ButCH2CO2H and Et3N (2 : 2.5 : 2 : 1 : 9) in MeCN/MeOH. Rather surprisingly, the copper(II)/yttrium(III) analogue has a sli…

Inorganic ChemistryLanthanideCrystallographyTrigonal bipyramidal molecular geometrychemistry.chemical_compoundchemistryPyridinechemistry.chemical_elementMoleculeAntiferromagnetismYttriumCarboxylateMagnetic susceptibilityDalton Transactions
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