Search results for "SULFUR"

showing 10 items of 545 documents

Non-Classical Transformation of Benzendiazonium Hydrogen Sulfates. Access to 1,3-Dimethylisochromeno[4,3-c]pyrazol-5(1H)-one, a Potential Benzodiazep…

2013

The compound 2-((1,3-dimethyl-1H-pyrazol-5-yl)(methyl)carbamoyl)benzene-diazonium hydrogen sulfate (10) was reacted with copper sulfate and sodium chloride, in the presence of ascorbic acid as reducing agent, to afford a mixture of the chlorinated epimers 4′-chloro-2,2′,5′-trimethyl-2′,4′-dihydrospiro[isoindoline-1,3′-pyrazol]-3-one (18) and (19), the epimers 4′-hydroxy-2,2′,5′-trimethyl-2′,4′-dihydrospiro[isoindoline-1,3′-pyrazol]-3-one (20) and (21), and N-(1,3-dimethyl-1H-pyrazol-5-yl)benzamide (22). Under the foregoing conditions, diazonium salt 10 affords neither the 2-chloro-N-(1,3-dimethyl-1H-pyrazol-5-yl)-N-methylbenzamide (23) nor the tricyclic derivative 24, the classical products…

Reducing agentGABA AgentsSodiumPharmaceutical Sciencechemistry.chemical_elementSalt (chemistry)Sulfuric Acid EstersLigandsMedicinal chemistryArticleSandmeyer reactionAnalytical Chemistrylcsh:QD241-441chemistry.chemical_compoundlcsh:Organic chemistryisochromeno[43-c]pyrazol-5(1H)-oneDrug DiscoverySandmeyer reactionOrganic chemistryPhysical and Theoretical ChemistryBenzamide15-hydrogen atom transferchemistry.chemical_classificationheterocyclesChemistryOrganic ChemistrySettore CHIM/06 - Chimica OrganicaDiazonium CompoundsAscorbic acidPschorr reactionReceptors GABA-ASettore CHIM/08 - Chimica FarmaceuticaIsocoumarinsChemistry (miscellaneous)Molecular MedicinePyrazolesEpimerCrystallizationisochromeno[43-<i>c</i>]pyrazol-5(1<i>H</i>)-oneDerivative (chemistry)heterocycles; Pschorr reaction; Sandmeyer reaction; 15-hydrogen atom transfer; isochromeno[43-c]pyrazol-5(1H)-oneheterocycleMolecules
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Respiratory epithelium exposed to sulfur dioxide--functional and ultrastructural alterations.

1995

The value of morphological investigations of airway mucosa should be compared to a functional method when estimating the toxicity of airborne pollutants. In 34 guinea pig tracheas, mucociliary activity was measured using a modified light beam reflex method before and following exposure to sulfur dioxide for 30 minutes in concentrations ranging between 7.5 and 37.5 mg/m3. Exposure to air served as a control. Simultaneously, specimens were taken for light and electron microscopy. Mucociliary activity decreased from 8.4 +/- 2.9 Hz (control exposure) to 4.0 +/- 2.9 Hz following exposure to 7.5 mg/m3, to 3.4 +/- 2.7 Hz at 15 mg/m3 sulfur dioxide, to 1.8 +/- 2.2 Hz at 22.5 mg/m3 sulfur dioxide, t…

Respiratory MucosaPathologymedicine.medical_specialtyGuinea PigsEpitheliumlaw.inventionGuinea pigchemistry.chemical_compoundlawEdemaMedicineAnimalsSulfur DioxideCiliaSulfur dioxideMucous MembraneDose-Response Relationship Drugbusiness.industryMolecular biologyTracheaMicroscopy ElectronOtorhinolaryngologychemistryMucociliary ClearanceToxicityUltrastructureRespiratory epitheliumElectron microscopemedicine.symptombusinessThe Laryngoscope
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Šķērssaistīta sulfurēta poli(ēter ēter ketona) membrānas un to īpašības

2018

Šķērssaistīta sulfurēta poli(ēter ēter ketona) membrānas un to īpašības. Sinitsa N., vadītājs asoc. prof., Dr. Chem. Vaivars G. Maģistra darbs, 43 lappuses, 28 attēli, 4 tabulas, 36 literatūras avoti, 2 pielikumi. Latviešu valodā. Maģistra darba ietvaros tika veikta poli(ēter ēter ketona) sulfurēšana ar hlorsulfonskābi un sērskābi un iegūto polimēru modificēšana, izmantojot dažādas šķērsaistīšanas metodes. No iegūtiem šķērssaistītiem polimēriem tika izgatavotas membrānas, kurām pētīja termiskās un mehāniskās īpašības, kā arī uzbriešanas pakāpi ūdens vidē un ūdens uzņemšanu. Membrānu morfoloģijas izvērtēšanu veica ar skenējošo elektronu mikroskopiju.

SULFURĒTS POLI(ĒTER ĒTER KETONS)SKENEJOŠĀ ELEKTRONU MIKROSKOPIJATERMOGRAVIMETRISKĀ ANALĪZEMEHĀNISKĀ IZTURĪBAŠĶĒRSSAISTĪŠANAĶīmija
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Transcriptomic and Proteomic Approach for Understanding the Molecular Basis of Adaptation of Saccharomyces cerevisiae to Wine Fermentation

2006

ABSTRACT Throughout alcoholic fermentation, Saccharomyces cerevisiae cells have to cope with several stress conditions that could affect their growth and viability. In addition, the metabolic activity of yeast cells during this process leads to the production of secondary compounds that contribute to the organoleptic properties of the resulting wine. Commercial strains have been selected during the last decades for inoculation into the must to carry out the alcoholic fermentation on the basis of physiological traits, but little is known about the molecular basis of the fermentative behavior of these strains. In this work, we present the first transcriptomic and proteomic comparison between …

Saccharomyces cerevisiae ProteinsProteomeTranscription GeneticSaccharomyces cerevisiaeSulfur metabolismWineSaccharomyces cerevisiaeEthanol fermentationBiologyApplied Microbiology and BiotechnologyGene Expression Regulation FungalHeat shock proteinFermentation in winemakingWineEcologyGene Expression ProfilingPhysiology and Biotechnologybiology.organism_classificationAdaptation PhysiologicalYeastBiochemistryFermentationFermentationHeat-Shock ResponseFood ScienceBiotechnologyApplied and Environmental Microbiology
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Urmylation and tRNA thiolation functions of ubiquitin-like Uba4·Urm1 systems are conserved from yeast to man

2015

AbstractThe ubiquitin-like protein Urm1 from budding yeast and its E1-like activator Uba4 have dual roles in protein urmylation and tRNA thiolation pathways. To study whether these are conserved among eukaryotes, we used gene shuffles to replace the yeast proteins by their human counterparts, hURM1 and hUBA4/MOCS3. As judged from biochemical and genetical assays, hURM1 and hUBA4 are functional in yeast, albeit at reduced efficiencies. They mediate urmylation of the peroxiredoxin Ahp1, a known urmylation target in yeast, and support tRNA thiolation. Similar to hUBA4, yeast Uba4 itself is modified by Urm1 and hURM1 suggesting target overlap between eukaryal urmylation pathways. In sum, our st…

Saccharomyces cerevisiae ProteinsUba4 (hUBA4/MOCS3)Saccharomyces cerevisiaeBiophysicstRNA thiolationSaccharomyces cerevisiaeBiochemistryUbiquitin-like urmylationRNA TransferUbiquitinStructural BiologyAnticodonGeneticsHumansUbiquitinsMolecular BiologyProtein urmylationGeneUrm1 (hURM1)Conserved SequenceSequence Homology Amino AcidbiologyActivator (genetics)TRNA thiolationCell Biologybiology.organism_classificationNucleotidyltransferasesYeastBiochemistrySulfurtransferasesbiology.proteinPeroxiredoxinHeLa CellsFEBS Letters
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Sulfur cycling and methanogenesis primarily drive microbial colonization of the highly sulfidic Urania deep hypersaline basin

2009

Urania basin in the deep Mediterranean Sea houses a lake that is &gt;100 m deep, devoid of oxygen, 6 times more saline than seawater, and has very high levels of methane and particularly sulfide (up to 16 mM), making it among the most sulfidic water bodies on Earth. Along the depth profile there are 2 chemoclines, a steep one with the overlying oxic seawater, and another between anoxic brines of different density, where gradients of salinity, electron donors and acceptors occur. To identify and differentiate the microbes and processes contributing to the turnover of organic matter and sulfide along the water column, these chemoclines were sampled at a high resolution. Bacterial cell numbers…

SalinitySulfideMethanogenesisMolecular Sequence Datageosphere-biosphere interactionchemistry.chemical_elementGEO/01 - PALEONTOLOGIA E PALEOECOLOGIA03 medical and health sciencesWater columnelement cyclingMediterranean SeaSeawater14. Life underwaterEcosystemComputingMilieux_MISCELLANEOUS030304 developmental biology2. Zero hungerchemistry.chemical_classification[SDU.OCEAN]Sciences of the Universe [physics]/Ocean AtmosphereManganese0303 health sciencesNitratesMultidisciplinaryBacteriabiology030306 microbiologyEcologyWaterdeep anoxic hypersaline lake15. Life on landbiology.organism_classificationArchaeaSulfurAnoxic waters6. Clean waterOxygenRedox gradientchemistryDeep anoxic hypersaline lake; Element cycling; Geosphere-biosphere interaction; Mediterranean Sea; Microbial diversityEnvironmental chemistrymicrobial diversityPhysical SciencesSeawaterdeep anoxic hypersaline lake element cycling geosphere–biosphere interaction Mediterranean Sea microbial diversitySulfurArchaea
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Chiral Inversion of 1-Hydroxyethylpyrene Enantiomers Mediated by Enantioselective Sulfotransferases

1998

The benzylic alcohol 1-hydroxyethylpyrene (1-HEP) is activated to a mutagen by sulfotransferases. The sulfuric acid ester formed is difficult to detect, as it is rapidly hydrolysed back to the alcohol. Incubation of the individual enantiomers of 1-HEP with human hydroxysteroid sulfotransferase (hHST) or estrogen sulfotransferase (hEST), expressed in bacteria, led to the formation of the other enantiomer. The rates of sulfation were determined from the initial rates of chiral inversion of the alcohol, knowing that hydrolysis follows an SN1 mechanism and therefore produces racemic alcohol. hEST showed high enantioselectivity for S-1-HEP, whereas hHST strongly preferred the R-enantiomer. The r…

Salmonella typhimuriumSulfotransferaseStereochemistryChemistryPhosphoadenosine PhosphosulfateBiophysicsEnantioselective synthesisStereoisomerismStereoisomerismAlcoholCell BiologySulfuric Acid EstersBiochemistrychemistry.chemical_compoundSulfationHumansEstrogen SulfotransferaseHydroxysteroidSulfotransferasesEnantiomerMolecular BiologyBenzyl AlcoholsBiochemical and Biophysical Research Communications
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Bioavailability and food production of organosulfur compounds from edible Allium species

2019

Abstract Allium members are known for their wide use in culinary dishes and the content of their bioactive compounds. In this aspect, edible Allium members, such as garlic (A. sativum), onion (A. cepa), leeks (A. porrum), chives (A. schoenoprasum), and shallots (A. ascalonicum), have been widely studied with respect to their functional properties in vivo. Their beneficial effects on humans are closely associated with bioavailability of organosulfur compounds (OSCs) in allyl and methyl forms. However, the OSCs are thermally unstable, so it is important to identify critical processing types/parameters that have destructive effects on bioavailability of the OSCs, and possibly to avoid them in …

SativumbiologyChemistrybusiness.industryFood processingAlliumFood sciencebiology.organism_classificationbusinessBeneficial effectsOrganosulfur compoundsBioavailability
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4-(3H)-quinazolinones N-3 substituted with a five membered heterocycle: A promising scaffold towards bioactive molecules

2020

Abstract The quinazolinone nucleus represents, among the class of fused heterocycles, a very important scaffold to obtain molecules with biological activities. A review of literature revealed how such kind of fused heterocycles, coming from natural or synthetic source, are associated with a wide range of biological activities. This review is mainly directed towards the 4-(3H)-quinazolinones N-3 substituted with a five membered heterocycle in which all the possible combinations of nitrogen, sulfur and oxygen atoms are present.

ScaffoldNitrogenBioactive moleculesAnti-Inflammatory AgentsAntitubercular Agentschemistry.chemical_elementAntineoplastic Agents01 natural sciencesAntioxidants03 medical and health scienceschemistry.chemical_compoundAnti-Infective AgentsDrug DiscoveryAnimalsHumansMoleculeBenzothiazolesQuinazolinoneQuinazolinones030304 developmental biologyPharmacology0303 health sciencesMolecular Structure010405 organic chemistryOrganic ChemistryN-3 substituted-4-(3H)-quinazolinones five membered heterocycle bioactive systemGeneral MedicineSettore CHIM/08 - Chimica FarmaceuticaSulfurCombinatorial chemistryBronchodilator Agents0104 chemical sciencesOxygenThiazolesOxygen atomchemistryAnticonvulsantsSulfurEuropean Journal of Medicinal Chemistry
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NanoSIMS: insights into the organization of the proteinaceous scaffold within Hexactinellid sponge spicules.

2010

The giant basal spicules (GBS) from Monorhaphis chuni (Porifera [sponges], Hexactinellida) represent the largest biosilica structures on Earth and can reach lengths of 300 cm (diameter of 1.1 cm). The amorphous silica of the inorganic matrix is formed enzymatically by silicatein. During this process, the enzyme remains trapped inside the lamellar-organized spicules. In order to localize the organic silicatein scaffold, the inside of a lamella has been analyzed by nano-secondary ion mass spectrometry (NanoSIMS). It is shown that the GBSs are composed of around 245 concentrically arranged individual siliceous lamellae. These surround an internal siliceous axial cylinder. The lamellae adjacent…

ScaffoldSpiculebiologyHexactinellidOrganic ChemistryMatrix (biology)biology.organism_classificationSilicon DioxideBiochemistryCarbonMass SpectrometryPoriferaCrystallographySponge spiculeLamella (surface anatomy)Chemical engineeringMolecular MedicineAnimalsInorganic matrixAmorphous silicaMolecular BiologySulfurChembiochem : a European journal of chemical biology
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