Search results for "Small Intestine"

showing 10 items of 94 documents

Glucagon-like peptide-2 modulates neurally evoked mucosal chloride secretion in guinea pig small intestine in vitro

2009

Glucagon-like peptide-2 (GLP-2) is an important neuroendocrine peptide in intestinal physiology. It influences digestion, absorption, epithelial growth, motility, and blood flow. We studied involvement of GLP-2 in intestinal mucosal secretory behavior. Submucosal-mucosal preparations from guinea pig ileum were mounted in Ussing chambers for measurement of short-circuit current ( Isc) as a surrogate for chloride secretion. GLP-2 action on neuronal release of acetylcholine was determined with ELISA. Enteric neuronal expression of the GLP-2 receptor (GLP-2R) was studied with immunohistochemical methods. Application of GLP-2 (0.1–100 nM) to the serosal or mucosal side of the preparations evoke…

MaleTime FactorsPhysiologyVasoactive intestinal peptideHormones and SignalingFluorescent Antibody TechniqueSettore BIO/09 - FisiologiaEnteric Nervous SystemMembrane PotentialsIntestinal mucosaGlucagon-Like Peptide 2Receptors GlucagonNeuropeptide YIntestinal MucosaNeurotransmitter Agentsdigestive oral and skin physiologyGastroenterologygastrointestinal hormoneGlucagon-like peptide-2ImmunohistochemistrySomatostatinmedicine.anatomical_structureenteric nervous system; gastrointestinal hormones; intestine; mucosal secretionGlucagon-Like Peptide-2 ReceptorSomatostatinhormones hormone substitutes and hormone antagonistsVasoactive Intestinal Peptideendocrine systemmedicine.medical_specialtyGuinea PigsMotilityEnzyme-Linked Immunosorbent AssayIleumIn Vitro TechniquesBiologyCholine O-AcetyltransferaseChloridesIleumPhysiology (medical)Internal medicinemedicineAnimalsintestineIntestinal SecretionsHepatologymucosal secretionAcetylcholineElectric StimulationSmall intestineEndocrinologyGlucagon-Like Peptide-2 Receptor
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Labetalol absorption kinetics: Rat small intestine and colon studies

2006

Labetalol is a widely used drug for the management of hypertension, which is preferably administered by the oral route despite its low bioavailability. The objective of this study is to ascertain the mechanisms underlying its absorption as an approach to help in predicting the influence of dosage changes, possible drug-drug and drug-fruit juice interactions. Perfusion experiments have been performed in rats in two sites of absorption: the intestine and the colon. The nonlinearity of the process has been established by means of the assay of a wide range of concentrations (2-2000 microM). Fitting of the concentration versus time data allows the estimation of passive diffusion constant in the …

MalebiologyColonChemistryPharmaceutical ScienceAbsorption (skin)PharmacologyIntestinal absorptionSmall intestineRatsBioavailabilitymedicine.anatomical_structureIntestinal AbsorptionPharmacokineticsIntestine Smallmedicinebiology.proteinAnimalsLabetalolEffluxRats WistarLabetalolmedicine.drugP-glycoproteinJournal of Pharmaceutical Sciences
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CD36 Displays Features of a Lipid-Sensor Involved in Chylomicron Processing in the Rodent Small Intestine

2010

International audience; The membrane glycoprotein CD36 binds nanomolar concentrations of long-chain fatty acids (LCFA) and is highly expressed on the luminal surface of enterocytes. CD36 deficiency reduces chylomicron production through unknown mechanisms.In this report, we provide novel insights into the potential underlying mechanisms. Our in vivo data demonstrated that CD36 gene deletion in mice did not affect LCFA uptake and their subsequent esterification into triglycerides by the intestinal mucosa at micellar LCFA concentrations prevailing in the intestine. In rodents, CD36 protein early disappeared from the luminal side of intestinal villi during the post-prandial period but only whe…

medicine.medical_specialtyRodent030309 nutrition & dietetics[SDV]Life Sciences [q-bio]CD36030209 endocrinology & metabolismGastroenterology03 medical and health sciences0302 clinical medicineInternal medicinebiology.animalparasitic diseasesInternal Medicinemedicine0303 health sciencesbiologyChemistryGeneral MedicineSmall intestineCell biologymedicine.anatomical_structurebiology.proteinlipids (amino acids peptides and proteins)Cardiology and Cardiovascular Medicine[SDV.AEN]Life Sciences [q-bio]/Food and NutritionChylomicronAtherosclerosis Supplements
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Cisplatin increases the release of 5-hydroxytryptamine (5-HT) from the isolated vascularly perfused small intestine of the guinea-pig: Involvement of…

1991

Isolated segments of the guinea-pig small intestine were vascularly perfused and the release of 5-hydroxytryptamine (5-HT) and 5-hydroxyindoleacetic acid (5-HIAA) into the portal venous effluent determined by high pressure liquid chromatography with electrochemical detection. Release of acetylcholine from isolated superfused intestinal segments was determined as outflow of [3H]radioactivity from preparations preincubated with [3H]choline. Cisplatin (3 microM) increased the outflow of 5-HT and 5-HIAA by about 90%. At 30 and 100 microM cisplatin decreased the outflow of 5-HT and its metabolite by 40%-50%. The stimulatory effect of cisplatin was consistently observed only when the bicarbonate-…

MaleSerotoninmedicine.medical_specialtymedicine.drug_classMetaboliteGuinea PigsTetrodotoxinIn Vitro Techniqueschemistry.chemical_compoundInternal medicineIntestine SmallEnterochromaffin CellsmedicineAnimalsReceptor5-HT receptorPharmacologyCisplatinDose-Response Relationship DrugImidazolesGeneral MedicineHydroxyindoleacetic AcidReceptor antagonistOndansetronAcetylcholineSmall intestinePerfusionEndocrinologymedicine.anatomical_structurechemistryReceptors SerotoninFemaleHexamethoniumCisplatinAcetylcholinemedicine.drugNaunyn-Schmiedeberg's Archives of Pharmacology
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Microbiota Depletion Promotes Human Rotavirus Replication in an Adult Mouse Model

2021

Intestinal microbiota-virus-host interaction has emerged as a key factor in mediating enteric virus pathogenicity. With the aim of analyzing whether human gut bacteria improve the inefficient replication of human rotavirus in mice, we performed fecal microbiota transplant (FMT) with healthy infants as donors in antibiotic-treated mice. We showed that a simple antibiotic treatment, irrespective of FMT, resulted in viral shedding for 6 days after challenge with the human rotavirus G1P[8] genotype Wa strain (RVwa). Rotavirus titers in feces were also significantly higher in antibiotic-treated animals with or without FMT but they were decreased in animals subject to self-FMT, where a partial re…

Rotavirus0301 basic medicinePermissivenessmiceQH301-705.5Virus RNA030106 microbiologyPopulationMicrobiologiaMedicine (miscellaneous)Antibiòticsmedicine.disease_causeGeneral Biochemistry Genetics and Molecular BiologyVirusArticlevirus sheddingMicrobiologyMice03 medical and health sciencesAntigenAntibioticsRotavirusLactobacillusantibioticmedicinemicrobiotaBiology (General)Viral sheddingeducationFecesInfectivityeducation.field_of_studyInnate immune systembiologyMicrobiotaVirus sheddingbiology.organism_classificationSmall intestine030104 developmental biologymedicine.anatomical_structurerotavirusBiomedicines
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Calcium transport in rat small intestine in vitro and in vivo

1972

Intestinal calcium (Ca) transport was studied in the rat jejunum by the in vitro perfusion technique of Fisher and Parsons and in the tied loop in vivo. Mucosal uptake and absorption of Ca was examined under the following conditions: rising intraluminal Ca-concentrations (0.5–128 meq/l); inhibition of energy dependent metabolism (2,4-dinitrophenol, N2, low temperature); net water flow, out of or into the intestinal lumen; addition of strontium (Sr); pretreatment with low Ca-diet and with 6-methyl-prednisolone. The concentration-dependent Ca absorption curve rose steeply at low Ca-concentrations but changed to a slowly rising straight line above 16 meq/l Ca++. In contrast, Ca uptake into the…

Calcium IsotopesAbsorption (pharmacology)medicine.medical_specialtyWater flowPrednisolonechemistry.chemical_elementIn Vitro TechniquesBiologyCalciumIn vivoInternal medicineSolvent dragIntestine SmallmedicineAnimalsIntestinal MucosaPharmacologyBiological TransportRats Inbred StrainsGeneral MedicineMetabolismIn vitroSmall intestineDietRatsJejunummedicine.anatomical_structureEndocrinologyIntestinal AbsorptionchemistryStrontiumCalciumFemaleDinitrophenolsNaunyn-Schmiedeberg's Archives of Pharmacology
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Intestinal absorption pathway of gamma-aminobutyric acid in rat small intestine.

1994

Intestinal absorption of gamma-aminobutyric acid (GABA), as a model compound for gamma-aminoacids, has not been extensively studied from the kinetic viewpoint. Since data from our laboratory suggested that some competition arises between intestinal absorption of beta-alanine and GABA and since our intent was to maintain the aqueous stagnant diffusion layer in order to approach absorption tests to in vivo physiological conditions, a rat jejunum in situ study was undertaken in order to gain an insight into the mechanism of GABA absorption. In the present paper, results from assays using isotonic perfusion solutions with starting GABA concentrations ranging from 1 to 50 mM are reported. They s…

Absorption (pharmacology)MalePharmaceutical ScienceMichaelis–Menten kineticsAminobutyric acidIntestinal absorptionDiffusionNon-competitive inhibitionBody WaterIn vivoIntestine SmallmedicineAnimalsPharmacology (medical)Rats WistarChromatography High Pressure Liquidgamma-Aminobutyric AcidPharmacologyAlanineChemistryGeneral MedicineMembrane transportSmall intestineRatsmedicine.anatomical_structureSpectrometry FluorescenceBiochemistryIntestinal AbsorptionBiophysicsBiopharmaceuticsdrug disposition
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Balanced Bcl-3 expression in murine CD4+T cells is required for generation of encephalitogenic Th17 cells

2017

The function of NF-κB family members is controlled by multiple mechanisms including the transcriptional regulator Bcl-3, an atypical member of the IκB family. By using a murine model of conditional Bcl-3 overexpression specifically in T cells, we observed impairment in the development of Th2, Th1 and Th17 cells. High expression of Bcl-3 promoted CD4+ T-cell survival, but at the same time suppressed proliferation in response to TCR stimulation, resulting in reduced CD4+ T-cell expansion. As a consequence, T cell specific overexpression of Bcl-3 led to reduced inflammation in the small intestine of mice applied with anti-CD3 in a model of gut inflammation. Moreover, impaired Th17-cell develop…

0301 basic medicineT cellMultiple sclerosisImmunologyT-cell receptorStimulationInflammationNF-κBBiologymedicine.diseaseSmall intestineCell biology03 medical and health scienceschemistry.chemical_compound030104 developmental biologymedicine.anatomical_structurechemistryImmunologymedicineTranscriptional regulationImmunology and Allergymedicine.symptomEuropean Journal of Immunology
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Link between Intestinal CD36 Ligand Binding and Satiety Induced by a High Protein Diet in Mice

2012

International audience; CD36 is a ubiquitous membrane glycoprotein that binds long-chain fatty acids. The presence of a functional CD36 is required for the induction of satiety by a lipid load and its role as a lipid receptor driving cellular signal has recently been demonstrated. Our project aimed to further explore the role of intestinal CD36 in the regulation of food intake. Duodenal infusions of vehicle or sulfo-N-succinimidyl-oleate (SSO) was performed prior to acute infusions of saline or Intralipid (IL) in mice. Infusion of minute quantities of IL induced a decrease in food intake (FI) compared to saline. Infusion of SSO had the same effect but no additive inhibitory effect was obser…

CD36 AntigensMaleTime FactorsAnatomy and Physiologymedicine.medical_treatmentCD36[SDV]Life Sciences [q-bio]lcsh:MedicineOleic AcidsLigandsSatiety ResponseBiochemistryJejunumFood-intakeEatingMiceOleoylethanolamidechemistry.chemical_compound0302 clinical medicineIntestinal Mucosalcsh:ScienceReceptorSalineAnimal Management2. Zero hunger0303 health sciencesMultidisciplinaryAgricultureLipidsIntestinesmedicine.anatomical_structureSatiety Response030220 oncology & carcinogenesisChain Fatty-AcidsMedicineProtein BindingResearch ArticleReceptormedicine.medical_specialtySuccinimidesTransportBiologyBody-weightAbsorption03 medical and health sciencesInternal medicinemedicineAnimalsCholesterol UptakeBiologyNutrition030304 developmental biologyEvolutionary Biologylcsh:ROleoylethanolamideGluconeogenesisProteinsSmall intestineDietMice Inbred C57BLEndocrinologyGene Expression RegulationGluconeogenesischemistryImmunologybiology.proteinRatVeterinary Sciencelcsh:QZoology[SDV.AEN]Life Sciences [q-bio]/Food and Nutrition
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Influence of Chronic Alcohol Intake on Intestinal Taurine and Antipyrine Transport in Pregnant Rats

1998

Taurine is a nonessential amino acid that plays a critical role in development. However, biosynthetic capacity is almost negligible in the fetus and must be supplied by the mother. Therefore, when maternal taurine status is depressed during gestation, fetal tissue taurine concentrations can also be compromised. In the present study, the effect of chronic alcohol intake on the intestinal transport of taurine during pregnancy has been investigated by an in vitro technique that allows measurement of the unidirectional influx of the amino acid across the intact rat mid jejunum. The influence of alcohol intake on the passive component of the intestinal transport was also investigated with antipy…

Taurinemedicine.medical_specialtyFetusEthanolLiquid dietMedicine (miscellaneous)ToxicologyIntestinal absorptionSmall intestineJejunumPsychiatry and Mental healthchemistry.chemical_compoundmedicine.anatomical_structureEndocrinologychemistryIntestinal mucosaInternal medicinemedicineAlcoholism: Clinical and Experimental Research
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