Search results for "Steroid"

showing 10 items of 1005 documents

The Influence of Brassinosteroid, a Growth-promoting Steroidal Lactone, on Development and CO2-fixation Capacity of Intact Wheat and Mustard Seedlings

1984

In 1970, Mitchell et al. isolated a lipoidal complex from the pollen of rape (Brassica napus L.). This complex, called “Brassins” was found to have partly powerful growth-promoting properties. The novel growth response of young bean plants in the second internode assay (Worley, Mitchell 1971; Mitchell, Gregory 1972) and other physiological changes following Brassin-treatment have been studied under several aspects (Krizek, Worley 1981; Gregory 1981).

chemistry.chemical_classificationGrowth promotingbiologyCarbon fixationBrassicabiology.organism_classificationmedicine.disease_causeMustard PlantHorticulturechemistry.chemical_compoundchemistryPollenBotanymedicineBrassinosteroidLactone
researchProduct

Nonsteroidal Antiinflammatory Agents, XVIII: C-5 Functionalized 6,7-Diphenyl-2,3-dihydro-1H-pyrrolizines as Inhibitors of Bovine Cyclooxygenase and 5…

1994

6-(4-Chlorophenyl)-7-phenyl-2,3-dihydro-1H-pyrrolizines with functional groups at position 5 of the heterocyclic moiety were synthesized and tested. To determine their antiinflammatory activity bovine blood was used as enzyme source for the cyclooxygenase and 5-lipoxygenase, respectively. The iminoxy acetic acid derivative and the iminotetrazole selectively inhibit the 5-lipoxygenase, all the other compounds show medium or low affinity to the active sites of cyclooxygenase and 5-lipoxygenase. In general all compounds inhibit 5-lipoxygenase more effectively than cyclooxygenase. Concerning the inhibition of 5-lipoxygenase the most active compounds found are equipotent to the corresponding pro…

chemistry.chemical_classificationHydroxamic acidbiologyBicyclic moleculeStereochemistryAnti-Inflammatory Agents Non-SteroidalPharmaceutical ScienceStructure-Activity Relationshipchemistry.chemical_compoundEnzymeModels ChemicalchemistryEnzyme inhibitorDrug DiscoveryArachidonate 5-lipoxygenasebiology.proteinAnimalsStructure–activity relationshipMoietyCattleCyclooxygenase InhibitorsPyrrolesLipoxygenase InhibitorsCyclooxygenaseArchiv der Pharmazie
researchProduct

Stable Expression of Heterologous Sulfotransferase in V79 Cells: Activation of Primary and Secondary Benzylic Alcohols

1994

Abstract A sulfotransferase (ST) capable of activating 1-hydroxymethylpyrene (HMP) and 9-hydroxymethylanthracene (HMA) to mutagens was purified from rat liver. This enzyme appeared to be identical with hydroxysteroid STa, whose cDNA was cloned and stably expressed in Chinese hamster V79 cells. Several primary and secondary benzylic alcohols derived from polycyclic aromatic hydrocarbons induced gene mutations, sister chromatid exchanges (SCE) and/or cytotoxicity in these cells.

chemistry.chemical_classificationSulfotransferasePolymers and PlasticsbiologyOrganic ChemistryHeterologousGene mutationbiology.organism_classificationChinese hamsterchemistry.chemical_compoundEnzymeBiochemistrychemistryComplementary DNAMaterials ChemistryHydroxysteroidCytotoxicityPolycyclic Aromatic Compounds
researchProduct

Three Spirostanol Glycosides from the Seeds of Hyoscyamus Niger L.

2006

Three steroidal glycosides of spirostane series have been isolated from the seeds of Hyoscyamus niger L.(Solanaceae). Their structures were determined on the basis of chemical evidence and extensive spectroscopic methods including one-dimensional, two-dimensional NMR and MS analysis. In the genus Hyoscyamus the given compounds have been found out for the first time.

chemistry.chemical_classificationbiologyChemistryProcess Chemistry and TechnologyGlycosideGeneral. Including alchemyGeneral Chemistrybiology.organism_classificationsteroidal glycosideHyoscyamusChemistryNMR analysisQD1-65BotanyEnvironmental ChemistryHyoscyamus nigerQD1-999Chemistry Journal of Moldova
researchProduct

ChemInform Abstract: Non-Steroidal Antiinflammatory Agents. Part 22. Pyrrolidino-enaminones with an Acetic Acid Function at C-3: Synthesis and Inhibi…

2010

chemistry.chemical_classificationbiologyStereochemistryGeneral MedicineNon steroidalPyrrole derivativesAcetic acidchemistry.chemical_compoundEnzymechemistryArachidonate 5-lipoxygenasebiology.proteinOrganic chemistryCyclooxygenaseFunction (biology)ChemInform
researchProduct

Saponins as immunoadjuvants and immunostimulants

1999

Saponins are either triterpene or steroid glycosides widely distributed in the plant and animal kingdom and include a large number of biologically active compounds. Most of them have surface-active and cholesterol-binding properties.

chemistry.chemical_classificationbiologyTraditional medicineQuillaja saponariaChemistrymedicine.medical_treatmentGlycosideBiological activitySimian immunodeficiency virusmedicine.disease_causebiology.organism_classificationSteroidTriterpenemedicine
researchProduct

Biologically and Pharmacologically Active Saponins from Plants: Recent Advances

2000

Saponins as triterpene or steroid glycosides were well known in ancient times for their detergent, haemolytic and fish toxic activities, properties which are correlated with the amphiphilic character of the molecules and their ability to complex cholesterol.

chemistry.chemical_classificationchemistry.chemical_compoundchemistryBiochemistryTriterpeneCholesterolmedicine.medical_treatmentAmphiphilemedicineGlycosideFish <Actinopterygii>Oleanolic acidSteroid
researchProduct

Crystal structure of an epoxysterol: 9α,11α-epoxy-5α-cholest-7-ene-3β,5,6α-triol 3,6-diacetate

2017

The title compound is a polyoxygenated ep­oxy steroid that crystallizes in the P212121 space group.

chemistry.chemical_classificationcrystal structurehydrogen bondCrystallography010405 organic chemistryHydrogen bondGeneral ChemistryCrystal structure010402 general chemistryCondensed Matter PhysicsRing (chemistry)01 natural sciencesResearch Communications0104 chemical sciencesCrystalCrystallographychemistry.chemical_compoundchemistryQD901-999MoleculeGeneral Materials ScienceTriolEne reactionAlkylsteroidsActa Crystallographica Section E Crystallographic Communications
researchProduct

ChemInform Abstract: Nonsteroidal Antiinflammatory Agents. Part 18. C-5 Functionalized 6,7- Diphenyl-2,3-dihydro-1H-pyrrolizines as Inhibitors of Bov…

2010

chemistry.chemical_compoundNonsteroidalchemistrybiologyArachidonate 5-lipoxygenasebiology.proteinGeneral MedicineCyclooxygenasePharmacologyChemInform
researchProduct

ChemInform Abstract: Non-Steroidal Antiinflammatory Agents. Part 21. 2-Aryl-pyrrolo(2,1-b) benzothiazoles as Selective or Dual Inhibitors of Cyclooxy…

2010

chemistry.chemical_compoundbiologychemistryStereochemistryArylArachidonate 5-lipoxygenasebiology.proteinGeneral MedicineCyclooxygenaseNon steroidalChemInform
researchProduct