Search results for "Terpenoid"

showing 10 items of 221 documents

Effect of selected triterpenoids on chronic dermal inflammation.

1997

The activity of four natural triterpenoids on a 12-O-tetradecanoylphorbol-13-acetate multiple-dose model of skin chronic inflammation was studied. Erythrodiol and ursolic acid were significantly effective. The most important features concerning structure-activity relationship and previous data on the effect of these triterpenoids on other inflammatory conditions are discussed.

Anti-Inflammatory AgentsDrug Evaluation PreclinicalInflammationPharmacologyDermatitis ContactDexamethasonechemistry.chemical_compoundMiceTriterpenoidDermisUrsolic acidTriterpeneEdemamedicineAnimalsOleanolic AcidBetulinic AcidDexamethasonePharmacologychemistry.chemical_classificationintegumentary systembusiness.industryTriterpenesmedicine.anatomical_structurechemistryImmunologyTetradecanoylphorbol AcetateFemalemedicine.symptombusinessPentacyclic Triterpenesmedicine.drugEuropean journal of pharmacology
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Zanhasaponins A and B, Antiphospholipase A2 Saponins from an Antiinflammatory Extract of Zanha africana Root Bark

1997

A MeOH extract from Z. africana was examined for topical antiinflammatory activity and proved to be active against arachidonic acid (AA) acute edema, 12-O-tetradecanoylphorbol 13-acetate (TPA)-induced chronic inflammation, and oxazolone delayed-type hypersensitivity in mice. The extract also showed significant inhibitory activity of Naja naja phospholipase A2 when a polarographic method was used. Two oleanane-type triterpene saponins, zanhasaponins A (1) and B (2), and the cyclitol pinitol (4), isolated from the extract, were active as inhibitors of PLA2. A further saponin, zanhasaponin C (3) was inactive in this assay.

Anti-Inflammatory AgentsSaponinPharmaceutical SciencePharmacognosyDermatitis ContactPhospholipases AAnalytical ChemistryMicechemistry.chemical_compoundPhospholipase A2Adjuvants ImmunologicTriterpeneDrug DiscoveryAnimalsEdemaEnzyme InhibitorsPeroxidaseSkinPharmacologychemistry.chemical_classificationintegumentary systembiologyTraditional medicineOrganic ChemistryOxazoloneGlycosideSaponinsTriterpenesTerpenoidPhospholipases A2Complementary and alternative medicinechemistryBiochemistryvisual_artvisual_art.visual_art_mediumbiology.proteinTetradecanoylphorbol AcetateMolecular MedicineFemaleBarkArachidonic acidJournal of Natural Products
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Synthesis and biological evaluation of (+)-labdadienedial, derivatives and precursors from (+)-sclareolide

2010

Labdadienedial and a series of C15,C16-functionalized derivatives were synthesized from commercial (+)-sclareolide and evaluated for their cytotoxic, antimycotic, and antiviral activities. Their precursors were similarly evaluated.

Antifungal AgentsStereochemistryAntineoplastic AgentsHerpesvirus 1 HumanAntiviral AgentsChemical synthesisInhibitory Concentration 50chemistry.chemical_compoundChlorocebus aethiopsDrug Discoveryotorhinolaryngologic diseasesAnimalsHumansCytotoxicityVero CellsPharmacologyOrganic ChemistryFungifood and beveragesSclareolideBiological activityGeneral MedicineCombinatorial chemistryTerpenoidIn vitrostomatognathic diseaseschemistrylipids (amino acids peptides and proteins)DiterpenesDiterpeneEnantiomerHeLa CellsEuropean Journal of Medicinal Chemistry
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SKRINING FITOKIMIA DAN UJI AKTIVITAS ANTIOKSIDAN DAN ANTITUMOR 20 TUMBUHAN OBAT ASAL KABUPATEN MANOKWARI

2008

<strong><em>Flavanoid, steroid, and terpenoid contents of 20 Manokwari medicinal plants were analyzed.  The antioxidant activity, total phenolic contents and antitumor activity of 20 Manokwari medicinal plants were also evaluated. The result shows that 83% positif to flavanoid test, 59% positif to terpenoid test and only 25% positif steroid. Antioxidant activity and total phenolic contents evaluated using Ferric Thiocianate (FTC) and Folin-Ciocalteu methods respectively. Antioxidant activity and total phenolic contents of medicinal plants were extracted by the traditional method, boiling in water and also in 80% methanol. Twenty plants evaluated in both exstracts have significan…

Antitumor activityAntioxidantTraditional medicineChemistrymedicine.medical_treatmentmedicineMedicinal plantsTerpenoidSteroidJurnal Natural
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The Diterpenoids of the Genus Elaeoselinum (Apiaceae) and their Biological Properties

2008

The natural kaurane, beyerane and atisane diterpenoids isolated from the genus Elaeoselinum (Apiaceae)and their semi-synthetic derivatives are reviewed. Published 13C NMR spectroscopic data and biological properties of these diterpenes are also reported.

ApiaceaebiologyGenusElaeoselinumChemistryBiological propertyOrganic ChemistryBotanyditerpenoids Eleoselinum biological propertiesSettore BIO/15 - Biologia Farmaceuticabiology.organism_classificationCurrent Organic Chemistry
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Floral volatiles in a sapromyiophilous plant and their importance in attracting house fly pollinators

2015

Floral scent in sapromyiophilous plants often consists of complex blends with not only fetid (e.g., sulfides) but also sweet (e.g., terpenoids) volatile organic compounds and a recent study suggests that both groups of compounds are involved in pollinator attraction. However, little is known about the number and identity of compounds involved in pollinator attraction in these deceptive plants that mimic breeding sites of fly pollinators. In the present paper, we studied flower volatiles of sapromyiophilous Periploca laevigata and their capability to elicit biological responses in one of the pollinator species, Musca domestica. Floral volatiles were collected by dynamic headspace and analyse…

Arthropod AntennaeSettore BIO/07 - EcologiaPollinationBiologyBiochemistryGas Chromatography-Mass Spectrometrychemistry.chemical_compoundPollinatorHousefliesBotanyOlfactometryAnimalsPeriplocaPollinationEcology Evolution Behavior and SystematicsVolatile Organic CompoundsGeneral Medicinebiology.organism_classificationOlfactory PerceptionAttractionTerpenoidApocynaceaeSettore AGR/11 - Entomologia Generale E ApplicatachemistryOlfactometerApocynaceae Behaviour Electrophysiology Floral scent Musca domestica Muscidae Periploca Pollination SapromyophilousSettore BIO/03 - Botanica Ambientale E ApplicataGas chromatographyDimethyl trisulfide
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Analytical characterisation of the biodeterioration of diterpenoid labdanic varnishes used in pictorial techniques: Sandarac and Manila copal

2014

Abstract The deterioration produced by fungal and bacterial growth on the sandarac and Manila copal, diterpenoid varnishes traditionally used as art materials, was evaluated by gas chromatography–mass spectrometry (GC–MS), and pyrolysis–gas chromatography–mass spectrometry (Py–GC–MS). Test specimens, coated with a solidified thin layer of the studied varnishes, were inoculated and incubated with selected fungi and bacteria obtained from collections and oil paintings affected by biodeterioration, and analysed by the above mentioned techniques. Significant changes were detected, showing evidence of deterioration processes caused or favoured by some of the studied microorganisms.

BiomaterialsChromatographyChemistryMicroorganismThin layerBotanySandaracGas chromatography–mass spectrometryBacterial growthWaste Management and DisposalMicrobiologyTerpenoidInternational Biodeterioration & Biodegradation
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Hirsutane-Type Sesquiterpenes with Uncommon Modifications from Three Basidiomycetes

2010

From three basidiomycetes, Xeromphalina sp., Stereum sp., and Pleurocybella porrigens, six triquinane sesquiterpenes with unprecendented modifications and a rearranged sesquiterpene related to coriolin C have been isolated. Their isolation, structure elucidation, and biological evaluation are described.

Bridged-Ring CompoundsPolycyclic SesquiterpenesAntifungal AgentsBacteriaMolecular StructurebiologyStereochemistryXeromphalinaBasidiomycotaOrganic ChemistryFungibiology.organism_classificationSesquiterpenePleurocybella porrigensTerpenoidAnti-Bacterial Agentschemistry.chemical_compoundchemistryOrganic chemistryStereumSesquiterpenesBiological evaluationThe Journal of Organic Chemistry
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Environmental and Biochemical Factors Controlling the in Vitro Emergence of Somatic Embryos in European Spindle Tree (Euonymus europaeus L)

2000

The European spindle tree (Euonymus europaeus L. Celastraceae) is a shrubby tree widely distributed in temperate regions of western European countries from the northern part of France to St. Petersburg and the western part of Russia. The Celastraceae comprises 55 genera, including at least 850 known species of trees and shrubs which are found in tropical and temperate regions. Various secondary metabolites are elaborated in the family including steroids, triterpenoids, sesquiterpene, peptide ore alkaloids. The spindle tree is commonly found in quickset hedges and small broad-leaved forests when the soil is deep, moist, clayey and chalky. The leaves are relatively small (3–4 cm long) simple …

CelastraceaeTriterpenoidSomatic embryogenesisbiologyEcotypevisual_artBotanyvisual_art.visual_art_mediumTemperate climateEuropean Spindle-TreeBarkEuonymus europaeusbiology.organism_classification
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Spiroterpenoids from Hypericum reflexum

1993

Abstract Two new spiroterpenoids, hyperireflexolide A and B, were isolated from Hypericum reflexum . Their structures and stereochemistry were established by spectroscopic methods, including 13 C NMR, DEPT and HMQC, and X-ray data.

ChemistryStereochemistryX ray dataPlant ScienceGeneral MedicineHorticultureDEPTCarbon-13 NMRMolecular BiologyBiochemistryTerpenoidHypericum reflexumPhytochemistry
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