Search results for "Xanthydrol"

showing 4 items of 4 documents

Determination of N-acetyl-l-glutamine in urine by HPLC

1986

The determination of N-acetyl-l-glutamine (AC-GLN) in urine of rats after derivatization with xanthydrol by HPLC is described. The urine samples were collected from two groups of rats, one group fed normal nutrition, the other treated with AC-GLN. About 5 mM/l AC-GLN was detected in urine of untreated animals, whereas the excretion of the other group was in the range of 50 mM/l corresponding to about 50 wt.-% of the given AC-GLN.

Excretionchemistry.chemical_compoundChromatographyChemistryClinical BiochemistryN-acetyl-L-glutamineGeneral Materials ScienceGeneral MedicineUrineXanthydrolDerivatizationHigh-performance liquid chromatographyAnalytical ChemistryFresenius' Zeitschrift für analytische Chemie
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Regioselective proton-catalyzed diarylmethylation of indoles with 9H-xanthydrol, dibenzosuberenol, and bis[4-dimethylaminophenyl]methanol

1988

3-Isopropylindole (4) is xanthenylated both at N-1 (stereocontrolled major reaction), C-2, and on the phenyl nucleus of the indole skeleton by xanthydrol (1). Other carbinols such as dibenzosuberenol (2) and bis[4-dimethylaminophenyl]methanol (3) with lower electrophilic SN1 activities than 1 do not react with 4 but do react very selectively with simple methylindoles to form diarylmethylated derivatives.

Indole testchemistry.chemical_compoundAcid catalysisBicyclic moleculeChemistryOrganic ChemistryElectrophileRegioselectivityOrganic chemistryMethanolXanthydrolMedicinal chemistryCatalysisJournal of Heterocyclic Chemistry
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Mechanismus und Reaktionswege der Xanthenylierung an ambidenten nukleophilen Arzneistoffen

1986

Am Beispiel der ambidenten nukleophilen Arzneistoffe 4-Aminobenzolsulfonamid (3), Indometacin (7) und Phenylbutazon (10) werden Aralkylierungen mit dem SN1-aktiven Reagens Xanthydrol (1) vorgestellt. Mechanism and Reaction Path of the Xanthenylation of Ambident Nucleophilic Drugs The aralkylation of ambident nucleophilic drugs, e.g. 4-aminobenzenesulfonamide (3), indometacine (7) and phenylbutazone (10), with SN1-active xanthydrol (1) is described.

chemistry.chemical_classificationchemistry.chemical_compoundSN1 reactionNucleophileBicyclic moleculechemistryStereochemistryDrug DiscoveryPharmaceutical ScienceReaction pathXanthydrolSulfonamideArchiv der Pharmazie
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ChemInform Abstract: Regioselective Proton-Catalyzed Diarylmethylation of Indoles with 9H-Xanthydrol, Dibenzosuberenol, and Bis(4-dimethylaminophenyl…

1989

3-Isopropylindole (4) is xanthenylated both at N-1 (stereocontrolled major reaction), C-2, and on the phenyl nucleus of the indole skeleton by xanthydrol (1). Other carbinols such as dibenzosuberenol (2) and bis[4-dimethylaminophenyl]methanol (3) with lower electrophilic SN1 activities than 1 do not react with 4 but do react very selectively with simple methylindoles to form diarylmethylated derivatives.

Indole testchemistry.chemical_compoundProtonchemistryElectrophileRegioselectivityGeneral MedicineMethanolXanthydrolMedicinal chemistryCatalysisChemInform
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