Search results for "biophysics"

showing 10 items of 3515 documents

Investigation of Isoindolo[2,1-a] quinoxaline-6-imines as Topoisomerase I Inhibitors with Molecular Modeling Methods

2017

Background: Isoindolo[2,1-alpha] quinoxalines constitute an important class of compounds which demonstrated potent antiproliferative activity against different human tumor cell lines and topoisomerase I inhibitors. In particular, their water soluble imine or iminium salts recently synthesized showed potent growth inhibitory effect on NCI-60 tumor cell line panel and biological studies performed on the most active compounds demonstrated that they cause DNA damage via topoisomerase I poisoning. Objective: Herein, we investigate with molecular modeling methods, the common features responsible for topoisomerase I inhibition of the water-soluble isoindolo[2,1-alpha] quinoxalin-6-imines, by compa…

0301 basic medicine030103 biophysicsMolecular modelStereochemistryDNA damageAntineoplastic AgentsIsoindolesTopoisomerase-I InhibitorCrystallography X-RayaromatechinStructure-Activity Relationship03 medical and health scienceschemistry.chemical_compoundQuinoxalinetopotecanantiproliferativeCell Line TumorNeoplasmsQuinoxalinesquinoxalineDrug DiscoveryHumansCell Proliferationbiologypharmacophore modelTopoisomeraseIminiumGeneral MedicineSettore CHIM/08 - Chimica FarmaceuticaMolecular Docking SimulationTopoisomerase IindenoisoquinolineDNA Topoisomerases Type IchemistryDocking (molecular)dockingbiology.proteinMolecular MedicineTopoisomerase I; quinoxaline; antiproliferative; topotecan; aromatechin; indenoisoquinoline; docking; pharmacophore modelIminesTopoisomerase I InhibitorsPharmacophore
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X-ray response of CdZnTe detectors grown by the vertical Bridgman technique: Energy, temperature and high flux effects

2016

Abstract Nowadays, CdZnTe (CZT) is one of the key materials for the development of room temperature X-ray and gamma ray detectors and great efforts have been made on both the device and the crystal growth technologies. In this work, we present the results of spectroscopic investigations on new boron oxide encapsulated vertical Bridgman (B-VB) grown CZT detectors, recently developed at IMEM-CNR Parma, Italy. Several detectors, with the same electrode layout (gold electroless contacts) and different thicknesses (1 and 2.5 mm), were realized: the cathode is a planar electrode covering the detector surface (4.1×4.1 mm2), while the anode is a central electrode (2×2 mm2) surrounded by a guard-rin…

0301 basic medicine030103 biophysicsNuclear and High Energy PhysicsHigh fluxDigital pulse shape analysi01 natural sciencesBoron oxide encapsulated vertical Bridgmanlaw.invention03 medical and health scienceslaw0103 physical sciencesPolarization (electrochemistry)InstrumentationPhysicsX-ray and gamma ray detectors010308 nuclear & particles physicsbusiness.industryCdZnTe detectorsCdZnTe detectorEnergy-resolved photon counting detectorSettore FIS/01 - Fisica SperimentaleDetectorGamma raySettore FIS/07 - Fisica Applicata(Beni Culturali Ambientali Biol.e Medicin)CathodePhoton countingAnodeFull width at half maximumElectrodeEnergy-resolved photon counting detectorsOptoelectronicsDigital pulse shape analysisbusinessNuclear Instruments and Methods in Physics Research Section A: Accelerators, Spectrometers, Detectors and Associated Equipment
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Digital fast pulse shape and height analysis on cadmium-zinc-telluride arrays for high-flux energy-resolved X-ray imaging.

2017

Cadmium-zinc-telluride (CZT) arrays with photon-counting and energy-resolving capabilities are widely proposed for next-generation X-ray imaging systems. This work presents the performance of a 2â...mm-thick CZT pixel detector, with pixel pitches of 500 and 250â...μm, dc coupled to a fast and low-noise ASIC (PIXIE ASIC), characterized only by the preamplifier stage. A custom 16-channel digital readout electronics was used, able to digitize and process continuously the signals from each output ASIC channel. The digital system performs on-line fast pulse shape and height analysis, with a low dead-time and reasonable energy resolution at both low and high fluxes. The spectroscopic response …

0301 basic medicine030103 biophysicsNuclear and High Energy PhysicsMaterials sciencePreamplifierInstrumentationenergy-resolved photon counting detectordigital pulse shape analysienergy-resolved photon counting detectors01 natural sciencesCharge sharing03 medical and health scienceschemistry.chemical_compoundOpticshigh flux0103 physical sciencesInstrumentationX-ray and ?-ray detectorsNuclear and High Energy Physiccharge sharingRadiationdigital pulse shape analysisPixel010308 nuclear & particles physicsbusiness.industryCdZnTe detectorsCdZnTe detectorSettore FIS/01 - Fisica SperimentaleDetectorX-ray and γ-ray detectorBiasingSettore FIS/07 - Fisica Applicata(Beni Culturali Ambientali Biol.e Medicin)Cadmium zinc telluridechemistryDirect couplingbusinessJournal of synchrotron radiation
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Dual-polarity pulse processing and analysis for charge-loss correction in cadmium–zinc–telluride pixel detectors

2018

Charge losses at the inter-pixel gap are typical drawbacks in cadmium–zinc–telluride (CZT) pixel detectors. In this work, an original technique able to correct charge losses occurring after the application of charge-sharing addition (CSA) is presented. The method, exploiting the strong relation between the energy after CSA and the beam position at the inter-pixel gap, allows the recovery of charge losses and improvements in energy resolution. Sub-millimetre CZT pixel detectors were investigated with both uncollimated radiation sources and collimated synchrotron X-rays, at energies below and above the K-shell absorption energy of the CZT material. The detectors are DC coupled to fast and low…

0301 basic medicine030103 biophysicsNuclear and High Energy PhysicsMaterials sciencePreamplifierPhysics::Instrumentation and Detectors01 natural sciencesCollimated lightCharge sharinglaw.invention03 medical and health scienceschemistry.chemical_compoundOpticslawcharge losse0103 physical sciencesInstrumentationenergy-resolved photon-counting detectorsNuclear and High Energy Physiccharge lossescharge sharingRadiationPixel010308 nuclear & particles physicsbusiness.industryCdZnTe detectorsCdZnTe detectorDetectorSettore FIS/01 - Fisica Sperimentaleenergy-resolved photon-counting detectorSynchrotronSettore FIS/07 - Fisica Applicata(Beni Culturali Ambientali Biol.e Medicin)Cadmium zinc tellurideX-ray and gamma-ray detectorschemistryDirect couplingbusinessX-ray and gamma-ray detector
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Clinical effect of diode laser on peri-implant tissues during non-surgical peri-implant mucositis therapy: Randomized controlled clinical study

2019

Background: The aim of this study is to evaluate the response to the non-surgical treatment of peri-implant mucositis using the diode laser as an adjuvant therapy in patients with implant-supported restorations, in terms of clinical variables, with respect to those patients in whom conventional non-surgical therapy is used. Material and Methods: Randomized controlled clinical trial with simple blind 3 months follow-up. Two groups of patients were established, the non-surgical mechanical debridement of the affected implants was performed in the control group (n = 34) and the diode laser therapy was also performed in the test group (n = 34). The implant was considered the study subject; the v…

0301 basic medicine030103 biophysicsPeri-implant mucositisBleeding on probingDentistryOdontología03 medical and health sciences0302 clinical medicineLáseresStatistical significanceAdjuvant therapymedicineMucositisTecnología médicaGeneral DentistryImplantes dentalesbusiness.industryResearch030206 dentistrymedicine.disease:CIENCIAS MÉDICAS [UNESCO]Clinical trialUNESCO::CIENCIAS MÉDICASAnalysis of varianceImplantmedicine.symptomOral SurgerybusinessJournal of Clinical and Experimental Dentistry
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Hands On: Using Tryptophan Fluorescence Spectroscopy to Study Protein Structure

2019

Fluorescence spectroscopy is well suited to obtain information about the structure and function of proteins. The major advantage of this spectroscopic technique is the pronounced dependence of the fluorescence emission characteristics of fluorophores on their distinct local environment and the rather inexpensive equipment required. In particular, the use of intrinsic tryptophan fluorescence offers the possibility to study structure and function of proteins without the need to modify the protein. While fluorescence spectroscopy is technically not demanding, a number of factors can artificially alter the results. In this article, we systematically describe the most common applications in fluo…

0301 basic medicine030103 biophysicsQuenching (fluorescence)ChemistryTryptophanFluorescenceFluorescence spectroscopy03 medical and health sciences030104 developmental biologyProtein structureTryptophan fluorescenceBiophysicsLocal environmentSpectroscopy
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Generation of oxysterols formed by free radicals and enzymes by electrochemical oxidation

2016

International audience; It is commonly accepted that cholesterol oxide derivatives, also named oxysterols, are 27 carbon-atom molecules deriving either from enzymatic and non-enzymatic oxidation of cholesterol. Most of these compounds can be synthesized by more or less difficult and time consuming chemical reactions, and some of them have been discovered before the identification of the enzymes [mainly cytochrome P450 enzymes (CYP enzymes)] involved in their biosynthesis. A wide range of biological activities depends on oxysterols. Some oxysterols are also involved in the synthesis of cholesterol metabolites which have various properties. The paper by Weber et al. in this issue of European …

0301 basic medicine030103 biophysicsRadical[ SDV.AEN ] Life Sciences [q-bio]/Food and NutritionChemical reactionIndustrial and Manufacturing EngineeringEditorial Material03 medical and health scienceschemistry.chemical_compoundBiosynthesisIn vivopolycyclic compoundsMoleculechemistry.chemical_classificationbiologyCholesterolCytochrome P450General ChemistryOxysterols[SDV.AEN] Life Sciences [q-bio]/Food and NutritionEnzymeElectrochemical oxidationchemistryBiochemistrybiology.proteinlipids (amino acids peptides and proteins)Food ScienceBiotechnology
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The effect of photodynamic therapy and polymer solution containing nano-particles of Ag /ZnO on push-out bond strength of the sealers AH-Plus and MTA…

2017

BACKGROUND The aim of this in vitrostudy was to examine and compare the effect of photodynamic therapy and solution containing nano particles Ag/ZnO on adhesion of endodontic sealers to dentinal walls of human root canal. MATERIAL AND METHODS Ninty single-rooted human teeth were selected and their clinical crown was cut from the cemento-enamel junction zone. Canals were prepared by RaCe rotary system and the smear layer was removed using 17% EDTA and 5.25% NaOCl. Samples were randomly divided into two groups of AH Plus and MTA Fillapex based on the sealer type and each group based on antimicrobial method was divided into two sub-groups of photodynamic therapy and polymer containing nano par…

0301 basic medicine030103 biophysicsScanning electron microscopeRoot canalmedicine.medical_treatmentSmear layerNanoparticleDentistryPhotodynamic therapyOperative Dentistry and Endodontics03 medical and health sciences0302 clinical medicineMTA-FillapexPush outmedicineGeneral DentistryBond strengthbusiness.industryChemistryResearch030206 dentistry:CIENCIAS MÉDICAS [UNESCO]medicine.anatomical_structureUNESCO::CIENCIAS MÉDICASbusinessNuclear chemistry
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"The human use of human beings": Interdisciplinarity, transdisciplinarity and all that in biophysics and beyond.

2017

Abstract Biophysics, just by looking at its name, indicates an interdisciplinary scientific activity, although the notion of interdisciplinarity, as such, seems to be not widely or specifically discussed by biophysicists. The same seems to have happened as well in the early stages of the development of cybernetics, notably in Norbert Wiener's writings. This situation seems to contrast with what has happened in subsequent developments of cybernetics ideas, notably in general system theory and cognitive sciences. After a few general reflections on the notion of interdisciplinarity, its sophisticated variants and the path leading to the birth of cognitive science, we shall refer to Wiener's th…

0301 basic medicine030103 biophysicsSettore INF/01 - InformaticaChemistryOrganic ChemistryInterdisciplinarityBiophysicsSettore MAT/01 - Logica MatematicaHistory 20th CenturyBiochemistry03 medical and health sciencesBiophysicHuman useTransdisciplinarityWienerBiophysicsCyberneticsHumansCyberneticSocial responsibilityCyberneticsScientific activityHumanInterdisciplinarityBiophysical chemistry
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UVER and UV index at high altitude in Northwestern Argentina

2016

Measurements of ultraviolet erythemal radiation (UVER) made during two years at three sites located at altitudes over 1000 m a.s.l. in Northwestern Argentina (Salta, San Carlos, and El Rosal) have been used to estimate and analyze the UV Index (UVI) and the cumulative doses at these locations. For the UVER irradiance, data of January (maximum values) and June (minimum values) have been analyzed as representative of the year for all locations. The UVI reaches extreme (> 11) values in > 20% of the analyzed days in Salta (1190 m a.s.l.), while these are reached in San Carlos (1611 m a.s.l.) and El Rosal (3355 m a.s.l.) in > 40% of the analyzed days. Finally, the cumulative doses over an averag…

0301 basic medicine030103 biophysicsVeterinary medicineMeteorologyUltraviolet erythemal radiation (UVER)Ultraviolet RaysBiophysicsIrradianceArgentinaRadiation DosageCumulative dosesCiencias de la Tierra y relacionadas con el Medio Ambiente03 medical and health sciencesRadiation MonitoringHigh altitudeRadiology Nuclear Medicine and imagingSouthern HemisphereRadiationRadiological and Ultrasound TechnologyAltitudeEffects of high altitude on humansUltraviolet index (UVI)Southern hemisphereEnvironmental scienceMeteorología y Ciencias AtmosféricasCIENCIAS NATURALES Y EXACTAS
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