Search results for "carbamate"

showing 10 items of 219 documents

Effects of several muscarinic agonists on cardiac performance and the release of noradrenaline from sympathetic nerves of the perfused rabbit heart

1972

Summary 1 The effects of several muscarinic agonists on atrial tension development, ventricular rate and noradrenaline release from terminal sympathetic fibres evoked by electrical nerve stimulation (SNS) and 1,1-dimethyl-4-phenylpiperazinium (DMPP) were measured in isolated perfused rabbit hearts. 2 Hexamethonium, in a concentration which almost abolished the release of noradrenaline by DMPP, had no effect on the release produced by SNS, confirming that the stimulation was postganglionic. 3 The order of potency for inhibition of atrial tension development was N-methyl-1,2,5,6, tetrahydro-nicotinic acid prop-2-yne ester (MH-1)>oxotremorine > acetylcholine > methacholine > carbachol > furtre…

AtropineMalemedicine.medical_specialtySympathetic Nervous SystemCarbacholAutopharmacologyHexamethonium CompoundsIn Vitro TechniquesPharmacologyNorepinephrinechemistry.chemical_compoundHeart RateInternal medicineMuscarinic acetylcholine receptormedicineOxotremorineAnimalsMethacholine CompoundsPharmacologyChemistryOxotremorinePilocarpineHeartAcetylcholineElectric StimulationPerfusionQuaternary Ammonium CompoundsAtropineEndocrinologyParasympathomimeticsPilocarpineCarbacholFemaleMethacholineHexamethoniumCarbamatesRabbitsDimethylphenylpiperazinium IodideAcetylcholinemedicine.drugBritish Journal of Pharmacology
researchProduct

Analysis of pesticides in fruits by pressurized liquid extraction and liquid chromatography-ion trap-triple stage mass spectrometry.

2005

A multi-residue method using pressurized liquid extraction (PLE) and liquid chromatography-quadrupole ion trap-triple stage mass spectrometry (LC-IT-MS(3)) has been developed for determining trace levels of pesticides in fruits. The selected pesticides can be distinguished in: benzimidazoles and azoles, organophosphorus, carbamates, neonicotinoids, and acaricides. PLE has been optimized to extract these pesticide residues from oranges and peaches by studying the effect of experimental variables on PLE efficiency. Samples were extracted at high temperature and pressure (75 degrees C and 1500psi) using ethyl acetate as extraction solvent and acidic alumina as drying agent. The recoveries obta…

AzolesEthyl acetateAcetatesMass spectrometryBiochemistryHigh-performance liquid chromatographySensitivity and SpecificityAnabasineMass SpectrometryAnalytical Chemistrychemistry.chemical_compoundOrganophosphorus Compoundsmedia_common.cataloged_instanceEuropean unionPesticidesmedia_commonResidue (complex analysis)ChromatographyPesticide residueChemistryOrganic ChemistryExtraction (chemistry)Pesticide ResiduesTemperatureReproducibility of ResultsGeneral MedicineFruitBenzimidazolesIon trapCarbamatesChromatography LiquidJournal of chromatography. A
researchProduct

CCDC 1564495: Experimental Crystal Structure Determination

2017

Related Article: Fernando Rabasa-Alcañiz, Javier Torres, María Sánchez-Roselló, Tomás Tejero, Pedro Merino, Santos Fustero, Carlos del Pozo|2017|Adv.Synth.Catal.|359|3752|doi:10.1002/adsc.201700975

Benzyl [(3aR5S9bR)-7-fluoro-3-methyl-9b-(trifluoromethyl)-133a459bhexahydronaphtho[21-c]isoxazol-5-yl](hydroxy)carbamateSpace GroupCrystallographyCrystal SystemCrystal StructureCell ParametersExperimental 3D Coordinates
researchProduct

Effects of thrombin and of the phospholipase C inhibitor, D609, on the vascularity of the chick chorioallantoic membrane.

2000

Abstract Microvascular corrosion casting was used to assess the effects of thrombin and D609, a phospholipase C inhibitor, on the vascularity of the chick embryo chorioallantoic membrane (CAM). Discs containing vehicle, thrombin or D609 were placed on the CAM of fertilized white Leghorn eggs on Day 9 of gestation and vascularity was assessed on Day 11. Thrombin caused significant increases in the numbers (43%), diameters (5%) and lengths (17%), of both pre- and postcapillaries (first-order vessels by centripetal ordering). Conversely, D609 caused a decrease in the numbers (27%), lengths (12%) and diameters (8%) of first-order vessels. D609 decreased the total vascular volume of first- to th…

Bridged-Ring Compoundsmedicine.medical_specialtyanimal structuresAngiogenesisPhosphodiesterase InhibitorsNeovascularization PhysiologicChick EmbryoBiologyHemostaticsMicrocirculationThrombinVascularityAllantoisThiocarbamatesInternal medicinemedicineAnimalsOvumPharmacologyBlood VolumePhospholipase CThrombinThionesChorionNorbornanesChorioallantoic membraneEndocrinologymedicine.anatomical_structureType C PhospholipasesCirculatory systemMicroscopy Electron Scanningmedicine.symptommedicine.drugBlood vesselGeneral pharmacology
researchProduct

Multi-elemental determination of heavy elements in plastics using X-ray fluorescence after destruction of the polymer by molten sodium hydroxide

1992

In this paper a method is proposed for the multielemental analysis of Sb(III), Ba, Cd, Cr(III), Hg, Pb and As(III) in plastics, using X-ray fluorescence after alkaline decomposition and preconcentration by (co)precipitation. The organic matrix is destroyed by decomposition with sodium hydroxide melted in a silver crucible by the open system technique, using sodium nitrate as auxiliary oxidant. The variables which influence preconcentration are optimized: digestion time, pH, salinity, carrier and sodium diethyldithiocarbamate (DDTC) and sodium rhodizonate (R) as precipitants. The calibration curves were linear up to 200 μg of the element present, except for lead (150 μg) antimony(III) (100 μ…

Calibration curveSodiumInorganic chemistrychemistry.chemical_elementX-ray fluorescenceBariumBiochemistryAnalytical Chemistrychemistry.chemical_compoundchemistryAntimonySodium nitrateSodium hydroxideSodium diethyldithiocarbamateFresenius' Journal of Analytical Chemistry
researchProduct

The Endocannabinoid System Promotes Astroglial Differentiation by Acting on Neural Progenitor Cells

2006

Endocannabinoids exert an important neuromodulatory role via presynaptic cannabinoid CB1receptors and may also participate in the control of neural cell death and survival. The function of the endocannabinoid system has been extensively studied in differentiated neurons, but its potential role in neural progenitor cells remains to be elucidated. Here we show that the CB1receptor and the endocannabinoid-inactivating enzyme fatty acid amide hydrolase are expressed, bothin vitroandin vivo, in postnatal radial glia (RC2+cells) and in adult nestin type I (nestin+GFAP+) neural progenitor cells. Cell culture experiments show that CB1receptor activation increases progenitor proliferation and differ…

Cannabinoid receptorCellular differentiationMorpholinesApoptosisNerve Tissue ProteinsBiologyNaphthalenesHippocampusAmidohydrolasesNestinMiceIntermediate Filament ProteinsReceptor Cannabinoid CB1Cannabinoid Receptor ModulatorsGlial Fibrillary Acidic ProteinAnimalsProgenitor cellEnzyme InhibitorsNeural cellCells CulturedProgenitorMice KnockoutNeuronsCannabinoidsmusculoskeletal neural and ocular physiologyGeneral NeuroscienceStem CellsCell DifferentiationArticlesNestinEndocannabinoid systemNeural stem cellBenzoxazinesRatsnervous systemAstrocytesBenzamideslipids (amino acids peptides and proteins)CarbamatesNeurosciencepsychological phenomena and processesEndocannabinoids
researchProduct

Cholinesterase Activity and Hematological Parameters as Biomarkers of Sublethal Molinate Exposure in Anguilla anguilla

2000

Cholinesterase (ChE) activity was measured in plasma, whole blood [using 5,5'-dithiobis(2-nitrobenzoic acid) and 2-PDS as chromophores], brain, and whole eyes of Anguilla anguilla exposed to a sublethal concentration of 11.15 mg/L (one-third of the 96-h LC(50)) of the carbamate herbicide molinate. ChE activity was evaluated after 6, 24, 48, 72, and 96 h of pesticide exposure. Results indicated that ChE activity in eel tissues decreased as time of exposure increased, especially in eel blood. Eels exposed to molinate were transferred to a pesticide-free water for a recovery period of 4 days and ChE activity was also evaluated. Results indicated that ChE activity for those animals with preexpo…

CarbamateHealth Toxicology and Mutagenesismedicine.medical_treatmentPhysiologyHematocritToxicologyThiocarbamatesAnguillidaeBlood plasmamedicineAnimalsCholinesterasesCholinesteraseWhole bloodBlood CellsEelsintegumentary systembiologymedicine.diagnostic_testHerbicidesPublic Health Environmental and Occupational HealthAzepinesBlood ProteinsGeneral Medicinebiology.organism_classificationPollutionBlood proteinsToxicitybiology.proteinCarbamatesCholinesterase InhibitorsBiomarkersEcotoxicology and Environmental Safety
researchProduct

Comparison of basal cytotoxicity of seven carbamates in CHO-K1 cells

2006

The cytotoxic effects of seven carbamate pesticides, aldicarb, aldicarb sulfone, aldicarb sulfoxide, benfuracarb, pirimicarb, propoxur and thiobencarb, were compared in Chinese hamster ovary (CHO-K1) cell line of Circetulus griseus. The endpoints evaluated were lysosomal function by neutral red assay and mitochondrial integrity by 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyltetrazolium bromide (MTT assay). The carbamates tested were evaluated in both serum-free medium and in serum-containing medium. Results demonstrate that CHO-K1 lysosomes appeared more susceptible to propoxur, aldicarb and its metabolites than mitochondria. Aldicarb was the most toxic carbamate pesticide tested on CHO-K1 cel…

CarbamateNeutral redAldicarbHealth Toxicology and Mutagenesismedicine.medical_treatmentChinese hamster ovary cellPropoxurBiologyPirimicarbPollutionchemistry.chemical_compoundchemistryBiochemistrymedicineEnvironmental ChemistryMTT assayCytotoxicityToxicological & Environmental Chemistry
researchProduct

Novel examples of the N-methyl effect on cyclisations of N-Boc derivatives of amino alcohols. A theoretical study

2004

New examples of the N-methyl effect on the cyclisation of N-tert-butoxycarbonyl derivatives of amino alcohols are reported. Ab initio studies for the displacement step with formation of the five-membered heterocycle indicate that the increase of the nucleophile character of the carbonyl oxygen of the carbamate group with the N-methyl substitution is responsible for the acceleration of the cyclisation step.

CarbamateNucleophileStereochemistryChemistrymedicine.medical_treatmentOrganic ChemistryDrug DiscoveryThorpe–Ingold effectAb initiomedicineBiochemistryTetrahedron
researchProduct

EFFECTS OF THIOBENCARB HERBICIDE TO AN ALGA (NANNOCHLORIS OCULATA) AND THE CLADOCERAN (DAPHNIA MAGNA)

2001

Chronic toxicity studies were conducted with an algae (Nannochloris oculata) and the cladoceran (Daphnia magna) to determine their relative sensitivities to the thiocarbamate herbicide thiobencarb (S-4-chlorobenzyl diethylthiocarbamate). Most of the algal populations were initially affected by exposure to the herbicide. Thiobencarb concentrations higher than 0.5 mg/L significantly reduced algal densities after 24-h exposure. The 24-h static EC50 in D. magna was 3.01 mg/L. The sublethal effects of 0.3, 0.37, 0.5, 0.75, and 1.5 mg/L of thiobencarb concentrations on the survival, reproduction, and growth of D. magna were monitored for 21 days. The parameters used to determined the effect of th…

CarbamateTime Factorsmedicine.medical_treatmentDaphnia magnaBranchiopodaSensitivity and SpecificityRandom AllocationAnimal scienceChlorophytaThiocarbamatesBotanymedicineAnimalsEcotoxicologyChronic toxicityreproductive and urinary physiologyEC50Population DensityDose-Response Relationship DrugbiologyHerbicidesfungiGeneral MedicinePesticidebiology.organism_classificationSurvival AnalysisPollutionFertilityDaphniaCladoceraFood ScienceJournal of Environmental Science and Health, Part B
researchProduct