Search results for "chemical and pharmacologic phenomena"

showing 10 items of 616 documents

Switch between tyrosinase and catecholoxidase activity of scorpion hemocyanin by allosteric effectors

2008

AbstractPhenoloxidases and hemocyanins have similar type 3 copper centers although they perform different functions. Hemocyanins are oxygen carriers, while phenoloxidases (tyrosinase/catecholoxidase) catalyze the initial step in melanin synthesis. Tyrosinases catalyze two subsequent reactions, whereas catecholoxidases catalyze only the second one. Recent results indicate that hemocyanins can also function as phenoloxidases and here we show for the first time that hemocyanin can be converted to phenoloxidase. Furthermore, its substrate specificity can be switched between catecholoxidase and tyrosinase activity depending on effectors such as hydroxymethyl-aminomethan (Tris) and Mg2+-ions. Thi…

TrisStereochemistrymedicine.medical_treatmentTyrosinaseDopamineAllosteric regulationActivated hemocyaninBiophysicsMagnesium ChlorideTyramineType 3 copper proteinchemical and pharmacologic phenomenaBiochemistryCatalysisSubstrate SpecificityScorpionschemistry.chemical_compoundEnzyme activatorAllosteric RegulationStructural BiologyHemolymphHemolymphGeneticsmedicineAnimalsCatechol oxidaseMolecular BiologyScorpion Pandinus imperatorbiologyMonophenol MonooxygenaseSpectrum AnalysisActive siteCatecholoxidaseHemocyaninCell BiologyEnzyme ActivationchemistryBiochemistryHemocyaninsbiology.proteinTyrosinaseCatechol OxidaseFEBS Letters
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Mycobacterium tuberculosis Immune Response in Patients With Immune-Mediated Inflammatory Disease

2021

Subjects with immune-mediated inflammatory diseases (IMID), such as rheumatoid arthritis (RA), have an intrinsic higher probability to develop active-tuberculosis (TB) compared to the general population. The risk ranges from 2.0 to 8.9 in RA patients not receiving therapies. According to the WHO, the RA prevalence varies between 0.3% and 1% and is more common in women and in developed countries. Therefore, the identification and treatment of TB infection (TBI) in this fragile population is important to propose the TB preventive therapy. We aimed to study the M. tuberculosis (Mtb) specific T-cell response to find immune biomarkers of Mtb burden or Mtb clearance in patients with different TB …

TuberculosisImmunologyPopulationchemical and pharmacologic phenomenaDiseaseMycobacterium tuberculosisImmune systemmedicineM. tuberculosisImmunology and AllergyCytotoxic T celleducationIFN-γCD27Original Researcheducation.field_of_studybiologybusiness.industryRC581-607bacterial infections and mycosesmedicine.diseasebiology.organism_classificationtuberculosisRheumatoid arthritisImmunologyTumor necrosis factor alphaImmunologic diseases. Allergybusinessimmune-mediated inflammatory disease
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Plasmacytoid dendritic cells are inefficient in activation of human regulatory T cells

2011

BACKGROUND: Dendritic cells (DC) play a key role in initiation and regulation of immune responses. Plasmacytoid DC (pDC), a small subset of DC, characterized as type-I interferon producing cells, are critically involved in anti-viral immune responses, but also mediate tolerance by induction of regulatory T cells (Treg). In this study, we compared the capacity of human pDC and conventional DC (cDC) to modulate T cell activity in presence of Foxp3(+) Treg. PRINCIPAL FINDINGS: In coculture of T effector cells (Teff) and Treg, activated cDC overcome Treg anergy, abrogate their suppressive function and induce Teff proliferation. In contrast, pDC do not break Treg anergy but induce Teff prolifera…

Tumor ImmunologyT cellImmune CellsImmunology610 Medizinlcsh:MedicineAntigen-Presenting Cellschemical and pharmacologic phenomenaAutoimmunityBiologyLymphocyte ActivationT-Lymphocytes RegulatoryFlow cytometryImmunomodulationImmune systemInterferonNeutralization Tests610 Medical sciencesmedicineCytotoxic T cellHumanslcsh:ScienceBiologyImmune ResponseCell ProliferationMultidisciplinarymedicine.diagnostic_testCell growthT Cellslcsh:RFOXP3hemic and immune systemsForkhead Transcription FactorsDendritic CellsImmunologic SubspecialtiesCoculture TechniquesCell biologymedicine.anatomical_structureLymphocyte activationCytokinesMedicinelcsh:QClinical ImmunologyInflammation Mediatorsmedicine.drugResearch Article
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dsRNA induces apoptosis through an atypical death complex associating TLR3 to caspase-8

2012

Toll-like receptor 3 (TLR3) is a pattern-recognition receptor known to initiate an innate immune response when stimulated by double-stranded RNA (dsRNA). Components of TLR3 signaling, including TIR domain-containing adapter inducing IFN-α (TRIF), have been demonstrated to contribute to dsRNA-induced cell death through caspase-8 and receptor interacting protein (RIP)1 in various human cancer cells. We provide here a detailed analysis of the caspase-8 activating machinery triggered in response to Poly(I:C) dsRNA. Engagement of TLR3 by dsRNA in both type I and type II lung cancer cells induces the formation of an atypical caspase-8-containing complex that is devoid of classical death receptors…

Ubiquitin-Protein LigasesvirusesApoptosischemical and pharmacologic phenomenaInhibitor of Apoptosis ProteinsCell Line TumorHumansFADDMolecular BiologyRNA Double-StrandedDeath domainCaspase 8Original PaperbiologyUbiquitinationRNA-Binding Proteinshemic and immune systemsMDA5Cell BiologyTNF Receptor-Associated Factor 2Fas receptorTRADDBaculoviral IAP Repeat-Containing 3 ProteinTNF Receptor-Associated Death Domain ProteinToll-Like Receptor 3Cell biologyNuclear Pore Complex ProteinsUbiquitin ligase complexDeath-inducing signaling complexTLR3biology.proteinSignal TransductionCell Death & Differentiation
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Corporate social responsibility and managerial compensation: further evidence from spanish listed companies

2021

Ongoing regulatory efforts aim to link managerial compensation with a firm’s performance. However, little is known about whether and how Corporate Social Responsibility (CSR) goals are considered in the design of the managerial compensation scheme. This paper addresses this research question by analyzing a sample of Spanish listed firms for the period spanning 2013–2018. The outcomes of the regressions suggest that there is a positive relationship between CSR and the managerial compensation, but this relationship is significant only with lower levels of CSR. The study also reveals that CSR is positively associated with the proportion of equity-based compensation and, therefore, negatively a…

Value (ethics)media_common.quotation_subjectGeography Planning and DevelopmentTJ807-830Accountingchemical and pharmacologic phenomenaManagement Monitoring Policy and LawTD194-195:CIENCIAS ECONÓMICAS [UNESCO]Renewable energy sources0502 economics and businessGE1-350Research questionmedia_common050208 financeExecutive compensationcorporate social responsibilityEnvironmental effects of industries and plantsRenewable Energy Sustainability and the Environmentbusiness.industryCompensation (psychology)Corporate governance05 social sciencesEquity (finance)UNESCO::CIENCIAS ECONÓMICASBuilding and Constructionceo compensationcompensation structureCEO compensationmanagerial compensationEnvironmental sciencesCashCorporate social responsibilitybusinessexecutive compensation050203 business & management
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Foxp3 and gata3 polymorphisms, vitamin d3 and multiple sclerosis

2021

Background: Regulatory T cells (Tregs) alterations have been implicated in the pathogenesis of Multiple Sclerosis (MS). Recently, a crucial role of the X-Linked Forkhead Box P3 (FoxP3) for the development and the stability of Tregs has emerged, and FOXP3 gene polymorphisms have been associated with the susceptibility to autoimmune diseases. The expression of Foxp3 in Tregs is regulated by the transcription factor GATA binding-protein 3 (GATA3) and vitamin D3. The aim of this retrospective case-control study was to investigate the potential association between FOXP3 and GATA3 genetic variants, Vitamin D3, and MS risk. Methods: We analyzed two polymorphisms in the FOXP3 gene (rs3761547 and rs…

VitaminFOXP3chemical and pharmacologic phenomenaSingle-nucleotide polymorphismArticlelcsh:RC321-571Multiple sclerosis03 medical and health scienceschemistry.chemical_compound0302 clinical medicineGeneticPolymorphism (computer science)GATA3Vitamin D and neurologymedicineAlleleVitamin Dlcsh:Neurosciences. Biological psychiatry. Neuropsychiatry030304 developmental biology0303 health sciencesbusiness.industryGeneral NeuroscienceMultiple sclerosisGATA3FOXP3hemic and immune systemsmedicine.diseasechemistryImmunologybusinessPolymorphisms030217 neurology & neurosurgery
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UNDERSTANDING OF REACTIONAL SEQUENCES AND LIMITING STAGES DURING TRICALCIUM ALUMINATE HYDRATION WITH AND WITHOUT GYPSUM.

2007

International audience; The tricalcium aluminate reacts very quickly with water to form calcium hydroaluminates while the addition of calcium sulphate, leads to the formation of ettringite, with a slower process. The systematic study of the systems: “C3A” and “C3A-sulphate” by isothermal microcalorimetry and a follow up of ionic concentrations of diluted system suspensions made it possible to understand the sequence of the reactions and the limiting stages in both systems. In all cases, as it is in contact with the solution, the C3A dissolves what leads to the instantaneous precipitation of a certain quantity of calcium hydroaluminate. In case of only C3A hydration, there is then a decrease…

[CHIM.MATE] Chemical Sciences/Material chemistry[ CHIM.MATE ] Chemical Sciences/Material chemistrychemical and pharmacologic phenomena[CHIM.MATE]Chemical Sciences/Material chemistry
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Dacarbazine mediate antimelanoma effects via NK cells.

2013

International audience; Melanoma is a highly chemoresistant and metastatic tumor that, in the absence of BRAF mutations, is generally treated with the alkylating agent dacarbazine (DTIC). We discovered that DTIC upregulates the expression of NKG2D ligands on tumor cells, leading to the activation of natural killer (NK) and CD8(+) T cells. These observations underscore the immunogenic properties of DTIC and provide a rationale to combine DTIC with immunotherapeutic agents.

[SDV.IMM] Life Sciences [q-bio]/ImmunologyDacarbazineImmunologyNkg2d ligandsTumor cellschemical and pharmacologic phenomenadacarbazineNK cellsMetastatic tumorNKG2DmedicinemelanomaImmunology and Allergy[ SDV.IMM ] Life Sciences [q-bio]/ImmunologyB16Author's Viewbusiness.industryMelanomamedicine.diseaseNKG2D3. Good healthOncologyImmunologyCancer research[SDV.IMM]Life Sciences [q-bio]/ImmunologybusinessCD8medicine.drug
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Unveiling the Different Reactivity of Bent and Linear Three-Atom-Components Participating in [3 + 2] Cycloaddition Reactions

2021

The reactivity of a series of pairs of bent and linear three-atom-component (B-TACs and L-TACs) participating in [3 + 2] cycloaddition (32CA) reactions towards ethylene and electrophilic dicyanoethylene (DCE) have been studied within the Molecular Electron Density Theory. While the pseudodiradical structure of B-TACs changes to that of pseudoradical or carbenoid L-TACs upon dehydrogenation, zwitterionic B-TACs remain unchanged. Conceptual Density Functional Theory (CDFT) indices characterize five of the nine TACs as strong nucleophiles participating in polar reactions towards electrophilic ethylenes. The activation energies of the 32CA reactions with electrophilic DCE range from 0.5 to 22.0…

analytical_chemistry[3 + 2] cycloaddition reactionsOrganic chemistrychemical and pharmacologic phenomena010402 general chemistry01 natural sciencesQD241-441stomatognathic systemNucleophileComputational chemistrySingle bondReactivity (chemistry)skin and connective tissue diseasesCarbenoid010405 organic chemistryChemistrymolecular electron density theoryRegioselectivity16. Peace & justiceCycloaddition0104 chemical sciencesreactivitystomatognathic diseasesbent and linear three-atom-componentsregioselectivityElectrophileDensity functional theoryOrganics
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Extracellular Vesicles and Tumor-Immune Escape: Biological Functions and Clinical Perspectives

2020

The modulation of the immune system is one of the hallmarks of cancer. It is now widely described that cancer cells are able to evade the immune response and thus establish immune tolerance. The exploration of the mechanisms underlying this ability of cancer cells has always attracted the scientific community and is the basis for the development of new promising cancer therapies. Recent evidence has highlighted how extracellular vesicles (EVs) represent a mechanism by which cancer cells promote immune escape by inducing phenotypic changes on different immune cell populations. In this review, we will discuss the recent findings on the role of tumor-derived extracellular vesicles (TEVs) in re…

animal diseasesCellProgrammed Cell Death 1 Receptorchemical and pharmacologic phenomenapd-1/pd-l1 axisReviewBiologyCatalysisImmune toleranceInorganic Chemistrylcsh:ChemistryExtracellular VesiclesImmune systemNeoplasmsmedicineImmune ToleranceAnimalsHumansPhysical and Theoretical ChemistryMolecular Biologylcsh:QH301-705.5SpectroscopyMechanism (biology)Organic ChemistryCancerGeneral Medicinebiochemical phenomena metabolism and nutritionimmune checkpointsmedicine.diseasePhenotypeComputer Science ApplicationsCell biologyextracellular vesicles (evs) cancer immune toleranceThe Hallmarks of Cancermedicine.anatomical_structurelcsh:Biology (General)lcsh:QD1-999Cancer cellbacteriaTumor EscapeImmune checkpointImmunotherapyextracellular vesicles (EVs)cancer immune toleranceInternational Journal of Molecular Sciences
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