Search results for "cycles"

showing 10 items of 306 documents

Chemostratigraphy, magnetostratigraphy, chronology, palaeoenvironments and correlations.

2013

4 pages

Paleomagnetismglaciationcycles[ SDU.STU.ST ] Sciences of the Universe [physics]/Earth Sciences/StratigraphyCarbonCretaceousOxygenQuaternaryPleistoceneValanginianpaleoclimate[SDU.STU.ST] Sciences of the Universe [physics]/Earth Sciences/StratigraphyWeissert excursionisotopes
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Parasite specificity in Podarcis bocagei and P. carbonelli (Lacertidae) from NW Portugal: a host-parasite history

2015

Host parasite specificity is related to several factors including the type of life cycle of the parasite, the habitat occupied by both parasites and hosts, and the food habits of the hosts. In this work, gastrointestinal helminths in two congeneric lacertid lizards, Podarcis bocagei and Podarcis carbonelli living in sintopy, have been analysed. Out of four helminth species found, three of them, the trematode Brachylaima sp., the cestode Oochoristica gallica and the nematode Skrjabinelazia hoffmanni, have indirect life cycles while the nematode Spauligodon carbonelli has a direct life cycle. Heteroxenous helminths showed low host specificity whereas S. carbonelli may be placed at an intermed…

Parasitic life cyclesbiologyEcologyZoologybiology.organism_classificationPodarcis bocageiNematodeparasitic diseasesPodarcis carbonelliHelminthsParasite hostingLacertidaeGeneral Materials ScienceBrachylaimaBasic and Applied Herpetology
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Heterocyclic Scaffolds for the Treatment of Alzheimer's Disease

2016

Background: The treatment and diagnosis of Alzheimer’s Disease (AD) are two of the most urgent goals for research around the world. The cognitive decline is generally associated with the elevated levels of extracellular senile plaques, intracellular neurofibril- lary tangles (NFTs), and with a progressive shutdown of the cholinergic basal forebrain neurons transmission. Even if several key targets are under fervent investigation in the cure of AD, till now, the only approved therapeutic strategy is the treatment of symptoms by using cholinesterases inhibitors. It has been demonstrated that both acetylcholinesterase (AChE) and butyrylcholinesterase (BuChE) enzymes are not only responsible of…

Pathologymedicine.medical_specialtyTau proteinDisease010402 general chemistry01 natural scienceschemistry.chemical_compoundAlzheimer DiseaseHeterocyclic CompoundsDrug DiscoverymedicineAnimalsHumansSenile plaquesCognitive declineButyrylcholinesterasePharmacologybiologyMolecular Structure010405 organic chemistryChemistryAcetylcholinesterase0104 chemical sciencesbiology.proteinCholinergicNeuroscienceAmyloid precursor protein secretaseAlzheimer’s disease amyloid-peptide secretase acetylcholinesterase tau protein heterocycles
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Fluorinated Heterocyclic Compounds. A Photochemical Approach to a Synthesis of Polyfluoroaryl-1,2,4-triazoles.

2005

The reaction of some fluorinated 1,2,4-oxadiazoles in the presence of methylamine or propylamine has been investigated. The irradiation in methanol or acetonitrile leads with acceptable yields to the corresponding fluorinated 1- methyl- or 1-propyl-1,2,4-triazole.

PharmacologyFLUORO HETEROCYCLESMethylamineOrganic ChemistryQUINAZOLIN-4-ONES124-Triazole124-OXADIAZOLESPropylamineSettore CHIM/06 - Chimica OrganicaGeneral MedicineEXPEDIENT ROUTEPhotochemistryMedicinal chemistryAnalytical Chemistrychemistry.chemical_compound124-TRIAZOLESchemistryTriazole derivativesOrganic chemistry5-MEMBERED HETEROCYCLESIrradiationMethanolAcetonitrilePHOTOINDUCED MOLECULAR-REARRANGEMENTSChemInform
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Fluorinated Heterocyclic Compounds. A Photochemical Approach to a Synthesis of Fluorinated Quinazolin-4-ones

2004

An efficient and generalized photochemical methodology for the preparation of fluorinated quinazolin-4-ones is described. Depending on the starting substrate, quinazolin-4-ones bearing a perfluoroalkyl- or perfluoroaryl- substituent in position 2 or fluorine atoms on any positions of the benzo-fused moiety can easily be obtained. 5-Aryl-3-perfluoroalkylpentafluorophenyl- or 5-polyfluoroaryl-3-phenyl(methyl)-1,2,4-oxadiazoles, respectively, can be considered as ideal precursors that can be transformed into the target quinazolin-4-ones by irradiation in the presence of triethylamine (TEA) (at λ = 313 nm) or pyrene (at λ = 365 nm) in dry methanol or acetonitrile as solvent. Some mechanistic co…

PharmacologyFLUORO HETEROCYCLESOrganic Chemistrychemistry.chemical_elementSettore CHIM/06 - Chimica OrganicaGeneral MedicinePhotochemistryPhotoinduced electron transferAnalytical ChemistrySolventchemistry.chemical_compoundchemistryFluorinePyreneMoietyMethanolAcetonitrileTriethylaminePHOTOINDUCED MOLECULAR-REARRANGEMENTSHETEROCYCLES
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Photochemistry of 1,2,4-oxadiazoles. A DFT study on photoinduced competitive rearrangements of 3-amino- and 3-N-methylamino-5-perfluoroalkyl-1,2,4-ox…

2006

The photoinduced competitive rearrangements of 5-perfluoroalkyl-3-amino(N-alkylamino)-1,2,4-oxadia- zoles have been investigated by DFT calculations and UV-vis spectroscopy. The observed product selectivity depends on the number of hydrogen atoms present in the amino moiety and involves two or three possible routes: (i) ring contraction-ring expansion (RCRE), (ii) internal-cyclization isomerization (ICI), or (iii) C(3)-N(2) migration-nucleophilic attack-cyclization (MNAC). UV absorption and fluorescence spectra of the reactants, and vertical excitation energy values, calculated by time dependent DFT, support the involvement of a neutral singlet excited state in the photoexcitation process. …

PhotochemistryUltraviolet RaysFluorescence spectrometryReaction intermediatePhotochemistryDENSITY-FUNCTIONAL THEORYSinglet stateHUMAN 5-HT1B RECEPTORBASIS-SETSOxadiazolesRING-PHOTOISOMERIZATIONMolecular StructureChemistryOrganic ChemistryEXPEDIENT ROUTETautomerTransition statePhotoexcitationMOLECULAR-ORBITAL METHODSModels ChemicalLUORINATED HETEROCYCLIC-COMPOUNDSAROMATICITY INDEXExcited state5-MEMBERED HETEROCYCLESEXCITATION-ENERGIESIsomerization
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FUSED NITROGEN HETEROCYCLES AS PROMISING SMALL MOLECULES FOR THE TREATMENT OF CANCER

2020

Photodynamic therapy photosensitizing nitrogen heterocycles CDK inhibitors antiproliferative activitySettore CHIM/08 - Chimica Farmaceutica
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A 16 channel high resolution (<11 ps RMS) Time-to-Digital Converter in a Field Programmable Gate Array

2012

A 16-channel Time-to-Digital Converter (TDC) was implemented in a general purpose Field-Programmable Gate Array (FPGA). The fine time calculations are achieved by using the dedicated carry-chain lines. The coarse counter defines the coarse time stamp. In order to overcome the negative effects of temperature and power supply dependency bin-by-bin calibration is applied. The time interval measurements are done using 2 channels. The time resolution of channels are calculated for 1 clock cycle and a minimum of 10.3 ps RMS on two channels, yielding 7.3 ps RMS (10.3 ps/√2) on a single channel is achieved.

PhysicsCycles per instructionbusiness.industryElectrical engineeringPower (physics)Time-to-digital converterOpticsGate arrayCalibrationTimestampbusinessField-programmable gate arrayInstrumentationMathematical PhysicsCommunication channelJournal of Instrumentation
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Nilpotence of orbits under monodromy and the length of Melnikov functions

2021

Abstract Let F ∈ ℂ [ x , y ] be a polynomial, γ ( z ) ∈ π 1 ( F − 1 ( z ) ) a non-trivial cycle in a generic fiber of F and let ω be a polynomial 1-form, thus defining a polynomial deformation d F + e ω = 0 of the integrable foliation given by F . We study different invariants: the orbit depth k , the nilpotence class n , the derivative length d associated with the couple ( F , γ ) . These invariants bind the length l of the first nonzero Melnikov function of the deformation d F + e ω along γ . We analyze the variation of the aforementioned invariants in a simple but informative example, in which the polynomial F is defined by a product of four lines. We study as well the relation of this b…

PhysicsPure mathematicsSequencePolynomialConjectureMelnikov functionAbelian integrals010102 general mathematicsStatistical and Nonlinear PhysicsIterated integralsCondensed Matter Physics01 natural sciencesNilpotence classFoliationDisplacement functionLimit cyclesMonodromySimple (abstract algebra)[MATH.MATH-MP]Mathematics [math]/Mathematical Physics [math-ph]Product (mathematics)0103 physical sciences010307 mathematical physics0101 mathematicsOrbit (control theory)ComputingMilieux_MISCELLANEOUS
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rac-(E,trans)-4-Bromo-10,10-dimethyl-9,11-dioxabicyclo[6.3.0]undec-4-ene

2020

In the title compound, a cyclooctene ring in a twist-boat conformation and a dioxolane ring with a distorted envelope conformation are annulated in a trans configuration. Alternating strands of single enantiomers build up the crystal. Within the strands, the molecules are connected by weak C—H...O hydrogen bonds.

Physics::Biological PhysicsQuantitative Biology::Biomoleculescrystal structureheterocyclesChemistrybrominelcsh:QD901-999Crystal structuremedium-sized ringlcsh:CrystallographyMedicinal chemistryEne reactionIUCrData
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