Search results for "magnetic resonance spectroscopy"

showing 10 items of 1362 documents

Reaction of complex ligands: Part 95. Chromium tricarbonyl complexes of polysubstituted naphthohydroquinones: regioselective synthesis via [3+2+1]-be…

2003

Abstract A series of polysubstituted naphthohydroquinoid tricarbonyl chromium complexes were prepared by chromium mediated [3+2+1]-benzannulation of Fischer-type carbene complexes with alkynes. The kinetics and the thermodynamic data of the η6-η6-haptotropic rearrangements were investigated by in-situ NMR spectroscopy. The free activation energies ΔG# range from 23 to 26 kcal mol−1 and only slightly depend on the bulk and the donor/acceptor properties of the substituents. Equilibrium of metal migration was observed for naphthohydroquinone complexes bearing methoxy substituents at the non-hyroquinoid ring (ring A). In complexes bearing methyl groups or only hydrogen substituents at ring A th…

ChemistryStereochemistryOrganic ChemistryDiastereomerRegioselectivityHexafluorobenzenechemistry.chemical_elementNuclear magnetic resonance spectroscopyRing (chemistry)BiochemistryMedicinal chemistryInorganic Chemistrychemistry.chemical_compoundChromiumReaction rate constantMaterials ChemistryPhysical and Theoretical ChemistryCarbeneJournal of Organometallic Chemistry
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Über polygermane

1986

Abstract The synthesis of GePh4 and Ge2Ph6 by Grignard reaction in THF or ether/toluene leads to the by-products Ge3Ph8 (up to 11%) and Ge4Ph10 (up to 18%) which is dependant on using an excess of Mg. A quantitative analysis of the resulting products by HPLC and a semipreparative separation by column, flash, and HPL chromatography is described. The crystal structures of Ge3Ph8 (R = 0.075) and Ge4Ph10 · 2C6H6 (R = 0.054) have been determined. Ge4Ph10 has Ci symmetry and both chain conformations are well staggered (49–70° for Ge3Ph8, 53–66° for Ge4Ph10). The GeGe distances and GeGeGe angles are 244 pm and 121° (Ge3Ph8), and 246 pm and 118° (Ge4Ph10).

ChemistryStereochemistryOrganic ChemistryGrignard reactionEtherNuclear magnetic resonance spectroscopyCrystal structureBiochemistryMedicinal chemistryTolueneHigh-performance liquid chromatographyInorganic Chemistrychemistry.chemical_compoundX-ray crystallographyMaterials ChemistryMoleculePhysical and Theoretical ChemistryJournal of Organometallic Chemistry
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Interaction of methylmercury(II) with the bifunctional ligand o-diphenylphosphinobenzoate, dpb. Synthesis and characterization of [(dpb)HgMe] and [(d…

1998

Abstract The complex [(dpb)HgMe] (1) is obtained by reaction of MeHg(OH) with o-diphenylphosphinobenzoic acid (Hdpb); alternatively the solvate [(dpb)HgMe] · 0.5H2O · 0.5C5H5N (1bis) can be prepared by reacting MeHgCl with Hdpb and pyridine. The derivative [(dpbo)HgMe] (2), where dpbo is o-diphenylphosphinoxidebenzoate, is formed by reaction of 1 or 1bis solutions with atmospheric oxygen. Crystal data for 1bis: monoclinic, space group P2/n, a=10.413(4), b=9.831(3), c=20.674(3) A, β=102.51(3)°, Z=2. Crystal data for 2: triclinic, space group P1, a=11.535(2), b=12.897(5), c=13.275(7) A, α=88.31(4), β=73.65(4), γ=85.27(4)°, Z=2. In 1bis the mercury atom displays a distorted linear fashion, bei…

ChemistryStereochemistryOrganic ChemistryNuclear magnetic resonance spectroscopyCrystal structureTriclinic crystal systemBiochemistryInorganic Chemistrychemistry.chemical_compoundCrystallographyPyridineMaterials ChemistryMoietyMoleculePhysical and Theoretical ChemistryBifunctionalMethyl groupJournal of Organometallic Chemistry
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Metal ion complexation by tetraester derivatives of bridged calix [4] arenes

1992

A series of bridged calix [4] arenes (5–10 methylene groups in the bridge) were synthesized and transformed into their tetraester derivatives by reaction with ethyl bromoacetate. The stability constants for complexes of the tetraester derivatives with sodium, potassium and silver cations, determined in methanol by spectroscopic or potentiometric techniques, show a drastic decrease (more than 105 for Na +) for the shorter methylene chains. 1H NMR studies demonstrate a conformational rearrangement of the calixarene part to fourfold symmetry to be necessary for the complexation of a cation, which is prevented by the shorter chains. This is further confirmed by the X-ray structure of a tetraest…

ChemistryStereochemistryOrganic ChemistryPotentiometric titrationNuclear magnetic resonance spectroscopyCrystal structureMedicinal chemistryEthyl bromoacetatechemistry.chemical_compoundCalixareneProton NMRPhysical and Theoretical ChemistryMethyleneMonoclinic crystal systemJournal of Physical Organic Chemistry
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Dynamic formation of hybrid peptidic capsules by chiral self-sorting and self-assembly.

2014

Owing to their versatility and biocompatibility, peptide-based self-assembled structures constitute valuable targets for complex functional designs. It is now shown that artificial capsules based on β-barrel binding motifs can be obtained by means of dynamic covalent chemistry (DCC) and self-assembly. Short peptides (up to tetrapeptides) are reversibly attached to resorcinarene scaffolds. Peptidic capsules are thus selectively formed in either a heterochiral or a homochiral way by simultaneous and spontaneous processes, involving chiral sorting, tautomerization, diastereoselective induction of inherent chirality, and chiral self-assembly. Self-assembly is shown to direct the regioselectivit…

ChemistryStereochemistryProton Magnetic Resonance SpectroscopySupramolecular chemistryDynamic covalent chemistryRegioselectivityStereoisomerismGeneral ChemistryGeneral MedicineResorcinareneInherent chiralityTautomerCatalysisSelf-assemblyChirality (chemistry)Peptidesta116Angewandte Chemie (International ed. in English)
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Ferrocenyl-functionalized tetranuclear gold(I) and gold(I)-copper(I) complexes based on tridentate phosphanes

2013

Tetranuclear AuI–FeII dimetallic and AuI–CuI–FeII trimetallic complexes bearing ferrocenyl (Fc) groups have been assembled by using two triphosphane ligands, namely, (PPh2CH2)2PPh (dpmp) and (PPh2)3CH (tppm). The compositions and structural type of the clusters are dependent on the stereochemistry of the P donor ligands. The complexes [tppmAu3Cu(C2R)3]PF6 [R = Fc (1) and 4-C6H4-Fc (2)] adopt a trigonal pyramidal {Au3Cu} arrangement of the coordinating metal core, whereas for the compounds with the linear triphosphane [Au4(dpmp)2(C2R)2](PF6)2 [R = Fc (3) and 4-C6H4-Fc (4)], a planar rhomboidal {Au4} framework was found. Clusters 1–4 were characterized by NMR spectroscopy and ESI-MS measureme…

ChemistryStereochemistrychemistry.chemical_elementTrigonal pyramidal molecular geometryNuclear magnetic resonance spectroscopyElectrochemistryRedoxCopperInorganic ChemistryMetalElectron transferchemistry.chemical_compoundCrystallographyTriphosphanevisual_artvisual_art.visual_art_mediumta116European journal of inorganic chemistry
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Organoelement derivatives of steroids: synthesis and structural characterization of diorganotin chloride adducts of hormones

1986

Abstract Ten new diorganotin dichloride adducts of hormones of the type R 2 SnCl 2 ·2L [where R = Me, Et, n-Bu, Oct and Ph; L = 4-androsten-17s-ol-3-one ( A ); 5-androsten-3s-ol-17-one ( B ); 4-androsten-17α- methyl-17s-ol-3-one ( C ) and 3,17-dihydroxy-5- pregnene-20-one ( D )] have been prepared and characterized at 297 K and 223 K. Spectroscopic measurements (IR; Raman; 1 H, 13 C, 119 Sn NMR) suggest the dissociation or fast ligand exchange in solution at 297 K. Hexa-coordinated adducts with bonding through carbonyl oxygen and trans -R groups in octahedral geometry are formulated at 223 K.

ChemistryStereochemistrymedicine.medical_treatmentchemistry.chemical_elementNuclear magnetic resonance spectroscopyChlorideOxygenDissociation (chemistry)AdductSteroidInorganic Chemistrysymbols.namesakeOctahedral molecular geometryMaterials ChemistrymedicinesymbolsPhysical and Theoretical ChemistryRaman spectroscopymedicine.drugInorganica Chimica Acta
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Measurements of Tumor Blood Flow Using Intraperitoneal Deuterium and 2H-NMR Spectroscopy

1992

Tumors usually have a sparse, disorganized, and inefficient vascular network that leaves a large fraction of the tumor cells in an oxygen deprived and hostile metabolic microenvironment. Hence tumor blood flow, or more correctly nutritive perfusion, has important interactions with treatment efficacy. For example, hypoxic tumor cells, which occur in tumors with low blood flow, are less susceptible to radiation and are probably responsible for most radiation treatment failures (Adams, 1981). Similarly, cytotoxic drug delivery could be predicted by blood flow measurements, with clear implications regarding the expected success of chemotherapy. Thus, the ability to conveniently measure tumor bl…

ChemotherapyHypoxic tumorDeuteriumVascular networkCytotoxic drugChemistrymedicine.medical_treatmentmedicineAnalytical chemistryCancer researchNuclear magnetic resonance spectroscopyBlood flowPerfusion
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Sesterterpenes and macrolide derivatives from the endophytic fungus Aplosporella javeedii.

2020

Abstract Five sesterterpenes (1–5) including two new compounds (1 and 2), as well as a new (6) and a known macrolide (7) were isolated from the endophytic fungus Aplosporella javeedii. The structures of the new compounds were elucidated by analysis of their 1D and 2D NMR and HRMS data as well as by comparison with the literature. Compound 4 and its acetyl derivatives 4a, 4b, 4c which were prepared by acetylation of 4 exhibited moderate cytotoxicity against the mouse lymphoma cell line L5178Y with IC50 values ranging from 6.2 to 12.8 μM, respectively. Moreover, 4a and 4c exhibited also cytotoxicity against human leukemia (Jurkat J16) and lymphoma (Ramos) cell lines. Compound 7 showed strong …

ChinaStaphylococcus aureusSesterterpenesAntineoplastic AgentsApoptosismedicine.disease_cause01 natural sciencesJurkat cellsSesterterpenesMiceStructure-Activity RelationshipAscomycotaCell Line TumorDrug DiscoverymedicineEndophytesAnimalsHumansCytotoxicityPharmacologyMolecular Structure010405 organic chemistryChemistryGeneral MedicineMolecular biology0104 chemical sciencesAnti-Bacterial Agents010404 medicinal & biomolecular chemistryStaphylococcus aureusCell cultureAcetylationBrassicaceaeMacrolidesAntibacterial activityTwo-dimensional nuclear magnetic resonance spectroscopyFitoterapia
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Marine Isonitriles and Their Related Compounds.

2016

Marine isonitriles represent the largest group of natural products carrying the remarkable isocyanide moiety. Together with marine isothiocyanates and formamides, which originate from the same biosynthetic pathways, they offer diverse biological activities and in spite of their exotic nature they may constitute potential lead structures for pharmaceutical development. Among other biological activities, several marine isonitriles show antimalarial, antitubercular, antifouling and antiplasmodial effects. In contrast to terrestrial isonitriles, which are mostly derived from α-amino acids, the vast majority of marine representatives are of terpenoid origin. An overview of all known marine isoni…

ChinaisothiocyanatesMagnetic Resonance SpectroscopyStereochemistrycarbonimidic dichloridesmalariaPharmaceutical ScienceReviewBiology010402 general chemistry01 natural sciencesantibioticsStructure-Activity RelationshipDrug DiscoveryOrganic chemistryHumansSeawaterPharmacology Toxicology and Pharmaceutics (miscellaneous)lcsh:QH301-705.5isonitriles010405 organic chemistryTerpenesmarine natural productsformamides0104 chemical scienceslcsh:Biology (General)Marine drugs
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