Search results for "triazol"

showing 10 items of 598 documents

1,1′-[2,3,5,6-Tetramethyl-p-phenylenebis(methyleneoxy)]di-1H-benzotriazole

2009

The complete molecule of the title compound, C(24)H(24)N(6)O(2), is generated by a crystallographic inversion centre. The benzotriazole rings form dihedral angles of 2.10 (7)° with the central aromatic ring. The crystal packing is consolidated by π-π inter-actions, with centroid-centroid distances of 3.6234 (10) Å, together with weak C-H⋯π inter-actions.

Crystalchemistry.chemical_compoundBenzotriazoleChemistryMoleculeGeneral Materials ScienceGeneral ChemistryDihedral angleCondensed Matter PhysicsBioinformaticsRing (chemistry)Organic PapersMedicinal chemistryActa Crystallographica Section E Structure Reports Online
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1-(2,3,5,6-Tetramethylbenzyloxy)-1H-benzotriazole

2009

In the title compound, C17H19N3O, the benzotriazole ring is essentially planar, with a maximum deviation of 0.0069 (15) Å. The mean plane of the benzotriazole ring forms a dihedral angle of 13.16 (4)° with the mean plane of the benzene ring. The crystal packing is stabilized by π–π stacking interactions, with a centroid–centroid distance of 3.8077 (12) Å, together with weak C—H...π interactions. Molecules are stacked along the a axis.

CrystallographyBenzotriazolebiologyPlane (geometry)StackingGeneral ChemistryDihedral angleCondensed Matter PhysicsBioinformaticsRing (chemistry)biology.organism_classificationOrganic PapersCrystalchemistry.chemical_compoundCrystallographychemistryQD901-999TetraGeneral Materials ScienceBenzeneActa Crystallographica Section E Structure Reports Online
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N-(5-Amino-1H-1,2,4-triazol-3-yl)pyridine-2-carboxamide

2013

The title compound, C8H8N6O, was obtained by the reaction of 3,5-diamino-1,2,4-triazole with ethyl 2-picolinate in a glass oven. The dihedral angles formed between the plane of the amide group and the pyridine and triazole rings are 11.8 (3) and 5.8 (3)°, respectively. In the crystal, an extensive system of classical N—H...N and N—H...O hydrogen bonds generate an infinite three-dimensional network.

CrystallographyChemistryHydrogen bondmedicine.drug_classTriazoleCarboxamideGeneral ChemistryDihedral angleCondensed Matter PhysicsBioinformaticsOrganic PapersMedicinal chemistryCrystalchemistry.chemical_compoundQD901-999AmidePyridinemedicineGeneral Materials ScienceActa Crystallographica Section E Structure Reports Online
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A C(π-hole)⋯Cl-Zn tetrel interaction driving a metal-organic supramolecular assembly

2020

A brominated pyrimidinyl triazolopyridine ligand (bptpy) forms a C(π-hole)⋯Cl-Zn tetrel interaction that plays a determining role in the formation of supramolecular layers through chain assembly in 18 membered metallacycle [(ZnCl2)2(μ-bptpy)2] crystals. Supramolecular chains are formed through C-H⋯X interactions. The observed interactions are supported by DFT calculations using model dimers. This journal is

CrystallographyChemistryLigandSupramolecular chemistryGeneral Materials ScienceTriazolopyridineGeneral ChemistryMetallacycleCondensed Matter PhysicsSupramolecular assemblyCrystEngComm 22: 6979-6982 (2020)
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Synthesis and crystal structures of two novel triazolopyridine compounds solved by local L.S. minimizations from powder diffraction data

2014

The heteroaryl-substituted triazolopyridines 3-phenyl-7-(pyrazin-2-yl)-[1,2,3]triazolo[1,5-a]pyridine (2) and 3-[6-(pyridazin-3-yl)-pyridin-2-yl]-[1,2,3]triazolo[1,5-a]pyridine (4) have been synthesized and characterized (by HRMS, IR,1H and13C NMR, XRPD, melting point). The crystal structures have been solved from laboratory powder X-ray diffraction data with the direct-space strategy TALP for molecular compounds based on fast local least-squares minimizations. The crystal structure confirmed the formation of the tridentate compound4from a ring chain isomerization process. The almost planar arrangement of atoms in both the structures favors the presence of intermolecularπ–πinteractions, alt…

CrystallographyRadiationMaterials scienceGeneral Materials ScienceTriazolopyridineCrystal structureCondensed Matter PhysicsInstrumentationPowder diffractionPowder Diffraction
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1-[2-(2,4-Dichloro­phenyl)­pent­yl]-1H-1,2,4-triazole

2009

The title compound, C13H15Cl2N3, also known as penconazole, crystallizes as a racemate. The dihedral angle between the benzene and triazole rings is 24.96 (13)°. In the crystal structure, molecules are linked into chains running parallel to the c axis by intermolecular C—H...N hydrogen-bonding interactions.

CrystallographyTriazole124-TriazoleGeneral ChemistryCrystal structureDihedral angleCondensed Matter PhysicsBioinformaticsMedicinal chemistryOrganic Paperschemistry.chemical_compoundchemistryQD901-999General Materials ScienceBenzeneActa Crystallographica Section E: Structure Reports Online
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New polynuclear 4,4ˈ-bis-1,2,4-triazole Fe(II) spin crossover compounds

2001

L'interet porte aux materiaux moleculaires du Fe(II) presentant une transition entre un etat haut-spin (HS, S = 2) et un etat bas-spin (LS, S = 0), sous l'effet d'une variation de temperature, de pression ou d'une irradiation lumineuse, n'a cesse de croitre au cours de ces dix dernieres annees [1-4]. La famille des composes du Fe(II) a base de derives du 1,2,4-triazole substitues par un groupe R sur l'azote 4 a ete tres etudiee pour ses proprietes de transition de spin (TS), qui pourraient permettre des applications en electronique moleculaire [5-15, 29, 32, 36, 37]. Nous avons recemment presente le premier compose a TS possedant une structure tridimensionnelle (figure 2). Ce compose de for…

Crystallographychemistry.chemical_compoundChemistryStereochemistrySpin crossoverTriazole derivatives124-TriazoleGeneral ChemistryComptes Rendus de l'Académie des Sciences - Series IIC - Chemistry
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Nanowire iron(III) coordination polymer based on 1,2,4-triazolo[1,5-a]pyrimidine and chloride ligands

2019

Abstract The neutral ligand 1,2,4-triazolo[1,5-a]pyrimidine (tp) has been employed to prepare a new coordination compound of Fe(III), [FeCl3(tp)2]n (1). Compound 1 was investigated by single crystal X-ray diffraction and found to be a coordination polymer forming a ladder structure based on metal–ligand interactions, while H-bonding and aromatic interactions contribute to the supramolecular self-assembly into a 3D nanostructured material. The polymeric assembly is retained also in solution, where a metallo-supramolecular polymer based on coordinative metal–ligand binding is present, as shown by dynamic light scattering (DLS) measurements. The redox properties of the Fe(III) coordination pol…

Cyclic voltammetryCoordination polymer124-Triazolo[15-a]pyrimidineSupramolecular chemistry010402 general chemistry01 natural sciencesCoordination complexInorganic Chemistrychemistry.chemical_compoundDynamic light scatteringSolid state structureMaterials ChemistryPhysical and Theoretical Chemistrychemistry.chemical_classification010405 organic chemistryLigandSelf-assemblyPolymer0104 chemical sciencesCrystallographyScanning probe microscopychemistrySettore CHIM/03 - Chimica Generale E Inorganica124-Triazolo[15-a]pyrimidine Solid state structure Cyclic voltammetry Self-assembly Scanning probe microscopySelf-assemblySingle crystalPolyhedron
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ω-Hetarilbutānskābes atvasinājumu iegūšana pretvēža aktivitātes noteikšanai: pieclocekļu heterocikli ar trim heteroatomiem.

2022

ω-Hetarilbutānskābes atvasinājumu iegūšana pretvēža aktivitātes noteikšanai: pieclocekļu heterocikli ar trim heteroatomiem. Fiļipčuks M., zinātniskais vadītājs Dr. chem. Kļimenkovs I. Bakalaura darbs, 37 lappuses, 35 attēli, 1 tabula, 33 literatūras avoti, 19 pielikumi. Latviešu valodā. Bakalaura darba ietvaros tika izpētītas un aprakstītas diaizvietotu pieclocekļu heterociklisko savienojumu ar trim heteroatomiem iegūšanas iespējas.

DIAIZVIETOTI 124-TRIAZOLICIKLIZĀCIJADIAZIVIETOTI OKSADIAZOLIDIACILHIDRAZĪDIĶīmija
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Cytotoxic Activity of Organotin(IV) Derivatives with Triazolopyrimidine Containing Exocyclic Oxygen Atoms

2020

In this study cytotoxicity of organotin(IV) compounds with 1,2,4-triazolo[1,5-a]pyrimidines, Me3Sn(5tpO) (1), n-Bu3Sn(5tpO) (2), Me3Sn(mtpO) (3), n-Bu3Sn(mtpO) (4), n-Bu3Sn(HtpO2) (5), Ph3Sn(HtpO2) (6) where 5HtpO = 4,5-dihydro-5-oxo-[1,2,4]triazolo-[1,5-a]pyrimidine, HmtpO = 4,7-dihydro-5-methyl-7-oxo-[1,2,4]triazolo-[1,5-a]pyrimidine, and H2tpO2 = 4,5,6,7-tetrahydro-5,7- dioxo-[1,2,4]triazolo-[1,5-a]-pyrimidine, was assessed on three different human tumor cell lines: HCT-116 (colorectal carcinoma), HepG2 (hepatocarcinoma) and MCF-7 (breast cancer). While 1 and 3 were inactive, compounds 2, 4, 5 and 6 inhibited the growth of the three tumor cell lines with IC50 values in the submicromolar …

DenticityCellPharmaceutical Science01 natural sciencesAnalytical Chemistrychemistry.chemical_compoundDrug DiscoveryOrganotin CompoundstriazolopyrimidineCytotoxicityMembrane Potential MitochondrialCytotoxinsapoptosisBiological activityHep G2 CellsG2 Phase Cell Cycle CheckpointsGene Expression Regulation Neoplasticmedicine.anatomical_structureChemistry (miscellaneous)Mitochondrial MembranesMCF-7 CellsMolecular MedicineCyclin-Dependent Kinase Inhibitor p21crystal structurein vitro anticancer activityPyrimidineCell SurvivalStereochemistryorganotin(iv)010402 general chemistryArticlelcsh:QD241-441Inhibitory Concentration 50Structure-Activity Relationshiplcsh:Organic chemistrymedicineHumansPhysical and Theoretical ChemistryMetallodrug010405 organic chemistryLigandOrganic ChemistryTriazolesHCT116 CellsapoptosiG1 Phase Cell Cycle Checkpoints0104 chemical sciencesPyrimidineschemistrymetallodrugsCell cultureApoptosisDrug DesignTumor Suppressor Protein p53Reactive Oxygen SpeciesMolecules
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