6533b821fe1ef96bd127b04f
RESEARCH PRODUCT
The Concise Guide To Pharmacology 2021/22: G Protein-Coupled Receptors
Nigel J. M. BirdsallStephen J LolaitHans-jürgen WesterPaul L. ChazotSadashiva S. KarnikSimon D. HardingCeline ValantStephen P.h. AlexanderOlivier CivelliZsolt CsabaMastgugu HoriuchiKhuraijam Dhanachandra SinghTheodore L. GoodfriendMorley D. HollenbergDuuamene NyimanuShlomo MelmedG. Enrico RovatiXavier NorelLeigh A. StoddartKlemens KaupmannRobyn MacraeNicholas D. HollidayDeborah L. SegaloffJusto P. CastañoTony NgoGordon DentJean-martin BeaulieuThomas L WilliamsAntonia CianciulliPaweł KozielewiczXaria X. LiJyrki P. KukkonenCraig A. McardleJohn D. LeePhilippe RondardSteven D. DouglasHubert VaudryKhaled A. Al-hosainiNan ChiangBernhard BettlerGiovanni TulipanoCorinne BousquetKaren J. GregoryCraig GerardRobert T. JensenStefan SchulzRithwik RamachandranRoss A. D. BathgateDeepa JonnalagaddaDavid M. ThalTakio KitazawaManisha RayBice ChiniThomas UngerMarta FumagalliJean-pierre VilardagaDonald T. WardRoger G. PertweeStefan OffermannsMarvin C. GershengornMarc ParmentierPieter TimmermansEamonn KellyYukihiko SugimotoHamiyet UnalVincenzo MitoloAlistair MathieEmma L. VealeAndrew L. GundlachAnthony P. DavenportMark T. QuinnJérôme LeprinceChrista E. MüllerGeoffrey BurnstockAkos HeinemannJacqueline R. KempRichard D. YeBernard MouillacRoger J. SummersRaul R. GainetdinovGirolamo CalòPhilip N. MurphyAmelie LuppKalyan C. TirupulaWalter G. ThomasJulien HansonAhsan HusainKatie LeachLucie H. ClappHans Bräuner-osborneGunnar SchulteKenneth E. BernsteinJean MazellaTorsten SchönebergSatoru EguchiMartin C. MichelMaria Antonietta PanaroKevin J. CattRainer K. ReinscheidHans-jürgen KreienkampWayne R. AlexanderEmanuel EscherAnne Marie O'carrollMagnus BäckLaurence J. MillerJane F. ArmstrongChiara RuzzaTrent M. WoodruffDaniel HoyerChengcan YaoMaria P. AbbracchioJohn A. PetersGary B. WillarsJean-philippe PinDavid VaudryDebbie L. HayFrançois BoulayDavide LeccaEric R. ProssnitzArthur ChristopoulosVictoria A. BlahoYasuyuki KiharaCharles KennedyChristopher SouthanLászló HunyadyPascal DournaudFernand GobeilCyril GoudetCharles N. SerhanClaes DahlgrenJörg HamannTobias LangenhanRalf JockersNicholas M. BarnesJean-louis NahonRichard L. HaugerAdam J. PawsonGareth J. SangerTung FongSusan E. LeemanElena FaccendaEdward J. FilardoValerie P. TanMarc De GasparoJi Ming WangJamie A. DaviesJerold ChunStefania CerutiTadashi InagamiRéjean CoutureKenneth A. JacobsonPatrick VanderheydenAdriaan P. IjzermanJanet J. MaguireChristopher S. Walkersubject
RMCytoplasmic and NuclearComputer scienceDatabases PharmaceuticalHumans; Ion Channels; Ligands; Receptors Cytoplasmic and Nuclear; Receptors G-Protein-Coupled; Databases Pharmaceutical; PharmacologyReceptors Cytoplasmic and NuclearIN-VITRO CHARACTERIZATIONPharmacologyLigandsIon ChannelsNORSlaw.inventionReceptors G-Protein-CoupledG-Protein-CoupledDatabases03 medical and health sciencesCALCIUM-SENSING RECEPTOR0302 clinical medicineDELTA-OPIOID RECEPTORlawSummary informationReceptorsHumansHISTAMINE H-3 RECEPTORFATTY-ACID RECEPTORMETABOTROPIC GLUTAMATE-RECEPTOR030304 developmental biologyG protein-coupled receptorPharmacologyGONADOTROPIN-RELEASING-HORMONE0303 health sciencesClinical pharmacologyFORMYL PEPTIDE RECEPTORMUSCARINIC ACETYLCHOLINE-RECEPTOR3. Good health317 Pharmacy030220 oncology & carcinogenesisPharmaceuticalNEGATIVE ALLOSTERIC MODULATORCatalytic receptorsdescription
The Concise Guide to PHARMACOLOGY 2021/22 is the fifth in this series of biennial publications. The Concise Guide provides concise overviews, mostly in tabular format, of the key properties of nearly 1900 human drug targets with an emphasis on selective pharmacology (where available), plus links to the open access knowledgebase source of drug targets and their ligands (www.guidetopharmacology.org), which provides more detailed views of target and ligand properties. Although the Concise Guide constitutes over 500 pages, the material presented is substantially reduced compared to information and links presented on the website. It provides a permanent, citable, point-in-time record that will survive database updates. The full contents of this section can be found at http://onlinelibrary.wiley.com/doi/bph.15538. G protein-coupled receptors are one of the six major pharmacological targets into which the Guide is divided, with the others being: ion channels, nuclear hormone receptors, catalytic receptors, enzymes and transporters. These are presented with nomenclature guidance and summary information on the best available pharmacological tools, alongside key references and suggestions for further reading. The landscape format of the Concise Guide is designed to facilitate comparison of related targets from material contemporary to mid-2021, and supersedes data presented in the 2019/20, 2017/18, 2015/16 and 2013/14 Concise Guides and previous Guides to Receptors and Channels. It is produced in close conjunction with the Nomenclature and Standards Committee of the International Union of Basic and Clinical Pharmacology (NC-IUPHAR), therefore, providing official IUPHAR classification and nomenclature for human drug targets, where appropriate.
| year | journal | country | edition | language |
|---|---|---|---|---|
| 2021-10-01 |