ChemInform Abstract: Synthesis of 5-Substituted 2,3-Dihydrobenzofurans in a One-Pot Oxidation/Cyclization Reaction.

6533b835fe1ef96bd129fdba

RESEARCH PRODUCT

ChemInform Abstract: Synthesis of 5-Substituted 2,3-Dihydrobenzofurans in a One-Pot Oxidation/Cyclization Reaction.

Christian Duchamp Natali Henriques Patrizia Diana Alessandra Montalbano Roland Barret Eugenio Lo Piccolo Eugenio Lo Piccolo Thierry Lomberget Fabien Baragona Fabien Baragona

subject

Chemistry Organic chemistry General Medicine Cycloaddition Quinone

description

The oxidation of N-protected p-aminophenol derivatives to quinone imides is combined with cycloaddition towards azadiene (II) in a one-pot reaction to give dihydrobenzofuran derivatives in moderate to good yields.

year	journal	country	edition	language
2012-02-16	ChemInform

https://doi.org/10.1002/chin.201211081

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