Search results for "Chemotype"

showing 10 items of 24 documents

Comprehending and improving cannabis specialized metabolism in the systems biology era

2020

Cannabis sativa is a source of food, fiber and specialized metabolites such as cannabinoids, with psychoactive and pharmacological effects. Due to its expanding and increasingly-accepted use in medicine, cannabis cultivation is acquiring more importance and less social stigma. Humans initiated different domestication episodes whose later spread gave rise to a plethora of landrace cultivars. At present, breeders cross germplasms from different gene pools depending on their specific use. The fiber (hemp) and drug (marijuana) types of C. sativa differ in their cannabinoid chemical composition phenotype (chemotype) and also in the accumulation of terpenoid compounds that constitute a strain’s p…

0106 biological sciences0301 basic medicineSystems biologymedicine.medical_treatmentPlant ScienceComputational biology01 natural sciencesGenomeTerpene03 medical and health sciencesCannabinoid chemotypeGeneticsmedicineCannabisbiologyChemotypeCannabinoidsTerpenesSystems Biologyfood and beveragesGeneral Medicinebiology.organism_classificationTerpenoidMarijuanaPlant BreedingMetabolic pathway030104 developmental biologyCannabinoidCannabisHempAgronomy and Crop ScienceMetabolic Networks and Pathways010606 plant biology & botanyPlant Science
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Efficacy of sea fennel (Crithmum maritimum L., Apiaceae) essential oils against Culex quinquefasciatus Say and Spodoptera littoralis (Boisd.)

2017

The effective management of insect pests and vectors still represents a major challenge in current entomology. Culex quinquefasciatus Say is a key vector of lymphatic filariasis, Rift Valley fever, West Nile, St. Louis encephalitis and Western equine encephalitis virus. Recently, the importance of the eco-friendly control of C. quinquefasciatus larval population using plant-borne biopesticides, including essential oils (EOs), has been stressed. Spodoptera littoralis (Boisd.) also known as tobacco cutworm, is one of the most destructive moth agricultural pests in tropic and sub-tropic regions. Despite the fact that sea fennel (Crithmum maritimum L., Apiaceae) is considered as a promising bio…

0106 biological sciencesBiopesticides[SDV]Life Sciences [q-bio]Population01 natural sciencesEssential oillaw.inventionSpodoptera littoralichemistry.chemical_compoundCulex quinquefasciatulawCrithmumBotanyBiopesticides; Crithmum maritimum; Culex quinquefasciatus; Essential oil; Spodoptera littoralis14. Life underwatereducationSpodoptera littoralisEssential oilDillapioleeducation.field_of_studyApiaceaebiologyChemotype010405 organic chemistryCrithmum maritimumCulex quinquefasciatusSpodoptera littoralisbiology.organism_classificationCulex quinquefasciatus0104 chemical scienceschemistry13. Climate actionBiopesticideAgronomy and Crop Science010606 plant biology & botany
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Artemisia arborescens essential oil composition, enantiomeric distribution and antimicrobial activity from different wild populations from the Medite…

2016

International audience; Aerial parts of Artemisiaarborescens were collected from different sites of the Mediterranean area (southwestern Algeria and southern Italy) and the chemical composition of their essential oil (EO) extracted by hydrodistillation was studied by both gas chromatography (GC) equipped with an enantioselective capillary column and GC/mass spectrometry (GC/MS). The EOs obtained were tested against several Listeriamonocytogenes strains. Using GC and GC/MS, 41 compounds were identified, accounting for 96.0-98.8% of the total EO. All EOs showed a similar terpene profile, which was rich in chamazulene, -thujone, and camphor. However, the concentration of such compounds varied …

0106 biological sciencesListeriaBioengineeringMicrobial Sensitivity TestsSettore MED/42 - Igiene Generale E Applicata01 natural sciencesBiochemistry[ CHIM ] Chemical Scienceslaw.inventionTerpeneCamphorchemistry.chemical_compoundlawBotanyOils Volatile[CHIM]Chemical SciencesFood scienceMolecular BiologyEssential oilVolatile compositionbiologyChemotypeMediterranean RegionChemistryChamazuleneBiological activityStereoisomerismGeneral ChemistryGeneral Medicinebiology.organism_classificationArtemisia arborescensEnantiomeric distributionListeria monocytogenesAnti-Bacterial Agents0104 chemical sciences010404 medicinal & biomolecular chemistrySettore MED/18 - Chirurgia GeneraleArtemisiaItalyAlgeriaGram-negative bacteriaMolecular MedicineArtemisiaGas chromatographyEnantiomeric distribution Biological activity Gram-negative bacteria Volatile composition Listeria monocytogenes.010606 plant biology & botanySettore AGR/16 - Microbiologia Agraria
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Agronomic Evaluation and Chemical Characterization of Sicilian Salvia sclarea L. Accessions

2020

Clary sage (Salvia sclarea L.), known for its aromatic and medicinal properties, belongs to the Lamiaceae family. Although the species grows wild throughout Sicily, knowledge of its production and qualitative properties is limited. The aim of this study was to evaluate the agronomic behavior of the species over two years of testing and to characterize the chemical properties of its wild counterparts in order to identify the most promising accessions for cropping or for use in breeding programs. Tests were carried out during 2008, 2009, and 2010. During the first year, the plot was established. Subsequently, the main parameters for bio-agronomic evaluation were taken in 2009 and 2010. Regard…

0106 biological sciencesMediterranean climateRange (biology)Linalyl acetate01 natural sciencesessential oillaw.inventionlcsh:Agriculturechemistry.chemical_compoundlawSalvia sclareaclary sagearomatic plant specieEssential oilbiologyChemotypeSAGEaromatic plant specieslcsh:S04 agricultural and veterinary sciencesbiology.organism_classificationSettore AGR/02 - Agronomia E Coltivazioni ErbaceeHorticulturechemistry040103 agronomy & agriculture0401 agriculture forestry and fisheriesLamiaceaeAgronomy and Crop Science010606 plant biology & botanybiometric and agronomic characteristicsAgronomy
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Essential oil variability in a collection of Ocimum basilicum L. (basil) cultivars.

2016

Ocimum basilicum L. (Lamiaceae) is an aromatic plant of great tradition in the Mediterranean area. Its economic importance is growing up determining an expansion of cultivation. This paper evaluated the morphological traits, the chemical profiles, and antibacterial activity of 21 cultivars of basil belonging to Ê»Genoveseʼ, Ê»Napoletanoʼ, and Ê»Purple basilʼ types. The cultivars were characterized by different growth rate and morphological traits. The chemical composition of the oils analyzed by GC and GC/MS analysis, supported by the PCA analysis, underlined the strong influence of chemotype. It is noteworthy that estragole, never present in Genovese and purple basil types, occurred in …

0106 biological sciencesfood.ingredientPCA analysisBioengineeringMicrobial Sensitivity TestsBiologyGram-Positive Bacteria01 natural sciencesBiochemistrychemistry.chemical_compoundStructure-Activity Relationship0404 agricultural biotechnologyfoodLinaloolMethyl eugenolOcimum basilicum LBiomorphological characteristicAnti-Bacterial AgentBotanyGram-Negative BacteriaAntibacterial activitiesOils VolatileBiomorphological characteristicsMolecular BiologyEssential-oil constituentChemotypeDose-Response Relationship DrugMicrobial Sensitivity TestChemistry (all)Basilicumfood and beveragesEssential-oil constituents04 agricultural and veterinary sciencesGeneral ChemistryGeneral MedicineOcimumbiology.organism_classification040401 food scienceAnti-Bacterial AgentsEugenolchemistryOcimum basilicumMolecular MedicineAntibacterial activitieEstragoleLamiaceaeAntibacterial activities; Biomorphological characteristics; Essential-oil constituents; Ocimum basilicum L.; PCA analysisPCA analysi010606 plant biology & botany
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Assessment of production and qualitative characteristics of different populations of Salvia sclarea L. found in Sicily (Italy)

2021

Salvia sclarea L. is an important industrial crop, valued for its herbal-aromatic properties and high quality essential oils, that is used in food, pharmaceuticals and cosmetics. In this study, carried out from 2009 to 2010, the morphological and production characteristics and essential oil content and composition of three Sicilian populations were studied. In particular, the composition of essential oils extracted from primary and secondary inflorescences using steam distillation was assessed. Morphological, production and qualitative data from the three populations were subjected to analysis of variance and cluster analysis. Regarding the quality of the oils, only the most prevalent compo…

0106 biological sciencesspike yieldPopulation<i>Salvia sclarea</i> L.; spike yield; primary and secondary inflorescences; local populations; essential oil principal componentsBiologyLinalyl acetateSalvia sclarea L.01 natural scienceslaw.inventionSteam distillationchemistry.chemical_compoundLinaloollawSalvia sclarealocal populationseducationEssential oilprimary and secondary inflorescenceseducation.field_of_studyChemotypeS<i>Salvia sclarea</i> L.Agricultureessential oil principal components0104 chemical sciencesSettore AGR/02 - Agronomia E Coltivazioni Erbacee010404 medicinal & biomolecular chemistryHorticultureInflorescencechemistrylocal populationprimary and secondary inflorescenceAgronomy and Crop Science010606 plant biology & botany
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The Nonvolatile and Volatile Metabolites of Prangos ferulacea and Their Biological Properties

2019

Abstract Prangos ferulacea (L.) Lindl. (Fam. Apiaceae), an orophilous species of eastern Mediterranean and western Asia, possesses a number of biological properties that are worthy of exploitation in different fields. Phytochemical investigations revealed the presence of coumarins, prenyl-coumarins, and furano-coumarins as the main constituents of this species, as well as several flavonoids. Among prenyl-coumarins, osthol is a promising apoptotic agent quite selective toward cancer cells. In addition, the essential oils have been extensively investigated, and several chemotypes have been identified. This work reviews the literature on this species published between 1965 and 2018, describes …

Anti-Infective AgentPrangos ferulaceaPharmaceutical Science01 natural sciencesAntioxidantsAnalytical Chemistrylaw.inventionchemistry.chemical_compoundAnti-Infective AgentslawDrug Discoveryheterocyclic compoundsAnalgesicsbiologyTraditional medicinePhytochemicalprenyl-coumarinsMolecular MedicineAntioxidantfurano-coumarinOstholHumanCoumarinessential oilBiological propertyAnimalsHumansHypoglycemic AgentsVolatile metabolitesEssential oilPharmacologyPrangos ferulaceacoumarinsApiaceaeHypoglycemic AgentChemotypeAnimalPlant Extracts010405 organic chemistryOrganic ChemistryPrangos ferulacea; Apiaceae; coumarins; prenyl-coumarins; furano-coumarinsSettore CHIM/06 - Chimica Organicabiology.organism_classification0104 chemical sciencesprenyl-coumarin010404 medicinal & biomolecular chemistryComplementary and alternative medicinechemistrySettore BIO/03 - Botanica Ambientale E ApplicataAnalgesicApiaceaefurano-coumarinsPlanta Medica
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Discovery of new G-quadruplex binding chemotypes

2013

We report here on the discovery and preliminary evaluation of a novel non-macrocyclic low molecular weight quadruplex-stabilizing chemotype. The lead compounds, based on a furan core, show high G-quadruplex stabilisation and selectivity as well as potent in vitro anti-proliferative activity.

Cell SurvivalAntineoplastic Agents010402 general chemistryG-quadruplex01 natural sciencesArticleCatalysis03 medical and health scienceschemistry.chemical_compoundCell Line TumorFuranMaterials ChemistryHumansheterocyclic compoundsFuransCell survival030304 developmental biologyG quadruplex binding0303 health sciencesG-quadruplexChemotypeChemistryCircular DichroismMetals and AlloysGeneral ChemistryCombinatorial chemistryIn vitro3. Good health0104 chemical sciencesSurfaces Coatings and FilmsElectronic Optical and Magnetic MaterialsG-QuadruplexesCeramics and CompositesSelectivityChem. Commun.
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Chemical Composition and Antimicrobial Activity of the Essential Oils from Three Chemotypes of Origanum vulgare L. ssp. hirtum (Link) Ietswaart Growi…

2009

Essential oils obtained from inflorescences of three Origanum vulgare L.ssp. hirtum (Link) Ietswaart samples, growing wild in different locations in Campania (Southern Italy), were analysed. Three chemotypes were found: the first, with a prevalence of carvacrol/thymol; the second, characterized by the prevalence of thymol/alpha-terpineol; the third, featuring a prevalence of linalyl acetate and linalool. This chemical study attempts to provide a contribution in shedding light on the relationship between chemical composition and biotypes and/or chemotypes in Origanum vulgare ssp. hirtum. The essential oils were also evaluated for their antibacterial activity against 10 selected microorganism…

Chromatography GasAcyclic MonoterpenescarvacrolPharmaceutical ScienceCyclohexane MonoterpenesMicrobial Sensitivity TestsLinalyl acetateCymenesArticleGas Chromatography-Mass SpectrometryAnalytical Chemistrylcsh:QD241-441chemistry.chemical_compoundOriganum vulgare ssp. hirtumantibacterial activitylcsh:Organic chemistryLinaloolOriganumthymolCyclohexenesDrug DiscoveryBotanyOils VolatilePlant OilsCarvacrollinalyl acetatePhysical and Theoretical ChemistryThymolessential oil compositionBacteriabiologyChemotypeOrganic ChemistryOriganum vulgare ssp. hirtum; essential oil composition; thymol; carvacrol; linalyl acetate; antibacterial activityOriganumbiology.organism_classificationAntimicrobialAnti-Bacterial AgentsItalychemistryChemistry (miscellaneous)MonoterpenesCymenesMolecular MedicineMolecules
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Bioactive Constituents of Juniperus turbinata Guss. from La Maddalena Archipelago.

2018

A comprehensive phytochemical study of Juniperus turbinata (Cupressaceae) collected from La Maddalena Archipelago (Sardinia, Italy) is reported. Both the essential oil and the ethanolic extract obtained from the aerial parts were analyzed. The essential oil appears to belong to a new chemotype compared to other Mediterranean juniper accessions, as it was favored by geographic isolation of the isles. It showed a low content of monoterpene hydrocarbons and -terpineol, ent-manoyl oxide, 1,10-di-epi-cubenol as the major constituents. The ethanolic fraction contained mainly diterpenoids. Among these, 15-formyloxyimbricatolic acid (7) is a new natural product since it has hitherto been obtained o…

CupressaceaeFree RadicalsDPPHMonoterpeneJuniperus turbinata; biological activity; essential oil; imbricataloic acid; polar compoundsPhytochemicalsMolecular ConformationBioengineeringbiological activityAmentoflavonePhytochemical01 natural sciencesBiochemistryessential oilimbricataloic acidAntioxidantslaw.inventionchemistry.chemical_compoundStructure-Activity RelationshiplawCell Line TumorOils VolatileHumanspolar compoundMolecular BiologyEssential oilCell ProliferationbiologyChemotypeTraditional medicineDose-Response Relationship Drug010405 organic chemistryCupressaceaeGeneral ChemistryGeneral Medicinebiology.organism_classificationAntineoplastic Agents Phytogenic0104 chemical sciences010404 medicinal & biomolecular chemistrychemistryPhytochemicalItalyMolecular MedicineTroloxAntioxidantDrug Screening Assays AntitumorFree RadicalJuniperus turbinataHumanChemistrybiodiversity
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