Search results for "DAP"

showing 10 items of 3579 documents

Structural Basis of the High Affinity Interaction between the Alphavirus Nonstructural Protein-3 (nsP3) and the SH3 Domain of Amphiphysin-2

2016

We show that a peptide from Chikungunya virus nsP3 protein spanning residues 1728–1744 binds the amphiphysin-2 (BIN1) Src homology-3 (SH3) domain with an unusually high affinity (Kd 24 nM). Our NMR solution complex structure together with isothermal titration calorimetry data on several related viral and cellular peptide ligands reveal that this exceptional affinity originates from interactions between multiple basic residues in the target peptide and the extensive negatively charged binding surface of amphiphysin-2 SH3. Remarkably, these arginines show no fixed conformation in the complex structure, indicating that a transient or fluctuating polyelectrostatic interaction accounts for this …

0301 basic medicinenuclear magnetic resonance (NMR)Amino Acid MotifsStatic ElectricityPeptideTarget peptidePlasma protein bindingViral Nonstructural ProteinsBiologyhost-pathogen interactionBiochemistrySH3 domainsrc Homology Domainsamphiphysin SH3Structure-Activity Relationship03 medical and health sciencesProtein structuredynaminHumansShort linear motifprotein structureNuclear Magnetic Resonance BiomolecularMolecular BiologySrc homology 3 domain (SH3 domain)Adaptor Proteins Signal Transducingchemistry.chemical_classificationTumor Suppressor Proteinsta1182Nuclear ProteinsIsothermal titration calorimetryCell Biologyintrinsically disordered protein030104 developmental biologychemistryBiochemistrynsP3Protein Structure and FoldingAmphiphysinBiophysicsPeptidesChikungunya virusProtein BindingJournal of Biological Chemistry
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Lack of Hypothalamus Polysialylation Inducibility Correlates With Maladaptive Eating Behaviors and Predisposition to Obesity

2018

This original research article (6 p.) is part of the research topic . Specialty section: This article was submitted to Neuroenergetics, Nutrition and Brain Health, a section of the journal Frontiers in Nutrition.; International audience; High variability exists in individual susceptibility to develop overweight in an obesogenic environment and the biological underpinnings of this heterogeneity are poorly understood. In this brief report, we show in mice that the vulnerability to diet-induced obesity is associated with low level of polysialic acid-neural cell adhesion molecule (PSA-NCAM), a factor of neural plasticity, in the hypothalamus. As we previously shown that reduction of hypothalami…

0301 basic medicineobesityfood intakePSA-NCAMEndocrinology Diabetes and Metabolismmedia_common.quotation_subject[SDV]Life Sciences [q-bio][SDV.NEU.NB]Life Sciences [q-bio]/Neurons and Cognition [q-bio.NC]/Neurobiologybrainmaladaptive eating behaviorlcsh:TX341-641BiologyOverweightEnergy homeostasis03 medical and health sciencesNeuroplasticitymedicineFood and Nutritionhypothalamusmedia_commonNutritionOriginal ResearchNutrition and Dieteticssynaptic plasticitycomportement alimentairepolysialylation[SDV.NEU.NB] Life Sciences [q-bio]/Neurons and Cognition [q-bio.NC]/NeurobiologyNeurosciencesAppetitemedicine.diseaseprise alimentaireObesity3. Good health[SDV] Life Sciences [q-bio]food intake;obesity;maladaptive eating behavior;synaptic plasticity;PSA-NCAM;polysialylation;brain;hypothalamusEating disordersobésité030104 developmental biologynervous systemHypothalamusNeurons and CognitionSynaptic plasticityAlimentation et Nutritionplasticité synaptiquecerveaumedicine.symptomlcsh:Nutrition. Foods and food supplyNeuroscienceFood ScienceFrontiers in Nutrition
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Anti-proliferative and apoptosis-inducing effect of theabrownin against non-small cell lung adenocarcinoma A549 cells

2016

With the highest cancer incidence rate, lung cancer, especially non-small cell lung cancer (NSCLC), is the leading cause of cancer death in the world. Tea (leaves of Camellia sinensis) has been widely used as a traditional beverage beneficial to human health, including anti-NSCLC activity. Theabrownin (TB) is one major kind of tea pigment responsible for the beneficial effects of tea liquor. However, its effect on NSCLC is unknown. The aim of the present study was to evaluate anti-proliferative and apoptosis-inducing effect of TB on NSCLC (A549) cells, using MTT assay, morphological observation (DAPI staining), in situ terminal deoxynucleotidyl transferase dUTP nick end labeling (TUNEL) ass…

0301 basic medicinep53ApoptosisBiology03 medical and health scienceschemistry.chemical_compound0302 clinical medicineA549 cellsPharmacology (medical)MTT assayDAPIOriginal ResearchPharmacologyA549 cellTUNEL assayCell growthTheabrowninlcsh:RM1-950Molecular biologylung cancer030104 developmental biologyReal-time polymerase chain reactionlcsh:Therapeutics. PharmacologyTerminal deoxynucleotidyl transferasechemistryApoptosis030220 oncology & carcinogenesisA549 cells;Frontiers in Pharmacology
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Expert Opinion on Three Phage Therapy Related Topics: Bacterial Phage Resistance, Phage Training and Prophages in Bacterial Production Strains

2018

Phage therapy is increasingly put forward as a "new" potential tool in the fight against antibiotic resistant infections. During the "Centennial Celebration of Bacteriophage Research" conference in Tbilisi, Georgia on 26-29 June 2017, an international group of phage researchers committed to elaborate an expert opinion on three contentious phage therapy related issues that are hampering clinical progress in the field of phage therapy. This paper explores and discusses bacterial phage resistance, phage training and the presence of prophages in bacterial production strains while reviewing relevant research findings and experiences. Our purpose is to inform phage therapy stakeholders such as po…

0301 basic medicinephage therapyPhage therapyprophagemedicine.medical_treatmentviruses030106 microbiologylcsh:QR1-502Resistance (psychoanalysis)adaptationlcsh:MicrobiologyBacteriophageresistance03 medical and health sciencesAntibiotic resistanceVirologyPolitical sciencemedicineBacteriophageProphageComputingMilieux_MISCELLANEOUSbiologybusiness.industryConference ReportregulationPublic relationsResearch findingsbiology.organism_classification[SDV.MP.BAC]Life Sciences [q-bio]/Microbiology and Parasitology/Bacteriology3. Good healthInfectious DiseasesExpert opinionproductionbusinessViruses
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STRIPAK Members Orchestrate Hippo and Insulin Receptor Signaling to Promote Neural Stem Cell Reactivation

2019

Summary Adult stem cells reactivate from quiescence to maintain tissue homeostasis and in response to injury. How the underlying regulatory signals are integrated is largely unknown. Drosophila neural stem cells (NSCs) also leave quiescence to generate adult neurons and glia, a process that is dependent on Hippo signaling inhibition and activation of the insulin-like receptor (InR)/PI3K/Akt cascade. We performed a transcriptome analysis of individual quiescent and reactivating NSCs harvested directly from Drosophila brains and identified the conserved STRIPAK complex members mob4, cka, and PP2A (microtubule star, mts). We show that PP2A/Mts phosphatase, with its regulatory subunit Widerbors…

0301 basic medicinereactivationendocrine systemMitosisNerve Tissue ProteinsProtein Serine-Threonine KinasesBiologyArticleGeneral Biochemistry Genetics and Molecular BiologyAnimals Genetically ModifiedPhosphatidylinositol 3-Kinases03 medical and health sciences0302 clinical medicineNeural Stem CellsAnimalsDrosophila ProteinsquiescenceProtein Phosphatase 2lcsh:QH301-705.5Protein kinase BCells CulturedPI3K/AKT/mTOR pathwayTissue homeostasisAdaptor Proteins Signal TransducingCell ProliferationHippo signaling pathwayGene Expression ProfilingHippo signalingInR/PI3K/Akt signalingfungiIntracellular Signaling Peptides and ProteinsBrainSTRIPAK membersProtein phosphatase 2Receptor InsulinNeural stem cellCell biologyDrosophila melanogaster030104 developmental biologylcsh:Biology (General)nervous systemHippo signalingSingle-Cell AnalysisTranscriptomeProto-Oncogene Proteins c-akt030217 neurology & neurosurgeryAdult stem cellCell Reports
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Ocular Clocks: Adapting Mechanisms for Eye Functions and Health

2018

Vision is a highly rhythmic function adapted to the extensive changes in light intensity occurring over the 24-hour day. This adaptation relies on rhythms in cellular and molecular processes, which are orchestrated by a network of circadian clocks located within the retina and in the eye, synchronized to the day/night cycle and which, together, fine-tune detection and processing of light information over the 24-hour period and ensure retinal homeostasis. Systematic or high throughput studies revealed a series of genes rhythmically expressed in the retina, pointing at specific functions or pathways under circadian control. Conversely, knockout studies demonstrated that the circadian clock re…

0301 basic medicineretinavisiongenetic structuresPeriod (gene)[SDV.NEU.NB]Life Sciences [q-bio]/Neurons and Cognition [q-bio.NC]/NeurobiologyCircadian clockCLOCK ProteinsGene ExpressionContext (language use)melatoninReviewBiologyrhythm03 medical and health scienceschemistry.chemical_compoundCircadian ClocksmedicineAnimalsHumansCircadian rhythmOcular Physiological PhenomenaComputingMilieux_MISCELLANEOUSRetinaAdaptation OcularRetinalphotoreceptorCircadian RhythmCLOCKLight intensity030104 developmental biologymedicine.anatomical_structurecircadianchemistrysense organsdopamineNeuroscienceInvestigative Ophthalmology & Visual Science
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Genome-wide scan of fat-tail sheep identifies signals of selection for fat deposition and adaptation

2018

Fat tail in sheep represents a valuable energy reserve for facing future climate changes. The identification of genes with a role in the fat-tail phenotype may contribute to understanding the physiology of fat deposition and the mechanisms of adaptation. Genotypic data obtained with the OvineSNP50K array in 13 thin-tail sheep breeds from Italy were used to identify selection signatures of fat tail through pairwise thin- versus fat-tail sheep breed comparisons, with the following fat-tail breeds of the Mediterranean area: two unique Italian fat-tail breeds (Barbaresca and Laticauda), a Barbary sheep breed from Libya, Ossimi breed from Egypt, Cyprus Fat-Tail and Chios from the Greek islands …

0301 basic medicinesheepGenomicsadaptationfat-tailBarbaresca03 medical and health sciencesSettore AGR/17 - Zootecnica Generale E Miglioramento Geneticobiology.animalLaticaudagenomicsbiologyadaptation; fat-tail; genomics; sheep; Food Science; Animal Science and Zoology0402 animal and dairy science04 agricultural and veterinary sciencesBarbary sheepbiology.organism_classification040201 dairy & animal sciencePhenotypeBreed030104 developmental biologyfat-tail adaptation genomics sheepEvolutionary biologyGenetic markerAnimal Science and ZoologyAdaptationFood Science
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Constrained evolvability of interferon suppression in an RNA virus.

2016

AbstractInnate immunity responses controlled by interferon (IFN) are believed to constitute a major selective pressure shaping viral evolution. Viruses encode a variety of IFN suppressors, but these are often multifunctional proteins that also play essential roles in other steps of the viral infection cycle, possibly limiting their evolvability. Here, we experimentally evolved a vesicular stomatitis virus (VSV) mutant carrying a defect in the matrix protein (M∆51) that abolishes IFN suppression and that has been previously used in the context of oncolytic virotherapy. Serial transfers of this virus in normal, IFN-secreting cells led to a modest recovery of IFN blocking capacity and to weak …

0301 basic medicineviruses030106 microbiologyAdaptation BiologicalBiologyVirus ReplicationModels BiologicalVirusArticleCell Line03 medical and health sciencesViral ProteinsRNA Virus InfectionsInterferonmedicineHumansRNA VirusesPhosphorylationMultidisciplinaryViral matrix proteinInterferon SuppressionGenetic Variationbiology.organism_classificationVirologyBiological EvolutionImmunity InnateOncolytic virus030104 developmental biologyViral replicationVesicular stomatitis virusViral evolutionMutationInterferonsmedicine.drugScientific reports
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Sleep, alertness and alertness management among commercial airline pilots on short-haul and long-haul flights

2016

Item does not contain fulltext Airline pilots' sleep and on-duty alertness are important focus areas in commercial aviation. Until now, studies pertaining to this topic have mainly focused on specific characteristics of flights and thus a comprehensive picture of the matter is not well established. In addition, research knowledge of what airline pilots actually do to maintain their alertness while being on duty is scarce. To address these gaps in research knowledge, we conducted a field study on a representative sample of the airline pilots of a medium-sized airline. The sample consisted of 90 pilots, of whom 30 flew long-haul (LH) routes, 30 short-haul (SH) routes, and 30 flew both. A tota…

030110 physiology0301 basic medicineEngineeringAircraftAviationCruiseHuman Factors and ErgonomicsAviation safety03 medical and health sciences0302 clinical medicineAeronauticsSleep Disorders Circadian RhythmWork Schedule TolerancemedicineHumansSafety Risk Reliability and QualitySimulationFatigueFinlandOccupational Healthta515Work Health and PerformanceSleep Stagesbusiness.industryPublic Health Environmental and Occupational HealthAlertness managementCivil aviationawiationAlertnessAdaptation PhysiologicalSleep deprivationAlertnessPilotsCommercial aviationSleep DeprivationSleep Stagesmedicine.symptombusinessAviationSleep030217 neurology & neurosurgeryPsychomotor Performance
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The best way to assess visually induced motion sickness in a fixed-base driving simulator

2017

Abstract Objective Driving simulator usage is becoming more widespread, yet many users still experience substantial motion sickness-like symptoms induced by optical flow, called visually induced motion sickness (VIMS). The Fast Motion sickness Scale (FMS) allows for continuous on-line assessment of VIMS. Using mixed models for ordinal data, this study investigated how to optimally analyze FMS data, and then used the resulting models to examine the development of symptoms over time in detail. Additionally, the study explored the impact of specific VIMS-inducing road elements. Methods Twenty-eight healthy young adults without prior simulator experience completed six courses on two days in a f…

030110 physiology0301 basic medicineOrdinal dataMixed modelmedicine.medical_specialtyComputer science05 social sciencesDriving simulatorOptical flowPoison controlTransportationAdaptation (eye)medicine.diseaseInterval Scale03 medical and health sciencesMotion sicknessPhysical medicine and rehabilitationAutomotive Engineeringmedicine0501 psychology and cognitive sciences050107 human factorsApplied PsychologySimulationCivil and Structural EngineeringTransportation Research Part F: Traffic Psychology and Behaviour
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