Search results for "Hesperidin"

showing 7 items of 17 documents

Bond strength and elemental analysis of oxidized dentin bonded to resin modified glass ionomer based restorative material

2019

Background This study aimed to investigate the influence of hesperidin application on the bonding of resin-modified glass ionomer-based restorative material to dentin treated with oxygen-induced endodontic irrigants. Material and Methods One hundred human permanent molars were categorized into five groups (n= 20/group), treated with various irrigants as follows: Group C; distilled water (control group), Group SH; 5.25% NaOCl, Group SH+H; 5.25% NaOCl + 5 % hesperidin, Group HP; 10% H2O2, Group HP+H; 10% H2O2 + 5 % hesperidin. Specimens were bonded with RMGI based restorative material. For each group, half of the specimens were evaluated for µSBS by a universal testing machine and the other h…

MolarUniversal testing machineChemistryBond strengthResearch0206 medical engineeringGlass ionomer cement030206 dentistry02 engineering and technology:CIENCIAS MÉDICAS [UNESCO]020601 biomedical engineeringOperative Dentistry and Endodontics03 medical and health sciencesHesperidinchemistry.chemical_compound0302 clinical medicinemedicine.anatomical_structureDistilled waterstomatognathic systemElemental analysisUNESCO::CIENCIAS MÉDICASDentinmedicineGeneral DentistryNuclear chemistry
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Modeling anti-allergic natural compounds by molecular topology.

2013

Molecular topology has been applied to the search of QSAR models able to identify the anti-allergic activity of a wide group of heterogeneous compounds. Through the linear discriminant analysis and artificial neural networks, correct classification percentages above 85% for both the training set and the test set have been obtained. After carrying out a virtual screening with a natural product library, about thirty compounds with theoretical anti-allergic activity have been selected. Among them, hesperidin, naringin, salinomycin, sorbitol, curcumol, myricitrin, diosmin and kinetin stand out. Some of these compounds have already been referenced as having anti-allergic activity.

Virtual screeningQuantitative structure–activity relationshipStereochemistryOrganic ChemistryDiosminDiscriminant AnalysisQuantitative Structure-Activity RelationshipGeneral MedicineComputational biologyLinear discriminant analysisModels BiologicalComputer Science Applicationschemistry.chemical_compoundHesperidinchemistryArtificial IntelligenceTest setDrug DiscoveryAnti-Allergic AgentsmedicineHumansNeural Networks ComputerMyricitrinNaringinmedicine.drugCombinatorial chemistryhigh throughput screening
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Cytotoxicity of the crude extract and constituents of the bark of Fagara tessmannii towards multi-factorial drug resistant cancer cells.

2019

Abstract Ethnopharmacological relevance Fagara tessmannii Engl. is an African medicinal plant used in Cameroonian traditional medicine to treat various types of cancers. Aim of the study This work was designed to determine the cytotoxicity of the crude extract (FTB), fractions (FTBa-d) and compounds isolated from the bark of Fagara tessmannii, namely lupeol (1), fagaramide (2), zanthoxyline (3), hesperidin (4), nitidine chloride (5), fagaridine chloride (6), and β-sitosterol-3-O-β-D-glucopyranoside (7). The study was extended to the mode of induction of apoptosis by FTB, compounds 5 and 6. Materials and methods The resazurin reduction assay was used to evaluate the cytotoxicity of samples. …

ZanthoxylumApoptosisFlow cytometry03 medical and health scienceschemistry.chemical_compoundHesperidinInhibitory Concentration 500302 clinical medicineCell Line TumorNeoplasmsDrug DiscoverymedicineHumansCytotoxicity030304 developmental biologyLupeolPharmacologychemistry.chemical_classificationMembrane Potential Mitochondrial0303 health sciencesReactive oxygen speciesmedicine.diagnostic_testPlant ExtractsCell CycleCell cycleMolecular biologyAntineoplastic Agents PhytogenicchemistryApoptosisDoxorubicinDrug Resistance Neoplasm030220 oncology & carcinogenesisCancer cellPlant BarkReactive Oxygen SpeciesJournal of ethnopharmacology
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Molecular topology: a useful tool for the search of new antibacterials.

2000

Molecular topology has been applied to find new lead antibacterial compounds. Among the selected compounds, hesperidin, neohesperidin and Mordant Brown 24 stand out, with minimum inhibitory concentrations 90, MIC90<0.3 mg / mL.

chemistry.chemical_classificationNeohesperidinMolecular modelBacteriamedicine.drug_classStereochemistryOrganic ChemistryClinical BiochemistryAntibioticsFlavonoidPharmaceutical ScienceMordantBiochemistryCombinatorial chemistryAnti-Bacterial AgentsHesperidinchemistry.chemical_compoundchemistryDrug DiscoverymedicineMolecular MedicineMolecular BiologyTopology (chemistry)Antibacterial agentBioorganicmedicinal chemistry letters
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Influence of solvents on the antioxidant property of flavonoids.

2003

In polyphenols redox systems, the solvent plays a fundamental role in the chemical behaviour of these compounds. Antioxidants can react in different ways with the prooxidant molecules. We have found differences in the antioxidant capacity of flavonoids such as naringin, neohesperidin, neoericitrin, hesperidin, narirutin didymin and the related flavones naringenin, hesperetin eriodictyol and isosakuratenin, when they are in the presence of radicals and solved in water or in an alcohol mixture.

chemistry.chemical_classificationNeohesperidinNaringeninFlavonoidsNarirutinFree RadicalsHesperetinEriodictyolFlavonesAntioxidantschemistry.chemical_compoundHesperidinchemistrySolventsOrganic chemistryReactive Oxygen SpeciesNaringinOxidation-ReductionFood ScienceDie Nahrung
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Ruta chalepensis L. (Rutaceae) leaf extract: chemical composition, antioxidant and hypoglicaemic activities.

2017

Ruta chalepensis L. (Rutaceae) leaf extract was investigated for its chemical profile and antioxidant and hypoglycaemic properties. The antioxidant effects were investigated by 2,2-diphenyl-1-picrylhydrazyl (DPPH), Chi-carotene bleaching, and metal chelating activity assays. The carbohydrate-hydrolysing enzymes inhibition assay was used to test the hypoglycaemic potential. R. chalepensis showed a high content of hesperidin and rutin with values of 591.9 and 266.7 mg/g dry extract, respectively. The extract exhibited a promising protection of lipid peroxidation (IC50 value of 16.9 mu g/mL) and inhibited both alpha-amylase and alpha-glucosidase enzymes in a concentration-dependent manner. The…

leaveMetal chelating activityAntioxidantDPPHmedicine.medical_treatmentRutinHPLC analysiantioxidant activityPlant Science01 natural sciencesBiochemistryAntioxidantsAnalytical ChemistryLipid peroxidationRutinchemistry.chemical_compoundHesperidinEnzyme InhibitorEnzyme InhibitorsTraditional medicinebiologyHydrolysisbeta CaroteneRuta chalepensisAntioxidantPlant Leavehypoglycaemic activityPlant Extractalpha-AmylaseInhibitory Concentration 50PicratesRuta chalepensiBotanymedicineGlycoside Hydrolase InhibitorsGlycoside Hydrolase InhibitorRutaDose-Response Relationship Drug010405 organic chemistryPlant ExtractsHesperidinOrganic ChemistryBiphenyl CompoundsSettore CHIM/06 - Chimica Organicabiology.organism_classificationHydrolysi0104 chemical sciencesPlant Leaves010404 medicinal & biomolecular chemistryRutaceaechemistryBiphenyl CompoundPicrateLipid Peroxidationalpha-AmylasesNatural product research
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Deficit irrigation and maturation stage influence quality and flavonoid composition of ‘Valencia’ orange fruit

2016

BACKGROUND:Effects of continuous deficit irrigation (DI) and partial rootzone drying (PRD) treatments (50%ETc) in comparison with full irrigation (CI, 100% ETc) were investigated during ‘Valencia’ orange fruit maturation. Ultra-high-performance liquid chromatography/high-resolutionmass spectrometry was used to quantify hesperidin, narirutin, tangeritin, nobiletin, didymin and neoeriocitrin in the fruit juice and peel. RESULTS: No significant effect of irrigation was found on yield, juice soluble solids or acidity. Juice color was not influenced by irrigation or harvest date, whereas peel color increased during maturation and was more pronounced in CI and PRD fruits. Juice acidity reached a …

partial rootzone dryingSettore AGR/03 - Arboricoltura Generale E Coltivazioni ArboreeUHPLC/HESI-MShesperidinSettore CHIM/10 - Chimica Degli AlimentiCitrus sinensis; hesperidin; partial rootzone drying; peel color; soluble solids; UHPLC/HESI-MSpeel colorCitrus sinensisoluble solid
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