Search results for "Molecular imaging"

showing 10 items of 59 documents

Targeted tumor imaging of anti-CD20-polymeric nanoparticles developed for the diagnosis of B-cell malignancies

2015

Sara Capolla,1 Chiara Garrovo,2 Sonia Zorzet,1 Andrea Lorenzon,3 Enrico Rampazzo,4 Ruben Spretz,5 Gabriele Pozzato,6 Luis Núñez,7 Claudio Tripodo,8 Paolo Macor,1,9 Stefania Biffi2 1Department of Life Sciences, University of Trieste, 2Institute for Maternal and Child Health – IRCCS “Burlo Garofolo”, Trieste, 3Animal Care Unit, Cluster in Biomedicine (CBM scrl), Trieste, Italy; 4Department of Chemistry “G. Ciamician”, University of Bologna, Bologna, Italy; 5LNK Chemsolutions LLC, Lincoln, NE, USA; 6Department of Medical, Surgery and Health Sciences, University of Trieste, Trieste, Italy; 7Bio-Target, Inc., University of C…

Medicine (General)Active targeting; Optical imaging; Tumor accumulation; Animals; Antigens CD20; Cell Line Tumor; Humans; Leukemia B-Cell; Mice; Molecular Imaging; Nanoparticles; Polymers; Drug Delivery Systems; Bioengineering; Biophysics; Biomaterials; Drug Discovery3003 Pharmaceutical Science; Organic ChemistryTumor accumulationPolymersPharmaceutical SciencePharmacologyOptical imagingMiceDrug Delivery SystemsNanoparticleInternational Journal of NanomedicineDrug DiscoveryPolymerOriginal ResearchActive targeting; Optical imaging; Tumor accumulation; Animals; Antigens CD20; Cell Line Tumor; Humans; Leukemia B-Cell; Mice; Molecular Imaging; Nanoparticles; Polymers; Drug Delivery Systems; Biophysics; Bioengineering; Biomaterials; Organic Chemistry; Drug Discovery3003 Pharmaceutical ScienceTumorLeukemiaActive targetingtumor accumulationGeneral MedicineMolecular ImagingDrug deliverySystemic administrationPreclinical imagingHumanactive targetingMaterials scienceBiophysicsBioengineeringCell LineBiomaterialsoptical imagingR5-920In vivoCell Line TumormedicineLeukemia B-CellDistribution (pharmacology)AnimalsHumansCD20AntigensAnimalDrug Discovery3003 Pharmaceutical ScienceOrganic ChemistryB-CellCancermedicine.diseaseAntigens CD20BiomaterialTargeted drug deliveryBiophysicNanoparticlesMolecular imagingDrug Delivery System
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Subphthalocyanines: addressing water-solubility, nano-encapsulation, and activation for optical imaging of B16 melanoma cells

2014

Water-soluble disulfonato-subphthalocyanines (SubPcs) or hydrophobic nano-encapsulated SubPcs are efficient probes for the fluorescence imaging of cells. 20 nm large liposomes (TEM and DLS) incorporated about 13% SubPc. Moreover, some of these fluorophores were found to be pH activatable.

Models MolecularFluorescence-lifetime imaging microscopyNanostructureIndolesMelanoma ExperimentalIsoindoles010402 general chemistryPhotochemistryCrystallography X-Ray01 natural sciencesCatalysisMiceMaterials ChemistryMoleculeAnimals[CHIM]Chemical SciencesSolubilityFluorescent DyesLiposomeAqueous solutionMolecular Structure010405 organic chemistryChemistryMetals and AlloysWaterGeneral ChemistryHydrogen-Ion Concentration0104 chemical sciencesSurfaces Coatings and FilmsElectronic Optical and Magnetic MaterialsMolecular ImagingNanostructuresNano encapsulationSolubilityLiposomesCeramics and CompositesMolecular imaging
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Rapid hyperpolarization and purification of the metabolite fumarate in aqueous solution

2020

Significance Magnetic resonance imaging is hindered by inherently low sensitivity, which limits the method for the most part to observing water molecules in the body. Hyperpolarized molecules exhibit strongly enhanced MRI signals which opens the door for imaging low-concentration species in vivo. Biomolecules can be hyperpolarized and injected into a patient allowing for metabolism to be tracked in real time, greatly expanding the information available to the radiologist. Parahydrogen-induced polarization (PHIP) is a hyperpolarization method renowned for its low cost and accessibility, but is generally limited by low polarization levels, modest molecular concentrations, and contamination by…

Molar concentrationparahydrogen02 engineering and technologyBiosensing Techniques010402 general chemistry01 natural sciencesChemical reaction41003 medical and health sciences0302 clinical medicineFumaratesHyperpolarization (physics)Carbon-13 Magnetic Resonance SpectroscopyPolarization (electrochemistry)DissolutionhyperpolarizationBiomarker; Hyperpolarization; Metabolism; MRI; Parahydrogen; Fumarates; Molecular Imaging; Solutions; Water; Biosensing Techniques; Carbon-13 Magnetic Resonance Spectroscopychemistry.chemical_classificationParahydrogenMultidisciplinaryAqueous solutionChemistryBiomolecule500WaterBiomarker021001 nanoscience & nanotechnologyCombinatorial chemistryMolecular Imaging0104 chemical sciencesSolutionsSolventChemistryHyperpolarizationMetabolism030220 oncology & carcinogenesisReagentPhysical Sciencesbiomarkerddc:5000210 nano-technologymetabolismBiosensorMRI
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Gadolinium-chelating nanogels as MR contrast agents specifically targeting tumor cells

2014

Aims and objectives Methods and materials Results Conclusion Personal information References

Molecular imaging Diagnostic procedure MR-Functional imaging MR Contrast agentsMolecular genomics and proteomicsgenetic structuresMolecular imagingMRDiagnostic procedureContrast agentsMR-Functional imaging
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Development of functionalizable azaBODIPYs for the conception of theranostic agents and bimodal probes for imaging uses

2020

The in vivo use of optical imaging is still limited by the lack of near infrared emitting probes. This thesis work focuses on the optimization and valorization of a water-soluble fluorescent platform whose optical properties enable an in vivo use. Two distinct applications were investigated for this WazaBY (Water-soluble azaBODIPY) platform: use as a PET (or SPECT) / optical bimodal probe, and as a theranostic agent. Concerning the first project, we were able to develop a targetted SPECT/optical bimodal probe, which was radiometallated with indium 111. Using xenografted murine models, we were able to show a clear accumulation of the probe in the tumor 24 hours after injection. Moreover, the…

Near infrared fluorescenceAzaBODIPYImagerie moléculaireMolecular imagingMedical imagingFluorophoreBimodality probeSonde bimodale[CHIM.ORGA] Chemical Sciences/Organic chemistryImagerie médicaleFluorescence proche infrarouge
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Molecular in vivo imaging of gastric cancer in a human-murine xenograft model: targeting epidermal growth factor receptor

2012

Background The prognosis of gastric cancer depends on early diagnosis. Targeted therapies against epidermal growth factor receptors (EGFRs) are currently emerging for the treatment of gastric cancer. Objective To specifically visualize gastric cancer by using monoclonal antibodies targeting EGFR1 as molecular probes for in vivo molecular confocal laser endomicroscopy (mCLE) in a human-murine xenograft model. Design Prospective in vivo animal study. Setting Animal laboratory. Interventions Human gastric carcinoma xenografts were examined in 26 nude mice by using mCLE after injection of fluorescently labeled antibodies. Nine mice received low-dose anti-EGFR1 antibodies, 7 mice cetuximab, and …

Pathologymedicine.medical_specialtymedicine.drug_classCetuximabMice NudeAntineoplastic AgentsAntibodies Monoclonal HumanizedMonoclonal antibodyAntibodiesMiceStomach NeoplasmsEpidermal growth factorIn vivomedicineAnimalsHumansRadiology Nuclear Medicine and imagingEpidermal growth factor receptorFluorescent DyesMicroscopy ConfocalbiologyCetuximabbusiness.industryCarcinomaGastroenterologyAntibodies MonoclonalCancerFlow Cytometrymedicine.diseaseMolecular ImagingErbB ReceptorsDisease Models Animalbiology.proteinImmunohistochemistrybusinessPreclinical imagingmedicine.drugGastrointestinal Endoscopy
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Approaching ‘kit-type’ labelling with 68Ga : the DATA chelators.

2015

The DATA chelators are a novel class of tri-anionic ligands based on 6-amino-1,4-diazepine-triacetic acid, which have been introduced recently for the chelation of (68)Ga. Compared with macrocyclic chelators based on the cyclen scaffold (i.e., DOTA, DO3A, and DO2A derivatives), DATA chelators undergo quantitative radiolabelling more rapidly and under milder conditions. In this study, a systematic evaluation of the labelling of four DATA chelators--DATA(M), DATA(P), DATA(Ph), and DATA(PPh)--with (68)Ga is presented. The results highlight the extraordinary potential of this new class of chelators for application in molecular imaging using (68)Ga positron emission tomography (PET).

PharmacologyStereochemistryRadiopharmaceuticals.Organic ChemistryGallium-68Gallium RadioisotopesBiochemistryLigand designchemistry.chemical_compoundKineticsMacrocyclic ligandsCyclenchemistryLabellingIsotope LabelingDrug DiscoveryChelatesMolecular MedicineDOTAChelationGeneral Pharmacology Toxicology and PharmaceuticsMolecular imagingChelating Agents
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NODAPA-OH and NODAPA-(NCS)n: Synthesis, 68Ga-radiolabelling and in vitro characterisation of novel versatile bifunctional chelators for molecular ima…

2008

This report concerns synthesis, (68)Ga-radiolabelling and stability data of 1,4,7-triazacyclononane-1,4-diacetic acid-7-p-isothio-cyanatophenyl-acetic acid (NODAPA-NCS), 1,4,7-triazacyclononane-1-acetic acid-4,7-di-p-isothiocyanatophenyl-acetic acid (NODAPA-(NCS)(2)) and 1,4,7-triazacyclononane-1,4-diacetic acid-7-p-hydroxyphenyl-acetic acid (NODAPA-OH), versatile bifunctional chelators with potential for molecular imaging. Protein binding and exemplified conjugation are also reported.

PhenylacetatesStereochemistryChemistry PharmaceuticalClinical BiochemistryLysinePharmaceutical ScienceGallium RadioisotopesIn Vitro TechniquesBiochemistryChemical synthesisHeterocyclic Compounds 1-Ringchemistry.chemical_compoundHeterocyclic CompoundsDrug DiscoveryChelationBifunctionalMolecular BiologyChelating AgentsPhenylacetatesRadioisotopesOrganic ChemistryHydrogen-Ion ConcentrationModels ChemicalchemistryAminosugarDrug DesignIsotope LabelingPositron-Emission TomographyMolecular MedicineChemical stabilityMolecular imagingBioorganic & Medicinal Chemistry Letters
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Molecular Imaging in the Regenerating Post Pneumonectomy Lung

2012

Pneumonectomymedicine.medical_specialtyLungmedicine.anatomical_structurebusiness.industrymedicine.medical_treatmentMedicineSurgeryRadiologyMolecular imagingbusinessJournal of Surgical Research
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Data for: Synthesis and evaluation of 89Zr-labeled and long-lived GLP-1 receptor agonists for PET imaging

2020

Appendix B. PET imaging 3D rendered images. 1. PET 3D of 4-89Zr 2. PET 3D of 5-89Zr

Positron Emission TomographyMolecular Imaging
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